| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| INSR | 3BU5A | P06213 | 1014 | 1310 | 1382.0 | ATP:60300 | ATPlike | Active | DFGin | 6.6591 | 13.9339 | BLAminus | -128.64, -166.6 | 44.54, 89.54 | -102.81, 23.91 | 295.82, 99.34 | -57.5, -34.18 | in-in | in | 8.2612 | Saltbr-in | 3.1304 | HRD-in | -68.86, -51.91 | 77.02, -10.33 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8444 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.0, 102.51 | APE9-dihe-in | -127.85, 151.44 | APE8-dihe-in | -79.76, 69.1 | APE8-rot-na | 32.47 | APE67-dihe-in | -66.77, -8.03 | -57.27, -41.89 | APE12-dist-na | 15.9367 | APE11-dist-na | 11.7238 | APE10-dist-na | 11.3004 | APE9-dist-in | 7.4014 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.1 | 0.196 | 0.239 | A | 306.0 | 294.0 | 3 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 3bu5 | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 4XLVA | P06213 | 1001 | 1310 | 1382.0 | ACP:61301 | ATPlike | Active | DFGin | 6.3572 | 13.4037 | BLAminus | -129.47, -169.61 | 59.33, 81.3 | -99.86, 10.75 | 301.2, 100.62 | -50.37, -35.15 | in-in | in | 8.1751 | Saltbr-in | 2.4413 | HRD-in | -74.09, -41.95 | 72.32, -7.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0293 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -31.8, 98.01 | APE9-dihe-in | -128.43, 131.43 | APE8-dihe-in | -62.62, 111.75 | APE8-rot-na | 18.22 | APE67-dihe-in | -71.49, -19.39 | -64.21, -23.54 | APE12-dist-na | 14.7406 | APE11-dist-na | 10.5509 | APE10-dist-na | 11.0271 | APE9-dist-in | 6.6146 | Y992F,C1008S | PTR999,PTR1185,PTR1189,PTR1190 | PTR999,PTR1185,PTR1189,PTR1190 | XRAY | 2.3 | 0.207 | 0.266 | A | 328.0 | 310.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4xlv | TYR_INSR_HUMAN | TYR | 1.7e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | AF-P06213-K1A | P06213 | 1015 | 1300 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.4423 | 13.5827 | BLAminus | -131.7, -172.45 | 45.37, 86.41 | -94.16, 16.44 | 302.88, 99.36 | -59.84, -31.96 | in-in | in | 8.2467 | Saltbr-in | 2.6737 | HRD-in | -73.51, -42.55 | 67.15, -19.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9665 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -58.18, 137.66 | APE9-dihe-in | -134.51, 139.18 | APE8-dihe-in | -78.44, 64.7 | APE8-rot-na | 35.42 | APE67-dihe-in | -75.31, -12.73 | -45.13, -39.55 | APE12-dist-na | 15.053 | APE11-dist-na | 10.9693 | APE10-dist-na | 10.1027 | APE9-dist-in | 7.0405 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 286.0 | 286.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | AF-P06213-K1 | TYR_INSR_HUMAN | TYR | 1.1e-96 | 329.0 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | AF-P06213-K3A | P06213 | 1015 | 1300 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 5.9245 | 13.0713 | BLAminus | -130.69, -170.6 | 46.9, 83.67 | -94.17, 11.86 | 307.8, 94.97 | -60.63, -30.18 | in-in | in | 8.0541 | Saltbr-in | 2.702 | HRD-in | -75.97, -44.42 | 67.04, -12.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9161 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -52.4, 144.11 | APE9-dihe-in | -144.36, 141.94 | APE8-dihe-in | -80.35, 60.58 | APE8-rot-na | 36.98 | APE67-dihe-in | -71.25, -11.2 | -43.91, -40.1 | APE12-dist-na | 15.2124 | APE11-dist-na | 11.3383 | APE10-dist-na | 9.8636 | APE9-dist-in | 6.7768 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 286.0 | 286.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | AF-P06213-K3 | TYR_INSR_HUMAN | TYR | 1.1e-96 | 329.0 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 1GAGA | P06213 | 1008 | 1310 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.4716 | 14.3547 | BLAminus | -139.79, -163.29 | 39.42, 88.74 | -105.4, 34.47 | 300.89, 100.42 | -68.02, -37.48 | in-in | in | 8.2108 | Saltbr-in | 3.0518 | HRD-in | -70.91, -47.43 | 72.33, -9.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8081 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.0, 110.5 | APE9-dihe-in | -118.5, 144.45 | APE8-dihe-in | -78.32, 65.87 | APE8-rot-na | 35.19 | APE67-dihe-in | -59.72, -1.72 | -33.26, -57.54 | APE12-dist-na | 15.007 | APE11-dist-na | 10.7529 | APE10-dist-na | 9.8952 | APE9-dist-in | 6.9259 | C1008S,Y1011F | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.7 | 0.214 | 0.269 | A | 306.0 | 303.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1gag | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 1RQQA | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.3041 | 13.6548 | BLAminus | -139.27, -172.16 | 50.78, 88.11 | -102.35, 26.03 | 306.58, 94.08 | -57.3, -43.84 | in-in | in | 7.8446 | Saltbr-in | 2.7395 | HRD-in | -71.1, -43.22 | 70.05, -11.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9269 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -79.1, 113.79 | APE9-dihe-in | -119.85, 145.04 | APE8-dihe-in | -81.27, 63.72 | APE8-rot-na | 35.79 | APE67-dihe-in | -62.06, -15.17 | -39.6, -48.57 | APE12-dist-na | 14.863 | APE11-dist-na | 10.6827 | APE10-dist-na | 9.7658 | APE9-dist-in | 6.8912 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.6 | 0.229 | 0.277 | A | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1rqq | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 1RQQB | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.4257 | 13.7866 | BLAminus | -137.51, -169.29 | 49.47, 88.05 | -100.38, 24.24 | 303.21, 103.09 | -57.34, -45.05 | in-in | in | 7.8496 | Saltbr-in | 3.2513 | HRD-in | -70.29, -44.51 | 70.11, -13.