CMGC_GSK3B (Glycogen synthase kinase-3 beta)

Total number of chains: 188
Active chains: 153
Family: CMGC
Uniprot: GSK3B_HUMAN
Kinase Domain Residues: 56 - 340
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 185 98.4% AF-P49841-K1A
DFGin ABAminus 2 1.1% 6Y9SA
DFGin None 1 0.5% 8QJIA

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PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
4NM5A 24 383 420.0 ADP:60401 ATPlike Active DFGin 6.55 14.006 BLAminus -136.16, -177.73 61.88, 88.47 -108.64, 28.76 287.87, 80.78 -73.66, -15.44 in-in in 8.619 Saltbr-in 2.673 HRD-in -65.83, -43.73 64.82, 15.23 in-in-in SNCiii in-in ActLoopNT-in 2.839 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.92, 173.97 APE9-dihe-na 66.26, 147.02 APE8-dihe-in -77.1, 152.8 APE8-rot-in 293.28 APE67-dihe-inflip 82.03, -25.76 -52.23, 150.7 APE12-dist-in 13.279 APE11-dist-in 11.599 APE10-dist-in 6.949 APE9-dist-in 3.238 None None None XRAY 2.3 0.185 0.232 A 377 360 0 0 0 0 [[56, 340]] 1.0 4nm5 CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4NM7A 25 383 420.0 ADP:60401 ATPlike Active DFGin 6.515 13.993 BLAminus -137.35, -178.06 62.82, 88.6 -107.3, 24.56 288.41, 80.2 -69.84, -12.63 in-in in 8.818 Saltbr-in 2.743 HRD-in -66.5, -46.64 67.84, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.829 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 172.54 APE9-dihe-na 68.99, 153.43 APE8-dihe-in -86.9, 151.79 APE8-rot-in 300.04 APE67-dihe-inflip 84.67, -25.93 -50.38, 146.2 APE12-dist-in 13.355 APE11-dist-in 11.678 APE10-dist-in 6.905 APE9-dist-in 3.21 None None None XRAY 2.3 0.185 0.234 A 377 354 2 0 0 0 [[56, 340]] 1.0 4nm7 CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4NM3A 6 383 420.0 ADP:60409 ATPlike Active DFGin 6.475 13.947 BLAminus -129.98, -178.05 63.17, 87.87 -103.96, 21.26 289.38, 80.04 -65.46, -16.35 in-in in 8.806 Saltbr-in 2.726 HRD-in -69.81, -46.77 71.59, 6.75 in-in-in SNCiii in-in ActLoopNT-in 2.75 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.34, 169.99 APE9-dihe-na 69.15, 146.37 APE8-dihe-in -83.47, 151.55 APE8-rot-in 296.54 APE67-dihe-inflip 86.0, -31.11 -49.79, 146.79 APE12-dist-in 13.269 APE11-dist-in 11.484 APE10-dist-in 6.907 APE9-dist-in 3.112 None SEP9 SEP9 XRAY 2.1 0.197 0.242 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nm3 CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1J1BA 35 388 420.0 ANP:60430 ATPlike Active DFGin 6.767 13.788 BLAminus -136.8, -178.88 61.6, 83.12 -97.64, 25.1 286.09, 80.4 -68.7, -13.11 in-in in 8.566 Saltbr-in 2.59 HRD-in -71.16, -45.98 70.36, 3.88 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.52, 175.26 APE9-dihe-na 75.44, 133.64 APE8-dihe-in -75.76, 147.49 APE8-rot-in 306.57 APE67-dihe-inflip 98.15, -33.72 -56.43, 141.52 APE12-dist-in 13.056 APE11-dist-in 10.974 APE10-dist-in 5.893 APE9-dist-in 3.112 None None None XRAY 1.8 0.216 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1b CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1J1BB 23 386 420.0 ANP:60930 ATPlike Active DFGin 6.609 13.669 BLAminus -136.4, -177.03 61.49, 81.88 -98.08, 27.2 288.49, 82.07 -71.33, -13.14 in-in in 8.457 Saltbr-in 2.713 HRD-in -67.51, -45.87 68.87, 6.43 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.88, 174.17 APE9-dihe-na 76.18, 138.08 APE8-dihe-in -76.12, 141.41 APE8-rot-in 301.11 APE67-dihe-inflip 98.0, -37.59 -54.78, 144.25 APE12-dist-in 12.978 APE11-dist-in 11.066 APE10-dist-in 6.011 APE9-dist-in 3.174 None None None XRAY 1.8 0.216 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1b CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1J1CA 35 388 420.0 ADP:60430 ATPlike Active DFGin 6.812 13.93 BLAminus -139.24, -179.75 62.79, 82.17 -97.34, 25.19 286.68, 82.3 -65.83, -19.9 in-in in 8.601 Saltbr-in 2.647 HRD-in -68.65, -43.85 68.34, 7.36 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.05, 172.96 APE9-dihe-na 78.17, 130.85 APE8-dihe-in -73.54, 145.97 APE8-rot-in 310.16 APE67-dihe-inflip 99.09, -35.01 -54.43, 141.28 APE12-dist-in 13.077 APE11-dist-in 11.067 APE10-dist-in 5.926 APE9-dist-in 3.2 None None None XRAY 2.1 0.218 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1c CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1J1CB 23 386 420.0 ADP:60930 ATPlike Active DFGin 6.694 13.709 BLAminus -138.27, -179.99 63.33, 82.68 -100.46, 28.2 289.88, 80.26 -70.45, -13.94 in-in in 8.52 Saltbr-in 2.738 HRD-in -67.92, -43.36 67.59, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.71, 170.27 APE9-dihe-na 78.71, 139.86 APE8-dihe-in -81.56, 140.05 APE8-rot-in 302.5 APE67-dihe-inflip 101.62, -36.53 -50.52, 137.44 APE12-dist-in 12.868 APE11-dist-in 11.128 APE10-dist-in 6.025 APE9-dist-in 3.208 None None None XRAY 2.1 0.218 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1c CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8XN6A 35 384 420.0 ANP:501 ATPlike Active DFGin 6.682 13.862 BLAminus -137.72, 173.39 67.73, 84.48 -99.84, 22.57 287.77, 80.54 -65.33, -24.58 in-in in 8.463 Saltbr-in 2.63 HRD-in -71.05, -47.88 67.82, 15.5 in-in-in SNCiii in-in ActLoopNT-in 3.054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.0, 164.43 APE9-dihe-na 85.44, 135.36 APE8-dihe-in -74.2, 151.55 APE8-rot-in 291.81 APE67-dihe-in -69.28, -17.83 -36.59, -67.98 APE12-dist-in 12.907 APE11-dist-in 10.787 APE10-dist-in 5.68 APE9-dist-in 3.182 None None None XRAY 2.4 0.194 0.242 A 421 350 0 0 0 0 [[56, 340]] 1.0 8xn6 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1PYXA 35 386 420.0 ANP:1001 ATPlike Active DFGin 6.584 13.622 BLAminus -138.81, -178.07 65.18, 79.92 -98.83, 26.07 289.95, 78.27 -73.24, -7.6 in-in in 8.373 Saltbr-in 2.765 HRD-in -67.79, -47.84 71.28, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.12, 170.17 APE9-dihe-na 80.64, 129.74 APE8-dihe-in -63.79, 140.05 APE8-rot-in 299.48 APE67-dihe-in -56.43, -21.61 -20.65, -80.28 APE12-dist-in 12.903 APE11-dist-in 10.937 APE10-dist-in 5.784 APE9-dist-in 3.15 None None None XRAY 2.4 0.206 0.233 A 422 343 9 0 0 0 [[56, 340]] 1.0 1pyx CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1PYXB 35 383 420.0 ANP:2001 ATPlike Active DFGin 6.593 13.718 BLAminus -140.94, -178.47 65.26, 79.98 -98.11, 22.32 290.75, 76.51 -68.32, -7.73 in-in in 8.488 Saltbr-in 2.666 HRD-in -69.98, -47.18 70.83, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.3, 169.41 APE9-dihe-na 81.27, 131.24 APE8-dihe-in -66.67, 140.79 APE8-rot-in 300.74 APE67-dihe-in -56.9, -22.2 -20.58, -79.9 APE12-dist-in 12.838 APE11-dist-in 10.861 APE10-dist-in 5.718 APE9-dist-in 3.132 None None None XRAY 2.4 0.206 0.233 B 422 338 11 0 0 0 [[56, 340]] 1.0 1pyx CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
AF-P49841-K1A 48 348 420.0 No_ligand No_ligand Active DFGin 6.784 14.069 BLAminus -132.22, 178.4 62.95, 68.76 -81.18, 15.79 285.47, 79.99 -60.59, -34.48 in-in in 8.475 Saltbr-in 2.71 HRD-in -72.93, -43.95 66.08, 11.33 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.31, 173.16 APE9-dihe-na 65.7, 144.93 APE8-dihe-in -63.41, 136.54 APE8-rot-in 298.96 APE67-dihe-in -66.32, -15.33 -50.7, -49.59 APE12-dist-in 13.45 APE11-dist-in 11.989 APE10-dist-in 6.996 APE9-dist-in 3.127 None None None AF2 -1.0 1.0 1.0 A 301 301 0 0 0 0 [[56, 340]] 1.0 AF-P49841-K1 CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
AF-P49841-K3A 48 348 420.0 No_ligand No_ligand Active DFGin 6.524 13.884 BLAminus -137.65, -179.24 64.43, 60.31 -74.11, 11.79 288.76, 87.67 -59.53, -33.87 in-in in 8.232 Saltbr-in 2.675 HRD-in -76.11, -42.33 64.92, 19.4 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, -179.86 APE9-dihe-na 61.35, 145.02 APE8-dihe-in -62.21, 135.58 APE8-rot-in 295.17 APE67-dihe-in -63.79, -15.52 -52.47, -50.54 APE12-dist-in 13.486 APE11-dist-in 11.995 APE10-dist-in 7.07 APE9-dist-in 3.244 None None None AF2 -1.0 1.0 1.0 A 301 301 0 0 0 0 [[56, 340]] 1.0 AF-P49841-K3 CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2QA 35 383 420.0 No_ligand No_ligand Active DFGin 7.052 14.715 BLAminus -137.83, -179.15 61.41, 79.74 -96.27, 22.19 285.08, 78.46 -63.78, -22.81 in-in in 9.6 Saltbr-in 2.835 HRD-in -68.59, -45.76 72.18, 9.73 in-in-in SNCiii in-in ActLoopNT-in 2.932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.17, 171.92 APE9-dihe-na 79.53, 140.67 APE8-dihe-in -94.64, 154.44 APE8-rot-in 291.59 APE67-dihe-inflip 92.14, -26.46 -46.09, 133.9 APE12-dist-in 12.819 APE11-dist-in 10.688 APE10-dist-in 5.811 APE9-dist-in 3.156 None None None XRAY 1.68 0.174 0.202 A 359 349 0 0 0 0 [[56, 340]] 1.0 9x2q CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2QC 36 383 420.0 No_ligand No_ligand Active DFGin 7.21 15.088 BLAminus -133.92, -175.86 59.44, 76.77 -92.13, 23.3 281.6, 76.88 -64.8, -22.26 in-in in 9.585 Saltbr-in 2.881 HRD-in -73.13, -43.06 72.53, 6.24 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -80.09, 170.02 APE9-dihe-na 80.69, 143.27 APE8-dihe-in -98.08, 153.35 APE8-rot-in 292.56 APE67-dihe-inflip 91.66, -29.76 -46.15, 133.94 APE12-dist-in 12.831 APE11-dist-in 10.762 APE10-dist-in 5.787 APE9-dist-in 3.164 None None None XRAY 1.68 0.174 0.202 C 359 344 4 0 0 0 [[56, 340]] 1.0 9x2q CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2UA 35 382 420.0 No_ligand No_ligand Active DFGin 6.928 15.007 BLAminus -133.34, -178.44 58.79, 78.89 -95.7, 26.22 286.38, 80.77 -67.47, -21.14 in-in in 9.819 Saltbr-in 2.904 HRD-in -68.71, -46.18 69.43, 14.55 in-in-in SNCiii in-in ActLoopNT-in 2.926 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.25, 174.16 APE9-dihe-na 72.67, 147.17 APE8-dihe-in -96.66, 153.81 APE8-rot-in 303.03 APE67-dihe-inflip 89.84, -29.57 -56.61, 146.99 APE12-dist-in 12.872 APE11-dist-in 10.763 APE10-dist-in 6.052 APE9-dist-in 3.212 None None None XRAY 2.07 0.198 0.233 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2u CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2UB 35 382 420.0 No_ligand No_ligand Active DFGin 7.031 15.039 BLAminus -142.07, -178.25 60.15, 75.53 -94.78, 27.78 287.55, 76.1 -71.78, -16.86 in-in in 9.544 Saltbr-in 3.111 HRD-in -69.92, -46.99 71.31, 12.91 in-in-in SNCiii in-in ActLoopNT-in 2.857 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.99, 177.06 APE9-dihe-na 70.96, 140.3 APE8-dihe-in -91.49, 155.78 APE8-rot-in 299.08 APE67-dihe-inflip 86.39, -30.22 -56.97, 152.43 APE12-dist-in 12.801 APE11-dist-in 10.684 APE10-dist-in 6.083 APE9-dist-in 3.216 None None None XRAY 2.07 0.198 0.233 B 359 346 2 0 0 0 [[56, 340]] 1.0 9x2u CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2WA 35 382 420.0 No_ligand No_ligand Active DFGin 7.002 14.662 BLAminus -137.11, -172.55 57.37, 78.08 -92.78, 22.6 285.25, 77.53 -65.29, -22.08 in-in in 9.426 Saltbr-in 2.69 HRD-in -70.87, -42.87 69.61, 6.59 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.52, 174.16 APE9-dihe-na 78.0, 143.92 APE8-dihe-in -99.28, 152.84 APE8-rot-in 293.19 APE67-dihe-inflip 94.63, -26.01 -40.27, 130.65 APE12-dist-in 12.851 APE11-dist-in 10.695 APE10-dist-in 5.869 APE9-dist-in 3.149 None None None XRAY 1.92 0.179 0.209 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2w CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2WC 36 381 420.0 No_ligand No_ligand Active DFGin 7.232 15.121 BLAminus -131.33, -174.54 58.27, 79.41 -92.24, 20.59 282.51, 74.33 -64.49, -19.25 in-in in 9.502 Saltbr-in 2.925 HRD-in -70.18, -47.01 71.8, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.863 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.09, 172.17 APE9-dihe-na 81.56, 146.73 APE8-dihe-in -102.37, 154.39 APE8-rot-in 287.29 APE67-dihe-inflip 98.99, -30.15 -43.41, 127.27 APE12-dist-in 12.772 APE11-dist-in 10.661 APE10-dist-in 5.82 APE9-dist-in 3.147 None None None XRAY 1.92 0.179 0.209 C 359 343 3 0 0 0 [[56, 340]] 1.0 9x2w CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2XA 35 382 420.0 No_ligand No_ligand Active DFGin 7.096 14.802 BLAminus -134.71, -177.87 61.9, 80.09 -94.66, 24.51 284.3, 79.87 -70.56, -15.85 in-in in 9.585 Saltbr-in 2.845 HRD-in -72.18, -43.18 72.48, 8.24 in-in-in SNCiii in-in ActLoopNT-in 2.908 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.7, 174.99 APE9-dihe-na 74.21, 144.04 APE8-dihe-in -99.9, 155.52 APE8-rot-in 294.34 APE67-dihe-inflip 98.06, -28.28 -45.69, 131.32 APE12-dist-in 12.91 APE11-dist-in 10.817 APE10-dist-in 5.923 APE9-dist-in 3.137 None None None XRAY 1.79 0.178 0.207 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2x CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2XC 35 382 420.0 No_ligand No_ligand Active DFGin 7.055 15.211 BLAminus -133.52, -175.85 56.94, 77.42 -93.62, 21.48 281.91, 76.2 -62.69, -19.85 in-in in 9.611 Saltbr-in 2.837 HRD-in -74.39, -45.42 70.67, 10.42 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.32, 172.59 APE9-dihe-na 78.39, 148.01 APE8-dihe-in -102.94, 151.91 APE8-rot-in 298.64 APE67-dihe-inflip 95.53, -30.76 -39.02, 129.93 APE12-dist-in 12.904 APE11-dist-in 10.761 APE10-dist-in 5.918 APE9-dist-in 3.224 None None None XRAY 1.79 0.178 0.207 C 359 348 0 0 0 0 [[56, 340]] 1.0 9x2x CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2YA 35 382 420.0 No_ligand No_ligand Active DFGin 7.05 14.658 BLAminus -140.01, -179.57 60.44, 76.66 -91.5, 22.26 284.52, 79.37 -66.64, -18.87 in-in in 9.354 Saltbr-in 2.946 HRD-in -71.93, -44.87 72.02, 8.24 in-in-in SNCiii in-in ActLoopNT-in 2.972 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.33, 176.92 APE9-dihe-na 74.96, 144.91 APE8-dihe-in -97.18, 152.76 APE8-rot-in 297.41 APE67-dihe-inflip 94.26, -28.73 -49.99, 137.38 APE12-dist-in 12.914 APE11-dist-in 10.749 APE10-dist-in 5.852 APE9-dist-in 3.129 None None None XRAY 1.96 0.182 0.205 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2y CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2YB 37 382 420.0 No_ligand No_ligand Active DFGin 7.168 15.426 BLAminus -135.79, -176.64 57.44, 76.44 -90.64, 22.98 280.99, 76.17 -68.43, -15.63 in-in in 9.632 Saltbr-in 2.646 HRD-in -70.95, -47.52 72.95, 6.25 in-in-in SNCiii in-in ActLoopNT-in 2.831 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.29, 173.98 APE9-dihe-na 78.55, 143.82 APE8-dihe-in -97.73, 153.79 APE8-rot-in 303.29 APE67-dihe-inflip 99.44, -30.41 -47.09, 134.37 APE12-dist-in 12.869 APE11-dist-in 10.666 APE10-dist-in 5.798 APE9-dist-in 3.151 None None None XRAY 1.96 0.182 0.205 B 359 346 0 0 0 0 [[56, 340]] 1.0 9x2y CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1GNGA 36 385 420.0 No_ligand No_ligand Active DFGin 6.885 14.064 BLAminus -143.26, -176.0 52.72, 77.37 -90.17, 24.13 284.09, 64.37 -57.11, -28.67 in-in in 7.904 Saltbr-in 2.916 HRD-in -73.29, -39.28 60.06, 11.92 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.61, 159.4 APE9-dihe-na 81.31, 139.52 APE8-dihe-in -59.26, 125.44 APE8-rot-in 312.57 APE67-dihe-in -52.62, -25.58 -28.83, -64.47 APE12-dist-in 13.55 APE11-dist-in 11.957 APE10-dist-in 7.016 APE9-dist-in 3.111 None PTR216 PTR216 XRAY 2.6 0.196 0.262 A 378 350 0 0 0 0 [[56, 340]] 1.0 1gng CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1GNGB 28 384 420.0 No_ligand No_ligand Active DFGin 7.075 14.143 BLAminus -137.26, -174.12 57.41, 76.0 -92.3, 24.73 292.83, 74.1 -62.54, -16.26 in-in in 8.103 Saltbr-in 2.801 HRD-in -56.65, -46.78 67.13, 3.53 in-in-in SNCiii in-in ActLoopNT-in 3.053 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.46, 162.71 APE9-dihe-na 73.79, 160.3 APE8-dihe-in -71.09, 143.31 APE8-rot-in 306.45 APE67-dihe-in -62.51, -22.51 -44.24, -51.03 APE12-dist-in 13.461 APE11-dist-in 11.737 APE10-dist-in 7.233 APE9-dist-in 3.292 None PTR216 PTR216 XRAY 2.6 0.196 0.262 B 378 357 0 0 0 0 [[56, 340]] 1.0 1gng CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1H8FA 35 386 420.0 No_ligand No_ligand Active DFGin 7.005 14.467 BLAminus -132.29, -174.92 54.46, 76.42 -91.57, 20.83 287.85, 73.58 -61.47, -17.91 in-in in 8.812 Saltbr-in 2.63 HRD-in -65.88, -45.02 68.7, 5.89 in-in-in SNCiii in-in ActLoopNT-in 3.03 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.85, 172.29 APE9-dihe-na 81.77, 142.51 APE8-dihe-in -88.0, 149.96 APE8-rot-in 300.12 APE67-dihe-in -68.04, -14.11 -16.17, -79.65 APE12-dist-in 12.877 APE11-dist-in 10.874 APE10-dist-in 5.794 APE9-dist-in 3.089 None None None XRAY 2.8 0.22 0.256 A 352 352 0 0 0 0 [[56, 340]] 1.0 1h8f CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1H8FB 35 384 420.0 No_ligand No_ligand Active DFGin 7.053 14.488 BLAminus -137.11, -175.26 54.49, 79.79 -96.15, 19.99 284.33, 74.24 -61.84, -16.45 in-in in 8.784 Saltbr-in 2.631 HRD-in -65.99, -45.44 68.05, 7.58 in-in-in SNCiii in-in ActLoopNT-in 2.992 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.76, 172.7 APE9-dihe-na 81.11, 140.51 APE8-dihe-in -87.0, 149.5 APE8-rot-in 302.15 APE67-dihe-in -67.01, -11.3 -16.16, -82.04 APE12-dist-in 12.875 APE11-dist-in 10.843 APE10-dist-in 5.761 APE9-dist-in 3.101 None None None XRAY 2.8 0.22 0.256 B 352 350 0 0 0 0 [[56, 340]] 1.0 1h8f CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1I09A 25 384 420.0 No_ligand No_ligand Active DFGin 6.914 14.149 BLAminus -130.79, -175.77 55.31, 78.24 -94.52, 21.05 292.59, 69.56 -64.23, -6.99 in-in in 8.521 Saltbr-in 2.763 HRD-in -66.04, -49.2 76.06, -6.11 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.67, -13.88 APE9-dihe-na -95.25, 153.25 APE8-dihe-in -66.11, 146.74 APE8-rot-in 277.64 APE67-dihe-in -57.92, -5.44 -43.43, -74.88 APE12-dist-in 12.968 APE11-dist-in 11.16 APE10-dist-in 5.972 APE9-dist-in 3.334 None None None XRAY 2.7 0.242 0.274 A 420 338 22 0 0 0 [[56, 340]] 1.0 1i09 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U2ZA 35 382 420.0 L7C:401 Type1 Active DFGin 7.044 14.328 BLAminus -133.1, 179.76 62.32, 79.84 -96.99, 23.84 285.42, 79.62 -65.82, -25.41 in-in in 8.558 Saltbr-in 2.764 HRD-in -73.49, -48.13 70.69, 16.81 in-in-in SNCiii in-in ActLoopNT-in 2.907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.38, 169.05 APE9-dihe-na 81.0, 139.13 APE8-dihe-in -79.34, 150.41 APE8-rot-in 288.38 APE67-dihe-inflip 98.4, -32.71 -58.44, 134.12 APE12-dist-in 13.138 APE11-dist-in 11.05 APE10-dist-in 5.888 APE9-dist-in 3.092 None None None XRAY 2.21 0.248 0.266 A 348 345 3 0 0 0 [[56, 340]] 1.0 7u2z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U2ZB 35 382 420.0 L7C:401 Type1 Active DFGin 7.083 14.316 BLAminus -133.0, 179.81 61.72, 80.12 -97.27, 23.94 285.32, 79.23 -65.78, -25.41 in-in in 8.516 Saltbr-in 2.765 HRD-in -73.41, -48.27 70.6, 17.33 in-in-in SNCiii in-in ActLoopNT-in 2.912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.19, 168.84 APE9-dihe-na 80.53, 139.96 APE8-dihe-in -79.72, 154.04 APE8-rot-in 288.98 APE67-dihe-in -82.66, -15.29 -42.95, -55.79 APE12-dist-in 13.132 APE11-dist-in 11.082 APE10-dist-in 5.892 APE9-dist-in 3.099 None None None XRAY 2.21 0.248 0.266 B 348 348 0 0 0 0 [[56, 340]] 1.0 7u2z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3F7ZB 35 383 420.0 34O:63000 Type1 Active DFGin 7.022 13.878 BLAminus -136.68, -179.55 57.9, 84.9 -98.68, 23.48 283.23, 74.81 -68.95, -21.14 in-in in 8.424 Saltbr-in 2.704 HRD-in -69.78, -45.02 65.34, 14.6 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.88, 179.92 APE9-dihe-na 68.48, 153.11 APE8-dihe-in -69.08, 139.27 APE8-rot-in 289.99 APE67-dihe-in -60.9, -22.52 -35.36, -58.5 APE12-dist-in 13.646 APE11-dist-in 11.954 APE10-dist-in 6.778 APE9-dist-in 3.248 None PTR216 PTR216 XRAY 2.4 0.206 0.253 B 350 339 10 0 0 0 [[56, 340]] 1.0 3f7z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3SD0B 35 383 420.0 TSK:400 Type1 Active DFGin 7.188 14.024 BLAminus -142.24, -171.3 46.91, 83.25 -91.85, 32.36 285.89, 73.19 -82.63, -8.9 in-in in 8.235 