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.947 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.8, 112.61 | APE9-dihe-in | -120.76, 146.23 | APE8-dihe-in | -80.75, 64.53 | APE8-rot-na | 38.22 | APE67-dihe-in | -64.56, -12.7 | -44.47, -42.91 | APE12-dist-na | 14.8782 | APE11-dist-na | 10.7174 | APE10-dist-na | 9.7472 | APE9-dist-in | 6.8619 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.6 | 0.229 | 0.277 | B | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1rqq | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 2AUHA | P06213 | 1011 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.1405 | 13.65 | ABAminus | -136.58, -4.55 | -122.41, 138.22 | -136.1, 17.13 | 297.74, 110.36 | -54.48, -33.89 | in-in | in | 8.4039 | Saltbr-in | 2.705 | HRD-in | -71.8, -48.89 | 72.15, -21.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9571 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -107.66, 123.66 | APE9-dihe-in | -133.04, 151.36 | APE8-dihe-in | -70.19, 59.35 | APE8-rot-na | 32.97 | APE67-dihe-in | -65.61, -7.78 | -36.89, -48.67 | APE12-dist-na | 15.4002 | APE11-dist-na | 11.1462 | APE10-dist-na | 9.8774 | APE9-dist-in | 6.7568 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 3.2 | 0.223 | 0.254 | A | 306.0 | 300.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2auh | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 2B4SB | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.4787 | 13.8198 | ABAminus | -125.78, 6.45 | -136.21, 138.63 | -137.01, 36.1 | 305.43, 85.48 | -62.07, -22.25 | in-in | in | 8.0452 | Saltbr-in | 3.5864 | HRD-in | -75.2, -47.87 | 71.7, -18.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7912 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -84.64, 128.11 | APE9-dihe-in | -127.63, 149.14 | APE8-dihe-in | -79.25, 69.85 | APE8-rot-na | 37.38 | APE67-dihe-in | -66.83, -13.89 | -42.23, -45.27 | APE12-dist-na | 15.0347 | APE11-dist-na | 11.2888 | APE10-dist-na | 10.9363 | APE9-dist-in | 7.457 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.3 | 0.208 | 0.239 | B | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2b4s | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 2B4SD | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5924 | 14.0884 | ABAminus | -130.66, 15.42 | -144.64, 123.77 | -125.26, 40.8 | 306.28, 76.94 | -64.15, -16.22 | in-in | in | 7.9815 | Saltbr-in | 2.648 | HRD-in | -75.91, -45.41 | 68.78, -17.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8804 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.77, 132.95 | APE9-dihe-in | -133.75, 151.9 | APE8-dihe-in | -79.94, 78.72 | APE8-rot-na | 36.75 | APE67-dihe-in | -73.63, -5.75 | -50.54, -37.22 | APE12-dist-na | 14.815 | APE11-dist-na | 11.4645 | APE10-dist-na | 11.398 | APE9-dist-in | 7.4086 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.3 | 0.208 | 0.239 | D | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2b4s | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 3BU6A | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9823 | 14.0035 | ABAminus | -127.49, -6.05 | -146.78, 128.5 | -126.39, 29.26 | 301.19, 85.56 | -62.37, -9.3 | in-in | in | 8.2511 | Saltbr-in | 3.5603 | HRD-in | -76.09, -48.83 | 72.52, -10.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8848 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.83, 102.44 | APE9-dihe-in | -128.25, 150.85 | APE8-dihe-in | -77.03, 62.98 | APE8-rot-na | 32.44 | APE67-dihe-in | -72.83, -9.55 | -48.55, -39.5 | APE12-dist-na | 16.1225 | APE11-dist-na | 12.0764 | APE10-dist-na | 11.7461 | APE9-dist-in | 7.7403 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 1.95 | 0.202 | 0.239 | A | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 3bu6 | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 1IR3A | P06213 | 1008 | 1310 | 1382.0 | ANP:60300 | ATPlike | Inactive | DFGin | 6.1283 | 14.366 | BLAminus | -133.72, -168.17 | 47.48, 85.02 | -100.33, 24.62 | 303.32, 104.39 | -58.78, -39.74 | in-out | in | 8.9234 | Saltbr-out | 4.3926 | HRD-in | -68.06, -49.87 | 71.52, -7.17 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9018 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.98, 116.19 | APE9-dihe-in | -117.81, 138.98 | APE8-dihe-in | -77.82, 71.42 | APE8-rot-na | 34.55 | APE67-dihe-in | -66.85, -13.55 | -40.74, -47.32 | APE12-dist-na | 14.5115 | APE11-dist-na | 10.4265 | APE10-dist-na | 9.7642 | APE9-dist-in | 6.771 | C1008S,Y1011F | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 1.9 | 0.194 | 0.226 | A | 306.0 | 303.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1ir3 | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 3BU3A | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8314 | 14.3175 | BLAminus | -125.34, -173.11 | 49.37, 91.34 | -105.76, 28.79 | 293.31, 96.09 | -61.52, -23.48 | in-out | in | 8.3343 | Saltbr-out | 3.6427 | HRD-in | -77.13, -47.35 | 74.01, -9.17 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8876 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -87.87, 102.94 | APE9-dihe-in | -129.84, 150.89 | APE8-dihe-in | -79.69, 65.67 | APE8-rot-na | 33.39 | APE67-dihe-in | -69.85, -9.41 | -51.56, -40.22 | APE12-dist-na | 15.8144 | APE11-dist-na | 11.5839 | APE10-dist-na | 11.082 | APE9-dist-in | 7.3699 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 1.65 | 0.203 | 0.22 | A | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 3bu3 | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 2Z8CA | P06213 | 1011 | 1310 | 1382.0 | S91:60001 | Type1 | Inactive | DFGin | 6.401 | 12.923 | BLAminus | -126.28, -180.0 | 45.53, 101.6 | -113.26, 32.07 | 305.0, 102.45 | -55.7, -35.78 | in-out | in | 7.4783 | Saltbr-out | 3.6266 | HRD-in | -88.34, -29.28 | 53.1, 14.66 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8483 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -65.92, 127.58 | APE9-dihe-in | -136.04, 148.74 | APE8-dihe-in | -92.61, 86.13 | APE8-rot-na | 40.99 | APE67-dihe-in | -57.55, -15.17 | -59.74, -44.88 | APE12-dist-na | 14.522 | APE11-dist-na | 10.6018 | APE10-dist-na | 9.7643 | APE9-dist-in | 6.8834 | C1008S,Y1011F | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 3.25 | 0.217 | 0.292 | A | 303.0 | 300.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2z8c | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 1I44A | P06213 | 1013 | 1310 | 1382.0 | ACP:60300 | ATPlike | Inactive | DFGin | 6.6413 | 13.7197 | None | -58.16, -57.88 | -145.23, -170.38 | -78.54, 6.88 | 58.45, 76.71 | 123.48, 176.59 | in-out | in | 9.122 | Saltbr-out | 5.8952 | HRD-in | -61.91, -52.97 | 77.04, -9.75 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -75.06 | APE8-dihe-out | -68.29, 48.19 | APE8-rot-na | 34.45 | APE67-dihe-in | -67.23, -7.11 | -39.74, -51.28 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.6829 | C1008S,Y1011F,D1188A | None | None | XRAY | 2.4 | 0.21 | 0.268 | A | 306.0 | 282.0 | 16 | 30 | 14 | 16 | [[1023, 1292]] | 1.0 | 1i44 | TYR_INSR_HUMAN | TYR | 3.4e-96 | 327.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 1P14A | P06213 | 1005 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 7.6107 | 15.3442 | None | -93.61, -127.04 | -78.93, 153.19 | -166.81, 155.93 | 65.2, 94.97 | -69.26, 999.0 | in-out | in | 9.2508 | Saltbr-out | 5.4695 | HRD-in | -68.39, -55.7 | 74.95, -11.95 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 51.41 | APE8-rot-na | 37.98 | APE67-dihe-in | -68.35, -7.74 | -43.78, -43.88 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1008S,D1159N | None | None | XRAY | 1.9 | 0.225 | 0.24 | A | 306.0 | 287.0 | 19 | 30 | 11 | 19 | [[1023, 1292]] | 1.0 | 1p14 | TYR_INSR_HUMAN | TYR | 5e-96 | 326.9 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 4IBMA | P06213 | 1009 | 1309 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 5.6235 | 15.3135 | None | -76.0, 163.85 | -44.82, 128.63 | -69.67, 135.99 | 297.32, 165.57 | 60.17, 44.87 | out-out | out | 10.6453 | Saltbr-out | 7.271 | HRD-in | -68.74, -46.51 | 75.22, -15.25 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.6653 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.2, 121.44 | APE9-dihe-in | -109.91, 120.82 | APE8-dihe-in | -81.27, 70.1 | APE8-rot-na | 28.73 | APE67-dihe-in | -71.57, -11.47 | -57.01, -32.73 | APE12-dist-na | 18.7378 | APE11-dist-na | 15.2744 | APE10-dist-na | 11.5056 | APE9-dist-in | 7.3145 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | A | 306.0 | 301.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 4IBMB | P06213 | 1014 | 1310 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 6.943 | 16.4452 | None | -69.6, 155.55 | -45.67, 125.47 | -61.25, 129.45 | 282.72, 8.49 | 78.34, 8.83 | in-out | in | 9.4175 | Saltbr-out | 5.034 | HRD-in | -66.87, -50.14 | 74.82, -11.33 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.2219 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.04, 122.58 | APE9-dihe-in | -120.44, 134.35 | APE8-dihe-in | -81.79, 69.08 | APE8-rot-na | 32.76 | APE67-dihe-in | -70.68, -10.48 | -58.86, -32.74 | APE12-dist-na | 19.958 | APE11-dist-na | 16.3087 | APE10-dist-na | 12.6646 | APE9-dist-in | 7.3059 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | B | 306.0 | 294.0 | 3 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 5E1SA | P06213 | 1010 | 1310 | 1382.0 | 5JA:61301 | Type1 | Inactive | DFGin | 6.8652 | 15.0896 | None | -82.55, -126.51 | -82.76, 146.74 | -146.5, 173.12 | 61.91, 96.0 | -67.13, 97.4 | in-out | in | 8.8331 | Saltbr-out | 6.372 | HRD-in | -66.03, -52.34 | 70.18, -7.85 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 142.88 | APE8-dihe-in | -78.62, 65.27 | APE8-rot-na | 31.33 | APE67-dihe-in | -70.73, -11.27 | -48.96, -36.84 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.3247 | None | None | None | XRAY | 2.264 | 0.215 | 0.262 | A | 308.0 | 284.0 | 17 | 30 | 13 | 17 | [[1023, 1292]] | 1.0 | 5e1s | TYR_INSR_HUMAN | TYR | 5.6e-96 | 326.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 3EKKA | P06213 | 1007 | 1309 | 1382.0 | GS2:60001 | Type1 | Inactive | DFGin | 6.9318 | 15.2617 | None | -91.44, -126.11 | -77.81, 134.04 | -139.23, 999.0 | 58.35, 102.32 | 999.0, 999.0 | in-out | in | 9.2869 | Saltbr-out | 5.3303 | HRD-in | -69.72, -54.17 | 78.3, -13.96 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -25.52 | APE9-dihe-in | -83.53, 136.03 | APE8-dihe-in | -85.94, 70.21 | APE8-rot-na | 27.34 | APE67-dihe-in | -74.98, -12.32 | -58.97, -28.