Saltbr-in 2.887 HRD-in -76.13, -44.58 70.79, 3.58 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.6, 179.93 APE9-dihe-na 74.21, 152.1 APE8-dihe-in -107.68, 155.88 APE8-rot-in 296.61 APE67-dihe-in -78.55, -3.01 -13.04, -81.61 APE12-dist-in 13.018 APE11-dist-in 11.099 APE10-dist-in 6.151 APE9-dist-in 3.156 None None None XRAY 2.7 0.179 0.254 B 350 349 0 0 0 0 [[56, 340]] 1.0 3sd0 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6HK3B 35 384 420.0 G8B:401 Type1 Active DFGin 6.788 13.641 BLAminus -137.2, -177.06 49.94, 95.88 -103.42, 19.32 279.02, 79.18 -69.5, -12.66 in-in in 8.168 Saltbr-in 2.602 HRD-in -82.47, -44.32 66.17, 21.49 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.65, -179.5 APE9-dihe-na 72.73, 150.58 APE8-dihe-in -63.57, 140.77 APE8-rot-in 271.9 APE67-dihe-in -55.77, -29.98 -51.2, -52.31 APE12-dist-in 13.408 APE11-dist-in 11.642 APE10-dist-in 6.365 APE9-dist-in 3.249 None PTR216 PTR216 XRAY 2.35 0.206 0.234 B 350 350 0 0 0 0 [[56, 340]] 1.0 6hk3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6HK4A 35 384 420.0 G8E:408 Type1 Active DFGin 6.928 13.508 BLAminus -141.9, -175.7 56.05, 83.18 -94.87, 22.99 284.64, 79.88 -61.73, -17.34 in-in in 8.371 Saltbr-in 2.656 HRD-in -76.65, -40.11 61.36, 16.95 in-in-in SNCiii in-in ActLoopNT-in 2.923 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.26, 167.76 APE9-dihe-na 63.34, 157.04 APE8-dihe-in -69.05, 135.63 APE8-rot-in 300.42 APE67-dihe-in -54.24, -34.87 -29.95, -58.61 APE12-dist-in 13.233 APE11-dist-in 11.745 APE10-dist-in 7.162 APE9-dist-in 3.192 None PTR216 PTR216 XRAY 2.5 0.212 0.249 A 350 350 0 0 0 0 [[56, 340]] 1.0 6hk4 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6HK4B 35 384 420.0 G8E:409 Type1 Active DFGin 6.943 13.541 BLAminus -140.37, -179.48 60.09, 87.67 -101.02, 22.8 284.5, 76.31 -75.88, -10.96 in-in in 8.208 Saltbr-in 2.506 HRD-in -82.4, -45.58 68.54, 13.94 in-in-in SNCiii in-in ActLoopNT-in 2.905 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.02, 172.84 APE9-dihe-na 63.46, 139.74 APE8-dihe-in -57.57, 136.79 APE8-rot-in 295.89 APE67-dihe-in -60.79, -29.87 -46.27, -47.23 APE12-dist-in 13.268 APE11-dist-in 11.678 APE10-dist-in 6.898 APE9-dist-in 3.074 None PTR216 PTR216 XRAY 2.5 0.212 0.249 B 350 350 0 0 0 0 [[56, 340]] 1.0 6hk4 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5F94A 36 381 420.0 3UO:401 Type1 Active DFGin 6.941 13.785 BLAminus -132.23, -171.99 59.12, 80.79 -95.82, 23.07 289.16, 72.98 -56.52, -34.28 in-in in 8.486 Saltbr-in 2.711 HRD-in -71.8, -46.49 68.5, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.784 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.99, 174.92 APE9-dihe-na 77.27, 148.67 APE8-dihe-in -101.45, 151.47 APE8-rot-in 289.94 APE67-dihe-inflip 89.58, -29.34 -36.24, 131.42 APE12-dist-in 12.915 APE11-dist-in 10.912 APE10-dist-in 5.952 APE9-dist-in 3.109 None None None XRAY 2.51 0.191 0.226 A 350 346 0 0 0 0 [[56, 340]] 1.0 5f94 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5F94B 37 385 420.0 3UO:401 Type1 Active DFGin 6.921 13.903 BLAminus -131.5, -174.71 60.13, 82.54 -97.18, 23.01 287.88, 72.62 -56.23, -35.38 in-in in 8.398 Saltbr-in 2.89 HRD-in -70.35, -45.36 66.02, 7.89 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.68, 174.32 APE9-dihe-na 79.06, 151.27 APE8-dihe-in -105.02, 147.7 APE8-rot-in 292.84 APE67-dihe-inflip 87.17, -28.31 -40.05, 137.25 APE12-dist-in 12.887 APE11-dist-in 10.901 APE10-dist-in 5.866 APE9-dist-in 3.193 None None None XRAY 2.51 0.191 0.226 B 350 349 0 0 0 0 [[56, 340]] 1.0 5f94 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5F95A 36 383 420.0 3UP:401 Type1 Active DFGin 6.851 14.121 BLAminus -131.03, -172.49 54.11, 85.8 -99.54, 23.42 287.04, 73.17 -58.21, -30.13 in-in in 8.492 Saltbr-in 2.642 HRD-in -68.05, -46.73 71.39, 6.88 in-in-in SNCiii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.52, 167.77 APE9-dihe-na 81.86, 152.62 APE8-dihe-in -108.33, 161.23 APE8-rot-in 296.59 APE67-dihe-in -81.75, 2.56 -4.13, -93.98 APE12-dist-in 13.1 APE11-dist-in 11.087 APE10-dist-in 6.378 APE9-dist-in 3.262 None None None XRAY 2.525 0.204 0.242 A 350 345 3 0 0 0 [[56, 340]] 1.0 5f95 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5F95B 36 385 420.0 3UP:401 Type1 Active DFGin 7.029 14.131 BLAminus -130.15, -170.55 52.93, 82.9 -96.95, 23.47 283.9, 71.07 -57.67, -29.42 in-in in 8.524 Saltbr-in 2.241 HRD-in -68.94, -45.23 69.65, 6.25 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.14, 169.18 APE9-dihe-na 82.46, 143.88 APE8-dihe-in -96.17, 168.5 APE8-rot-in 296.7 APE67-dihe-in -78.34, 2.06 -36.18, -73.12 APE12-dist-in 13.021 APE11-dist-in 11.027 APE10-dist-in 6.092 APE9-dist-in 3.21 None None None XRAY 2.525 0.204 0.242 B 350 338 12 0 0 0 [[56, 340]] 1.0 5f95 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U31A 36 385 420.0 L7I:402 Type1 Active DFGin 7.094 14.183 BLAminus -142.39, 178.42 62.99, 82.78 -98.0, 19.46 288.1, 81.67 -57.1, -32.73 in-in in 8.165 Saltbr-in 2.84 HRD-in -76.17, -49.99 76.15, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.54, -23.16 APE9-dihe-na -100.68, 154.06 APE8-dihe-in -79.73, 162.4 APE8-rot-in 294.75 APE67-dihe-in -75.9, -12.27 -44.4, -68.17 APE12-dist-in 13.102 APE11-dist-in 10.928 APE10-dist-in 5.909 APE9-dist-in 3.416 None None None XRAY 2.38 0.244 0.276 A 350 350 0 0 0 0 [[56, 340]] 1.0 7u31 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U31B 37 382 420.0 L7I:402 Type1 Active DFGin 7.049 14.287 BLAminus -143.88, 177.54 62.09, 82.63 -98.02, 19.8 287.95, 82.15 -57.33, -32.15 in-in in 8.377 Saltbr-in 2.717 HRD-in -76.73, -50.12 75.35, 8.49 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.33, 167.82 APE9-dihe-na 83.33, 132.28 APE8-dihe-in -83.68, 163.51 APE8-rot-in 292.75 APE67-dihe-in -76.54, -11.97 -40.44, -69.75 APE12-dist-in 13.108 APE11-dist-in 10.979 APE10-dist-in 5.927 APE9-dist-in 3.127 None None None XRAY 2.38 0.244 0.276 B 350 346 0 0 0 0 [[56, 340]] 1.0 7u31 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7SXJA 34 383 420.0 6VL:60401 Type1 Active DFGin 6.916 14.335 BLAminus -142.41, -179.99 59.67, 72.96 -86.59, 25.21 285.68, 73.81 -69.07, -21.65 in-in in 8.269 Saltbr-in 2.692 HRD-in -74.28, -41.7 68.05, 5.57 in-in-in SNCiii in-in ActLoopNT-in 2.943 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.32, 170.09 APE9-dihe-na 72.35, 148.74 APE8-dihe-in -71.51, 141.06 APE8-rot-in 303.21 APE67-dihe-in -59.11, -26.68 -51.44, -48.71 APE12-dist-in 13.503 APE11-dist-in 11.843 APE10-dist-in 7.042 APE9-dist-in 3.173 None PTR216 PTR216 XRAY 1.85 0.185 0.203 A 351 346 4 0 0 0 [[56, 340]] 1.0 7sxj CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7OY5A 35 385 420.0 39I:401 Type1 Active DFGin 6.926 14.033 BLAminus -126.76, 175.34 72.52, 92.63 -110.59, 33.29 286.05, 82.06 -75.35, -28.56 in-in in 8.688 Saltbr-in 2.936 HRD-in -72.48, -55.14 81.29, 7.92 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.43, 173.86 APE9-dihe-na 80.53, 146.3 APE8-dihe-in -94.81, 142.24 APE8-rot-in 295.61 APE67-dihe-inflip 101.01, -30.19 -44.76, 139.01 APE12-dist-in 12.924 APE11-dist-in 10.96 APE10-dist-in 5.893 APE9-dist-in 3.276 None None None XRAY 2.57 0.221 0.26 A 351 343 8 0 0 0 [[56, 340]] 1.0 7oy5 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7OY5B 35 383 420.0 39I:401 Type1 Active DFGin 7.115 14.145 BLAminus -131.55, -176.92 63.09, 57.6 -70.26, 11.8 285.25, 87.17 -66.04, -15.46 in-in in 8.495 Saltbr-in 3.027 HRD-in -75.85, -49.73 71.52, 4.36 in-in-in SNCiii in-in ActLoopNT-in 3.039 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.28, 172.83 APE9-dihe-na 79.24, 135.47 APE8-dihe-in -76.12, 154.7 APE8-rot-in 287.59 APE67-dihe-inflip 110.96, -34.61 -67.01, 135.0 APE12-dist-in 13.03 APE11-dist-in 10.958 APE10-dist-in 5.992 APE9-dist-in 3.008 None None None XRAY 2.57 0.221 0.26 B 351 344 5 0 0 0 [[56, 340]] 1.0 7oy5 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U33A 36 385 420.0 L7R:402 Type1 Active DFGin 7.023 14.049 BLAminus -140.49, 178.19 60.8, 84.54 -99.85, 16.49 288.62, 77.82 -50.41, -27.99 in-in in 8.511 Saltbr-in 2.774 HRD-in -71.53, -50.0 75.9, 8.27 in-in-in SNCiii in-in ActLoopNT-in 2.986 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.78, -39.59 APE9-dihe-na -85.32, 160.12 APE8-dihe-in -84.45, 147.1 APE8-rot-in 286.21 APE67-dihe-inflip 87.92, -34.06 -59.31, 147.18 APE12-dist-in 13.036 APE11-dist-in 10.991 APE10-dist-in 6.032 APE9-dist-in 3.262 None None None XRAY 2.6 0.233 0.264 A 351 350 0 0 0 0 [[56, 340]] 1.0 7u33 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U33B 37 382 420.0 L7R:402 Type1 Active DFGin 6.995 14.092 BLAminus -141.31, 178.2 60.97, 83.82 -100.06, 16.34 288.93, 78.7 -51.51, -27.59 in-in in 8.533 Saltbr-in 2.753 HRD-in -72.1, -49.87 75.78, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.62, 168.53 APE9-dihe-na 77.45, 140.58 APE8-dihe-in -89.54, 146.71 APE8-rot-in 285.53 APE67-dihe-in -82.12, -10.74 -0.24, -85.34 APE12-dist-in 13.035 APE11-dist-in 10.96 APE10-dist-in 6.029 APE9-dist-in 3.103 None None None XRAY 2.6 0.233 0.264 B 351 346 0 0 0 0 [[56, 340]] 1.0 7u33 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U36A 36 385 420.0 L7W:402 Type1 Active DFGin 7.055 14.057 BLAminus -140.39, -178.87 60.34, 89.59 -105.19, 18.12 284.52, 86.52 -57.6, -32.5 in-in in 8.453 Saltbr-in 3.019 HRD-in -77.18, -47.14 70.51, 17.98 in-in-in SNCiii in-in ActLoopNT-in 2.959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.43, -45.81 APE9-dihe-na -84.57, 153.41 APE8-dihe-in -68.83, 161.86 APE8-rot-in 280.03 APE67-dihe-in -82.26, -16.89 -53.14, -56.37 APE12-dist-in 12.87 APE11-dist-in 10.758 APE10-dist-in 5.812 APE9-dist-in 3.189 None None None XRAY 2.75 0.24 0.275 A 351 350 0 0 0 0 [[56, 340]] 1.0 7u36 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7U36B 37 382 420.0 L7W:402 Type1 Active DFGin 7.056 14.071 BLAminus -141.26, -179.45 60.58, 88.51 -105.71, 18.11 283.81, 87.44 -57.54, -31.03 in-in in 8.498 Saltbr-in 2.991 HRD-in -77.32, -47.05 68.98, 19.83 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -102.55, 163.3 APE9-dihe-na 90.09, 132.18 APE8-dihe-in -72.41, 162.37 APE8-rot-in 279.62 APE67-dihe-in -81.75, -17.56 -53.5, -56.42 APE12-dist-in 12.856 APE11-dist-in 10.778 APE10-dist-in 5.79 APE9-dist-in 3.107 None None None XRAY 2.75 0.24 0.275 B 351 346 0 0 0 0 [[56, 340]] 1.0 7u36 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
2OW3A 35 385 420.0 BIM:387 Type1 Active DFGin 6.854 14.088 BLAminus -145.58, -177.16 62.63, 79.7 -96.04, 38.01 299.18, 104.83 -72.62, -36.62 in-in in 8.34 Saltbr-in 2.838 HRD-in -75.79, -46.9 63.78, 27.01 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.84, 153.8 APE9-dihe-na 77.18, 154.82 APE8-dihe-in -72.33, 143.1 APE8-rot-in 299.46 APE67-dihe-in -64.33, -22.16 -49.08, -49.27 APE12-dist-in 13.724 APE11-dist-in 12.363 APE10-dist-in 7.515 APE9-dist-in 3.784 None PTR216 PTR216 XRAY 2.8 0.248 0.295 A 352 347 4 0 0 0 [[56, 340]] 1.0 2ow3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
2OW3B 35 386 420.0 BIM:387 Type1 Active DFGin 6.768 14.52 BLAminus -140.91, -178.82 62.87, 80.36 -94.83, 34.08 291.22, 81.94 -79.34, -15.72 in-in in 8.48 Saltbr-in 2.788 HRD-in -91.97, -42.45 64.4, 21.24 in-in-in SNCiii in-in ActLoopNT-in 2.877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.27, 157.33 APE9-dihe-na 81.52, 163.87 APE8-dihe-in -81.91, 157.75 APE8-rot-in 308.08 APE67-dihe-in -65.81, -19.16 -55.34, -61.54 APE12-dist-in 13.905 APE11-dist-in 12.542 APE10-dist-in 7.628 APE9-dist-in 3.538 None PTR216 PTR216 XRAY 2.8 0.248 0.295 B 352 352 0 0 0 0 [[56, 340]] 1.0 2ow3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3GB2A 35 383 420.0 G3B:999 Type1 Active DFGin 7.081 13.502 BLAminus -136.77, -176.86 57.81, 94.36 -109.09, 24.06 290.54, 74.85 -73.21, 4.88 in-in in 8.45 Saltbr-in 2.812 HRD-in -66.76, -55.55 72.33, 20.67 in-in-in SNCiii in-in ActLoopNT-in 2.859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.38, -175.57 APE9-dihe-na 67.46, 160.91 APE8-dihe-in -72.68, 139.68 APE8-rot-in 245.03 APE67-dihe-in -60.68, -25.16 -49.04, -51.42 APE12-dist-in 13.505 APE11-dist-in 11.973 APE10-dist-in 7.004 APE9-dist-in 3.287 None PTR216 PTR216 XRAY 2.4 0.225 0.289 A 353 341 8 0 0 0 [[56, 340]] 1.0 3gb2 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6TCUA 35 384 420.0 N1Q:401 Type1 Active DFGin 7.271 14.191 BLAminus -132.13, 178.03 59.16, 82.25 -93.13, 22.32 285.63, 78.52 -60.3, -31.7 in-in in 8.352 Saltbr-in 2.912 HRD-in -72.47, -46.38 65.88, 22.79 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.64, 162.18 APE9-dihe-na 73.42, 158.65 APE8-dihe-in -78.26, 138.24 APE8-rot-in 295.07 APE67-dihe-in -60.71, -25.87 -50.61, -49.17 APE12-dist-in 13.556 APE11-dist-in 11.943 APE10-dist-in 7.197 APE9-dist-in 3.24 None PTR216 PTR216 XRAY 2.14 0.204 0.24 A 355 350 0 0 0 0 [[56, 340]] 1.0 6tcu CMGC_GSK3B_HUMAN CMGC 1.9e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5T31A 35 381 420.0 6VL:501 Type1 Active DFGin 7.0 14.6 BLAminus -146.5, -178.72 58.09, 85.8 -94.81, 34.39 283.96, 70.89 -72.9, -29.06 in-in in 8.183 Saltbr-in 2.823 HRD-in -85.27, -37.65 59.13, 22.16 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.45, 179.68 APE9-dihe-na 63.71, 158.01 APE8-dihe-in -85.57, 141.47 APE8-rot-in 304.73 APE67-dihe-in -68.11, -24.88 -45.34, -45.1 APE12-dist-in 13.218 APE11-dist-in 11.545 APE10-dist-in 6.564 APE9-dist-in 3.195 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 A 420 335 12 0 0 0 [[56, 340]] 1.0 5t31 CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5T31B 36 382 420.0 6VL:501 Type1 Active DFGin 7.209 14.605 BLAminus -147.12, 178.9 61.54, 81.68 -96.09, 32.98 286.61, 73.16 -76.82, -18.6 in-in in 8.229 Saltbr-in 2.581 HRD-in -64.89, -47.6 63.02, 19.09 in-in-in SNCiii in-in ActLoopNT-in 3.018 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.39, 179.54 APE9-dihe-na 63.77, 153.96 APE8-dihe-in -75.26, 136.0 APE8-rot-in 291.41 APE67-dihe-in -61.67, -31.85 -41.28, -53.13 APE12-dist-in 13.381 APE11-dist-in 11.678 APE10-dist-in 6.473 APE9-dist-in 3.237 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 B 420 334 13 0 0 0 [[56, 340]] 1.0 5t31 CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7Z1GA 27 383 420.0 3NG:60401 Type1 Active DFGin 7.272 14.699 BLAminus -137.45, -179.93 52.32, 81.51 -93.1, 20.22 282.75, 78.65 -65.74, -16.48 in-in in 8.969 Saltbr-in 2.771 HRD-in -67.62, -47.44 74.98, 2.45 in-in-in SNCiii in-in ActLoopNT-in 2.926 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.67, 177.94 APE9-dihe-na 70.81, 142.84 APE8-dihe-in -95.23, 170.55 APE8-rot-in 305.08 APE67-dihe-inflip 72.5, -37.64 -53.01, 158.1 APE12-dist-in 12.785 APE11-dist-in 10.847 APE10-dist-in 5.858 APE9-dist-in 2.984 None None None XRAY 2.85 0.204 0.228 A 364 355 2 0 0 0 [[56, 340]] 1.0 7z1g CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7B6FA 36 382 420.0 SZW:401 Type1 Active DFGin 6.788 14.002 BLAminus -139.5, -179.55 63.73, 84.52 -97.59, 24.1 286.83, 79.42 -64.99, -20.21 in-in in 8.319 Saltbr-in 2.573 HRD-in -72.27, -45.59 68.3, 15.73 in-in-in SNCiii in-in ActLoopNT-in 2.861 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.61, 164.26 APE9-dihe-na 74.41, 146.1 APE8-dihe-in -66.85, 137.72 APE8-rot-in 301.31 APE67-dihe-in -60.67, -24.91 -43.57, -54.9 APE12-dist-in 13.468 APE11-dist-in 11.675 APE10-dist-in 7.087 APE9-dist-in 3.203 None PTR216 PTR216 XRAY 2.05 0.176 0.209 A 365 347 0 0 0 0 [[56, 340]] 1.0 7b6f CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8AUZA 27 381 420.0 O9C:402 Type1 Active DFGin 7.028 13.822 BLAminus -150.9, 179.1 54.07, 83.84 -94.84, 28.62 288.95, 81.72 -71.58, -10.75 in-in in 8.497 Saltbr-in 2.734 HRD-in -57.37, -52.37 73.76, 8.1 in-in-in SNCiii in-in ActLoopNT-in 3.155 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.43, 171.72 APE9-dihe-na 68.38, 153.94 APE8-dihe-in -73.1, 142.46 APE8-rot-in 305.9 APE67-dihe-in -60.73, -30.47 -42.52, -61.25 APE12-dist-in 13.255 APE11-dist-in 11.714 APE10-dist-in 7.025 APE9-dist-in 3.055 None PTR216 PTR216 XRAY 2.66 0.172 0.229 A 365 351 4 0 0 0 [[56, 340]] 1.0 8auz CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8AUZB 27 381 420.0 O9C:402 Type1 Active DFGin 7.099 13.907 BLAminus -145.47, 175.75 60.6, 82.78 -92.91, 28.92 286.05, 79.75 -73.75, -11.85 in-in in 8.586 Saltbr-in 2.697 HRD-in -55.14, -51.91 71.49, 10.11 in-in-in SNCiii in-in ActLoopNT-in 3.139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.91, 170.34 APE9-dihe-na 66.33, 153.39 APE8-dihe-in -70.91, 144.03 APE8-rot-in 280.02 APE67-dihe-in -59.87, -32.25 -43.58, -60.53 APE12-dist-in 13.172 APE11-dist-in 11.662 APE10-dist-in 6.924 APE9-dist-in 3.004 None PTR216 PTR216 XRAY 2.66 0.172 0.229 B 365 351 4 0 0 0 [[56, 340]] 1.0 8auz CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4AFJA 36 384 420.0 SJJ:1391 Type1 Active DFGin 6.937 13.715 BLAminus -130.67, 179.05 59.17, 87.64 -94.83, 20.23 280.89, 81.14 -65.73, -20.9 in-in in 8.572 Saltbr-in 2.652 HRD-in -69.53, -45.4 65.78, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.937 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.24, 160.98 APE9-dihe-na 76.37, 138.38 APE8-dihe-in -58.5, 130.27 APE8-rot-in 301.13 APE67-dihe-in -61.75, -23.96 -37.58, -52.92 APE12-dist-in 13.435 APE11-dist-in 11.681 APE10-dist-in 6.975 APE9-dist-in 3.193 None PTR216 PTR216 XRAY 1.98 0.179 0.216 A 367 344 5 0 0 0 [[56, 340]] 1.0 4afj CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4AFJB 34 384 420.0 SJJ:1392 Type1 Active DFGin 6.948 14.046 BLAminus -131.53, 179.02 57.76, 85.75 -93.28, 22.08 280.88, 83.41 -64.33, -20.8 in-in in 8.525 Saltbr-in 2.743 HRD-in -67.39, -46.66 68.06, 10.89 in-in-in SNCiii in-in ActLoopNT-in 2.877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.99, 165.35 APE9-dihe-na 75.2, 154.5 APE8-dihe-in -78.53, 128.88 APE8-rot-in 295.4 APE67-dihe-in -61.46, -24.46 -31.5, -55.04 APE12-dist-in 13.476 APE11-dist-in 11.582 APE10-dist-in 6.958 APE9-dist-in 3.146 None PTR216 PTR216 XRAY 1.98 0.179 0.216 B 367 347 4 0 0 0 [[56, 340]] 1.0 4afj CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3ZRKA 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.886 13.908 BLAminus -131.68, 179.96 63.1, 79.53 -95.35, 25.37 286.53, 78.64 -74.21, -8.59 in-in in 8.474 Saltbr-in 2.75 HRD-in -67.17, -50.87 73.03, 10.45 in-in-in SNCiii in-in ActLoopNT-in 2.841 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.35, 160.84 APE9-dihe-na 74.59, 142.57 APE8-dihe-in -61.86, 136.31 APE8-rot-in 305.46 APE67-dihe-in -59.75, -23.44 -46.23, -50.56 APE12-dist-in 13.377 APE11-dist-in 11.67 APE10-dist-in 7.003 APE9-dist-in 3.16 None PTR216 PTR216 XRAY 2.37 0.201 0.243 A 371 347 2 0 0 0 [[56, 340]] 1.0 3zrk CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3ZRKB 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.715 14.017 BLAminus -139.49, -177.28 57.97, 77.09 -90.4, 24.0 286.01, 81.23 -69.91, -16.36 in-in in 8.587 Saltbr-in 2.732 HRD-in -64.4, -48.95 71.37, 3.03 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.35, 163.72 APE9-dihe-na 73.35, 153.59 APE8-dihe-in -70.79, 138.65 APE8-rot-in 292.42 APE67-dihe-in -62.81, -26.76 -44.91, -48.41 APE12-dist-in 13.36 APE11-dist-in 11.482 APE10-dist-in 6.882 APE9-dist-in 3.161 None PTR216 PTR216 XRAY 2.37 0.201 0.243 B 371 349 0 0 0 0 [[56, 340]] 1.0 3zrk CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3ZRLA 36 385 420.0 ZRL:1390 Type1 Active DFGin 6.976 14.145 BLAminus -134.74, 178.82 66.15, 74.2 -88.14, 21.07 285.95, 79.46 -68.66, -8.3 in-in in 8.484 Saltbr-in 2.586 HRD-in -74.36, -46.11 75.3, 2.22 in-in-in