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.5248 | C1008S,D1159N | None | None | XRAY | 2.1 | 0.207 | 0.26 | A | 307.0 | 285.0 | 18 | 30 | 12 | 18 | [[1023, 1292]] | 1.0 | 3ekk | TYR_INSR_HUMAN | TYR | 5.1e-96 | 326.9 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 3EKNA | P06213 | 1011 | 1310 | 1382.0 | GS3:60001 | Type1 | Inactive | DFGin | 6.2472 | 13.3535 | None | -59.53, -41.76 | -156.68, -173.98 | -81.39, 6.66 | 55.61, 95.58 | 69.22, 37.13 | in-out | in | 8.4857 | Saltbr-out | 4.158 | HRD-in | -69.98, -55.95 | 75.05, -7.0 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.4799 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -63.36, -23.41 | APE9-dihe-in | -94.03, 128.42 | APE8-dihe-in | -84.32, 117.17 | APE8-rot-na | 4.91 | APE67-dihe-in | -79.33, -4.28 | -67.04, -22.99 | APE12-dist-na | 999.0 | APE11-dist-na | 13.7116 | APE10-dist-na | 9.2366 | APE9-dist-in | 4.8268 | C1008S,D1159N | None | None | XRAY | 2.2 | 0.214 | 0.274 | A | 307.0 | 297.0 | 3 | 30 | 27 | 3 | [[1023, 1292]] | 1.0 | 3ekn | TYR_INSR_HUMAN | TYR | 5.1e-96 | 326.9 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 5HHWA | P06213 | 1005 | 1310 | 1382.0 | 60O:1401 | Type1.5_Front | Inactive | DFGin | 6.5467 | 15.218 | None | -93.96, -126.86 | -75.33, 119.05 | -115.08, 17.9 | 55.03, 94.29 | -68.54, 168.98 | in-out | in | 9.6442 | Saltbr-out | 6.2026 | HRD-in | -63.14, -55.1 | 75.15, -13.24 | out-out-in | SNCooi | out-in | ActLoopNT-out | 12.985 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.8, 124.07 | APE9-dihe-in | -122.61, 132.0 | APE8-dihe-in | -80.76, 65.66 | APE8-rot-na | 27.91 | APE67-dihe-in | -68.74, -10.86 | -50.91, -39.07 | APE12-dist-na | 13.7099 | APE11-dist-na | 10.9449 | APE10-dist-na | 9.756 | APE9-dist-in | 7.5063 | C1008S,D1159N | None | None | XRAY | 1.79 | 0.172 | 0.198 | A | 307.0 | 306.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 5hhw | TYR_INSR_HUMAN | TYR | 5.5e-96 | 326.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 1IRKA | P06213 | 1008 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGout | 14.1104 | 8.254 | BBAminus | 170.32, 146.4 | -160.79, 149.25 | -78.89, -23.45 | 305.87, 140.64 | 112.61, 49.94 | in-out | in | 9.3136 | Saltbr-out | 5.9629 | HRD-in | -57.78, -53.43 | 77.45, -13.51 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.1823 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.89, 110.6 | APE9-dihe-in | -117.78, 141.32 | APE8-dihe-in | -78.03, 65.06 | APE8-rot-na | 33.68 | APE67-dihe-in | -72.48, -5.73 | -49.44, -39.24 | APE12-dist-na | 19.1925 | APE11-dist-na | 15.0441 | APE10-dist-na | 10.8154 | APE9-dist-in | 7.4582 | None | None | None | XRAY | 2.1 | 0.196 | 0.232 | A | 306.0 | 303.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1irk | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 3ETAA | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.7961 | 11.0134 | BBAminus | -132.13, -174.21 | -157.85, 103.42 | -76.03, -16.02 | 293.96, 86.44 | 92.76, -168.27 | in-in | in | 8.3215 | Saltbr-in | 2.7567 | HRD-in | -66.68, -47.32 | 76.44, -15.87 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8262 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -58.11, 133.17 | APE9-dihe-in | -138.51, 142.25 | APE8-dihe-in | -82.26, 68.13 | APE8-rot-na | 29.26 | APE67-dihe-in | -71.63, -9.4 | -61.34, -31.95 | APE12-dist-na | 14.3031 | APE11-dist-na | 10.2115 | APE10-dist-na | 6.0412 | APE9-dist-in | 7.1449 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | A | 317.0 | 293.0 | 1 | 30 | 29 | 1 | [[1023, 1292]] | 1.0 | 3eta | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 3ETAB | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.9171 | 11.1754 | BBAminus | -133.15, -176.66 | -152.04, 106.96 | -74.04, -41.1 | 283.79, 91.95 | 126.4, -175.96 | in-in | in | 8.351 | Saltbr-in | 3.1113 | HRD-in | -71.49, -47.77 | 78.43, -20.3 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8821 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.8, 131.91 | APE9-dihe-in | -139.37, 136.91 | APE8-dihe-in | -77.51, 68.63 | APE8-rot-na | 28.59 | APE67-dihe-in | -74.17, -10.01 | -54.55, -36.82 | APE12-dist-na | 14.3265 | APE11-dist-na | 10.1734 | APE10-dist-na | 5.8956 | APE9-dist-in | 7.247 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | B | 317.0 | 292.0 | 2 | 30 | 28 | 2 | [[1023, 1292]] | 1.0 | 3eta | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | 8DWNA | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -95.48, -147.03 | 167.35, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-out | in | 9.1838 | Saltbr-out | 6.0939 | HRD-in | -65.71, -54.25 | 86.56, -19.69 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.95, 141.67 | APE9-dihe-in | -121.95, 127.79 | APE8-dihe-in | -80.86, 78.35 | APE8-rot-na | 32.73 | APE67-dihe-in | -73.46, -9.67 | -56.68, -44.36 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.2005 | C1008S,Y1011F | PTR1185,PTR1189 | PTR1185,PTR1189 | XRAY | 2.15 | 0.195 | 0.247 | A | 306.0 | 286.0 | 11 | 30 | 19 | 11 | [[1023, 1292]] | 1.0 | 8dwn | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| INSR | INSR_HUMAN | 3BU5A | P06213 | 1014 | 1310 | 1382.0 | ATP:60300 | ATPlike | Active | DFGin | 6.6591 | 13.9339 | BLAminus | -128.64, -166.6 | 44.54, 89.54 | -102.81, 23.91 | 295.82, 99.34 | -57.5, -34.18 | in-in | in | 8.2612 | Saltbr-in | 3.1304 | HRD-in | -68.86, -51.91 | 77.02, -10.33 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8444 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.0, 102.51 | APE9-dihe-in | -127.85, 151.44 | APE8-dihe-in | -79.76, 69.1 | APE8-rot-na | 32.47 | APE67-dihe-in | -66.77, -8.03 | -57.27, -41.89 | APE12-dist-na | 15.9367 | APE11-dist-na | 11.7238 | APE10-dist-na | 11.3004 | APE9-dist-in | 7.4014 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.1 | 0.196 | 0.239 | A | 306.0 | 294.0 | 3 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 3bu5 | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 4XLVA | P06213 | 1001 | 1310 | 1382.0 | ACP:61301 | ATPlike | Active | DFGin | 6.3572 | 13.4037 | BLAminus | -129.47, -169.61 | 59.33, 81.3 | -99.86, 10.75 | 301.2, 100.62 | -50.37, -35.15 | in-in | in | 8.1751 | Saltbr-in | 2.4413 | HRD-in | -74.09, -41.95 | 72.32, -7.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0293 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -31.8, 98.01 | APE9-dihe-in | -128.43, 131.43 | APE8-dihe-in | -62.62, 111.75 | APE8-rot-na | 18.22 | APE67-dihe-in | -71.49, -19.39 | -64.21, -23.54 | APE12-dist-na | 14.7406 | APE11-dist-na | 10.5509 | APE10-dist-na | 11.0271 | APE9-dist-in | 6.6146 | Y992F,C1008S | PTR999,PTR1185,PTR1189,PTR1190 | PTR999,PTR1185,PTR1189,PTR1190 | XRAY | 2.3 | 0.207 | 0.266 | A | 328.0 | 310.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4xlv | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.7e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | AF-P06213-K1A | P06213 | 1015 | 1300 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.4423 | 13.5827 | BLAminus | -131.7, -172.45 | 45.37, 86.41 | -94.16, 16.44 | 302.88, 99.36 | -59.84, -31.96 | in-in | in | 8.2467 | Saltbr-in | 2.6737 | HRD-in | -73.51, -42.55 | 67.15, -19.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9665 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -58.18, 137.66 | APE9-dihe-in | -134.51, 139.18 | APE8-dihe-in | -78.44, 64.7 | APE8-rot-na | 35.42 | APE67-dihe-in | -75.31, -12.73 | -45.13, -39.55 | APE12-dist-na | 15.053 | APE11-dist-na | 10.9693 | APE10-dist-na | 10.1027 | APE9-dist-in | 7.0405 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 286.0 | 286.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | AF-P06213-K1 | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.1e-96 | 329.0 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | AF-P06213-K3A | P06213 | 1015 | 1300 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 5.9245 | 13.0713 | BLAminus | -130.69, -170.6 | 46.9, 83.67 | -94.17, 11.86 | 307.8, 94.97 | -60.63, -30.18 | in-in | in | 8.0541 | Saltbr-in | 2.702 | HRD-in | -75.97, -44.42 | 67.04, -12.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9161 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -52.4, 144.11 | APE9-dihe-in | -144.36, 141.94 | APE8-dihe-in | -80.35, 60.58 | APE8-rot-na | 36.98 | APE67-dihe-in | -71.25, -11.2 | -43.91, -40.1 | APE12-dist-na | 15.2124 | APE11-dist-na | 11.3383 | APE10-dist-na | 9.8636 | APE9-dist-in | 6.7768 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 286.0 | 286.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | AF-P06213-K3 | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.1e-96 | 329.0 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 1GAGA | P06213 | 1008 | 1310 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.4716 | 14.3547 | BLAminus | -139.79, -163.29 | 39.42, 88.74 | -105.4, 34.47 | 300.89, 100.42 | -68.02, -37.48 | in-in | in | 8.2108 | Saltbr-in | 3.0518 | HRD-in | -70.91, -47.43 | 72.33, -9.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8081 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.0, 110.5 | APE9-dihe-in | -118.5, 144.45 | APE8-dihe-in | -78.32, 65.87 | APE8-rot-na | 35.19 | APE67-dihe-in | -59.72, -1.72 | -33.26, -57.54 | APE12-dist-na | 15.007 | APE11-dist-na | 10.7529 | APE10-dist-na | 9.8952 | APE9-dist-in | 6.9259 | C1008S,Y1011F | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.7 | 0.214 | 0.269 | A | 306.0 | 303.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1gag | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 1RQQA | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.3041 | 13.6548 | BLAminus | -139.27, -172.16 | 50.78, 88.11 | -102.35, 26.03 | 306.58, 94.08 | -57.3, -43.84 | in-in | in | 7.8446 | Saltbr-in | 2.7395 | HRD-in | -71.1, -43.22 | 70.05, -11.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9269 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -79.1, 113.79 | APE9-dihe-in | -119.85, 145.04 | APE8-dihe-in | -81.27, 63.72 | APE8-rot-na | 35.79 | APE67-dihe-in | -62.06, -15.17 | -39.6, -48.57 | APE12-dist-na | 14.863 | APE11-dist-na | 10.6827 | APE10-dist-na | 9.7658 | APE9-dist-in | 6.8912 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.6 | 0.229 | 0.277 | A | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1rqq | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 1RQQB | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Active | DFGin | 6.4257 | 13.7866 | BLAminus | -137.51, -169.29 | 49.47, 88.05 | -100.38, 24.24 | 303.21, 103.09 | -57.34, -45.05 | in-in | in | 7.8496 | Saltbr-in | 3.2513 | HRD-in | -70.29, -44.51 | 70.11, -13.29 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.947 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.8, 112.61 | APE9-dihe-in | -120.76, 146.23 | APE8-dihe-in | -80.75, 64.53 | APE8-rot-na | 38.22 | APE67-dihe-in | -64.56, -12.7 | -44.47, -42.91 | APE12-dist-na | 14.8782 | APE11-dist-na | 10.7174 | APE10-dist-na | 9.7472 | APE9-dist-in | 6.8619 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.6 | 0.229 | 0.277 | B | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1rqq | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 2AUHA | P06213 | 1011 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.1405 | 13.65 | ABAminus | -136.58, -4.55 | -122.41, 138.22 | -136.1, 17.13 | 297.74, 110.36 | -54.48, -33.89 | in-in | in | 8.4039 | Saltbr-in | 2.705 | HRD-in | -71.8, -48.89 | 72.15, -21.21 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9571 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -107.66, 123.66 | APE9-dihe-in | -133.04, 151.36 | APE8-dihe-in | -70.19, 59.35 | APE8-rot-na | 32.97 | APE67-dihe-in | -65.61, -7.78 | -36.89, -48.67 | APE12-dist-na | 15.4002 | APE11-dist-na | 11.1462 | APE10-dist-na | 9.8774 | APE9-dist-in | 6.7568 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 3.2 | 0.223 | 0.254 | A | 306.0 | 300.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2auh | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 2B4SB | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.4787 | 13.8198 | ABAminus | -125.78, 6.45 | -136.21, 138.63 | -137.01, 36.1 | 305.43, 85.48 | -62.07, -22.25 | in-in | in | 8.0452 | Saltbr-in | 3.5864 | HRD-in | -75.2, -47.87 | 71.7, -18.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7912 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -84.64, 128.11 | APE9-dihe-in | -127.63, 149.14 | APE8-dihe-in | -79.25, 69.85 | APE8-rot-na | 37.38 | APE67-dihe-in | -66.83, -13.89 | -42.23, -45.27 | APE12-dist-na | 15.0347 | APE11-dist-na | 11.2888 | APE10-dist-na | 10.9363 | APE9-dist-in | 7.457 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.3 | 0.208 | 0.239 | B | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2b4s | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 2B4SD | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5924 | 14.0884 | ABAminus | -130.66, 15.42 | -144.64, 123.77 | -125.26, 40.8 | 306.28, 76.94 | -64.15, -16.22 | in-in | in | 7.9815 | Saltbr-in | 2.648 | HRD-in | -75.91, -45.41 | 68.78, -17.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8804 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.77, 132.95 | APE9-dihe-in | -133.75, 151.9 | APE8-dihe-in | -79.94, 78.72 | APE8-rot-na | 36.75 | APE67-dihe-in | -73.63, -5.75 | -50.54, -37.22 | APE12-dist-na | 14.815 | APE11-dist-na | 11.4645 | APE10-dist-na | 11.398 | APE9-dist-in | 7.4086 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 2.3 | 0.208 | 0.239 | D | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2b4s | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 3BU6A | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.9823 | 14.0035 | ABAminus | -127.49, -6.05 | -146.78, 128.5 | -126.39, 29.26 | 301.19, 85.56 | -62.37, -9.3 | in-in | in | 8.2511 | Saltbr-in | 3.5603 | HRD-in | -76.09, -48.83 | 72.52, -10.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8848 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.83, 102.44 | APE9-dihe-in | -128.25, 150.85 | APE8-dihe-in | -77.03, 62.98 | APE8-rot-na | 32.44 | APE67-dihe-in | -72.83, -9.55 | -48.55, -39.5 | APE12-dist-na | 16.1225 | APE11-dist-na | 12.0764 | APE10-dist-na | 11.7461 | APE9-dist-in | 7.7403 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 1.95 | 0.202 | 0.239 | A | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 3bu6 | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 1IR3A | P06213 | 1008 | 1310 | 1382.0 | ANP:60300 | ATPlike | Inactive | DFGin | 6.1283 | 14.366 | BLAminus | -133.72, -168.17 | 47.48, 85.02 | -100.33, 24.62 | 303.32, 104.39 | -58.78, -39.74 | in-out | in | 8.9234 | Saltbr-out | 4.3926 | HRD-in | -68.06, -49.87 | 71.52, -7.17 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.9018 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.98, 116.19 | APE9-dihe-in | -117.81, 138.98 | APE8-dihe-in | -77.82, 71.42 | APE8-rot-na | 34.55 | APE67-dihe-in | -66.85, -13.55 | -40.74, -47.32 | APE12-dist-na | 14.5115 | APE11-dist-na | 10.4265 | APE10-dist-na | 9.7642 | APE9-dist-in | 6.771 | C1008S,Y1011F | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 1.9 | 0.194 | 0.226 | A | 306.0 | 303.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1ir3 | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 3BU3A | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8314 | 14.3175 | BLAminus | -125.34, -173.11 | 49.37, 91.34 | -105.76, 28.79 | 293.31, 96.09 | -61.52, -23.48 | in-out | in | 8.3343 | Saltbr-out | 3.6427 | HRD-in | -77.13, -47.35 | 74.01, -9.17 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8876 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -87.87, 102.94 | APE9-dihe-in | -129.84, 150.89 | APE8-dihe-in | -79.69, 65.67 | APE8-rot-na | 33.39 | APE67-dihe-in | -69.85, -9.41 | -51.56, -40.22 | APE12-dist-na | 15.8144 | APE11-dist-na | 11.5839 | APE10-dist-na | 11.082 | APE9-dist-in | 7.3699 | C1008S | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 1.65 | 0.203 | 0.22 | A | 306.0 | 297.