SNCiii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.36, 158.14 APE9-dihe-na 75.43, 144.25 APE8-dihe-in -61.72, 142.08 APE8-rot-in 315.78 APE67-dihe-in -63.29, -26.99 -52.04, -46.88 APE12-dist-in 13.478 APE11-dist-in 11.716 APE10-dist-in 7.157 APE9-dist-in 3.171 None PTR216 PTR216 XRAY 2.48 0.188 0.249 A 371 348 2 0 0 0 [[56, 340]] 1.0 3zrl CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3ZRLB 36 384 420.0 ZRL:1390 Type1 Active DFGin 6.816 14.066 BLAminus -140.64, -176.21 56.19, 79.11 -88.83, 19.02 286.49, 80.49 -67.02, -13.2 in-in in 8.613 Saltbr-in 2.734 HRD-in -62.44, -47.89 69.81, 8.62 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.8, 160.71 APE9-dihe-na 76.77, 159.03 APE8-dihe-in -75.92, 142.27 APE8-rot-in 284.41 APE67-dihe-in -61.87, -25.02 -48.38, -50.46 APE12-dist-in 13.452 APE11-dist-in 11.697 APE10-dist-in 7.085 APE9-dist-in 3.218 None PTR216 PTR216 XRAY 2.48 0.188 0.249 B 371 349 0 0 0 0 [[56, 340]] 1.0 3zrl CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3ZRMA 36 383 420.0 ZRM:1388 Type1 Active DFGin 6.934 13.954 BLAminus -132.01, -179.16 64.76, 76.89 -91.07, 16.45 285.73, 79.52 -60.99, -14.53 in-in in 8.379 Saltbr-in 2.59 HRD-in -73.17, -48.0 77.03, 4.47 in-in-in SNCiii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.45, 164.9 APE9-dihe-na 71.3, 144.2 APE8-dihe-in -61.55, 140.83 APE8-rot-in 305.4 APE67-dihe-in -61.36, -25.73 -52.92, -47.77 APE12-dist-in 13.418 APE11-dist-in 11.733 APE10-dist-in 7.034 APE9-dist-in 3.184 None PTR216 PTR216 XRAY 2.49 0.19 0.247 A 371 346 2 0 0 0 [[56, 340]] 1.0 3zrm CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3ZRMB 36 384 420.0 ZRM:1389 Type1 Active DFGin 6.902 14.104 BLAminus -140.7, -177.64 59.24, 76.67 -89.43, 25.85 287.41, 78.75 -71.45, -17.33 in-in in 8.556 Saltbr-in 2.639 HRD-in -65.21, -46.92 71.38, 6.55 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.4, 163.13 APE9-dihe-na 76.6, 157.17 APE8-dihe-in -72.35, 137.17 APE8-rot-in 272.08 APE67-dihe-in -62.09, -20.43 -43.42, -53.94 APE12-dist-in 13.463 APE11-dist-in 11.697 APE10-dist-in 7.031 APE9-dist-in 3.11 None PTR216 PTR216 XRAY 2.49 0.19 0.247 B 371 349 0 0 0 0 [[56, 340]] 1.0 3zrm CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5K5NA 36 382 420.0 6QH:4001 Type1 Active DFGin 6.867 13.803 BLAminus -136.97, -178.03 58.54, 81.58 -94.06, 22.59 285.28, 80.04 -66.6, -22.76 in-in in 8.685 Saltbr-in 2.763 HRD-in -65.0, -45.17 61.7, 20.55 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.55, 163.97 APE9-dihe-na 70.72, 157.82 APE8-dihe-in -71.18, 131.1 APE8-rot-in 299.71 APE67-dihe-in -62.03, -24.12 -33.31, -56.32 APE12-dist-in 13.585 APE11-dist-in 11.966 APE10-dist-in 6.992 APE9-dist-in 3.201 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 A 370 332 12 0 0 0 [[56, 340]] 1.0 5k5n CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5K5NB 36 384 420.0 6QH:401 Type1 Active DFGin 6.968 13.745 BLAminus -135.06, -178.44 58.85, 83.42 -94.58, 20.58 286.7, 80.8 -64.41, -22.37 in-in in 8.869 Saltbr-in 2.795 HRD-in -64.71, -45.91 63.61, 14.11 in-in-in SNCiii in-in ActLoopNT-in 2.88 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.36, 162.07 APE9-dihe-na 75.01, 147.36 APE8-dihe-in -65.41, 124.62 APE8-rot-in 290.2 APE67-dihe-in -56.35, -27.77 -26.59, -62.75 APE12-dist-in 13.372 APE11-dist-in 11.994 APE10-dist-in 6.896 APE9-dist-in 3.109 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 B 370 335 11 0 0 0 [[56, 340]] 1.0 5k5n CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1R0EA 35 383 420.0 DFN:702 Type1 Active DFGin 7.211 13.978 BLAminus -134.01, -179.44 58.42, 85.11 -96.64, 20.85 278.46, 77.75 -63.57, -17.65 in-in in 8.372 Saltbr-in 2.716 HRD-in -68.9, -46.99 73.89, 15.3 in-in-in SNCiii in-in ActLoopNT-in 2.817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.99, 167.9 APE9-dihe-na 82.35, 148.07 APE8-dihe-in -104.61, 148.9 APE8-rot-in 290.93 APE67-dihe-inflip 91.63, -34.6 -37.68, 131.22 APE12-dist-in 13.098 APE11-dist-in 11.094 APE10-dist-in 6.24 APE9-dist-in 3.395 None None None XRAY 2.25 0.225 0.252 A 391 344 5 0 0 0 [[56, 340]] 1.0 1r0e CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1R0EB 35 383 420.0 DFN:501 Type1 Active DFGin 7.247 14.105 BLAminus -133.07, -177.02 55.1, 85.48 -97.08, 20.86 276.04, 78.13 -65.93, -17.26 in-in in 8.445 Saltbr-in 2.91 HRD-in -68.16, -44.28 70.07, 10.75 in-in-in SNCiii in-in ActLoopNT-in 2.884 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.79, 168.13 APE9-dihe-na 84.81, 147.78 APE8-dihe-in -104.27, 148.93 APE8-rot-in 288.7 APE67-dihe-inflip 91.14, -35.24 -35.52, 130.18 APE12-dist-in 13.079 APE11-dist-in 11.011 APE10-dist-in 6.177 APE9-dist-in 3.369 None None None XRAY 2.25 0.225 0.252 B 391 344 5 0 0 0 [[56, 340]] 1.0 1r0e CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q5KA 35 384 420.0 TMU:901 Type1 Active DFGin 6.988 13.863 BLAminus -136.18, -175.74 56.25, 81.9 -94.66, 24.16 283.53, 73.95 -64.32, -18.01 in-in in 8.227 Saltbr-in 2.549 HRD-in -67.21, -47.72 71.71, 7.94 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.63, 174.67 APE9-dihe-na 78.79, 134.14 APE8-dihe-in -77.03, 144.65 APE8-rot-in 302.42 APE67-dihe-inflip 99.66, -34.41 -53.93, 140.09 APE12-dist-in 12.905 APE11-dist-in 11.002 APE10-dist-in 5.832 APE9-dist-in 3.144 None None None XRAY 1.94 0.222 0.242 A 414 345 5 0 0 0 [[56, 340]] 1.0 1q5k CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q5KB 35 384 420.0 TMU:902 Type1 Active DFGin 6.985 13.773 BLAminus -138.67, -177.12 58.86, 79.46 -94.38, 28.16 285.34, 70.82 -69.41, -14.87 in-in in 8.132 Saltbr-in 2.832 HRD-in -69.04, -44.01 68.27, 5.21 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.05, 176.86 APE9-dihe-na 75.09, 135.72 APE8-dihe-in -79.59, 144.98 APE8-rot-in 303.4 APE67-dihe-inflip 93.62, -37.01 -50.51, 145.1 APE12-dist-in 12.931 APE11-dist-in 11.072 APE10-dist-in 5.846 APE9-dist-in 3.103 None None None XRAY 1.94 0.222 0.242 B 414 344 6 0 0 0 [[56, 340]] 1.0 1q5k CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3I4BA 25 385 420.0 Z48:501 Type1 Active DFGin 6.641 13.646 BLAminus -134.01, -176.44 58.71, 78.24 -93.71, 24.37 285.69, 79.56 -67.57, -20.03 in-in in 8.476 Saltbr-in 2.637 HRD-in -63.92, -46.73 77.65, -7.51 in-in-in SNCiii in-in ActLoopNT-in 2.95 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.08, 174.13 APE9-dihe-na 79.29, 137.44 APE8-dihe-in -92.27, 151.07 APE8-rot-in 303.5 APE67-dihe-inflip 83.63, -1.22 -43.52, 132.98 APE12-dist-in 13.009 APE11-dist-in 10.939 APE10-dist-in 5.839 APE9-dist-in 3.102 None None None XRAY 2.3 0.181 0.222 A 414 359 0 0 0 0 [[56, 340]] 1.0 3i4b CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3I4BB 36 382 420.0 Z48:501 Type1 Active DFGin 7.01 13.655 BLAminus -135.85, -175.31 58.14, 77.59 -93.89, 21.58 285.55, 84.81 -65.19, -18.79 in-in in 8.508 Saltbr-in 2.617 HRD-in -67.57, -44.79 75.92, -6.36 in-in-in SNCiii in-in ActLoopNT-in 2.941 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.93, 173.5 APE9-dihe-na 79.53, 137.7 APE8-dihe-in -93.51, 150.41 APE8-rot-in 299.4 APE67-dihe-inflip 78.16, -1.88 -37.33, 134.24 APE12-dist-in 13.043 APE11-dist-in 10.917 APE10-dist-in 5.828 APE9-dist-in 3.115 None None None XRAY 2.3 0.181 0.222 B 414 347 0 0 0 0 [[56, 340]] 1.0 3i4b CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3L1SA 25 384 420.0 Z92:421 Type1 Active DFGin 6.757 13.748 BLAminus -136.19, -175.27 59.75, 67.96 -82.46, 22.04 287.73, 86.13 -66.81, -21.63 in-in in 8.518 Saltbr-in 2.708 HRD-in -64.1, -46.34 73.45, -1.44 in-in-in SNCiii in-in ActLoopNT-in 2.949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 172.3 APE9-dihe-na 79.23, 137.51 APE8-dihe-in -89.89, 147.82 APE8-rot-in 303.47 APE67-dihe-inflip 83.2, -1.08 -42.22, 131.52 APE12-dist-in 13.007 APE11-dist-in 10.892 APE10-dist-in 5.894 APE9-dist-in 3.161 None None None XRAY 2.9 0.186 0.232 A 414 336 21 0 0 0 [[56, 340]] 1.0 3l1s CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3L1SB 36 382 420.0 Z92:422 Type1 Active DFGin 6.984 13.78 BLAminus -136.63, -175.36 61.34, 59.7 -75.09, 22.69 291.46, 84.75 -66.47, -23.35 in-in in 8.551 Saltbr-in 2.737 HRD-in -65.65, -45.98 77.68, -13.89 in-in-in SNCiii in-in ActLoopNT-in 2.937 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.08, 173.03 APE9-dihe-na 76.72, 137.31 APE8-dihe-in -89.1, 148.7 APE8-rot-in 302.46 APE67-dihe-inflip 83.32, 3.78 -42.62, 131.74 APE12-dist-in 13.014 APE11-dist-in 10.916 APE10-dist-in 6.149 APE9-dist-in 3.121 None None None XRAY 2.9 0.186 0.232 B 414 330 17 0 0 0 [[56, 340]] 1.0 3l1s CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
2JLDA 35 385 420.0 AG1:1385 Type1 Active DFGin 7.247 13.619 BLAminus -128.74, 174.0 65.55, 89.02 -101.06, 20.23 281.85, 78.64 -66.01, -16.46 in-in in 8.535 Saltbr-in 2.901 HRD-in -68.74, -48.89 74.29, 10.13 in-in-in SNCiii in-in ActLoopNT-in 2.846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -80.14, 165.31 APE9-dihe-na 82.65, 142.84 APE8-dihe-in -89.49, 145.54 APE8-rot-in 290.56 APE67-dihe-inflip 101.97, -33.31 -39.01, 124.35 APE12-dist-in 13.012 APE11-dist-in 11.005 APE10-dist-in 6.058 APE9-dist-in 3.239 None None None XRAY 2.35 0.192 0.227 A 420 349 2 0 0 0 [[56, 340]] 1.0 2jld CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
2JLDB 35 384 420.0 AG1:1385 Type1 Active DFGin 7.117 13.681 BLAminus -134.8, 174.83 62.6, 85.31 -97.62, 21.89 284.88, 76.87 -65.09, -17.38 in-in in 8.458 Saltbr-in 2.725 HRD-in -67.92, -46.43 70.86, 13.33 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.11, 167.47 APE9-dihe-na 84.04, 143.71 APE8-dihe-in -89.79, 148.89 APE8-rot-in 294.08 APE67-dihe-inflip 95.31, -31.23 -37.35, 123.61 APE12-dist-in 13.044 APE11-dist-in 10.951 APE10-dist-in 5.995 APE9-dist-in 3.203 None None None XRAY 2.35 0.192 0.227 B 420 349 1 0 0 0 [[56, 340]] 1.0 2jld CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3M1SB 35 384 420.0 DW1:421 Type1 Active DFGin 7.187 13.372 BLAminus -147.84, 174.37 70.86, 99.58 -120.24, 19.87 286.56, 80.37 -63.52, -14.18 in-in in 8.585 Saltbr-in 2.441 HRD-in -69.47, -49.47 71.23, 28.36 in-in-in SNCiii in-in ActLoopNT-in 3.091 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -106.87, 165.89 APE9-dihe-na 90.21, 134.65 APE8-dihe-in -74.2, 145.74 APE8-rot-in 300.21 APE67-dihe-in -72.41, -23.39 -22.57, -69.43 APE12-dist-in 12.944 APE11-dist-in 10.712 APE10-dist-in 5.899 APE9-dist-in 3.769 None None None XRAY 3.134 0.171 0.228 B 420 349 1 0 0 0 [[56, 340]] 1.0 3m1s CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3PUPA 35 382 420.0 OS1:421 Type1 Active DFGin 6.995 13.637 BLAminus -143.74, 172.61 64.16, 94.87 -107.49, 13.61 287.44, 72.72 -52.4, -32.47 in-in in 8.443 Saltbr-in 2.807 HRD-in -86.73, -34.2 66.44, 7.86 in-in-in SNCiii in-in ActLoopNT-in 2.857 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.24, -13.27 APE9-dihe-na -89.84, 168.85 APE8-dihe-in -94.34, 159.6 APE8-rot-in 296.79 APE67-dihe-in -69.26, -2.79 -42.9, -70.67 APE12-dist-in 13.056 APE11-dist-in 10.912 APE10-dist-in 6.171 APE9-dist-in 3.486 None None None XRAY 2.99 0.206 0.249 A 420 346 2 0 0 0 [[56, 340]] 1.0 3pup CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3PUPB 35 383 420.0 OS1:421 Type1 Active DFGin 6.987 13.646 BLAminus -146.61, 171.7 65.62, 100.17 -113.12, 21.06 287.13, 70.81 -60.05, -30.47 in-in in 8.479 Saltbr-in 2.972 HRD-in -88.21, -42.27 77.46, 8.13 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.13, -17.37 APE9-dihe-na -97.38, 160.84 APE8-dihe-in -100.44, 160.76 APE8-rot-in 282.35 APE67-dihe-in -75.14, -2.22 -49.84, -64.39 APE12-dist-in 13.107 APE11-dist-in 10.976 APE10-dist-in 6.5 APE9-dist-in 3.751 None None None XRAY 2.99 0.206 0.249 B 420 347 2 0 0 0 [[56, 340]] 1.0 3pup CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6B8JA 37 384 420.0 65C:502 Type1 Active DFGin 6.868 13.909 BLAminus -142.04, -175.4 56.86, 72.8 -87.54, 21.75 287.01, 61.58 -69.77, -16.08 in-in in 8.507 Saltbr-in 2.318 HRD-in -66.49, -42.97 62.67, 20.6 in-in-in SNCiii in-in ActLoopNT-in 2.821 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.37, 166.1 APE9-dihe-na 69.29, 116.74 APE8-dihe-in -38.51, 137.94 APE8-rot-in 299.43 APE67-dihe-in -65.74, -24.52 -56.45, -42.14 APE12-dist-in 13.685 APE11-dist-in 11.734 APE10-dist-in 7.018 APE9-dist-in 3.326 None PTR216 PTR216 XRAY 2.595 0.215 0.247 A 420 345 3 0 0 0 [[56, 340]] 1.0 6b8j CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6H0UA 36 383 420.0 FKB:501 Type1 Active DFGin 6.732 13.816 BLAminus -102.2, -173.91 62.01, 94.18 -105.02, 23.81 292.61, 84.27 -66.96, -25.5 in-in in 8.798 Saltbr-in 2.726 HRD-in -71.89, -49.13 79.92, 3.93 in-in-in SNCiii in-in ActLoopNT-in 2.966 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.85, 170.11 APE9-dihe-na 84.06, 143.45 APE8-dihe-in -90.7, 142.53 APE8-rot-in 301.69 APE67-dihe-in -73.12, -14.65 -13.27, -76.63 APE12-dist-in 12.955 APE11-dist-in 10.868 APE10-dist-in 5.76 APE9-dist-in 3.223 None None None XRAY 2.3 0.195 0.24 A 420 348 0 0 0 0 [[56, 340]] 1.0 6h0u CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6H0UB 36 383 420.0 FKB:501 Type1 Active DFGin 6.648 13.973 BLAminus -111.78, 175.04 68.36, 93.29 -102.83, 22.46 286.57, 84.56 -63.31, -24.15 in-in in 8.763 Saltbr-in 2.745 HRD-in -68.5, -49.8 75.08, 1.45 in-in-in SNCiii in-in ActLoopNT-in 2.851 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.21, 171.64 APE9-dihe-na 80.61, 138.7 APE8-dihe-in -91.3, 150.17 APE8-rot-in 304.68 APE67-dihe-inflip 101.55, -29.52 -53.44, 134.06 APE12-dist-in 12.722 APE11-dist-in 10.726 APE10-dist-in 5.704 APE9-dist-in 3.163 None None None XRAY 2.3 0.195 0.24 B 420 348 0 0 0 0 [[56, 340]] 1.0 6h0u CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6V6LA 37 384 420.0 QQA:501 Type1 Active DFGin 7.244 14.228 BLAminus -134.87, -179.15 59.4, 83.41 -98.99, 30.0 283.16, 72.37 -75.66, -20.38 in-in in 8.388 Saltbr-in 2.736 HRD-in -68.21, -49.19 67.93, 18.71 in-in-in SNCiii in-in ActLoopNT-in 3.016 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.84, 162.85 APE9-dihe-na 77.33, 149.16 APE8-dihe-in -69.69, 129.38 APE8-rot-in 287.88 APE67-dihe-in -58.07, -31.39 -36.48, -49.2 APE12-dist-in 13.461 APE11-dist-in 11.648 APE10-dist-in 6.953 APE9-dist-in 3.241 None PTR216 PTR216 XRAY 2.19 0.204 0.234 A 420 344 4 0 0 0 [[56, 340]] 1.0 6v6l CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3DU8A 35 382 420.0 553:553 Type1 Active DFGin 6.992 13.938 BLAminus -138.88, -177.6 60.76, 81.45 -97.52, 17.85 284.1, 81.79 -60.5, -23.71 in-in in 8.713 Saltbr-in 2.686 HRD-in -70.97, -44.22 68.9, 5.64 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.61, 170.6 APE9-dihe-na 82.17, 142.06 APE8-dihe-in -90.1, 145.24 APE8-rot-in 300.29 APE67-dihe-inflip 98.68, -34.99 -51.44, 136.14 APE12-dist-in 13.036 APE11-dist-in 10.944 APE10-dist-in 5.764 APE9-dist-in 3.152 None None None XRAY 2.2 0.215 0.246 A 422 336 12 0 0 0 [[56, 340]] 1.0 3du8 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3DU8B 35 385 420.0 553:553 Type1 Active DFGin 7.11 14.001 BLAminus -130.0, -177.1 64.69, 78.27 -91.27, 21.46 283.91, 80.88 -65.59, -20.64 in-in in 8.742 Saltbr-in 2.702 HRD-in -71.12, -43.48 71.58, 1.27 in-in-in SNCiii in-in ActLoopNT-in 2.992 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -75.13, 166.25 APE9-dihe-na 83.98, 139.39 APE8-dihe-in -88.38, 143.61 APE8-rot-in 294.95 APE67-dihe-inflip 93.54, -38.98 -56.03, 145.75 APE12-dist-in 13.05 APE11-dist-in 11.13 APE10-dist-in 5.901 APE9-dist-in 3.176 None None None XRAY 2.2 0.215 0.246 B 422 339 12 0 0 0 [[56, 340]] 1.0 3du8 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR5A 25 385 420.0 A1IE8:501 Type1 Active DFGin 7.063 14.321 BLAminus -141.02, 178.57 59.76, 86.64 -101.14, 27.38 287.09, 76.28 -70.78, -13.94 in-in in 8.363 Saltbr-in 2.867 HRD-in -72.5, -48.23 71.7, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.985 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.15, 177.99 APE9-dihe-na 68.95, 145.14 APE8-dihe-in -94.16, 151.35 APE8-rot-in 288.71 APE67-dihe-inflip 90.22, -34.5 -47.82, 143.36 APE12-dist-in 13.104 APE11-dist-in 11.105 APE10-dist-in 6.167 APE9-dist-in 3.186 None None None XRAY 2.3 0.204 0.235 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr5 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR5B 36 382 420.0 A1IE8:501 Type1 Active DFGin 7.068 14.397 BLAminus -143.23, 179.4 62.21, 84.47 -103.42, 28.19 287.66, 78.04 -72.31, -18.53 in-in in 8.684 Saltbr-in 2.965 HRD-in -72.41, -47.52 71.61, 14.06 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.66, -179.45 APE9-dihe-na 68.77, 147.4 APE8-dihe-in -97.67, 156.22 APE8-rot-in 283.57 APE67-dihe-inflip 84.77, -33.0 -49.59, 145.66 APE12-dist-in 13.056 APE11-dist-in 10.953 APE10-dist-in 5.986 APE9-dist-in 3.188 None None None XRAY 2.3 0.204 0.235 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr5 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR6A 25 385 420.0 A1IFO:501 Type1 Active DFGin 7.074 14.161 BLAminus -136.83, -174.79 60.55, 80.3 -97.86, 24.81 287.57, 77.74 -66.69, -16.26 in-in in 8.556 Saltbr-in 2.935 HRD-in -72.59, -48.06 71.15, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.992 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.91, 171.88 APE9-dihe-na 74.24, 144.89 APE8-dihe-in -96.08, 152.09 APE8-rot-in 291.49 APE67-dihe-inflip 90.67, -36.1 -52.14, 144.18 APE12-dist-in 13.022 APE11-dist-in 11.047 APE10-dist-in 6.124 APE9-dist-in 3.24 None None None XRAY 2.3 0.2 0.232 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr6 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR6B 36 382 420.0 A1IFO:501 Type1 Active DFGin 7.128 14.36 BLAminus -139.12, -179.31 63.06, 81.93 -99.98, 26.01 286.75, 75.51 -71.16, -14.75 in-in in 8.843 Saltbr-in 2.836 HRD-in -72.29, -48.89 71.91, 12.0 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.4, 172.1 APE9-dihe-na 77.09, 144.87 APE8-dihe-in -98.08, 154.15 APE8-rot-in 291.27 APE67-dihe-inflip 90.37, -33.63 -52.57, 140.86 APE12-dist-in 13.071 APE11-dist-in 10.957 APE10-dist-in 5.983 APE9-dist-in 3.22 None None None XRAY 2.3 0.2 0.232 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr6 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR7A 25 385 420.0 A1IFJ:501 Type1 Active DFGin 6.912 13.949 BLAminus -136.24, -176.42 58.55, 87.09 -104.67, 27.04 287.13, 78.6 -71.53, -14.0 in-in in 8.632 Saltbr-in 2.802 HRD-in -71.98, -46.0 72.36, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.987 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.42, 177.43 APE9-dihe-na 69.9, 145.82 APE8-dihe-in -94.03, 156.28 APE8-rot-in 289.17 APE67-dihe-inflip 91.05, -31.63 -52.45, 141.85 APE12-dist-in 13.108 APE11-dist-in 11.121 APE10-dist-in 6.121 APE9-dist-in 3.15 None None None XRAY 2.3 0.199 0.229 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr7 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR7B 36 382 420.0 A1IFJ:501 Type1 Active DFGin 6.99 13.952 BLAminus -139.3, -178.5 61.7, 87.08 -105.92, 24.05 284.91, 80.77 -70.11, -13.68 in-in in 8.593 Saltbr-in 2.71 HRD-in -71.41, -48.43 71.41, 11.5 in-in-in SNCiii in-in ActLoopNT-in 2.94 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.82, 177.23 APE9-dihe-na 70.05, 146.13 APE8-dihe-in -96.47, 160.58 APE8-rot-in 285.27 APE67-dihe-inflip 87.67, -29.95 -51.57, 140.33 APE12-dist-in 13.008 APE11-dist-in 11.007 APE10-dist-in 6.045 APE9-dist-in 3.156 None None None XRAY 2.3 0.199 0.229 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr7 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR8A 25 385 420.0 A1IE7:501 Type1 Active DFGin 6.991 14.325 BLAminus -138.39, -179.52 63.72, 81.82 -96.4, 23.65 287.29, 75.6 -66.3, -11.74 in-in in 8.553 Saltbr-in 2.906 HRD-in -71.33, -45.89 67.7, 10.94 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.78, 169.84 APE9-dihe-na 80.06, 148.59 APE8-dihe-in -102.16, 146.47 APE8-rot-in 284.89 APE67-dihe-inflip 97.34, -39.62 -53.84, 140.75 APE12-dist-in 13.081 APE11-dist-in 11.083 APE10-dist-in 6.012 APE9-dist-in 3.197 None None None XRAY 2.3 0.191 0.221 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr8 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR8B 36 383 420.0 A1IE7:501 Type1 Active DFGin 7.087 14.356 BLAminus -145.34, 175.42 68.0, 83.84 -100.29, 22.36 287.83, 75.27 -65.32, -15.0 in-in in 8.715 Saltbr-in 2.898 HRD-in -76.0, -49.5 72.49, 12.34 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.57, 172.15 APE9-dihe-na 78.67, 145.51 APE8-dihe-in -99.99, 146.48 APE8-rot-in 286.49 APE67-dihe-inflip 90.46, -36.44 -48.06, 141.27 APE12-dist-in 13.067 APE11-dist-in 10.852 APE10-dist-in 5.85 APE9-dist-in 3.153 None None None XRAY 2.3 0.191 0.221 B 442 348 0 0 0 0 [[56, 340]] 1.0 9fr8 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR9A 25 385 420.0 A1IE6:501 Type1 Active DFGin 7.037 14.325 BLAminus -140.22, -173.71 59.89, 84.2 -98.36, 22.56 286.21, 81.87 -68.06, -16.06 in-in in 8.462 Saltbr-in 2.928 HRD-in -72.09, -48.73 72.37, 5.47 in-in-in SNCiii in-in ActLoopNT-in 2.971 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.48, 176.45 APE9-dihe-na 79.51, 153.1 APE8-dihe-in -106.78, 146.27 APE8-rot-in 287.32 APE67-dihe-inflip 100.87, -37.49 -40.18, 126.82 APE12-dist-in 13.02 APE11-dist-in 11.03 APE10-dist-in 5.997 APE9-dist-in 3.173 None None None XRAY 2.55 0.197 0.234 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr9 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9FR9B 36 382 420.0 A1IE6:501 Type1 Active DFGin 6.97 14.413 BLAminus -146.13, 179.78 62.16, 86.8 -103.01, 25.64 284.6, 80.86 -74.54, -16.98 in-in in 8.76 Saltbr-in 3.487 HRD-in -67.74, -52.21 72.42, 13.09 in-in-in SNCiii in-in ActLoopNT-in 2.872 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.09, 170.35 APE9-dihe-na 79.85, 140.07 APE8-dihe-in -93.7, 153.67 APE8-rot-in 288.81 APE67-dihe-inflip 99.37, -31.56 -52.24, 133.09 APE12-dist-in 12.982 APE11-dist-in 10.81 APE10-dist-in 5.791 APE9-dist-in 3.181 None None None XRAY 2.55 0.197 0.234 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr9 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9HUKB 26 382 420.0 A1IXL:501 Type1 Active DFGin 7.463 14.062 BLAminus -139.0, -179.94 58.73, 94.97 -114.49, 25.32 285.15, 69.98 -63.61, -20.61 in-in in 8.13 Saltbr-in 3.28 HRD-in -69.2, -40.72 63.39, 20.78 in-in-in SNCiii in-in ActLoopNT-in 3.042 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.58, -178.87 APE9-dihe-na 67.27, 135.83 APE8-dihe-in -80.15, 163.62 APE8-rot-in 319.54 APE67-dihe-inflip 75.84, -27.97 -60.6, 162.6 APE12-dist-in 12.838 APE11-dist-in 10.744 APE10-dist-in 5.73 APE9-dist-in 3.212 None None None XRAY 3.5 0.219 0.25 B 442 357 0 0 0 0 [[56, 340]] 1.0 9huk CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9HULA 25 385 420.0 A1IXM:501 Type1 Active DFGin 7.07 13.943 BLAminus -137.8, -179.92 58.93, 93.22 -109.33, 21.24 284.01, 77.28 -66.77, -7.95 in-in in 8.344 Saltbr-in 2.923 HRD-in -67.44, -42.84 67.99, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.167 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.24, 178.29 APE9-dihe-na 68.13, 143.96 APE8-dihe-in -84.08, 162.04 APE8-rot-in 308.02 APE67-dihe-inflip 75.91, -35.84 -57.58, 161.58 APE12-dist-in 13.066 APE11-dist-in 11.024 APE10-dist-in 5.997 APE9-dist-in 3.163 None None None XRAY 2.9 0.218 0.244 A 442 361 0 0 0 0 [[56, 340]] 1.0 9hul CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9HULB 26 383 420.0 A1IXM:501 Type1 Active DFGin 7.218 13.9 BLAminus -141.92, -177.61 60.57, 66.5 -86.27, 21.98 288.8, 69.64 -66.75, -12.19 in-in in 8.268 Saltbr-in 2.748 HRD-in -68.36, -43.53 65.84, 14.02 in-in-in SNCiii in-in ActLoopNT-in 3.018 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.86, 177.51 APE9-dihe-na 70.81, 136.76 APE8-dihe-in -79.57, 164.11 APE8-rot-in 306.92 APE67-dihe-inflip 69.45, -30.71 -58.24, 165.67 APE12-dist-in 13.055 APE11-dist-in 10.975 APE10-dist-in 6.055 APE9-dist-in 3.14 None None None XRAY 2.9 0.218 0.244 B 442 358 0 0 0 0 [[56, 340]] 1.0 9hul CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9HV3A 25 385 420.0 A1IXN:501 Type1 Active DFGin 7.125 13.97 BLAminus -135.63, 170.17 69.98, 84.71 -102.55, 20.46 290.46, 80.59 -69.94, -0.25 in-in in 8.537 Saltbr-in 2.868 HRD-in -69.25, -48.0 72.7, 9.47 in-in-in SNCiii in-in ActLoopNT-in 2.935 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.1, 169.69 APE9-dihe-na 79.34, 142.23 APE8-dihe-in -80.23, 146.96 APE8-rot-in 316.9 APE67-dihe-inflip 78.3, -27.2 -49.89, 154.45 APE12-dist-in 13.123 APE11-dist-in 11.12 APE10-dist-in 6.197 APE9-dist-in 3.136 None None None XRAY 2.9 0.208 0.238 A 442 361 0 0 0 0 [[56, 340]] 1.0 9hv3 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9HV3B 25 382 420.0 A1IXN:501 Type1 Active DFGin 7.087 13.912 BLAminus -155.32, 174.2 63.74, 86.56 -102.98, 16.67 284.3, 76.87 -64.93, -6.56 in-in in 8.597 Saltbr-in 2.606 HRD-in -75.09, -41.25 66.67, 4.87 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.85, 168.81 APE9-dihe-na 83.21, 130.42 APE8-dihe-in -66.5, 151.79 APE8-rot-in 306.21 APE67-dihe-inflip 94.47, -29.15 -64.06, 143.12 APE12-dist-in 12.974 APE11-dist-in 10.879 APE10-dist-in 5.979 APE9-dist-in 3.017 None None None XRAY 2.9 0.208 0.238 B 442 358 0 0 0 0 [[56, 340]] 1.0 9hv3 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q3DA 35 385 420.0 STU:451 Type1 Active DFGin 7.206 14.411 BLAminus -139.48, 178.33 63.94, 87.17 -99.43, 23.77 282.58, 69.4 -66.25, -14.58 in-in in 8.701 Saltbr-in 2.855 HRD-in -65.74, -44.7 66.01, 11.52 in-in-in SNCiii in-in ActLoopNT-in 3.036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.53, 169.72 APE9-dihe-na 81.56, 143.56 APE8-dihe-in -91.54, 154.32 APE8-rot-in 294.67 APE67-dihe-inflip 96.36, -28.56 -51.12, 132.48 APE12-dist-in 13.074 APE11-dist-in 11.108 APE10-dist-in 6.087 APE9-dist-in 3.274 None None None XRAY 2.2 0.23 0.252 A 424 339 12 0 0 0 [[56, 340]] 1.0 1q3d CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q3DB 35 383 420.0 STU:452 Type1 Active DFGin 7.26 14.419 BLAminus -137.95, 177.39 64.41, 87.07 -97.99, 22.53 282.7, 70.11 -63.96, -17.29 in-in in 8.708 Saltbr-in 2.972 HRD-in -67.72, -45.35 66.86, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.75, 170.28 APE9-dihe-na 79.08, 144.81 APE8-dihe-in -89.94, 151.95 APE8-rot-in 299.26 APE67-dihe-inflip 101.61, -31.22 -54.51, 132.99 APE12-dist-in 13.085 APE11-dist-in 11.088 APE10-dist-in 6.146 APE9-dist-in 3.238 None None None XRAY 2.2 0.23 0.252 B 424 339 10 0 0 0 [[56, 340]] 1.0 1q3d CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q3WA 35 386 420.0 ATU:502 Type1 Active DFGin 7.146 13.952 BLAminus -137.77, 177.61 62.94, 83.24 -96.07, 24.67 288.22, 69.87 -66.71, -10.0 in-in in 8.322 Saltbr-in 2.924 HRD-in -67.11, -47.79 71.57, 6.31 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.32, 172.63 APE9-dihe-na 77.53, 136.48 APE8-dihe-in -79.93, 143.51 APE8-rot-in 298.62 APE67-dihe-in -62.35, -17.4 -13.52, -82.56 APE12-dist-in 13.075 APE11-dist-in 11.129 APE10-dist-in 5.964 APE9-dist-in 3.143 None None None XRAY 2.3 0.225 0.248 A 424 344 8 0 0 0 [[56, 340]] 1.0 1q3w CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q3WB 35 383 420.0 ATU:501 Type1 Active DFGin 7.09 14.27 BLAminus -140.46, 175.46 63.78, 84.76 -97.02, 22.89 286.31, 71.96 -64.9, -10.6 in-in in 8.547 Saltbr-in 2.792 HRD-in -67.92, -47.98 71.69, 6.95 in-in-in SNCiii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.2, 172.08 APE9-dihe-na 78.0, 136.99 APE8-dihe-in -80.5, 143.58 APE8-rot-in 301.78 APE67-dihe-in -64.47, -16.3 -12.81, -81.64 APE12-dist-in 13.069 APE11-dist-in 11.111 APE10-dist-in 5.938 APE9-dist-in 3.147 None None None XRAY 2.3 0.225 0.248 B 424 341 8 0 0 0 [[56, 340]] 1.0 1q3w CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q41A 35 386 420.0 IXM:451 Type1 Active DFGin 7.096 13.742 BLAminus -140.31, 177.95 63.36, 85.31 -97.68, 24.93 285.2, 72.61 -64.62, -16.75 in-in in 8.182 Saltbr-in 2.845 HRD-in -70.03, -43.74 69.02, 2.85 in-in-in SNCiii in-in ActLoopNT-in 3.007 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.85, 173.09 APE9-dihe-na 80.34, 135.13 APE8-dihe-in -75.55, 139.31 APE8-rot-in 298.19 APE67-dihe-in -65.33, -18.78 -13.64, -78.26 APE12-dist-in 13.068 APE11-dist-in 11.057 APE10-dist-in 5.915 APE9-dist-in 3.225 None None None XRAY 2.1 0.229 0.245 A 424 339 13 0 0 0 [[56, 340]] 1.0 1q41 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q41B 35 383 420.0 IXM:452 Type1 Active DFGin 7.094 13.894 BLAminus -139.75, 177.7 62.59, 85.88 -97.92, 24.85 285.3, 70.28 -63.82, -17.54 in-in in 8.388 Saltbr-in 2.83 HRD-in -70.82, -46.38 71.27, 6.28 in-in-in SNCiii in-in ActLoopNT-in 3.007 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.0, 171.76 APE9-dihe-na 82.35, 130.54 APE8-dihe-in -71.97, 140.37 APE8-rot-in 298.15 APE67-dihe-in -64.0, -13.46 -11.43, -84.5 APE12-dist-in 13.056 APE11-dist-in 11.055 APE10-dist-in 5.884 APE9-dist-in 3.236 None None None XRAY 2.1 0.229 0.245 B 424 343 6 0 0 0 [[56, 340]] 1.0 1q41 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q4LA 35 386 420.0 679:451 Type1 Active DFGin 6.944 13.754 BLAminus -138.39, -176.39 57.74, 86.06 -99.56, 21.29 285.7, 72.79 -65.03, -5.34 in-in in 8.524 Saltbr-in 3.007 HRD-in -67.11, -46.06 68.04, 16.48 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -95.21, 168.86 APE9-dihe-na 81.69, 129.23 APE8-dihe-in -70.09, 146.41 APE8-rot-in 291.03 APE67-dihe-inflip 104.98, -29.32 -58.42, 137.67 APE12-dist-in 13.117 APE11-dist-in 11.352 APE10-dist-in 6.301 APE9-dist-in 3.339 None None None XRAY 2.77 0.212 0.251 A 424 342 10 0 0 0 [[56, 340]] 1.0 1q4l CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1Q4LB 35 383 420.0 679:452 Type1 Active DFGin 7.169 13.649 BLAminus -140.11, -177.14 58.72, 87.12 -99.76, 20.01 285.14, 71.58 -64.5, -5.39 in-in in 8.339 Saltbr-in 2.673 HRD-in -67.89, -45.11 67.21, 17.1 in-in-in SNCiii in-in ActLoopNT-in 2.996 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.61, 167.87 APE9-dihe-na 83.04, 132.56 APE8-dihe-in -74.69, 156.93 APE8-rot-in 311.31 APE67-dihe-inflip 93.39, -29.64 -61.08, 141.61 APE12-dist-in 13.098 APE11-dist-in 11.322 APE10-dist-in 6.253 APE9-dist-in 3.349 None None None XRAY 2.77 0.212 0.251 B 424 337 12 0 0 0 [[56, 340]] 1.0 1q4l CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3Q3BA 35 386 420.0 55E:421 Type1 Active DFGin 6.859 13.89 BLAminus -146.51, -174.92 60.73, 82.19 -97.34, 22.93 287.93, 77.72 -66.67, -8.01 in-in in 8.46 Saltbr-in 2.718 HRD-in -65.09, -51.43 75.32, 0.61 in-in-in SNCiii in-in ActLoopNT-in 3.024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.28, 172.26 APE9-dihe-na 79.45, 140.83 APE8-dihe-in -87.39, 149.52 APE8-rot-in 308.45 APE67-dihe-in -68.31, -14.9 -12.45, -80.03 APE12-dist-in 13.004 APE11-dist-in 11.06 APE10-dist-in 6.186 APE9-dist-in 3.146 None None None XRAY 2.7 0.228 0.259 A 424 344 8 0 0 0 [[56, 340]] 1.0 3q3b CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3Q3BB 35 383 420.0 55E:421 Type1 Active DFGin 6.944 13.767 BLAminus -148.03, -175.09 60.19, 82.65 -96.08, 19.99 287.37, 77.74 -64.82, -9.3 in-in in 8.443 Saltbr-in 2.789 HRD-in -64.26, -50.5 74.85, 0.78 in-in-in SNCiii in-in ActLoopNT-in 3.048 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.17, 172.11 APE9-dihe-na 80.0, 136.06 APE8-dihe-in -78.43, 156.9 APE8-rot-in 303.64 APE67-dihe-in -69.77, -0.18 -23.17, -84.47 APE12-dist-in 12.996 APE11-dist-in 11.045 APE10-dist-in 6.179 APE9-dist-in 3.102 None None None XRAY 2.7 0.228 0.259 B 424 341 8 0 0 0 [[56, 340]] 1.0 3q3b CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4J1RA 36 383 420.0 I5R:502 Type1 Active DFGin 7.143 14.149 BLAminus -140.34, -172.16 50.83, 73.0 -88.1, 31.44 288.82, 75.41 -70.78, -20.52 in-in in 8.339 Saltbr-in 3.026 HRD-in -70.85, -43.96 67.49, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.918 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.66, 159.85 APE9-dihe-na 83.41, 158.3 APE8-dihe-in -70.39, 137.75 APE8-rot-in 276.14 APE67-dihe-in -62.89, -24.7 -48.3, -48.41 APE12-dist-in 13.466 APE11-dist-in 11.878 APE10-dist-in 7.006 APE9-dist-in 3.199 None PTR216 PTR216 XRAY 2.702 0.174 0.193 A 424 344 4 0 0 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4J1RB 36 384 420.0 I5R:502 Type1 Active DFGin 7.16 14.132 BLAminus -138.14, -172.1 51.97, 73.85 -90.74, 32.74 288.65, 76.48 -71.96, -19.84 in-in in 8.351 Saltbr-in 3.08 HRD-in -72.6, -39.29 60.47, 16.92 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.96, 157.32 APE9-dihe-na 86.27, 160.84 APE8-dihe-in -74.2, 139.51 APE8-rot-in 270.87 APE67-dihe-in -63.78, -23.12 -48.17, -50.06 APE12-dist-in 13.461 APE11-dist-in 11.633 APE10-dist-in 6.981 APE9-dist-in 3.199 None PTR216 PTR216 XRAY 2.702 0.174 0.193 B 424 347 2 0 0 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4J1RC 36 384 420.0 I5R:502 Type1 Active DFGin 7.154 14.145 BLAminus -137.53, -170.95 51.06, 74.57 -90.65, 33.09 289.21, 75.99 -73.08, -20.73 in-in in 8.344 Saltbr-in 3.009 HRD-in -71.61, -39.59 60.78, 16.42 in-in-in SNCiii in-in ActLoopNT-in 2.951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.54, 161.15 APE9-dihe-na 82.95, 157.27 APE8-dihe-in -71.13, 139.05 APE8-rot-in 271.75 APE67-dihe-in -63.34, -23.83 -48.75, -48.68 APE12-dist-in 13.475 APE11-dist-in 11.975 APE10-dist-in 7.027 APE9-dist-in 3.219 None PTR216 PTR216 XRAY 2.702 0.174 0.193 C 424 345 4 0 0 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4J1RD 36 384 420.0 I5R:502 Type1 Active DFGin 7.157 14.143 BLAminus -136.3, -170.0 51.29, 73.39 -89.98, 32.08 288.97, 75.59 -72.78, -18.14 in-in in 8.347 Saltbr-in 3.082 HRD-in -65.4, -45.24 73.44, 1.93 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.81, 157.82 APE9-dihe-na 85.66, 159.76 APE8-dihe-in -71.48, 137.15 APE8-rot-in 266.3 APE67-dihe-in -62.21, -25.06 -46.41, -50.2 APE12-dist-in 13.465 APE11-dist-in 11.902 APE10-dist-in 7.024 APE9-dist-in 3.117 None PTR216 PTR216 XRAY 2.702 0.174 0.193 D 424 346 3 0 0 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5HLNA 34 384 420.0 65C:501 Type1 Active DFGin 6.971 13.539 BLAminus -145.82, 177.83 61.52, 84.96 -98.63, 20.2 288.24, 74.65 -61.35, -16.22 in-in in 8.64 Saltbr-in 2.97 HRD-in -72.97, -42.53 59.11, 33.41 in-in-in SNCiii in-in ActLoopNT-in 2.966 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.08, -68.13 APE9-dihe-na -70.88, 179.27 APE8-dihe-in -73.41, 154.88 APE8-rot-in 283.39 APE67-dihe-in -59.67, -27.13 -52.94, -57.58 APE12-dist-in 13.109 APE11-dist-in 11.767 APE10-dist-in 7.214 APE9-dist-in 3.907 None PTR216 PTR216 XRAY 3.1 0.173 0.236 A 424 347 4 0 0 0 [[56, 340]] 1.0 5hln CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5HLPA 36 382 420.0 65A:501 Type1 Active DFGin 7.186 14.396 BLAminus -136.58, -178.8 62.45, 78.77 -95.76, 20.37 283.01, 75.68 -68.07, -12.1 in-in in 8.146 Saltbr-in 2.605 HRD-in -72.39, -43.73 64.36, 19.61 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.83, 176.24 APE9-dihe-na 71.02, 146.23 APE8-dihe-in -63.35, 144.14 APE8-rot-in 289.42 APE67-dihe-in -64.86, -21.95 -54.37, -48.38 APE12-dist-in 13.667 APE11-dist-in 11.819 APE10-dist-in 6.644 APE9-dist-in 3.298 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 A 424 339 8 0 0 0 [[56, 340]] 1.0 5hlp CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5HLPB 36 383 420.0 65A:501 Type1 Active DFGin 7.115 14.467 BLAminus -132.96, -174.02 57.79, 78.12 -94.26, 22.08 284.54, 74.66 -71.61, -17.17 in-in in 8.276 Saltbr-in 2.716 HRD-in -71.48, -47.76 70.66, 10.73 in-in-in SNCiii in-in ActLoopNT-in 2.837 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.37, 176.63 APE9-dihe-na 72.15, 149.52 APE8-dihe-in -67.13, 142.42 APE8-rot-in 293.57 APE67-dihe-in -63.1, -24.66 -49.41, -51.54 APE12-dist-in 13.356 APE11-dist-in 11.821 APE10-dist-in 6.581 APE9-dist-in 3.135 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 B 424 337 11 0 0 0 [[56, 340]] 1.0 5hlp CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5KPKA 35 384 420.0 6VK:500 Type1 Active DFGin 6.912 14.508 BLAminus -138.4, -178.64 58.08, 79.3 -90.22, 19.44 284.58, 73.09 -63.35, -18.32 in-in in 8.574 Saltbr-in 2.73 HRD-in -73.46, -47.41 66.88, 21.39 in-in-in SNCiii in-in ActLoopNT-in 2.95 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.73, 163.34 APE9-dihe-na 69.65, 162.27 APE8-dihe-in -73.86, 143.79 APE8-rot-in 303.06 APE67-dihe-in -60.34, -24.86 -54.25, -52.95 APE12-dist-in 13.597 APE11-dist-in 12.156 APE10-dist-in 7.487 APE9-dist-in 3.243 None PTR216 PTR216 XRAY 2.4 0.17 0.224 A 424 347 3 0 0 0 [[56, 340]] 1.0 5kpk CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5KPKB 35 383 420.0 6VK:500 Type1 Active DFGin 7.028 14.524 BLAminus -138.48, -175.82 55.16, 85.06 -97.98, 23.13 277.82, 78.64 -67.65, -21.76 in-in in 8.585 Saltbr-in 2.685 HRD-in -71.19, -45.78 65.3, 13.14 in-in-in SNCiii in-in ActLoopNT-in 3.004 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.69, 168.24 APE9-dihe-na 65.31, 163.84 APE8-dihe-in -77.16, 143.7 APE8-rot-in 304.59 APE67-dihe-in -57.42, -23.92 -54.57, -50.84 APE12-dist-in 13.693 APE11-dist-in 12.164 APE10-dist-in 7.395 APE9-dist-in 3.104 None PTR216 PTR216 XRAY 2.4 0.17 0.224 B 424 345 4 0 0 0 [[56, 340]] 1.0 5kpk CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5KPLA 36 384 420.0 6VL:500 Type1 Active DFGin 7.044 14.253 BLAminus -136.48, 178.55 58.11, 81.69 -92.72, 18.86 289.18, 73.73 -64.85, -20.41 in-in in 8.348 Saltbr-in 2.486 HRD-in -65.11, -50.47 69.64, 19.91 in-in-in SNCiii in-in ActLoopNT-in 3.088 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.42, 168.54 APE9-dihe-na 62.76, 158.29 APE8-dihe-in -78.28, 147.71 APE8-rot-in 310.05 APE67-dihe-in -62.4, -23.75 -53.92, -48.24 APE12-dist-in 13.434 APE11-dist-in 11.879 APE10-dist-in 7.137 APE9-dist-in 3.388 None PTR216 PTR216 XRAY 2.6 0.182 0.244 A 424 340 9 0 0 0 [[56, 340]] 1.0 5kpl CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5KPLB 36 383 420.0 6VL:500 Type1 Active DFGin 7.154 14.616 BLAminus -138.92, -172.41 52.88, 79.26 -88.95, 20.81 278.36, 73.5 -72.97, -16.23 in-in in 8.498 Saltbr-in 2.971 HRD-in -70.3, -40.66 56.94, 24.57 in-in-in SNCiii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.07, 160.76 APE9-dihe-na 66.33, 169.2 APE8-dihe-in -85.14, 144.57 APE8-rot-in 313.48 APE67-dihe-in -71.14, -21.99 -47.02, -47.87 APE12-dist-in 13.645 APE11-dist-in 11.859 APE10-dist-in 7.367 APE9-dist-in 3.38 None PTR216 PTR216 XRAY 2.6 0.182 0.244 B 424 340 8 0 0 0 [[56, 340]] 1.0 5kpl CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5KPMA 36 383 420.0 6VM:500 Type1 Active DFGin 7.179 14.152 BLAminus -127.54, 178.59 63.4, 85.66 -102.69, 28.41 287.99, 66.47 -62.48, -34.28 in-in in 8.406 Saltbr-in 2.669 HRD-in -73.98, -45.27 60.61, 25.04 in-in-in SNCiii in-in ActLoopNT-in 2.733 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.88, 162.98 APE9-dihe-na 64.81, 161.74 APE8-dihe-in -75.86, 141.16 APE8-rot-in 297.33 APE67-dihe-in -64.41, -17.12 -48.06, -52.48 APE12-dist-in 13.62 APE11-dist-in 11.838 APE10-dist-in 7.363 APE9-dist-in 3.261 None PTR216 PTR216 XRAY 2.69 0.178 0.24 A 424 345 3 0 0 0 [[56, 340]] 1.0 5kpm CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5KPMB 36 384 420.0 6VM:500 Type1 Active DFGin 7.141 14.638 BLAminus -142.12, 178.63 60.71, 81.6 -96.16, 22.05 281.72, 