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 3bu3 | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 2Z8CA | P06213 | 1011 | 1310 | 1382.0 | S91:60001 | Type1 | Inactive | DFGin | 6.401 | 12.923 | BLAminus | -126.28, -180.0 | 45.53, 101.6 | -113.26, 32.07 | 305.0, 102.45 | -55.7, -35.78 | in-out | in | 7.4783 | Saltbr-out | 3.6266 | HRD-in | -88.34, -29.28 | 53.1, 14.66 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8483 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -65.92, 127.58 | APE9-dihe-in | -136.04, 148.74 | APE8-dihe-in | -92.61, 86.13 | APE8-rot-na | 40.99 | APE67-dihe-in | -57.55, -15.17 | -59.74, -44.88 | APE12-dist-na | 14.522 | APE11-dist-na | 10.6018 | APE10-dist-na | 9.7643 | APE9-dist-in | 6.8834 | C1008S,Y1011F | PTR1185,PTR1189,PTR1190 | PTR1185,PTR1189,PTR1190 | XRAY | 3.25 | 0.217 | 0.292 | A | 303.0 | 300.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 2z8c | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 1I44A | P06213 | 1013 | 1310 | 1382.0 | ACP:60300 | ATPlike | Inactive | DFGin | 6.6413 | 13.7197 | None | -58.16, -57.88 | -145.23, -170.38 | -78.54, 6.88 | 58.45, 76.71 | 123.48, 176.59 | in-out | in | 9.122 | Saltbr-out | 5.8952 | HRD-in | -61.91, -52.97 | 77.04, -9.75 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -75.06 | APE8-dihe-out | -68.29, 48.19 | APE8-rot-na | 34.45 | APE67-dihe-in | -67.23, -7.11 | -39.74, -51.28 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.6829 | C1008S,Y1011F,D1188A | None | None | XRAY | 2.4 | 0.21 | 0.268 | A | 306.0 | 282.0 | 16 | 30 | 14 | 16 | [[1023, 1292]] | 1.0 | 1i44 | Homo sapiens | TYR_INSR_HUMAN | TYR | 3.4e-96 | 327.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 1P14A | P06213 | 1005 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGin | 7.6107 | 15.3442 | None | -93.61, -127.04 | -78.93, 153.19 | -166.81, 155.93 | 65.2, 94.97 | -69.26, 999.0 | in-out | in | 9.2508 | Saltbr-out | 5.4695 | HRD-in | -68.39, -55.7 | 74.95, -11.95 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 51.41 | APE8-rot-na | 37.98 | APE67-dihe-in | -68.35, -7.74 | -43.78, -43.88 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1008S,D1159N | None | None | XRAY | 1.9 | 0.225 | 0.24 | A | 306.0 | 287.0 | 19 | 30 | 11 | 19 | [[1023, 1292]] | 1.0 | 1p14 | Homo sapiens | TYR_INSR_HUMAN | TYR | 5e-96 | 326.9 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 4IBMA | P06213 | 1009 | 1309 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 5.6235 | 15.3135 | None | -76.0, 163.85 | -44.82, 128.63 | -69.67, 135.99 | 297.32, 165.57 | 60.17, 44.87 | out-out | out | 10.6453 | Saltbr-out | 7.271 | HRD-in | -68.74, -46.51 | 75.22, -15.25 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.6653 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.2, 121.44 | APE9-dihe-in | -109.91, 120.82 | APE8-dihe-in | -81.27, 70.1 | APE8-rot-na | 28.73 | APE67-dihe-in | -71.57, -11.47 | -57.01, -32.73 | APE12-dist-na | 18.7378 | APE11-dist-na | 15.2744 | APE10-dist-na | 11.5056 | APE9-dist-in | 7.3145 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | A | 306.0 | 301.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 4IBMB | P06213 | 1014 | 1310 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 6.943 | 16.4452 | None | -69.6, 155.55 | -45.67, 125.47 | -61.25, 129.45 | 282.72, 8.49 | 78.34, 8.83 | in-out | in | 9.4175 | Saltbr-out | 5.034 | HRD-in | -66.87, -50.14 | 74.82, -11.33 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.2219 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.04, 122.58 | APE9-dihe-in | -120.44, 134.35 | APE8-dihe-in | -81.79, 69.08 | APE8-rot-na | 32.76 | APE67-dihe-in | -70.68, -10.48 | -58.86, -32.74 | APE12-dist-na | 19.958 | APE11-dist-na | 16.3087 | APE10-dist-na | 12.6646 | APE9-dist-in | 7.3059 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | B | 306.0 | 294.0 | 3 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 5E1SA | P06213 | 1010 | 1310 | 1382.0 | 5JA:61301 | Type1 | Inactive | DFGin | 6.8652 | 15.0896 | None | -82.55, -126.51 | -82.76, 146.74 | -146.5, 173.12 | 61.91, 96.0 | -67.13, 97.4 | in-out | in | 8.8331 | Saltbr-out | 6.372 | HRD-in | -66.03, -52.34 | 70.18, -7.85 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 142.88 | APE8-dihe-in | -78.62, 65.27 | APE8-rot-na | 31.33 | APE67-dihe-in | -70.73, -11.27 | -48.96, -36.84 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.3247 | None | None | None | XRAY | 2.264 | 0.215 | 0.262 | A | 308.0 | 284.0 | 17 | 30 | 13 | 17 | [[1023, 1292]] | 1.0 | 5e1s | Homo sapiens | TYR_INSR_HUMAN | TYR | 5.6e-96 | 326.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 3EKKA | P06213 | 1007 | 1309 | 1382.0 | GS2:60001 | Type1 | Inactive | DFGin | 6.9318 | 15.2617 | None | -91.44, -126.11 | -77.81, 134.04 | -139.23, 999.0 | 58.35, 102.32 | 999.0, 999.0 | in-out | in | 9.2869 | Saltbr-out | 5.3303 | HRD-in | -69.72, -54.17 | 78.3, -13.96 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -25.52 | APE9-dihe-in | -83.53, 136.03 | APE8-dihe-in | -85.94, 70.21 | APE8-rot-na | 27.34 | APE67-dihe-in | -74.98, -12.32 | -58.97, -28.