76.19 -66.25, -7.91 in-in in 8.609 Saltbr-in 2.581 HRD-in -65.22, -49.2 64.23, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.34, 163.89 APE9-dihe-na 62.78, 158.8 APE8-dihe-in -77.09, 139.57 APE8-rot-in 302.93 APE67-dihe-in -64.17, -18.23 -41.12, -52.04 APE12-dist-in 13.559 APE11-dist-in 11.972 APE10-dist-in 7.47 APE9-dist-in 3.193 None PTR216 PTR216 XRAY 2.69 0.178 0.24 B 424 346 3 0 0 0 [[56, 340]] 1.0 5kpm CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4IQ6A 37 382 420.0 IQ6:501 Type1 Active DFGin 7.068 14.008 BLAminus -142.1, 176.37 68.23, 72.95 -88.9, 16.75 291.61, 92.77 -55.61, -37.28 in-in in 8.574 Saltbr-in 2.841 HRD-in -66.67, -43.42 72.45, -14.35 in-in-in SNCiii in-in ActLoopNT-in 3.012 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.44, 163.79 APE9-dihe-na 84.06, 140.31 APE8-dihe-in -95.86, 141.6 APE8-rot-in 294.32 APE67-dihe-inflip 102.08, -40.06 -38.49, 130.32 APE12-dist-in 13.214 APE11-dist-in 11.007 APE10-dist-in 6.193 APE9-dist-in 3.167 None None None XRAY 3.12 0.188 0.227 A 426 324 22 0 0 0 [[56, 340]] 1.0 4iq6 CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3SAYA 35 384 420.0 OFT:431 Type1 Active DFGin 6.924 14.208 BLAminus -134.06, -176.24 58.1, 80.75 -95.49, 24.69 285.79, 80.8 -58.99, -23.52 in-in in 8.765 Saltbr-in 2.683 HRD-in -76.77, -47.73 71.86, 15.98 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 177.68 APE9-dihe-na 70.36, 150.2 APE8-dihe-in -70.69, 142.5 APE8-rot-in 303.06 APE67-dihe-in -64.8, -21.63 -53.21, -43.25 APE12-dist-in 13.475 APE11-dist-in 11.768 APE10-dist-in 6.474 APE9-dist-in 3.141 None PTR216 PTR216 XRAY 2.231 0.202 0.23 A 430 348 2 0 0 0 [[56, 340]] 1.0 3say CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3SAYB 35 382 420.0 OFT:431 Type1 Active DFGin 7.095 14.208 BLAminus -125.43, -174.49 59.4, 82.08 -94.07, 22.41 283.95, 82.11 -68.04, -11.91 in-in in 8.776 Saltbr-in 2.596 HRD-in -71.92, -46.59 68.83, 6.83 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.5, 172.68 APE9-dihe-na 72.51, 152.54 APE8-dihe-in -66.45, 133.95 APE8-rot-in 293.34 APE67-dihe-in -62.41, -25.02 -42.21, -48.58 APE12-dist-in 13.503 APE11-dist-in 11.83 APE10-dist-in 6.704 APE9-dist-in 3.093 None PTR216 PTR216 XRAY 2.231 0.202 0.23 B 430 348 0 0 0 0 [[56, 340]] 1.0 3say CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4PTCA 36 381 420.0 2WE:501 Type1 Active DFGin 6.936 14.398 BLAminus -147.73, -174.11 62.98, 81.81 -100.26, 25.83 284.28, 79.03 -59.65, -43.28 in-in in 9.162 Saltbr-in 2.729 HRD-in -73.84, -45.42 69.86, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.77 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.04, 172.51 APE9-dihe-na 77.59, 144.28 APE8-dihe-in -89.54, 156.63 APE8-rot-in 297.82 APE67-dihe-inflip 95.7, -27.15 -58.15, 143.88 APE12-dist-in 13.05 APE11-dist-in 10.779 APE10-dist-in 6.004 APE9-dist-in 3.272 None None None XRAY 2.711 0.217 0.281 A 441 342 4 0 0 0 [[56, 340]] 1.0 4ptc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4PTCB 35 385 420.0 2WE:501 Type1 Active DFGin 7.213 14.605 BLAminus -123.82, -167.89 50.38, 80.91 -94.33, 28.59 284.85, 71.64 -64.12, -29.45 in-in in 8.924 Saltbr-in 2.402 HRD-in -67.43, -42.31 63.02, 14.07 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.89, 173.71 APE9-dihe-na 81.21, 152.66 APE8-dihe-in -112.25, 156.82 APE8-rot-in 292.56 APE67-dihe-inflip 100.85, -22.79 -44.26, 123.15 APE12-dist-in 13.083 APE11-dist-in 10.918 APE10-dist-in 5.89 APE9-dist-in 3.28 None None None XRAY 2.711 0.217 0.281 B 441 347 4 0 0 0 [[56, 340]] 1.0 4ptc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4PTEA 36 382 420.0 2WF:501 Type1 Active DFGin 6.932 14.017 BLAminus -141.21, 178.04 57.99, 89.39 -100.23, 24.26 286.38, 75.9 -68.08, -19.02 in-in in 8.716 Saltbr-in 2.635 HRD-in -73.56, -44.45 69.11, 4.74 in-in-in SNCiii in-in ActLoopNT-in 2.792 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.74, 175.98 APE9-dihe-na 75.98, 148.82 APE8-dihe-in -103.79, 152.51 APE8-rot-in 295.33 APE67-dihe-inflip 95.08, -28.26 -38.95, 126.56 APE12-dist-in 12.979 APE11-dist-in 10.89 APE10-dist-in 5.883 APE9-dist-in 3.088 None None None XRAY 2.033 0.17 0.195 A 441 341 6 0 0 0 [[56, 340]] 1.0 4pte CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4PTEB 36 385 420.0 2WF:501 Type1 Active DFGin 6.918 13.937 BLAminus -137.07, 179.43 58.52, 88.98 -101.38, 27.88 284.28, 76.88 -69.85, -20.65 in-in in 8.484 Saltbr-in 2.685 HRD-in -70.9, -46.61 73.05, 2.3 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.76, 178.59 APE9-dihe-na 72.73, 147.77 APE8-dihe-in -103.48, 150.66 APE8-rot-in 296.89 APE67-dihe-inflip 94.67, -27.57 -36.66, 125.81 APE12-dist-in 12.935 APE11-dist-in 10.88 APE10-dist-in 5.877 APE9-dist-in 3.154 None None None XRAY 2.033 0.17 0.195 B 441 347 3 0 0 0 [[56, 340]] 1.0 4pte CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4PTGA 36 382 420.0 2WG:501 Type1 Active DFGin 7.003 13.916 BLAminus -132.5, 179.85 66.28, 92.0 -106.7, 26.9 285.24, 77.28 -68.07, -25.88 in-in in 8.541 Saltbr-in 2.828 HRD-in -68.57, -44.88 68.54, 10.31 in-in-in SNCiii in-in ActLoopNT-in 2.939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.39, 169.96 APE9-dihe-na 80.02, 147.16 APE8-dihe-in -96.08, 142.52 APE8-rot-in 290.31 APE67-dihe-inflip 90.23, -35.22 -45.66, 142.01 APE12-dist-in 13.056 APE11-dist-in 11.019 APE10-dist-in 6.12 APE9-dist-in 3.284 None None None XRAY 2.361 0.173 0.211 A 441 333 14 0 0 0 [[56, 340]] 1.0 4ptg CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4PTGB 37 385 420.0 2WG:501 Type1 Active DFGin 6.951 13.863 BLAminus -136.28, -175.42 57.62, 87.0 -101.31, 27.32 285.42, 76.21 -67.67, -26.13 in-in in 8.437 Saltbr-in 2.705 HRD-in -71.07, -46.44 71.76, 6.12 in-in-in SNCiii in-in ActLoopNT-in 2.9 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.44, 175.88 APE9-dihe-na 76.35, 149.91 APE8-dihe-in -109.95, 151.08 APE8-rot-in 289.69 APE67-dihe-inflip 91.44, -30.76 -44.23, 136.59 APE12-dist-in 12.988 APE11-dist-in 11.009 APE10-dist-in 5.91 APE9-dist-in 3.16 None None None XRAY 2.361 0.173 0.211 B 441 332 17 0 0 0 [[56, 340]] 1.0 4ptg CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8DJCA 35 382 420.0 UAU:501 Type1 Active DFGin 7.107 13.645 BLAminus -130.93, 175.08 68.46, 84.27 -99.8, 25.87 290.84, 77.95 -66.29, -22.25 in-in in 8.442 Saltbr-in 2.699 HRD-in -67.33, -44.59 69.12, 7.74 in-in-in SNCiii in-in ActLoopNT-in 2.984 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 169.18 APE9-dihe-na 83.11, 139.06 APE8-dihe-in -86.29, 148.88 APE8-rot-in 301.44 APE67-dihe-inflip 95.96, -28.78 -50.91, 136.23 APE12-dist-in 12.912 APE11-dist-in 10.831 APE10-dist-in 5.804 APE9-dist-in 3.257 None None None XRAY 2.463 0.217 0.242 A 441 331 17 0 0 0 [[56, 340]] 1.0 8djc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8DJCB 35 385 420.0 UAU:501 Type1 Active DFGin 7.125 13.633 BLAminus -137.19, 179.71 59.65, 83.27 -96.94, 27.03 290.51, 79.22 -67.53, -21.56 in-in in 8.328 Saltbr-in 2.738 HRD-in -65.99, -44.91 69.53, 7.25 in-in-in SNCiii in-in ActLoopNT-in 2.986 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.05, 167.49 APE9-dihe-na 82.24, 138.29 APE8-dihe-in -85.04, 145.47 APE8-rot-in 300.63 APE67-dihe-inflip 98.12, -32.04 -46.91, 135.02 APE12-dist-in 12.942 APE11-dist-in 10.888 APE10-dist-in 5.944 APE9-dist-in 3.259 None None None XRAY 2.463 0.217 0.242 B 441 332 19 0 0 0 [[56, 340]] 1.0 8djc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8DJDA 36 383 420.0 U3E:501 Type1 Active DFGin 7.183 13.878 BLAminus -134.36, -179.72 59.88, 85.28 -97.18, 26.66 285.76, 75.79 -65.91, -27.91 in-in in 8.357 Saltbr-in 2.704 HRD-in -66.89, -45.93 70.71, 8.73 in-in-in SNCiii in-in ActLoopNT-in 2.974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -97.03, 169.31 APE9-dihe-na 77.5, 142.18 APE8-dihe-in -93.09, 155.03 APE8-rot-in 301.61 APE67-dihe-inflip 94.8, -31.52 -52.67, 137.81 APE12-dist-in 13.059 APE11-dist-in 11.039 APE10-dist-in 6.129 APE9-dist-in 3.198 None None None XRAY 2.205 0.209 0.222 A 441 338 10 0 0 0 [[56, 340]] 1.0 8djd CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8DJDB 36 384 420.0 U3E:501 Type1 Active DFGin 7.129 13.919 BLAminus -133.17, 179.77 59.91, 85.17 -97.09, 26.57 285.62, 75.36 -66.56, -27.45 in-in in 8.347 Saltbr-in 2.697 HRD-in -66.65, -46.07 70.85, 8.52 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.46, 170.54 APE9-dihe-na 79.57, 140.07 APE8-dihe-in -94.46, 154.56 APE8-rot-in 301.16 APE67-dihe-inflip 94.52, -31.07 -52.58, 138.22 APE12-dist-in 13.086 APE11-dist-in 11.08 APE10-dist-in 6.077 APE9-dist-in 3.217 None None None XRAY 2.205 0.209 0.222 B 441 341 8 0 0 0 [[56, 340]] 1.0 8djd CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8DJEA 36 384 420.0 U6S:501 Type1 Active DFGin 7.26 13.369 BLAminus -139.51, 175.88 67.17, 88.55 -102.31, 22.49 287.71, 78.25 -63.99, -27.99 in-in in 8.313 Saltbr-in 2.716 HRD-in -68.38, -45.52 70.24, 12.16 in-in-in SNCiii in-in ActLoopNT-in 2.893 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.85, 166.32 APE9-dihe-na 87.14, 140.36 APE8-dihe-in -88.6, 149.46 APE8-rot-in 293.07 APE67-dihe-inflip 99.13, -30.7 -44.53, 124.89 APE12-dist-in 12.957 APE11-dist-in 10.867 APE10-dist-in 6.044 APE9-dist-in 3.353 None None None XRAY 2.374 0.201 0.227 A 441 347 2 0 0 0 [[56, 340]] 1.0 8dje CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8DJEB 36 385 420.0 U6S:501 Type1 Active DFGin 7.239 13.421 BLAminus -137.87, 177.52 63.92, 86.56 -101.17, 24.78 290.39, 74.84 -68.33, -25.47 in-in in 8.265 Saltbr-in 2.736 HRD-in -65.34, -46.08 68.76, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.12, 167.71 APE9-dihe-na 84.3, 145.94 APE8-dihe-in -98.8, 148.34 APE8-rot-in 293.36 APE67-dihe-inflip 97.13, -37.27 -40.76, 129.94 APE12-dist-in 12.957 APE11-dist-in 10.932 APE10-dist-in 5.908 APE9-dist-in 3.263 None None None XRAY 2.374 0.201 0.227 B 441 343 7 0 0 0 [[56, 340]] 1.0 8dje CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8FF8A 36 382 420.0 XV0:501 Type1 Active DFGin 7.2 13.736 BLAminus -135.89, 175.65 65.86, 84.5 -97.83, 25.7 284.17, 77.94 -66.05, -27.44 in-in in 8.341 Saltbr-in 2.752 HRD-in -68.43, -43.4 70.29, 3.62 in-in-in SNCiii in-in ActLoopNT-in 2.842 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 167.87 APE9-dihe-na 84.02, 136.04 APE8-dihe-in -86.03, 151.96 APE8-rot-in 298.92 APE67-dihe-inflip 95.48, -31.71 -43.39, 129.41 APE12-dist-in 12.741 APE11-dist-in 10.753 APE10-dist-in 5.791 APE9-dist-in 3.211 None None None XRAY 2.33 0.198 0.217 A 441 347 0 0 0 0 [[56, 340]] 1.0 8ff8 CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8FF8B 36 385 420.0 XV0:501 Type1 Active DFGin 7.2 13.811 BLAminus -130.19, -175.53 57.72, 85.5 -98.92, 25.25 283.55, 78.69 -65.7, -29.77 in-in in 8.339 Saltbr-in 2.746 HRD-in -67.11, -43.98 70.41, 3.15 in-in-in SNCiii in-in ActLoopNT-in 2.825 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.86, 169.83 APE9-dihe-na 81.04, 142.01 APE8-dihe-in -96.19, 150.13 APE8-rot-in 300.46 APE67-dihe-inflip 95.56, -32.32 -40.34, 130.68 APE12-dist-in 12.779 APE11-dist-in 10.784 APE10-dist-in 5.825 APE9-dist-in 3.218 None None None XRAY 2.33 0.198 0.217 B 441 346 4 0 0 0 [[56, 340]] 1.0 8ff8 CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3F88A 35 383 420.0 3HT:999 Type1 Active DFGin 7.247 13.73 BLAminus -137.96, -171.11 53.2, 96.02 -109.46, 31.55 277.23, 77.74 -85.58, 3.2 in-in in 8.62 Saltbr-in 2.516 HRD-in -66.41, -48.84 71.78, 26.38 in-in-in SNCiii in-in ActLoopNT-in 3.141 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.98, 165.73 APE9-dihe-na 69.33, 171.05 APE8-dihe-in -86.85, 130.82 APE8-rot-in 314.66 APE67-dihe-in -71.94, -20.16 -24.55, -52.13 APE12-dist-in 13.547 APE11-dist-in 12.041 APE10-dist-in 7.341 APE9-dist-in 3.599 None PTR216 PTR216 XRAY 2.6 0.204 0.281 A 349 341 8 0 0 0 [[56, 340]] 1.0 3f88 CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3F88B 35 383 420.0 3HT:999 Type1 Active DFGin 7.0 13.651 BLAminus -143.93, 176.87 66.18, 95.41 -113.06, 21.86 281.61, 81.82 -72.47, -7.16 in-in in 8.765 Saltbr-in 2.671 HRD-in -64.13, -56.14 79.67, 28.55 in-in-in SNCiii in-in ActLoopNT-in 3.176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.92, 167.15 APE9-dihe-na 65.97, 165.61 APE8-dihe-in -80.57, 145.62 APE8-rot-in 308.56 APE67-dihe-in -71.31, -21.5 -44.75, -45.4 APE12-dist-in 13.509 APE11-dist-in 11.967 APE10-dist-in 7.257 APE9-dist-in 3.406 None PTR216 PTR216 XRAY 2.6 0.204 0.281 B 349 341 8 0 0 0 [[56, 340]] 1.0 3f88 CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACCA 35 385 420.0 7YG:1387 Type1 Active DFGin 7.183 13.581 BLAminus -136.28, 179.66 61.59, 88.25 -100.04, 20.56 281.3, 79.98 -65.9, -21.03 in-in in 8.347 Saltbr-in 2.762 HRD-in -66.74, -44.81 68.93, 1.06 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.14, 170.6 APE9-dihe-na 77.6, 138.09 APE8-dihe-in -85.62, 145.43 APE8-rot-in 296.7 APE67-dihe-inflip 94.96, -30.16 -47.88, 136.19 APE12-dist-in 13.034 APE11-dist-in 10.957 APE10-dist-in 5.889 APE9-dist-in 3.171 None None None XRAY 2.21 0.191 0.219 A 465 351 0 0 0 0 [[56, 340]] 1.0 4acc CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACCB 35 385 420.0 7YG:1386 Type1 Active DFGin 7.228 13.524 BLAminus -136.66, 179.59 61.79, 88.29 -99.73, 21.22 281.91, 80.18 -66.08, -22.29 in-in in 8.245 Saltbr-in 2.871 HRD-in -66.61, -45.06 69.24, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.27, 172.02 APE9-dihe-na 75.79, 137.96 APE8-dihe-in -86.62, 146.41 APE8-rot-in 295.61 APE67-dihe-inflip 93.46, -30.62 -49.23, 136.97 APE12-dist-in 13.056 APE11-dist-in 11.009 APE10-dist-in 5.912 APE9-dist-in 3.182 None None None XRAY 2.21 0.191 0.219 B 465 351 0 0 0 0 [[56, 340]] 1.0 4acc CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACDA 35 385 420.0 GR9:1385 Type1 Active DFGin 7.186 13.357 BLAminus -142.44, 176.49 66.05, 88.14 -100.25, 16.93 286.04, 81.9 -64.04, -24.03 in-in in 8.306 Saltbr-in 2.937 HRD-in -63.25, -48.42 73.67, 5.76 in-in-in SNCiii in-in ActLoopNT-in 2.883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.94, 167.01 APE9-dihe-na 78.77, 128.64 APE8-dihe-in -74.85, 143.25 APE8-rot-in 302.95 APE67-dihe-inflip 99.55, -31.6 -49.31, 132.99 APE12-dist-in 12.877 APE11-dist-in 10.868 APE10-dist-in 5.91 APE9-dist-in 3.21 None None None XRAY 2.6 0.18 0.226 A 465 351 0 0 0 0 [[56, 340]] 1.0 4acd CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACDB 35 385 420.0 GR9:1385 Type1 Active DFGin 7.141 13.377 BLAminus -142.06, 177.81 64.05, 89.32 -100.31, 16.47 285.95, 82.89 -62.46, -26.08 in-in in 8.223 Saltbr-in 2.941 HRD-in -62.52, -48.15 72.88, 6.33 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.53, 167.96 APE9-dihe-na 77.33, 127.92 APE8-dihe-in -74.4, 143.25 APE8-rot-in 302.61 APE67-dihe-inflip 99.75, -32.16 -47.58, 132.33 APE12-dist-in 12.928 APE11-dist-in 10.947 APE10-dist-in 5.956 APE9-dist-in 3.211 None None None XRAY 2.6 0.18 0.226 B 465 351 0 0 0 0 [[56, 340]] 1.0 4acd CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACGA 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.003 13.717 BLAminus -136.29, 179.17 66.16, 92.5 -104.82, 26.85 285.89, 83.54 -71.26, -31.7 in-in in 8.275 Saltbr-in 2.866 HRD-in -62.3, -47.68 71.35, 0.06 in-in-in SNCiii in-in ActLoopNT-in 2.99 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.26, 169.3 APE9-dihe-na 82.24, 136.71 APE8-dihe-in -91.92, 145.05 APE8-rot-in 294.1 APE67-dihe-inflip 97.4, -31.68 -47.8, 134.4 APE12-dist-in 12.946 APE11-dist-in 10.981 APE10-dist-in 5.928 APE9-dist-in 3.292 None None None XRAY 2.6 0.177 0.225 A 465 351 0 0 0 0 [[56, 340]] 1.0 4acg CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACGB 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.06 13.61 BLAminus -135.89, 178.4 67.23, 92.34 -105.78, 27.09 285.23, 82.98 -71.05, -30.43 in-in in 8.379 Saltbr-in 2.98 HRD-in -63.74, -47.68 70.98, 1.15 in-in-in SNCiii in-in ActLoopNT-in 2.973 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.69, 168.91 APE9-dihe-na 83.12, 137.88 APE8-dihe-in -91.66, 145.04 APE8-rot-in 292.39 APE67-dihe-inflip 98.28, -31.78 -48.39, 133.48 APE12-dist-in 12.918 APE11-dist-in 10.934 APE10-dist-in 5.917 APE9-dist-in 3.29 None None None XRAY 2.6 0.177 0.225 B 465 351 0 0 0 0 [[56, 340]] 1.0 4acg CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACHA 35 385 420.0 KDI:1386 Type1 Active DFGin 7.131 13.843 BLAminus -136.87, 179.55 65.58, 91.16 -104.2, 25.64 286.28, 84.07 -69.39, -35.2 in-in in 8.234 Saltbr-in 2.935 HRD-in -61.5, -48.36 72.42, -0.28 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.62, 166.44 APE9-dihe-na 83.56, 135.36 APE8-dihe-in -86.16, 143.31 APE8-rot-in 295.11 APE67-dihe-inflip 98.78, -32.06 -48.27, 133.26 APE12-dist-in 12.998 APE11-dist-in 11.059 APE10-dist-in 5.983 APE9-dist-in 3.322 None None None XRAY 2.6 0.231 0.252 A 465 351 0 0 0 0 [[56, 340]] 1.0 4ach CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4ACHB 35 385 420.0 KDI:1386 Type1 Active DFGin 7.081 13.716 BLAminus -136.91, 178.72 65.4, 91.31 -104.6, 25.63 285.26, 83.9 -68.47, -34.59 in-in in 8.36 Saltbr-in 2.938 HRD-in -60.93, -48.9 72.19, 0.38 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.1, 166.35 APE9-dihe-na 83.22, 136.77 APE8-dihe-in -87.16, 144.14 APE8-rot-in 294.96 APE67-dihe-inflip 98.6, -31.77 -49.65, 133.73 APE12-dist-in 12.935 APE11-dist-in 10.985 APE10-dist-in 5.938 APE9-dist-in 3.29 None None None XRAY 2.6 0.231 0.252 B 465 351 0 0 0 0 [[56, 340]] 1.0 4ach CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5OY4A 36 385 420.0 B4K:504 Type1.5_Back Active DFGin 6.999 13.822 BLAminus -130.87, 178.64 57.91, 86.19 -95.47, 21.04 282.05, 81.42 -63.36, -27.5 in-in in 8.088 Saltbr-in 2.722 HRD-in -68.24, -44.36 63.28, 15.03 in-in-in SNCiii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.23, 157.34 APE9-dihe-na 87.05, 159.63 APE8-dihe-in -83.83, 115.67 APE8-rot-in 295.36 APE67-dihe-in -60.03, -25.52 -23.01, -56.29 APE12-dist-in 13.558 APE11-dist-in 11.689 APE10-dist-in 7.058 APE9-dist-in 3.446 None PTR216 PTR216 XRAY 3.2 0.196 0.229 A 420 350 0 0 0 0 [[56, 340]] 1.0 5oy4 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4IQ6B 37 382 420.0 IQ6:501 Type1.5_Back Active DFGin 7.065 14.057 BLAminus -142.54, 175.49 69.06, 72.09 -88.69, 16.42 291.37, 92.47 -54.24, -38.91 in-in in 8.609 Saltbr-in 2.85 HRD-in -66.96, -42.68 72.42, -15.31 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.08, 167.69 APE9-dihe-na 81.68, 134.42 APE8-dihe-in -80.06, 146.43 APE8-rot-in 285.37 APE67-dihe-inflip 104.71, -27.8 -48.51, 126.71 APE12-dist-in 13.148 APE11-dist-in 10.908 APE10-dist-in 6.244 APE9-dist-in 3.115 None None None XRAY 3.12 0.188 0.227 B 426 332 14 0 0 0 [[56, 340]] 1.0 4iq6 CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6Y9SA 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.759 13.615 ABAminus -144.68, -36.37 -95.25, 102.78 -104.54, 22.52 286.7, 80.89 -71.31, -22.3 in-in in 8.469 Saltbr-in 2.731 HRD-in -69.96, -46.79 66.16, 22.69 in-in-out SNCiio in-out ActLoopNT-in 2.869 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.41, 160.13 APE9-dihe-na 78.21, 163.56 APE8-dihe-in -74.57, 133.14 APE8-rot-out 174.03 APE67-dihe-in -60.25, -21.67 -45.31, -52.5 APE12-dist-in 13.391 APE11-dist-in 11.634 APE10-dist-in 6.815 APE9-dist-in 3.217 None PTR216 PTR216 XRAY 2.03 0.204 0.249 A 350 344 5 0 0 0 [[56, 340]] 1.0 6y9s CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6Y9SB 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.466 13.644 ABAminus -142.08, -29.11 -101.71, 107.32 -109.34, 26.02 290.64, 79.47 -70.13, -24.37 in-in in 8.627 Saltbr-in 2.626 HRD-in -62.98, -47.75 66.63, 19.7 in-in-out SNCiio in-out ActLoopNT-in 2.871 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -149.54, 160.17 APE9-dihe-na 74.78, 156.26 APE8-dihe-in -72.21, 136.72 APE8-rot-out 179.96 APE67-dihe-in -63.91, -18.81 -47.88, -49.22 APE12-dist-in 13.498 APE11-dist-in 11.696 APE10-dist-in 6.94 APE9-dist-in 3.172 None PTR216 PTR216 XRAY 2.03 0.204 0.249 B 350 340 9 0 0 0 [[56, 340]] 1.0 6y9s CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4NM0A 26 383 420.0 ADP:60408 ATPlike Inactive DFGin 6.641 14.213 BLAminus -133.4, -174.33 56.9, 85.51 -105.72, 27.83 287.31, 80.39 -76.48, -2.57 in-in in 8.774 Saltbr-in 3.094 HRD-in -69.87, -45.12 67.03, 14.87 in-in-out SNCiio in-out ActLoopNT-in 2.927 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -71.29, 168.54 APE9-dihe-na 70.19, 144.11 APE8-dihe-in -96.47, 160.21 APE8-rot-out 64.82 APE67-dihe-inflip 78.46, -27.02 -43.67, 149.07 APE12-dist-in 13.091 APE11-dist-in 10.885 APE10-dist-in 6.571 APE9-dist-in 3.135 None None None XRAY 2.5 0.193 0.239 A 389 355 0 0 0 0 [[56, 340]] 1.0 4nm0 CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8XN6B 26 386 420.0 ANP:501 ATPlike Inactive DFGin 6.538 13.65 BLAminus -128.79, 173.26 73.68, 79.74 -95.9, 22.51 291.63, 80.46 -68.54, -21.83 in-in in 8.329 Saltbr-in 2.823 HRD-in -66.59, -53.03 79.09, 5.6 in-in-out SNCiio in-out ActLoopNT-in 2.951 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -88.32, 165.9 APE9-dihe-na 83.63, 132.42 APE8-dihe-in -59.67, 147.17 APE8-rot-out 189.94 APE67-dihe-in -64.51, -21.68 -60.38, -49.59 APE12-dist-in 13.024 APE11-dist-in 10.97 APE10-dist-in 5.846 APE9-dist-in 3.081 None None None XRAY 2.4 0.194 0.242 B 421 359 2 0 0 0 [[56, 340]] 1.0 8xn6 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9X2VA 35 383 420.0 PG6:502 Allosteric Inactive DFGin 6.894 14.046 BLAminus -136.47, 179.58 67.71, 81.15 -94.13, 21.93 285.02, 80.61 -69.61, -16.35 in-in in 8.707 Saltbr-in 2.796 HRD-in -72.8, -46.17 70.48, 11.06 in-in-out SNCiio in-out ActLoopNT-in 2.929 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_iiii APE10-dihe-na -102.48, 5.03 APE9-dihe-na -128.33, 167.55 APE8-dihe-out 50.5, 42.65 APE8-rot-in 319.92 APE67-dihe-in -79.33, -58.3 -90.94, -21.28 APE12-dist-in 10.275 APE11-dist-in 11.184 APE10-dist-in 7.71 APE9-dist-in 4.04 None None None XRAY 1.39 0.179 0.195 A 359 347 2 0 0 0 [[56, 340]] 1.0 9x2v CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1I09B 37 382 420.0 No_ligand No_ligand Inactive DFGin 6.861 14.025 BLAminus -135.93, 178.35 61.75, 84.0 -100.67, 24.72 288.55, 74.93 -64.65, -15.56 in-in in 8.483 Saltbr-in 2.711 HRD-in -62.69, -41.62 66.11, 9.61 in-in-out SNCiio in-out ActLoopNT-in 2.953 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.33, -45.22 APE9-dihe-na -71.78, 167.71 APE8-dihe-in -94.58, 171.33 APE8-rot-out 74.32 APE67-dihe-in -65.52, -17.17 -44.16, -80.97 APE12-dist-in 12.764 APE11-dist-in 11.113 APE10-dist-in 6.221 APE9-dist-in 3.37 None None None XRAY 2.7 0.242 0.274 B 420 341 5 0 0 0 [[56, 340]] 1.0 1i09 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6HK7A 36 382 420.0 G8N:403 Type1 Inactive DFGin 7.181 13.926 BLAminus -137.45, -171.56 51.7, 92.53 -104.06, 22.16 271.05, 85.97 -65.5, -26.28 in-in in 8.435 Saltbr-in 2.767 HRD-in -53.21, -66.83 89.97, 19.54 in-in-out SNCiio in-out ActLoopNT-in 2.957 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -85.73, 172.92 APE9-dihe-na 79.4, 146.18 APE8-dihe-in -92.07, 85.52 APE8-rot-in 243.21 APE67-dihe-out 35.1, -40.06 22.07, -158.21 APE12-dist-in 13.29 APE11-dist-in 11.446 APE10-dist-in 6.781 APE9-dist-in 3.32 None PTR216 PTR216 XRAY 3.2 0.204 0.286 A 347 347 0 0 0 0 [[56, 340]] 1.0 6hk7 CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7SXHA 37 383 420.0 D1E:501 Type1 Inactive DFGin 6.65 13.944 BLAminus -139.68, -175.41 60.2, 74.18 -88.43, 22.79 288.62, 86.11 -74.83, -15.81 in-in in 8.167 Saltbr-in 2.858 HRD-in -67.33, -47.27 70.7, 6.58 in-in-out SNCiio in-out ActLoopNT-in 2.863 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -126.8, 168.99 APE9-dihe-na 70.82, 157.42 APE8-dihe-in -70.74, 147.57 APE8-rot-out 190.63 APE67-dihe-in -58.92, -21.73 -57.82, -47.78 APE12-dist-in 13.771 APE11-dist-in 11.975 APE10-dist-in 7.371 APE9-dist-in 3.432 None PTR216 PTR216 XRAY 2.09 0.216 0.255 A 347 341 6 0 0 0 [[56, 340]] 1.0 7sxh CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3F7ZA 35 383 420.0 34O:63000 Type1 Inactive DFGin 7.116 13.818 BLAminus -134.47, 172.11 69.02, 81.68 -97.3, 19.46 284.39, 70.02 -68.92, -10.86 in-in in 8.485 Saltbr-in 2.575 HRD-in -62.81, -48.18 67.57, 12.21 in-in-out SNCiio in-out ActLoopNT-in 2.95 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -139.18, 179.1 APE9-dihe-na 69.89, 157.17 APE8-dihe-in -75.28, 142.37 APE8-rot-out 185.5 APE67-dihe-in -55.86, -28.19 -45.56, -57.07 APE12-dist-in 13.5 APE11-dist-in 12.029 APE10-dist-in 6.815 APE9-dist-in 3.314 None PTR216 PTR216 XRAY 2.4 0.206 0.253 A 350 339 10 0 0 0 [[56, 340]] 1.0 3f7z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3SD0A 35 384 420.0 TSK:400 Type1 Inactive DFGin 6.893 13.678 BLAminus -139.29, -172.59 62.67, 82.92 -94.93, 18.52 283.9, 73.87 -68.11, -17.74 in-in in 8.419 Saltbr-in 2.824 HRD-in -68.02, -47.17 76.6, 11.56 in-in-out SNCiio in-out ActLoopNT-in 2.8 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -82.28, 176.65 APE9-dihe-na 71.42, 130.7 APE8-dihe-in -100.53, 166.25 APE8-rot-out 29.1 APE67-dihe-inflip 91.12, -25.82 -31.67, 128.67 APE12-dist-in 12.91 APE11-dist-in 10.81 APE10-dist-in 5.779 APE9-dist-in 3.042 None None None XRAY 2.7 0.179 0.254 A 350 350 0 0 0 0 [[56, 340]] 1.0 3sd0 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3ZDIA 36 384 420.0 UGJ:61386 Type1 Inactive DFGin 7.09 14.011 BLAminus -139.08, 169.73 59.85, 93.36 -102.57, 31.03 284.51, 75.61 -74.44, -6.01 in-in in 8.719 Saltbr-in 2.774 HRD-in -66.47, -49.36 70.61, -12.05 in-in-out SNCiio in-out ActLoopNT-in 2.874 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.6, -176.4 APE9-dihe-na 57.27, -141.25 APE8-dihe-in -136.89, 135.85 APE8-rot-out 188.96 APE67-dihe-in -60.18, -28.67 -48.24, -43.31 APE12-dist-in 13.777 APE11-dist-in 12.116 APE10-dist-in 7.549 APE9-dist-in 3.094 None PTR216 PTR216 XRAY 2.645 0.204 0.242 A 350 349 0 0 0 0 [[56, 340]] 1.0 3zdi CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4B7TA 35 384 420.0 CWT:1385 Type1 Inactive DFGin 6.733 14.135 BLAminus -139.29, -173.55 55.51, 80.28 -97.98, 26.2 284.11, 78.64 -70.02, -22.23 in-in in 8.826 Saltbr-in 2.732 HRD-in -65.66, -45.08 68.98, -4.07 in-in-out SNCiio in-out ActLoopNT-in 3.022 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -80.96, 174.72 APE9-dihe-na 79.02, 153.66 APE8-dihe-in -90.72, 141.08 APE8-rot-out 219.61 APE67-dihe-inflip 82.28, -25.01 -65.77, 158.92 APE12-dist-in 13.15 APE11-dist-in 11.315 APE10-dist-in 6.552 APE9-dist-in 3.122 None None None XRAY 2.772 0.197 0.235 A 350 350 0 0 0 0 [[56, 340]] 1.0 4b7t CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6HK3A 35 384 420.0 G8B:401 Type1 Inactive DFGin 6.919 13.749 BLAminus -140.26, -177.42 53.43, 89.98 -101.44, 26.95 281.28, 77.81 -71.94, -4.92 in-in in 8.265 Saltbr-in 2.52 HRD-in -65.54, -43.12 59.71, 15.8 in-in-out SNCiio in-out ActLoopNT-in 2.931 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -120.05, -174.23 APE9-dihe-na 65.54, 142.28 APE8-dihe-in -62.37, 137.73 APE8-rot-out 183.0 APE67-dihe-in -57.53, -32.37 -39.19, -57.21 APE12-dist-in 13.389 APE11-dist-in 11.762 APE10-dist-in 6.421 APE9-dist-in 3.218 None PTR216 PTR216 XRAY 2.35 0.206 0.234 A 350 350 0 0 0 0 [[56, 340]] 1.0 6hk3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6Y9RA 35 384 420.0 OH8:401 Type1 Inactive DFGin 7.213 13.956 BLAminus -128.7, 177.14 64.74, 83.75 -99.31, 22.7 285.39, 75.74 -67.18, -22.12 in-in in 8.387 Saltbr-in 2.76 HRD-in -68.2, -47.94 70.12, 17.05 in-in-out SNCiio in-out ActLoopNT-in 2.97 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -147.41, 164.13 APE9-dihe-na 71.55, 162.91 APE8-dihe-in -81.0, 136.61 APE8-rot-out 173.09 APE67-dihe-in -62.95, -25.51 -45.24, -50.14 APE12-dist-in 13.684 APE11-dist-in 12.039 APE10-dist-in 7.353 APE9-dist-in 3.295 None PTR216 PTR216 XRAY 2.08 0.191 0.226 A 350 350 0 0 0 0 [[56, 340]] 1.0 6y9r CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1O9UA 35 384 420.0 ADZ:1386 Type1 Inactive DFGin 6.69 14.409 BLAminus -135.58, -170.77 57.68, 80.28 -97.17, 18.56 286.56, 73.24 -63.89, -4.57 in-in in 8.918 Saltbr-in 3.252 HRD-in -60.54, -48.22 66.04, 11.65 in-in-out SNCiio in-out ActLoopNT-in 2.965 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.51, 167.48 APE9-dihe-na 74.14, -178.83 APE8-dihe-in -103.59, 140.85 APE8-rot-out 179.41 APE67-dihe-in -52.99, -22.64 -16.1, -87.79 APE12-dist-in 13.762 APE11-dist-in 11.706 APE10-dist-in 7.362 APE9-dist-in 2.862 None PTR216 PTR216 XRAY 2.4 0.233 0.26 A 350 350 0 0 0 0 [[56, 340]] 1.0 1o9u CMGC_GSK3B_HUMAN CMGC 2.1e-69 240.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9PE9A 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.072 14.229 BLAminus -128.7, -179.96 59.31, 84.1 -97.11, 26.91 283.64, 74.63 -73.69, -18.15 in-in in 8.351 Saltbr-in 2.725 HRD-in -68.62, -45.57 65.7, 16.55 in-in-out SNCiio in-out ActLoopNT-in 2.925 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.94, 165.33 APE9-dihe-na 76.34, 152.28 APE8-dihe-in -69.82, 130.62 APE8-rot-out 176.66 APE67-dihe-in -58.68, -26.71 -39.69, -56.4 APE12-dist-in 13.28 APE11-dist-in 11.758 APE10-dist-in 7.093 APE9-dist-in 3.155 None PTR216 PTR216 XRAY 2.11 0.221 0.247 A 359 332 13 0 0 0 [[56, 340]] 1.0 9pe9 CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9PE9B 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.058 14.218 BLAminus -128.76, -179.81 59.6, 84.42 -97.78, 27.09 283.79, 74.38 -73.25, -17.71 in-in in 8.353 Saltbr-in 2.713 HRD-in -68.49, -44.82 64.55, 18.32 in-in-out SNCiio in-out ActLoopNT-in 2.94 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.27, 163.74 APE9-dihe-na 77.64, 152.05 APE8-dihe-in -69.14, 130.82 APE8-rot-out 177.12 APE67-dihe-in -58.92, -26.81 -39.96, -55.88 APE12-dist-in 13.36 APE11-dist-in 11.824 APE10-dist-in 7.161 APE9-dist-in 3.172 None PTR216 PTR216 XRAY 2.11 0.221 0.247 B 359 332 13 0 0 0 [[56, 340]] 1.0 9pe9 CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7Z1FA 28 383 420.0 3NG:60401 Type1 Inactive DFGin 7.172 14.387 BLAminus -140.61, -172.17 56.83, 67.31 -90.44, 24.59 283.96, 78.9 -70.58, -34.2 in-in in 8.589 Saltbr-in 2.706 HRD-in -70.71, -48.08 68.23, 20.67 in-in-out SNCiio in-out ActLoopNT-in 2.877 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -121.77, -56.1 APE9-dihe-na -73.95, 173.6 APE8-dihe-in -71.54, 133.95 APE8-rot-out 205.24 APE67-dihe-in -54.78, -22.55 -52.86, -47.6 APE12-dist-in 13.711 APE11-dist-in 11.921 APE10-dist-in 7.257 APE9-dist-in 3.478 None PTR216 PTR216 XRAY 3.0 0.224 0.249 A 364 354 2 0 0 0 [[56, 340]] 1.0 7z1f CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
7Z1FB 38 382 420.0 3NG:60401 Type1 Inactive DFGin 6.87 14.469 BLAminus -141.12, -171.82 52.8, 73.11 -90.49, 20.89 285.47, 81.84 -62.59, -35.1 in-in in 9.025 Saltbr-in 2.763 HRD-in -68.41, -52.97 70.54, 14.05 in-in-out SNCiio in-out ActLoopNT-in 3.039 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.34, -53.99 APE9-dihe-na -75.88, 165.71 APE8-dihe-in -64.92, 136.76 APE8-rot-out 179.7 APE67-dihe-in -58.44, -19.64 -54.95, -47.33 APE12-dist-in 13.527 APE11-dist-in 11.859 APE10-dist-in 7.154 APE9-dist-in 3.558 None PTR216 PTR216 XRAY 3.0 0.224 0.249 B 364 321 24 0 0 0 [[56, 340]] 1.0 7z1f CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8AV1A 27 381 420.0 O9L:406 Type1 Inactive DFGin 7.005 13.802 BLAminus -134.83, 176.12 61.29, 85.31 -97.92, 27.58 284.57, 74.39 -70.18, -20.31 in-in in 8.42 Saltbr-in 2.659 HRD-in -72.82, -53.06 75.09, 11.93 in-in-out SNCiio in-out ActLoopNT-in 2.811 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -162.3, 153.55 APE9-dihe-na 79.71, 140.85 APE8-dihe-in -55.94, 133.71 APE8-rot-out 187.25 APE67-dihe-in -61.14, -25.49 -46.06, -52.45 APE12-dist-in 13.268 APE11-dist-in 11.413 APE10-dist-in 6.884 APE9-dist-in 3.061 None PTR216 PTR216 XRAY 2.15 0.18 0.21 A 365 351 4 0 0 0 [[56, 340]] 1.0 8av1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8AV1B 27 381 420.0 O9L:405 Type1 Inactive DFGin 7.041 13.818 BLAminus -134.53, 176.17 61.15, 83.84 -96.42, 28.03 285.62, 75.68 -72.4, -19.61 in-in in 8.351 Saltbr-in 2.648 HRD-in -70.84, -52.05 73.58, 16.86 in-in-out SNCiio in-out ActLoopNT-in 2.809 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.36, 152.7 APE9-dihe-na 82.35, 142.4 APE8-dihe-in -57.42, 133.83 APE8-rot-out 184.71 APE67-dihe-in -59.68, -24.96 -48.86, -51.78 APE12-dist-in 13.26 APE11-dist-in 11.441 APE10-dist-in 6.85 APE9-dist-in 3.06 None PTR216 PTR216 XRAY 2.15 0.18 0.21 B 365 351 4 0 0 0 [[56, 340]] 1.0 8av1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6GN1A 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.94 14.335 BLAminus -135.29, 179.1 59.47, 89.49 -98.73, 29.98 286.18, 72.49 -75.74, -10.8 in-in in 8.608 Saltbr-in 3.04 HRD-in -74.24, -44.22 64.59, 22.98 in-in-out SNCiio in-out ActLoopNT-in 2.94 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -143.03, -18.16 APE9-dihe-na -103.04, 175.18 APE8-dihe-in -67.81, 136.03 APE8-rot-out 187.31 APE67-dihe-in -61.67, -27.65 -44.51, -52.79 APE12-dist-out 14.01 APE11-dist-in 12.355 APE10-dist-in 7.387 APE9-dist-in 3.587 None PTR216 PTR216 XRAY 2.6 0.224 0.259 A 368 340 8 0 0 0 [[56, 340]] 1.0 6gn1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6GN1B 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.944 14.317 BLAminus -135.3, 179.27 59.56, 89.49 -98.78, 30.1 286.37, 73.15 -75.82, -10.91 in-in in 8.622 Saltbr-in 3.034 HRD-in -74.17, -44.23 64.47, 22.86 in-in-out SNCiio in-out ActLoopNT-in 2.946 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -129.39, -14.9 APE9-dihe-na -108.68, -179.33 APE8-dihe-in -68.02, 134.54 APE8-rot-out 210.75 APE67-dihe-in -62.25, -27.68 -44.3, -51.95 APE12-dist-out 14.024 APE11-dist-in 12.183 APE10-dist-in 7.403 APE9-dist-in 3.7 None PTR216 PTR216 XRAY 2.6 0.224 0.259 B 368 340 8 0 0 0 [[56, 340]] 1.0 6gn1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
2O5KA 35 384 420.0 HBM:0 Type1 Inactive DFGin 6.721 13.939 BLAminus -127.34, -179.9 54.97, 85.31 -97.88, 27.22 279.56, 72.26 -63.78, -54.26 in-in in 8.352 Saltbr-in 3.376 HRD-in -66.17, -47.55 59.21, 39.45 in-in-out SNCiio in-out ActLoopNT-in 2.946 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_iiii APE10-dihe-na 170.93, -156.16 APE9-dihe-na 30.47, -152.36 APE8-dihe-out -134.5, -176.14 APE8-rot-in 306.82 APE67-dihe-in -73.05, -7.32 -59.58, -80.34 APE12-dist-in 12.679 APE11-dist-in 9.181 APE10-dist-in 5.885 APE9-dist-in 3.037 None None None XRAY 3.2 0.251 0.309 A 372 350 0 0 0 0 [[56, 340]] 1.0 2o5k CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
1UV5A 35 383 420.0 BRW:1383 Type1 Inactive DFGin 6.902 14.079 BLAminus -144.35, -177.14 59.35, 81.04 -94.26, 27.94 286.0, 72.94 -59.18, -36.48 in-in in 8.299 Saltbr-in 2.561 HRD-in -65.61, -42.55 70.5, 0.98 in-in-out SNCiio in-out ActLoopNT-in 2.884 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -98.47, 172.31 APE9-dihe-na 85.56, 133.89 APE8-dihe-in -66.16, 126.55 APE8-rot-out 191.14 APE67-dihe-in -61.71, -20.34 -21.78, -65.88 APE12-dist-in 12.763 APE11-dist-in 10.989 APE10-dist-in 5.715 APE9-dist-in 3.236 None None None XRAY 2.8 0.193 0.226 A 350 349 0 0 0 0 [[56, 340]] 1.0 1uv5 CMGC_GSK3B_HUMAN CMGC 7.4e-70 241.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6GJOA 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.176 14.254 BLAminus -136.61, 169.82 63.4, 86.22 -103.46, 25.41 276.6, 83.48 -69.91, -39.25 in-in in 8.636 Saltbr-in 2.81 HRD-in -57.84, -41.83 58.98, 16.97 in-in-out SNCiio in-out ActLoopNT-in 3.012 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.92, 162.15 APE9-dihe-na 71.93, 161.47 APE8-dihe-in -78.01, 132.19 APE8-rot-out 37.25 APE67-dihe-in -62.57, -18.8 -29.28, -56.31 APE12-dist-in 13.62 APE11-dist-in 11.862 APE10-dist-in 6.945 APE9-dist-in 3.445 None None None XRAY 2.91 0.218 0.237 A 414 349 0 0 0 0 [[56, 340]] 1.0 6gjo CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
6GJOB 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.478 14.251 BLAminus -136.82, 170.18 63.9, 83.46 -101.86, 22.92 278.62, 83.32 -68.81, -38.47 in-in in 8.405 Saltbr-in 3.084 HRD-in -57.78, -41.9 58.99, 17.22 in-in-out SNCiio in-out ActLoopNT-in 3.012 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.67, 163.61 APE9-dihe-na 73.76, 161.78 APE8-dihe-in -77.57, 137.96 APE8-rot-out 184.23 APE67-dihe-in -62.17, -20.4 -36.29, -55.68 APE12-dist-in 13.45 APE11-dist-in 11.784 APE10-dist-in 6.854 APE9-dist-in 3.437 None None None XRAY 2.91 0.218 0.237 B 414 343 6 0 0 0 [[56, 340]] 1.0 6gjo CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
3M1SA 35 385 420.0 DW1:421 Type1 Inactive DFGin 7.021 13.71 BLAminus -149.21, -179.05 55.83, 87.87 -101.26, 23.04 292.92, 65.81 -62.39, -0.11 in-in in 8.726 Saltbr-in 2.976 HRD-in -71.98, -44.05 63.65, 18.92 in-in-out SNCiio in-out ActLoopNT-in 3.032 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -100.39, 171.9 APE9-dihe-na 82.48, 144.37 APE8-dihe-in -94.3, 96.58 APE8-rot-in 285.71 APE67-dihe-out 116.42, -45.78 9.38, 103.41 APE12-dist-in 13.649 APE11-dist-in 11.709 APE10-dist-in 6.707 APE9-dist-in 3.445 None None None XRAY 3.134 0.171 0.228 A 420 348 3 0 0 0 [[56, 340]] 1.0 3m1s CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
9HUKA 25 385 420.0 A1IXL:501 Type1 Inactive DFGin 7.053 14.078 BLAminus -135.25, -177.02 57.0, 94.14 -110.6, 20.82 285.12, 72.82 -66.1, -13.46 in-out in 8.11 Saltbr-out 3.659 HRD-in -70.91, -39.46 63.28, 18.66 out-in-in SNCoii in-in ActLoopNT-in 3.157 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 179.26 APE9-dihe-na 68.03, 135.17 APE8-dihe-in -69.47, 168.34 APE8-rot-in 295.64 APE67-dihe-inflip 67.51, -44.25 -66.67, 175.58 APE12-dist-in 13.119 APE11-dist-in 10.946 APE10-dist-in 5.924 APE9-dist-in 3.202 None None None XRAY 3.5 0.219 0.25 A 442 361 0 0 0 0 [[56, 340]] 1.0 9huk CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4J71A 36 383 420.0 1JX:501 Type1 Inactive DFGin 6.929 14.034 BLAminus -134.37, 178.91 60.63, 80.22 -96.96, 24.92 284.72, 75.18 -68.29, -15.66 in-in in 8.448 Saltbr-in 3.096 HRD-in -74.9, -47.0 72.06, 4.98 in-in-out SNCiio in-out ActLoopNT-in 2.714 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.32, 163.35 APE9-dihe-na 76.45, 151.25 APE8-dihe-in -65.19, 140.55 APE8-rot-out 188.84 APE67-dihe-in -55.99, -28.06 -50.85, -54.43 APE12-dist-in 13.396 APE11-dist-in 11.896 APE10-dist-in 7.163 APE9-dist-in 2.998 None PTR216 PTR216 XRAY 2.31 0.191 0.234 A 424 348 0 0 0 0 [[56, 340]] 1.0 4j71 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4J71B 36 383 420.0 1JX:501 Type1 Inactive DFGin 7.043 13.832 BLAminus -140.62, 179.7 59.87, 90.62 -104.73, 25.33 288.76, 76.25 -66.71, -17.33 in-in in 8.331 Saltbr-in 2.896 HRD-in -77.92, -46.29 72.36, 3.7 in-in-out SNCiio in-out ActLoopNT-in 2.834 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.74, 169.96 APE9-dihe-na 69.52, 149.79 APE8-dihe-in -68.04, 134.18 APE8-rot-out 173.06 APE67-dihe-in -53.62, -29.43 -43.81, -55.09 APE12-dist-in 13.213 APE11-dist-in 11.957 APE10-dist-in 7.127 APE9-dist-in 2.974 None PTR216 PTR216 XRAY 2.31 0.191 0.234 B 424 348 0 0 0 0 [[56, 340]] 1.0 4j71 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5HLNB 37 383 420.0 65C:501 Type1 Inactive DFGin 6.848 13.332 BLAminus -143.06, -174.61 53.09, 90.34 -103.45, 33.01 288.97, 83.64 -74.69, -34.84 in-in in 8.996 Saltbr-in 2.604 HRD-in -68.15, -40.04 65.1, 19.28 in-in-out SNCiio in-out ActLoopNT-in 2.963 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -137.65, -62.86 APE9-dihe-na -78.36, 171.11 APE8-dihe-in -56.52, 151.93 APE8-rot-out 161.85 APE67-dihe-in -56.43, -28.42 -72.24, -45.62 APE12-dist-in 13.598 APE11-dist-in 11.834 APE10-dist-in 7.374 APE9-dist-in 3.416 None PTR216 PTR216 XRAY 3.1 0.173 0.236 B 424 347 0 0 0 0 [[56, 340]] 1.0 5hln CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
5OY4B 30 384 420.0 B4K:502 Type1.5_Back Inactive DFGin 7.008 13.741 BLAminus -131.51, 177.88 58.43, 85.84 -94.85, 21.53 281.4, 81.96 -63.5, -26.63 in-in in 7.965 Saltbr-in 2.751 HRD-in -68.43, -44.24 63.59, 14.9 in-in-out SNCiio in-out ActLoopNT-in 2.869 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -145.82, 158.71 APE9-dihe-na 86.22, 156.23 APE8-dihe-in -75.92, 122.37 APE8-rot-out 226.12 APE67-dihe-in -60.14, -24.48 -28.85, -54.97 APE12-dist-in 13.504 APE11-dist-in 11.621 APE10-dist-in 7.009 APE9-dist-in 3.404 None PTR216 PTR216 XRAY 3.2 0.196 0.229 B 420 354 1 0 0 0 [[56, 340]] 1.0 5oy4 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
8QJIA 36 381 420.0 VNG:401 Type1 Inactive DFGin 6.949 14.196 None -92.57, -90.5 -72.82, 155.73 -144.36, 17.02 276.05, 102.26 -73.85, -19.5 in-in in 8.384 Saltbr-in 2.694 HRD-in -65.27, -43.08 63.67, 22.78 in-in-out SNCiio in-out ActLoopNT-in 3.34 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -115.54, 179.17 APE9-dihe-na 65.4, 161.24 APE8-dihe-in -68.89, 150.02 APE8-rot-out 175.4 APE67-dihe-in -64.21, -18.12 -58.7, -47.99 APE12-dist-in 13.386 APE11-dist-in 12.002 APE10-dist-in 7.07 APE9-dist-in 3.447 None PTR216 PTR216 XRAY 3.02 0.253 0.289 A 364 340 6 0 0 0 [[56, 340]] 1.0 8qji CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
4DITA 35 387 420.0 0KD:501 Type1 None DFGin 6.805 13.948 BLAminus -145.37, 179.76 65.92, 81.37 -105.97, 22.54 288.96, 82.14 -68.29, -17.95 in-in in 8.825 Saltbr-in 2.717 HRD-in -69.87, -50.6 73.87, 5.2 in-in-none SNCiin in-none ActLoopNT-in 2.939 ActLoopCT-none nonTYR APEdihe_aannn APEdist_iinn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 14.5 999.0, 999.0 APE12-dist-in 13.489 APE11-dist-in 10.385 APE10-dist-none 999.0 APE9-dist-none 999.0 None PTR216 PTR216 XRAY 2.6 0.243 0.304 A 382 329 24 0 0 4 [[56, 340]] 1.0 4dit CMGC_GSK3B_HUMAN CMGC 2.4e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta

CMGC_GSK3B (Glycogen synthase kinase-3 beta)

Total number of chains: 204
Active chains: 159
Family: CMGC
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 200 98.0% AF-P49841-K1A
DFGin ABAminus 3 1.5% 5AIRA
DFGin None 1 0.5% 8QJIA

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GSK3B_HUMAN 4NM5A P49841 24 383 420.0 ADP:60401 ATPlike Active DFGin 6.55 14.006 BLAminus -136.16, -177.73 61.88, 88.47 -108.64, 28.76 287.87, 80.78 -73.66, -15.44 in-in in 8.619 Saltbr-in 2.673 HRD-in -65.83, -43.73 64.82, 15.23 in-in-in SNCiii in-in ActLoopNT-in 2.839 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.92, 173.97 APE9-dihe-na 66.26, 147.02 APE8-dihe-in -77.1, 152.8 APE8-rot-in 293.28 APE67-dihe-inflip 82.03, -25.76 -52.23, 150.7 APE12-dist-in 13.279 APE11-dist-in 11.599 APE10-dist-in 6.949 APE9-dist-in 3.238 None None None XRAY 2.3 0.185 0.232 A 377 360 0 0 0 0 [[56, 340]] 1.0 4nm5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4NM7A P49841 25 383 420.0 ADP:60401 ATPlike Active DFGin 6.515 13.993 BLAminus -137.35, -178.06 62.82, 88.6 -107.3, 24.56 288.41, 80.2 -69.84, -12.63 in-in in 8.818 Saltbr-in 2.743 HRD-in -66.5, -46.64 67.84, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.829 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 172.54 APE9-dihe-na 68.99, 153.43 APE8-dihe-in -86.9, 151.79 APE8-rot-in 300.04 APE67-dihe-inflip 84.67, -25.93 -50.38, 146.2 APE12-dist-in 13.355 APE11-dist-in 11.678 APE10-dist-in 6.905 APE9-dist-in 3.21 None None None XRAY 2.3 0.185 0.234 A 377 354 2 0 0 0 [[56, 340]] 1.0 4nm7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4NM3A P49841 6 383 420.0 ADP:60409 ATPlike Active DFGin 6.475 13.947 BLAminus -129.98, -178.05 63.17, 87.87 -103.96, 21.26 289.38, 80.04 -65.46, -16.35 in-in in 8.806 Saltbr-in 2.726 HRD-in -69.81, -46.77 71.59, 6.75 in-in-in SNCiii in-in ActLoopNT-in 2.75 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.34, 169.99 APE9-dihe-na 69.15, 146.37 APE8-dihe-in -83.47, 151.55 APE8-rot-in 296.54 APE67-dihe-inflip 86.0, -31.11 -49.79, 146.79 APE12-dist-in 13.269 APE11-dist-in 11.484 APE10-dist-in 6.907 APE9-dist-in 3.112 None SEP9 SEP9 XRAY 2.1 0.197 0.242 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nm3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1J1BA P49841 35 388 420.0 ANP:60430 ATPlike Active DFGin 6.767 13.788 BLAminus -136.8, -178.88 61.6, 83.12 -97.64, 25.1 286.09, 80.4 -68.7, -13.11 in-in in 8.566 Saltbr-in 2.59 HRD-in -71.16, -45.98 70.36, 3.88 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.52, 175.26 APE9-dihe-na 75.44, 133.64 APE8-dihe-in -75.76, 147.49 APE8-rot-in 306.57 APE67-dihe-inflip 98.15, -33.72 -56.43, 141.52 APE12-dist-in 13.056 APE11-dist-in 10.974 APE10-dist-in 5.893 APE9-dist-in 3.112 None None None XRAY 1.8 0.216 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1J1BB P49841 23 386 420.0 ANP:60930 ATPlike Active DFGin 6.609 13.669 BLAminus -136.4, -177.03 61.49, 81.88 -98.08, 27.2 288.49, 82.07 -71.33, -13.14 in-in in 8.457 Saltbr-in 2.713 HRD-in -67.51, -45.87 68.87, 6.43 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.88, 174.17 APE9-dihe-na 76.18, 138.08 APE8-dihe-in -76.12, 141.41 APE8-rot-in 301.11 APE67-dihe-inflip 98.0, -37.59 -54.78, 144.25 APE12-dist-in 12.978 APE11-dist-in 11.066 APE10-dist-in 6.011 APE9-dist-in 3.174 None None None XRAY 1.8 0.216 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1J1CA P49841 35 388 420.0 ADP:60430 ATPlike Active DFGin 6.812 13.93 BLAminus -139.24, -179.75 62.79, 82.17 -97.34, 25.19 286.68, 82.3 -65.83, -19.9 in-in in 8.601 Saltbr-in 2.647 HRD-in -68.65, -43.85 68.34, 7.36 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.05, 172.96 APE9-dihe-na 78.17, 130.85 APE8-dihe-in -73.54, 145.97 APE8-rot-in 310.16 APE67-dihe-inflip 99.09, -35.01 -54.43, 141.28 APE12-dist-in 13.077 APE11-dist-in 11.067 APE10-dist-in 5.926 APE9-dist-in 3.2 None None None XRAY 2.1 0.218 0.242 A 420 354 0 0 0 0 [[56, 340]] 1.0 1j1c Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1J1CB P49841 23 386 420.0 ADP:60930 ATPlike Active DFGin 6.694 13.709 BLAminus -138.27, -179.99 63.33, 82.68 -100.46, 28.2 289.88, 80.26 -70.45, -13.94 in-in in 8.52 Saltbr-in 2.738 HRD-in -67.92, -43.36 67.59, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.71, 170.27 APE9-dihe-na 78.71, 139.86 APE8-dihe-in -81.56, 140.05 APE8-rot-in 302.5 APE67-dihe-inflip 101.62, -36.53 -50.52, 137.44 APE12-dist-in 12.868 APE11-dist-in 11.128 APE10-dist-in 6.025 APE9-dist-in 3.208 None None None XRAY 2.1 0.218 0.242 B 420 364 0 0 0 0 [[56, 340]] 1.0 1j1c Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8XN6A P49841 35 384 420.0 ANP:501 ATPlike Active DFGin 6.682 13.862 BLAminus -137.72, 173.39 67.73, 84.48 -99.84, 22.57 287.77, 80.54 -65.33, -24.58 in-in in 8.463 Saltbr-in 2.63 HRD-in -71.05, -47.88 67.82, 15.5 in-in-in SNCiii in-in ActLoopNT-in 3.054 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.0, 164.43 APE9-dihe-na 85.44, 135.36 APE8-dihe-in -74.2, 151.55 APE8-rot-in 291.81 APE67-dihe-in -69.28, -17.83 -36.59, -67.98 APE12-dist-in 12.907 APE11-dist-in 10.787 APE10-dist-in 5.68 APE9-dist-in 3.182 None None None XRAY 2.4 0.194 0.242 A 421 350 0 0 0 0 [[56, 340]] 1.0 8xn6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1PYXA P49841 35 386 420.0 ANP:1001 ATPlike Active DFGin 6.584 13.622 BLAminus -138.81, -178.07 65.18, 79.92 -98.83, 26.07 289.95, 78.27 -73.24, -7.6 in-in in 8.373 Saltbr-in 2.765 HRD-in -67.79, -47.84 71.28, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.948 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.12, 170.17 APE9-dihe-na 80.64, 129.74 APE8-dihe-in -63.79, 140.05 APE8-rot-in 299.48 APE67-dihe-in -56.43, -21.61 -20.65, -80.28 APE12-dist-in 12.903 APE11-dist-in 10.937 APE10-dist-in 5.784 APE9-dist-in 3.15 None None None XRAY 2.4 0.206 0.233 A 422 343 9 0 0 0 [[56, 340]] 1.0 1pyx Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1PYXB P49841 35 383 420.0 ANP:2001 ATPlike Active DFGin 6.593 13.718 BLAminus -140.94, -178.47 65.26, 79.98 -98.11, 22.32 290.75, 76.51 -68.32, -7.73 in-in in 8.488 Saltbr-in 2.666 HRD-in -69.98, -47.18 70.83, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.3, 169.41 APE9-dihe-na 81.27, 131.24 APE8-dihe-in -66.67, 140.79 APE8-rot-in 300.74 APE67-dihe-in -56.9, -22.2 -20.58, -79.9 APE12-dist-in 12.838 APE11-dist-in 10.861 APE10-dist-in 5.718 APE9-dist-in 3.132 None None None XRAY 2.4 0.206 0.233 B 422 338 11 0 0 0 [[56, 340]] 1.0 1pyx Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN AF-P49841-K1A P49841 48 348 420.0 No_ligand No_ligand Active DFGin 6.784 14.069 BLAminus -132.22, 178.4 62.95, 68.76 -81.18, 15.79 285.47, 79.99 -60.59, -34.48 in-in in 8.475 Saltbr-in 2.71 HRD-in -72.93, -43.95 66.08, 11.33 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.31, 173.16 APE9-dihe-na 65.7, 144.93 APE8-dihe-in -63.41, 136.54 APE8-rot-in 298.96 APE67-dihe-in -66.32, -15.33 -50.7, -49.59 APE12-dist-in 13.45 APE11-dist-in 11.989 APE10-dist-in 6.996 APE9-dist-in 3.127 None None None AF2 -1.0 1.0 1.0 A 301 301 0 0 0 0 [[56, 340]] 1.0 AF-P49841-K1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN AF-P49841-K3A P49841 48 348 420.0 No_ligand No_ligand Active DFGin 6.524 13.884 BLAminus -137.65, -179.24 64.43, 60.31 -74.11, 11.79 288.76, 87.67 -59.53, -33.87 in-in in 8.232 Saltbr-in 2.675 HRD-in -76.11, -42.33 64.92, 19.4 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, -179.86 APE9-dihe-na 61.35, 145.02 APE8-dihe-in -62.21, 135.58 APE8-rot-in 295.17 APE67-dihe-in -63.79, -15.52 -52.47, -50.54 APE12-dist-in 13.486 APE11-dist-in 11.995 APE10-dist-in 7.07 APE9-dist-in 3.244 None None None AF2 -1.0 1.0 1.0 A 301 301 0 0 0 0 [[56, 340]] 1.0 AF-P49841-K3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2QA P49841 35 383 420.0 No_ligand No_ligand Active DFGin 7.052 14.715 BLAminus -137.83, -179.15 61.41, 79.74 -96.27, 22.19 285.08, 78.46 -63.78, -22.81 in-in in 9.6 Saltbr-in 2.835 HRD-in -68.59, -45.76 72.18, 9.73 in-in-in SNCiii in-in ActLoopNT-in 2.932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.17, 171.92 APE9-dihe-na 79.53, 140.67 APE8-dihe-in -94.64, 154.44 APE8-rot-in 291.59 APE67-dihe-inflip 92.14, -26.46 -46.09, 133.9 APE12-dist-in 12.819 APE11-dist-in 10.688 APE10-dist-in 5.811 APE9-dist-in 3.156 None None None XRAY 1.68 0.174 0.202 A 359 349 0 0 0 0 [[56, 340]] 1.0 9x2q Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2QC P49841 36 383 420.0 No_ligand No_ligand Active DFGin 7.21 15.088 BLAminus -133.92, -175.86 59.44, 76.77 -92.13, 23.3 281.6, 76.88 -64.8, -22.26 in-in in 9.585 Saltbr-in 2.881 HRD-in -73.13, -43.06 72.53, 6.24 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -80.09, 170.02 APE9-dihe-na 80.69, 143.27 APE8-dihe-in -98.08, 153.35 APE8-rot-in 292.56 APE67-dihe-inflip 91.66, -29.76 -46.15, 133.94 APE12-dist-in 12.831 APE11-dist-in 10.762 APE10-dist-in 5.787 APE9-dist-in 3.164 None None None XRAY 1.68 0.174 0.202 C 359 344 4 0 0 0 [[56, 340]] 1.0 9x2q Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2UA P49841 35 382 420.0 No_ligand No_ligand Active DFGin 6.928 15.007 BLAminus -133.34, -178.44 58.79, 78.89 -95.7, 26.22 286.38, 80.77 -67.47, -21.14 in-in in 9.819 Saltbr-in 2.904 HRD-in -68.71, -46.18 69.43, 14.55 in-in-in SNCiii in-in ActLoopNT-in 2.926 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.25, 174.16 APE9-dihe-na 72.67, 147.17 APE8-dihe-in -96.66, 153.81 APE8-rot-in 303.03 APE67-dihe-inflip 89.84, -29.57 -56.61, 146.99 APE12-dist-in 12.872 APE11-dist-in 10.763 APE10-dist-in 6.052 APE9-dist-in 3.212 None None None XRAY 2.07 0.198 0.233 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2u Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2UB P49841 35 382 420.0 No_ligand No_ligand Active DFGin 7.031 15.039 BLAminus -142.07, -178.25 60.15, 75.53 -94.78, 27.78 287.55, 76.1 -71.78, -16.86 in-in in 9.544 Saltbr-in 3.111 HRD-in -69.92, -46.99 71.31, 12.91 in-in-in SNCiii in-in ActLoopNT-in 2.857 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.99, 177.06 APE9-dihe-na 70.96, 140.3 APE8-dihe-in -91.49, 155.78 APE8-rot-in 299.08 APE67-dihe-inflip 86.39, -30.22 -56.97, 152.43 APE12-dist-in 12.801 APE11-dist-in 10.684 APE10-dist-in 6.083 APE9-dist-in 3.216 None None None XRAY 2.07 0.198 0.233 B 359 346 2 0 0 0 [[56, 340]] 1.0 9x2u Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2WA P49841 35 382 420.0 No_ligand No_ligand Active DFGin 7.002 14.662 BLAminus -137.11, -172.55 57.37, 78.08 -92.78, 22.6 285.25, 77.53 -65.29, -22.08 in-in in 9.426 Saltbr-in 2.69 HRD-in -70.87, -42.87 69.61, 6.59 in-in-in SNCiii in-in ActLoopNT-in 2.924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.52, 174.16 APE9-dihe-na 78.0, 143.92 APE8-dihe-in -99.28, 152.84 APE8-rot-in 293.19 APE67-dihe-inflip 94.63, -26.01 -40.27, 130.65 APE12-dist-in 12.851 APE11-dist-in 10.695 APE10-dist-in 5.869 APE9-dist-in 3.149 None None None XRAY 1.92 0.179 0.209 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2w Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2WC P49841 36 381 420.0 No_ligand No_ligand Active DFGin 7.232 15.121 BLAminus -131.33, -174.54 58.27, 79.41 -92.24, 20.59 282.51, 74.33 -64.49, -19.25 in-in in 9.502 Saltbr-in 2.925 HRD-in -70.18, -47.01 71.8, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.863 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.09, 172.17 APE9-dihe-na 81.56, 146.73 APE8-dihe-in -102.37, 154.39 APE8-rot-in 287.29 APE67-dihe-inflip 98.99, -30.15 -43.41, 127.27 APE12-dist-in 12.772 APE11-dist-in 10.661 APE10-dist-in 5.82 APE9-dist-in 3.147 None None None XRAY 1.92 0.179 0.209 C 359 343 3 0 0 0 [[56, 340]] 1.0 9x2w Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2XA P49841 35 382 420.0 No_ligand No_ligand Active DFGin 7.096 14.802 BLAminus -134.71, -177.87 61.9, 80.09 -94.66, 24.51 284.3, 79.87 -70.56, -15.85 in-in in 9.585 Saltbr-in 2.845 HRD-in -72.18, -43.18 72.48, 8.24 in-in-in SNCiii in-in ActLoopNT-in 2.908 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.7, 174.99 APE9-dihe-na 74.21, 144.04 APE8-dihe-in -99.9, 155.52 APE8-rot-in 294.34 APE67-dihe-inflip 98.06, -28.28 -45.69, 131.32 APE12-dist-in 12.91 APE11-dist-in 10.817 APE10-dist-in 5.923 APE9-dist-in 3.137 None None None XRAY 1.79 0.178 0.207 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2x Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2XC P49841 35 382 420.0 No_ligand No_ligand Active DFGin 7.055 15.211 BLAminus -133.52, -175.85 56.94, 77.42 -93.62, 21.48 281.91, 76.2 -62.69, -19.85 in-in in 9.611 Saltbr-in 2.837 HRD-in -74.39, -45.42 70.67, 10.42 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.32, 172.59 APE9-dihe-na 78.39, 148.01 APE8-dihe-in -102.94, 151.91 APE8-rot-in 298.64 APE67-dihe-inflip 95.53, -30.76 -39.02, 129.93 APE12-dist-in 12.904 APE11-dist-in 10.761 APE10-dist-in 5.918 APE9-dist-in 3.224 None None None XRAY 1.79 0.178 0.207 C 359 348 0 0 0 0 [[56, 340]] 1.0 9x2x Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2YA P49841 35 382 420.0 No_ligand No_ligand Active DFGin 7.05 14.658 BLAminus -140.01, -179.57 60.44, 76.66 -91.5, 22.26 284.52, 79.37 -66.64, -18.87 in-in in 9.354 Saltbr-in 2.946 HRD-in -71.93, -44.87 72.02, 8.24 in-in-in SNCiii in-in ActLoopNT-in 2.972 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.33, 176.92 APE9-dihe-na 74.96, 144.91 APE8-dihe-in -97.18, 152.76 APE8-rot-in 297.41 APE67-dihe-inflip 94.26, -28.73 -49.99, 137.38 APE12-dist-in 12.914 APE11-dist-in 10.749 APE10-dist-in 5.852 APE9-dist-in 3.129 None None None XRAY 1.96 0.182 0.205 A 359 348 0 0 0 0 [[56, 340]] 1.0 9x2y Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2YB P49841 37 382 420.0 No_ligand No_ligand Active DFGin 7.168 15.426 BLAminus -135.79, -176.64 57.44, 76.44 -90.64, 22.98 280.99, 76.17 -68.43, -15.63 in-in in 9.632 Saltbr-in 2.646 HRD-in -70.95, -47.52 72.95, 6.25 in-in-in SNCiii in-in ActLoopNT-in 2.831 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.29, 173.98 APE9-dihe-na 78.55, 143.82 APE8-dihe-in -97.73, 153.79 APE8-rot-in 303.29 APE67-dihe-inflip 99.44, -30.41 -47.09, 134.37 APE12-dist-in 12.869 APE11-dist-in 10.666 APE10-dist-in 5.798 APE9-dist-in 3.151 None None None XRAY 1.96 0.182 0.205 B 359 346 0 0 0 0 [[56, 340]] 1.0 9x2y Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1GNGA P49841 36 385 420.0 No_ligand No_ligand Active DFGin 6.885 14.064 BLAminus -143.26, -176.0 52.72, 77.37 -90.17, 24.13 284.09, 64.37 -57.11, -28.67 in-in in 7.904 Saltbr-in 2.916 HRD-in -73.29, -39.28 60.06, 11.92 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.61, 159.4 APE9-dihe-na 81.31, 139.52 APE8-dihe-in -59.26, 125.44 APE8-rot-in 312.57 APE67-dihe-in -52.62, -25.58 -28.83, -64.47 APE12-dist-in 13.55 APE11-dist-in 11.957 APE10-dist-in 7.016 APE9-dist-in 3.111 None PTR216 PTR216 XRAY 2.6 0.196 0.262 A 378 350 0 0 0 0 [[56, 340]] 1.0 1gng Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1GNGB P49841 28 384 420.0 No_ligand No_ligand Active DFGin 7.075 14.143 BLAminus -137.26, -174.12 57.41, 76.0 -92.3, 24.73 292.83, 74.1 -62.54, -16.26 in-in in 8.103 Saltbr-in 2.801 HRD-in -56.65, -46.78 67.13, 3.53 in-in-in SNCiii in-in ActLoopNT-in 3.053 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.46, 162.71 APE9-dihe-na 73.79, 160.3 APE8-dihe-in -71.09, 143.31 APE8-rot-in 306.45 APE67-dihe-in -62.51, -22.51 -44.24, -51.03 APE12-dist-in 13.461 APE11-dist-in 11.737 APE10-dist-in 7.233 APE9-dist-in 3.292 None PTR216 PTR216 XRAY 2.6 0.196 0.262 B 378 357 0 0 0 0 [[56, 340]] 1.0 1gng Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1H8FA P49841 35 386 420.0 No_ligand No_ligand Active DFGin 7.005 14.467 BLAminus -132.29, -174.92 54.46, 76.42 -91.57, 20.83 287.85, 73.58 -61.47, -17.91 in-in in 8.812 Saltbr-in 2.63 HRD-in -65.88, -45.02 68.7, 5.89 in-in-in SNCiii in-in ActLoopNT-in 3.03 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.85, 172.29 APE9-dihe-na 81.77, 142.51 APE8-dihe-in -88.0, 149.96 APE8-rot-in 300.12 APE67-dihe-in -68.04, -14.11 -16.17, -79.65 APE12-dist-in 12.877 APE11-dist-in 10.874 APE10-dist-in 5.794 APE9-dist-in 3.089 None None None XRAY 2.8 0.22 0.256 A 352 352 0 0 0 0 [[56, 340]] 1.0 1h8f Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1H8FB P49841 35 384 420.0 No_ligand No_ligand Active DFGin 7.053 14.488 BLAminus -137.11, -175.26 54.49, 79.79 -96.15, 19.99 284.33, 74.24 -61.84, -16.45 in-in in 8.784 Saltbr-in 2.631 HRD-in -65.99, -45.44 68.05, 7.58 in-in-in SNCiii in-in ActLoopNT-in 2.992 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.76, 172.7 APE9-dihe-na 81.11, 140.51 APE8-dihe-in -87.0, 149.5 APE8-rot-in 302.15 APE67-dihe-in -67.01, -11.3 -16.16, -82.04 APE12-dist-in 12.875 APE11-dist-in 10.843 APE10-dist-in 5.761 APE9-dist-in 3.101 None None None XRAY 2.8 0.22 0.256 B 352 350 0 0 0 0 [[56, 340]] 1.0 1h8f Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1I09A P49841 25 384 420.0 No_ligand No_ligand Active DFGin 6.914 14.149 