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.5248 | C1008S,D1159N | None | None | XRAY | 2.1 | 0.207 | 0.26 | A | 307.0 | 285.0 | 18 | 30 | 12 | 18 | [[1023, 1292]] | 1.0 | 3ekk | Homo sapiens | TYR_INSR_HUMAN | TYR | 5.1e-96 | 326.9 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 3EKNA | P06213 | 1011 | 1310 | 1382.0 | GS3:60001 | Type1 | Inactive | DFGin | 6.2472 | 13.3535 | None | -59.53, -41.76 | -156.68, -173.98 | -81.39, 6.66 | 55.61, 95.58 | 69.22, 37.13 | in-out | in | 8.4857 | Saltbr-out | 4.158 | HRD-in | -69.98, -55.95 | 75.05, -7.0 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.4799 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -63.36, -23.41 | APE9-dihe-in | -94.03, 128.42 | APE8-dihe-in | -84.32, 117.17 | APE8-rot-na | 4.91 | APE67-dihe-in | -79.33, -4.28 | -67.04, -22.99 | APE12-dist-na | 999.0 | APE11-dist-na | 13.7116 | APE10-dist-na | 9.2366 | APE9-dist-in | 4.8268 | C1008S,D1159N | None | None | XRAY | 2.2 | 0.214 | 0.274 | A | 307.0 | 297.0 | 3 | 30 | 27 | 3 | [[1023, 1292]] | 1.0 | 3ekn | Homo sapiens | TYR_INSR_HUMAN | TYR | 5.1e-96 | 326.9 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 5HHWA | P06213 | 1005 | 1310 | 1382.0 | 60O:1401 | Type1.5_Front | Inactive | DFGin | 6.5467 | 15.218 | None | -93.96, -126.86 | -75.33, 119.05 | -115.08, 17.9 | 55.03, 94.29 | -68.54, 168.98 | in-out | in | 9.6442 | Saltbr-out | 6.2026 | HRD-in | -63.14, -55.1 | 75.15, -13.24 | out-out-in | SNCooi | out-in | ActLoopNT-out | 12.985 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.8, 124.07 | APE9-dihe-in | -122.61, 132.0 | APE8-dihe-in | -80.76, 65.66 | APE8-rot-na | 27.91 | APE67-dihe-in | -68.74, -10.86 | -50.91, -39.07 | APE12-dist-na | 13.7099 | APE11-dist-na | 10.9449 | APE10-dist-na | 9.756 | APE9-dist-in | 7.5063 | C1008S,D1159N | None | None | XRAY | 1.79 | 0.172 | 0.198 | A | 307.0 | 306.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 5hhw | Homo sapiens | TYR_INSR_HUMAN | TYR | 5.5e-96 | 326.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 1IRKA | P06213 | 1008 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | DFGout | 14.1104 | 8.254 | BBAminus | 170.32, 146.4 | -160.79, 149.25 | -78.89, -23.45 | 305.87, 140.64 | 112.61, 49.94 | in-out | in | 9.3136 | Saltbr-out | 5.9629 | HRD-in | -57.78, -53.43 | 77.45, -13.51 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.1823 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.89, 110.6 | APE9-dihe-in | -117.78, 141.32 | APE8-dihe-in | -78.03, 65.06 | APE8-rot-na | 33.68 | APE67-dihe-in | -72.48, -5.73 | -49.44, -39.24 | APE12-dist-na | 19.1925 | APE11-dist-na | 15.0441 | APE10-dist-na | 10.8154 | APE9-dist-in | 7.4582 | None | None | None | XRAY | 2.1 | 0.196 | 0.232 | A | 306.0 | 303.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 1irk | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 3ETAA | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.7961 | 11.0134 | BBAminus | -132.13, -174.21 | -157.85, 103.42 | -76.03, -16.02 | 293.96, 86.44 | 92.76, -168.27 | in-in | in | 8.3215 | Saltbr-in | 2.7567 | HRD-in | -66.68, -47.32 | 76.44, -15.87 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8262 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -58.11, 133.17 | APE9-dihe-in | -138.51, 142.25 | APE8-dihe-in | -82.26, 68.13 | APE8-rot-na | 29.26 | APE67-dihe-in | -71.63, -9.4 | -61.34, -31.95 | APE12-dist-na | 14.3031 | APE11-dist-na | 10.2115 | APE10-dist-na | 6.0412 | APE9-dist-in | 7.1449 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | A | 317.0 | 293.0 | 1 | 30 | 29 | 1 | [[1023, 1292]] | 1.0 | 3eta | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 3ETAB | P06213 | 1017 | 1310 | 1382.0 | 351:62001 | Type2 | Inactive | DFGout | 15.9171 | 11.1754 | BBAminus | -133.15, -176.66 | -152.04, 106.96 | -74.04, -41.1 | 283.79, 91.95 | 126.4, -175.96 | in-in | in | 8.351 | Saltbr-in | 3.1113 | HRD-in | -71.49, -47.77 | 78.43, -20.3 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.8821 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.8, 131.91 | APE9-dihe-in | -139.37, 136.91 | APE8-dihe-in | -77.51, 68.63 | APE8-rot-na | 28.59 | APE67-dihe-in | -74.17, -10.01 | -54.55, -36.82 | APE12-dist-na | 14.3265 | APE11-dist-na | 10.1734 | APE10-dist-na | 5.8956 | APE9-dist-in | 7.247 | None | None | None | XRAY | 2.6 | 0.203 | 0.232 | B | 317.0 | 292.0 | 2 | 30 | 28 | 2 | [[1023, 1292]] | 1.0 | 3eta | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.6e-96 | 328.5 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| INSR | INSR_HUMAN | 8DWNA | P06213 | 1014 | 1310 | 1382.0 | No_ligand | No_ligand | Inactive | None | 999.0 | 999.0 | None | -95.48, -147.03 | 167.35, 999.0 | 999.0, 999.0 | 999.0, 999.0 | 999.0, 999.0 | in-out | in | 9.1838 | Saltbr-out | 6.0939 | HRD-in | -65.71, -54.25 | 86.56, -19.69 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -74.95, 141.67 | APE9-dihe-in | -121.95, 127.79 | APE8-dihe-in | -80.86, 78.35 | APE8-rot-na | 32.73 | APE67-dihe-in | -73.46, -9.67 | -56.68, -44.36 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.2005 | C1008S,Y1011F | PTR1185,PTR1189 | PTR1185,PTR1189 | XRAY | 2.15 | 0.195 | 0.247 | A | 306.0 | 286.0 | 11 | 30 | 19 | 11 | [[1023, 1292]] | 1.0 | 8dwn | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.4e-96 | 328.7 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|