BLAminus -130.79, -175.77 55.31, 78.24 -94.52, 21.05 292.59, 69.56 -64.23, -6.99 in-in in 8.521 Saltbr-in 2.763 HRD-in -66.04, -49.2 76.06, -6.11 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.67, -13.88 APE9-dihe-na -95.25, 153.25 APE8-dihe-in -66.11, 146.74 APE8-rot-in 277.64 APE67-dihe-in -57.92, -5.44 -43.43, -74.88 APE12-dist-in 12.968 APE11-dist-in 11.16 APE10-dist-in 5.972 APE9-dist-in 3.334 None None None XRAY 2.7 0.242 0.274 A 420 338 22 0 0 0 [[56, 340]] 1.0 1i09 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U2ZA P49841 35 382 420.0 L7C:401 Type1 Active DFGin 7.044 14.328 BLAminus -133.1, 179.76 62.32, 79.84 -96.99, 23.84 285.42, 79.62 -65.82, -25.41 in-in in 8.558 Saltbr-in 2.764 HRD-in -73.49, -48.13 70.69, 16.81 in-in-in SNCiii in-in ActLoopNT-in 2.907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.38, 169.05 APE9-dihe-na 81.0, 139.13 APE8-dihe-in -79.34, 150.41 APE8-rot-in 288.38 APE67-dihe-inflip 98.4, -32.71 -58.44, 134.12 APE12-dist-in 13.138 APE11-dist-in 11.05 APE10-dist-in 5.888 APE9-dist-in 3.092 None None None XRAY 2.21 0.248 0.266 A 348 345 3 0 0 0 [[56, 340]] 1.0 7u2z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U2ZB P49841 35 382 420.0 L7C:401 Type1 Active DFGin 7.083 14.316 BLAminus -133.0, 179.81 61.72, 80.12 -97.27, 23.94 285.32, 79.23 -65.78, -25.41 in-in in 8.516 Saltbr-in 2.765 HRD-in -73.41, -48.27 70.6, 17.33 in-in-in SNCiii in-in ActLoopNT-in 2.912 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.19, 168.84 APE9-dihe-na 80.53, 139.96 APE8-dihe-in -79.72, 154.04 APE8-rot-in 288.98 APE67-dihe-in -82.66, -15.29 -42.95, -55.79 APE12-dist-in 13.132 APE11-dist-in 11.082 APE10-dist-in 5.892 APE9-dist-in 3.099 None None None XRAY 2.21 0.248 0.266 B 348 348 0 0 0 0 [[56, 340]] 1.0 7u2z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3F7ZB P49841 35 383 420.0 34O:63000 Type1 Active DFGin 7.022 13.878 BLAminus -136.68, -179.55 57.9, 84.9 -98.68, 23.48 283.23, 74.81 -68.95, -21.14 in-in in 8.424 Saltbr-in 2.704 HRD-in -69.78, -45.02 65.34, 14.6 in-in-in SNCiii in-in ActLoopNT-in 2.869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.88, 179.92 APE9-dihe-na 68.48, 153.11 APE8-dihe-in -69.08, 139.27 APE8-rot-in 289.99 APE67-dihe-in -60.9, -22.52 -35.36, -58.5 APE12-dist-in 13.646 APE11-dist-in 11.954 APE10-dist-in 6.778 APE9-dist-in 3.248 None PTR216 PTR216 XRAY 2.4 0.206 0.253 B 350 339 10 0 0 0 [[56, 340]] 1.0 3f7z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3SD0B P49841 35 383 420.0 TSK:400 Type1 Active DFGin 7.188 14.024 BLAminus -142.24, -171.3 46.91, 83.25 -91.85, 32.36 285.89, 73.19 -82.63, -8.9 in-in in 8.235 Saltbr-in 2.887 HRD-in -76.13, -44.58 70.79, 3.58 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.6, 179.93 APE9-dihe-na 74.21, 152.1 APE8-dihe-in -107.68, 155.88 APE8-rot-in 296.61 APE67-dihe-in -78.55, -3.01 -13.04, -81.61 APE12-dist-in 13.018 APE11-dist-in 11.099 APE10-dist-in 6.151 APE9-dist-in 3.156 None None None XRAY 2.7 0.179 0.254 B 350 349 0 0 0 0 [[56, 340]] 1.0 3sd0 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6HK3B P49841 35 384 420.0 G8B:401 Type1 Active DFGin 6.788 13.641 BLAminus -137.2, -177.06 49.94, 95.88 -103.42, 19.32 279.02, 79.18 -69.5, -12.66 in-in in 8.168 Saltbr-in 2.602 HRD-in -82.47, -44.32 66.17, 21.49 in-in-in SNCiii in-in ActLoopNT-in 2.819 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.65, -179.5 APE9-dihe-na 72.73, 150.58 APE8-dihe-in -63.57, 140.77 APE8-rot-in 271.9 APE67-dihe-in -55.77, -29.98 -51.2, -52.31 APE12-dist-in 13.408 APE11-dist-in 11.642 APE10-dist-in 6.365 APE9-dist-in 3.249 None PTR216 PTR216 XRAY 2.35 0.206 0.234 B 350 350 0 0 0 0 [[56, 340]] 1.0 6hk3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6HK4A P49841 35 384 420.0 G8E:408 Type1 Active DFGin 6.928 13.508 BLAminus -141.9, -175.7 56.05, 83.18 -94.87, 22.99 284.64, 79.88 -61.73, -17.34 in-in in 8.371 Saltbr-in 2.656 HRD-in -76.65, -40.11 61.36, 16.95 in-in-in SNCiii in-in ActLoopNT-in 2.923 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.26, 167.76 APE9-dihe-na 63.34, 157.04 APE8-dihe-in -69.05, 135.63 APE8-rot-in 300.42 APE67-dihe-in -54.24, -34.87 -29.95, -58.61 APE12-dist-in 13.233 APE11-dist-in 11.745 APE10-dist-in 7.162 APE9-dist-in 3.192 None PTR216 PTR216 XRAY 2.5 0.212 0.249 A 350 350 0 0 0 0 [[56, 340]] 1.0 6hk4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6HK4B P49841 35 384 420.0 G8E:409 Type1 Active DFGin 6.943 13.541 BLAminus -140.37, -179.48 60.09, 87.67 -101.02, 22.8 284.5, 76.31 -75.88, -10.96 in-in in 8.208 Saltbr-in 2.506 HRD-in -82.4, -45.58 68.54, 13.94 in-in-in SNCiii in-in ActLoopNT-in 2.905 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.02, 172.84 APE9-dihe-na 63.46, 139.74 APE8-dihe-in -57.57, 136.79 APE8-rot-in 295.89 APE67-dihe-in -60.79, -29.87 -46.27, -47.23 APE12-dist-in 13.268 APE11-dist-in 11.678 APE10-dist-in 6.898 APE9-dist-in 3.074 None PTR216 PTR216 XRAY 2.5 0.212 0.249 B 350 350 0 0 0 0 [[56, 340]] 1.0 6hk4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5F94A P49841 36 381 420.0 3UO:401 Type1 Active DFGin 6.941 13.785 BLAminus -132.23, -171.99 59.12, 80.79 -95.82, 23.07 289.16, 72.98 -56.52, -34.28 in-in in 8.486 Saltbr-in 2.711 HRD-in -71.8, -46.49 68.5, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.784 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.99, 174.92 APE9-dihe-na 77.27, 148.67 APE8-dihe-in -101.45, 151.47 APE8-rot-in 289.94 APE67-dihe-inflip 89.58, -29.34 -36.24, 131.42 APE12-dist-in 12.915 APE11-dist-in 10.912 APE10-dist-in 5.952 APE9-dist-in 3.109 None None None XRAY 2.51 0.191 0.226 A 350 346 0 0 0 0 [[56, 340]] 1.0 5f94 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5F94B P49841 37 385 420.0 3UO:401 Type1 Active DFGin 6.921 13.903 BLAminus -131.5, -174.71 60.13, 82.54 -97.18, 23.01 287.88, 72.62 -56.23, -35.38 in-in in 8.398 Saltbr-in 2.89 HRD-in -70.35, -45.36 66.02, 7.89 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.68, 174.32 APE9-dihe-na 79.06, 151.27 APE8-dihe-in -105.02, 147.7 APE8-rot-in 292.84 APE67-dihe-inflip 87.17, -28.31 -40.05, 137.25 APE12-dist-in 12.887 APE11-dist-in 10.901 APE10-dist-in 5.866 APE9-dist-in 3.193 None None None XRAY 2.51 0.191 0.226 B 350 349 0 0 0 0 [[56, 340]] 1.0 5f94 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5F95A P49841 36 383 420.0 3UP:401 Type1 Active DFGin 6.851 14.121 BLAminus -131.03, -172.49 54.11, 85.8 -99.54, 23.42 287.04, 73.17 -58.21, -30.13 in-in in 8.492 Saltbr-in 2.642 HRD-in -68.05, -46.73 71.39, 6.88 in-in-in SNCiii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.52, 167.77 APE9-dihe-na 81.86, 152.62 APE8-dihe-in -108.33, 161.23 APE8-rot-in 296.59 APE67-dihe-in -81.75, 2.56 -4.13, -93.98 APE12-dist-in 13.1 APE11-dist-in 11.087 APE10-dist-in 6.378 APE9-dist-in 3.262 None None None XRAY 2.525 0.204 0.242 A 350 345 3 0 0 0 [[56, 340]] 1.0 5f95 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5F95B P49841 36 385 420.0 3UP:401 Type1 Active DFGin 7.029 14.131 BLAminus -130.15, -170.55 52.93, 82.9 -96.95, 23.47 283.9, 71.07 -57.67, -29.42 in-in in 8.524 Saltbr-in 2.241 HRD-in -68.94, -45.23 69.65, 6.25 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.14, 169.18 APE9-dihe-na 82.46, 143.88 APE8-dihe-in -96.17, 168.5 APE8-rot-in 296.7 APE67-dihe-in -78.34, 2.06 -36.18, -73.12 APE12-dist-in 13.021 APE11-dist-in 11.027 APE10-dist-in 6.092 APE9-dist-in 3.21 None None None XRAY 2.525 0.204 0.242 B 350 338 12 0 0 0 [[56, 340]] 1.0 5f95 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U31A P49841 36 385 420.0 L7I:402 Type1 Active DFGin 7.094 14.183 BLAminus -142.39, 178.42 62.99, 82.78 -98.0, 19.46 288.1, 81.67 -57.1, -32.73 in-in in 8.165 Saltbr-in 2.84 HRD-in -76.17, -49.99 76.15, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.54, -23.16 APE9-dihe-na -100.68, 154.06 APE8-dihe-in -79.73, 162.4 APE8-rot-in 294.75 APE67-dihe-in -75.9, -12.27 -44.4, -68.17 APE12-dist-in 13.102 APE11-dist-in 10.928 APE10-dist-in 5.909 APE9-dist-in 3.416 None None None XRAY 2.38 0.244 0.276 A 350 350 0 0 0 0 [[56, 340]] 1.0 7u31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U31B P49841 37 382 420.0 L7I:402 Type1 Active DFGin 7.049 14.287 BLAminus -143.88, 177.54 62.09, 82.63 -98.02, 19.8 287.95, 82.15 -57.33, -32.15 in-in in 8.377 Saltbr-in 2.717 HRD-in -76.73, -50.12 75.35, 8.49 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.33, 167.82 APE9-dihe-na 83.33, 132.28 APE8-dihe-in -83.68, 163.51 APE8-rot-in 292.75 APE67-dihe-in -76.54, -11.97 -40.44, -69.75 APE12-dist-in 13.108 APE11-dist-in 10.979 APE10-dist-in 5.927 APE9-dist-in 3.127 None None None XRAY 2.38 0.244 0.276 B 350 346 0 0 0 0 [[56, 340]] 1.0 7u31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7SXJA P49841 34 383 420.0 6VL:60401 Type1 Active DFGin 6.916 14.335 BLAminus -142.41, -179.99 59.67, 72.96 -86.59, 25.21 285.68, 73.81 -69.07, -21.65 in-in in 8.269 Saltbr-in 2.692 HRD-in -74.28, -41.7 68.05, 5.57 in-in-in SNCiii in-in ActLoopNT-in 2.943 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.32, 170.09 APE9-dihe-na 72.35, 148.74 APE8-dihe-in -71.51, 141.06 APE8-rot-in 303.21 APE67-dihe-in -59.11, -26.68 -51.44, -48.71 APE12-dist-in 13.503 APE11-dist-in 11.843 APE10-dist-in 7.042 APE9-dist-in 3.173 None PTR216 PTR216 XRAY 1.85 0.185 0.203 A 351 346 4 0 0 0 [[56, 340]] 1.0 7sxj Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7OY5A P49841 35 385 420.0 39I:401 Type1 Active DFGin 6.926 14.033 BLAminus -126.76, 175.34 72.52, 92.63 -110.59, 33.29 286.05, 82.06 -75.35, -28.56 in-in in 8.688 Saltbr-in 2.936 HRD-in -72.48, -55.14 81.29, 7.92 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.43, 173.86 APE9-dihe-na 80.53, 146.3 APE8-dihe-in -94.81, 142.24 APE8-rot-in 295.61 APE67-dihe-inflip 101.01, -30.19 -44.76, 139.01 APE12-dist-in 12.924 APE11-dist-in 10.96 APE10-dist-in 5.893 APE9-dist-in 3.276 None None None XRAY 2.57 0.221 0.26 A 351 343 8 0 0 0 [[56, 340]] 1.0 7oy5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7OY5B P49841 35 383 420.0 39I:401 Type1 Active DFGin 7.115 14.145 BLAminus -131.55, -176.92 63.09, 57.6 -70.26, 11.8 285.25, 87.17 -66.04, -15.46 in-in in 8.495 Saltbr-in 3.027 HRD-in -75.85, -49.73 71.52, 4.36 in-in-in SNCiii in-in ActLoopNT-in 3.039 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.28, 172.83 APE9-dihe-na 79.24, 135.47 APE8-dihe-in -76.12, 154.7 APE8-rot-in 287.59 APE67-dihe-inflip 110.96, -34.61 -67.01, 135.0 APE12-dist-in 13.03 APE11-dist-in 10.958 APE10-dist-in 5.992 APE9-dist-in 3.008 None None None XRAY 2.57 0.221 0.26 B 351 344 5 0 0 0 [[56, 340]] 1.0 7oy5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U33A P49841 36 385 420.0 L7R:402 Type1 Active DFGin 7.023 14.049 BLAminus -140.49, 178.19 60.8, 84.54 -99.85, 16.49 288.62, 77.82 -50.41, -27.99 in-in in 8.511 Saltbr-in 2.774 HRD-in -71.53, -50.0 75.9, 8.27 in-in-in SNCiii in-in ActLoopNT-in 2.986 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.78, -39.59 APE9-dihe-na -85.32, 160.12 APE8-dihe-in -84.45, 147.1 APE8-rot-in 286.21 APE67-dihe-inflip 87.92, -34.06 -59.31, 147.18 APE12-dist-in 13.036 APE11-dist-in 10.991 APE10-dist-in 6.032 APE9-dist-in 3.262 None None None XRAY 2.6 0.233 0.264 A 351 350 0 0 0 0 [[56, 340]] 1.0 7u33 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U33B P49841 37 382 420.0 L7R:402 Type1 Active DFGin 6.995 14.092 BLAminus -141.31, 178.2 60.97, 83.82 -100.06, 16.34 288.93, 78.7 -51.51, -27.59 in-in in 8.533 Saltbr-in 2.753 HRD-in -72.1, -49.87 75.78, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.62, 168.53 APE9-dihe-na 77.45, 140.58 APE8-dihe-in -89.54, 146.71 APE8-rot-in 285.53 APE67-dihe-in -82.12, -10.74 -0.24, -85.34 APE12-dist-in 13.035 APE11-dist-in 10.96 APE10-dist-in 6.029 APE9-dist-in 3.103 None None None XRAY 2.6 0.233 0.264 B 351 346 0 0 0 0 [[56, 340]] 1.0 7u33 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U36A P49841 36 385 420.0 L7W:402 Type1 Active DFGin 7.055 14.057 BLAminus -140.39, -178.87 60.34, 89.59 -105.19, 18.12 284.52, 86.52 -57.6, -32.5 in-in in 8.453 Saltbr-in 3.019 HRD-in -77.18, -47.14 70.51, 17.98 in-in-in SNCiii in-in ActLoopNT-in 2.959 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.43, -45.81 APE9-dihe-na -84.57, 153.41 APE8-dihe-in -68.83, 161.86 APE8-rot-in 280.03 APE67-dihe-in -82.26, -16.89 -53.14, -56.37 APE12-dist-in 12.87 APE11-dist-in 10.758 APE10-dist-in 5.812 APE9-dist-in 3.189 None None None XRAY 2.75 0.24 0.275 A 351 350 0 0 0 0 [[56, 340]] 1.0 7u36 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7U36B P49841 37 382 420.0 L7W:402 Type1 Active DFGin 7.056 14.071 BLAminus -141.26, -179.45 60.58, 88.51 -105.71, 18.11 283.81, 87.44 -57.54, -31.03 in-in in 8.498 Saltbr-in 2.991 HRD-in -77.32, -47.05 68.98, 19.83 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -102.55, 163.3 APE9-dihe-na 90.09, 132.18 APE8-dihe-in -72.41, 162.37 APE8-rot-in 279.62 APE67-dihe-in -81.75, -17.56 -53.5, -56.42 APE12-dist-in 12.856 APE11-dist-in 10.778 APE10-dist-in 5.79 APE9-dist-in 3.107 None None None XRAY 2.75 0.24 0.275 B 351 346 0 0 0 0 [[56, 340]] 1.0 7u36 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 2OW3A P49841 35 385 420.0 BIM:387 Type1 Active DFGin 6.854 14.088 BLAminus -145.58, -177.16 62.63, 79.7 -96.04, 38.01 299.18, 104.83 -72.62, -36.62 in-in in 8.34 Saltbr-in 2.838 HRD-in -75.79, -46.9 63.78, 27.01 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.84, 153.8 APE9-dihe-na 77.18, 154.82 APE8-dihe-in -72.33, 143.1 APE8-rot-in 299.46 APE67-dihe-in -64.33, -22.16 -49.08, -49.27 APE12-dist-in 13.724 APE11-dist-in 12.363 APE10-dist-in 7.515 APE9-dist-in 3.784 None PTR216 PTR216 XRAY 2.8 0.248 0.295 A 352 347 4 0 0 0 [[56, 340]] 1.0 2ow3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 2OW3B P49841 35 386 420.0 BIM:387 Type1 Active DFGin 6.768 14.52 BLAminus -140.91, -178.82 62.87, 80.36 -94.83, 34.08 291.22, 81.94 -79.34, -15.72 in-in in 8.48 Saltbr-in 2.788 HRD-in -91.97, -42.45 64.4, 21.24 in-in-in SNCiii in-in ActLoopNT-in 2.877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.27, 157.33 APE9-dihe-na 81.52, 163.87 APE8-dihe-in -81.91, 157.75 APE8-rot-in 308.08 APE67-dihe-in -65.81, -19.16 -55.34, -61.54 APE12-dist-in 13.905 APE11-dist-in 12.542 APE10-dist-in 7.628 APE9-dist-in 3.538 None PTR216 PTR216 XRAY 2.8 0.248 0.295 B 352 352 0 0 0 0 [[56, 340]] 1.0 2ow3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3GB2A P49841 35 383 420.0 G3B:999 Type1 Active DFGin 7.081 13.502 BLAminus -136.77, -176.86 57.81, 94.36 -109.09, 24.06 290.54, 74.85 -73.21, 4.88 in-in in 8.45 Saltbr-in 2.812 HRD-in -66.76, -55.55 72.33, 20.67 in-in-in SNCiii in-in ActLoopNT-in 2.859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.38, -175.57 APE9-dihe-na 67.46, 160.91 APE8-dihe-in -72.68, 139.68 APE8-rot-in 245.03 APE67-dihe-in -60.68, -25.16 -49.04, -51.42 APE12-dist-in 13.505 APE11-dist-in 11.973 APE10-dist-in 7.004 APE9-dist-in 3.287 None PTR216 PTR216 XRAY 2.4 0.225 0.289 A 353 341 8 0 0 0 [[56, 340]] 1.0 3gb2 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6TCUA P49841 35 384 420.0 N1Q:401 Type1 Active DFGin 7.271 14.191 BLAminus -132.13, 178.03 59.16, 82.25 -93.13, 22.32 285.63, 78.52 -60.3, -31.7 in-in in 8.352 Saltbr-in 2.912 HRD-in -72.47, -46.38 65.88, 22.79 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.64, 162.18 APE9-dihe-na 73.42, 158.65 APE8-dihe-in -78.26, 138.24 APE8-rot-in 295.07 APE67-dihe-in -60.71, -25.87 -50.61, -49.17 APE12-dist-in 13.556 APE11-dist-in 11.943 APE10-dist-in 7.197 APE9-dist-in 3.24 None PTR216 PTR216 XRAY 2.14 0.204 0.24 A 355 350 0 0 0 0 [[56, 340]] 1.0 6tcu Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.9e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5T31A P49841 35 381 420.0 6VL:501 Type1 Active DFGin 7.0 14.6 BLAminus -146.5, -178.72 58.09, 85.8 -94.81, 34.39 283.96, 70.89 -72.9, -29.06 in-in in 8.183 Saltbr-in 2.823 HRD-in -85.27, -37.65 59.13, 22.16 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.45, 179.68 APE9-dihe-na 63.71, 158.01 APE8-dihe-in -85.57, 141.47 APE8-rot-in 304.73 APE67-dihe-in -68.11, -24.88 -45.34, -45.1 APE12-dist-in 13.218 APE11-dist-in 11.545 APE10-dist-in 6.564 APE9-dist-in 3.195 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 A 420 335 12 0 0 0 [[56, 340]] 1.0 5t31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5T31B P49841 36 382 420.0 6VL:501 Type1 Active DFGin 7.209 14.605 BLAminus -147.12, 178.9 61.54, 81.68 -96.09, 32.98 286.61, 73.16 -76.82, -18.6 in-in in 8.229 Saltbr-in 2.581 HRD-in -64.89, -47.6 63.02, 19.09 in-in-in SNCiii in-in ActLoopNT-in 3.018 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.39, 179.54 APE9-dihe-na 63.77, 153.96 APE8-dihe-in -75.26, 136.0 APE8-rot-in 291.41 APE67-dihe-in -61.67, -31.85 -41.28, -53.13 APE12-dist-in 13.381 APE11-dist-in 11.678 APE10-dist-in 6.473 APE9-dist-in 3.237 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 B 420 334 13 0 0 0 [[56, 340]] 1.0 5t31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7Z1GA P49841 27 383 420.0 3NG:60401 Type1 Active DFGin 7.272 14.699 BLAminus -137.45, -179.93 52.32, 81.51 -93.1, 20.22 282.75, 78.65 -65.74, -16.48 in-in in 8.969 Saltbr-in 2.771 HRD-in -67.62, -47.44 74.98, 2.45 in-in-in SNCiii in-in ActLoopNT-in 2.926 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.67, 177.94 APE9-dihe-na 70.81, 142.84 APE8-dihe-in -95.23, 170.55 APE8-rot-in 305.08 APE67-dihe-inflip 72.5, -37.64 -53.01, 158.1 APE12-dist-in 12.785 APE11-dist-in 10.847 APE10-dist-in 5.858 APE9-dist-in 2.984 None None None XRAY 2.85 0.204 0.228 A 364 355 2 0 0 0 [[56, 340]] 1.0 7z1g Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7B6FA P49841 36 382 420.0 SZW:401 Type1 Active DFGin 6.788 14.002 BLAminus -139.5, -179.55 63.73, 84.52 -97.59, 24.1 286.83, 79.42 -64.99, -20.21 in-in in 8.319 Saltbr-in 2.573 HRD-in -72.27, -45.59 68.3, 15.73 in-in-in SNCiii in-in ActLoopNT-in 2.861 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.61, 164.26 APE9-dihe-na 74.41, 146.1 APE8-dihe-in -66.85, 137.72 APE8-rot-in 301.31 APE67-dihe-in -60.67, -24.91 -43.57, -54.9 APE12-dist-in 13.468 APE11-dist-in 11.675 APE10-dist-in 7.087 APE9-dist-in 3.203 None PTR216 PTR216 XRAY 2.05 0.176 0.209 A 365 347 0 0 0 0 [[56, 340]] 1.0 7b6f Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8AUZA P49841 27 381 420.0 O9C:402 Type1 Active DFGin 7.028 13.822 BLAminus -150.9, 179.1 54.07, 83.84 -94.84, 28.62 288.95, 81.72 -71.58, -10.75 in-in in 8.497 Saltbr-in 2.734 HRD-in -57.37, -52.37 73.76, 8.1 in-in-in SNCiii in-in ActLoopNT-in 3.155 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.43, 171.72 APE9-dihe-na 68.38, 153.94 APE8-dihe-in -73.1, 142.46 APE8-rot-in 305.9 APE67-dihe-in -60.73, -30.47 -42.52, -61.25 APE12-dist-in 13.255 APE11-dist-in 11.714 APE10-dist-in 7.025 APE9-dist-in 3.055 None PTR216 PTR216 XRAY 2.66 0.172 0.229 A 365 351 4 0 0 0 [[56, 340]] 1.0 8auz Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8AUZB P49841 27 381 420.0 O9C:402 Type1 Active DFGin 7.099 13.907 BLAminus -145.47, 175.75 60.6, 82.78 -92.91, 28.92 286.05, 79.75 -73.75, -11.85 in-in in 8.586 Saltbr-in 2.697 HRD-in -55.14, -51.91 71.49, 10.11 in-in-in SNCiii in-in ActLoopNT-in 3.139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.91, 170.34 APE9-dihe-na 66.33, 153.39 APE8-dihe-in -70.91, 144.03 APE8-rot-in 280.02 APE67-dihe-in -59.87, -32.25 -43.58, -60.53 APE12-dist-in 13.172 APE11-dist-in 11.662 APE10-dist-in 6.924 APE9-dist-in 3.004 None PTR216 PTR216 XRAY 2.66 0.172 0.229 B 365 351 4 0 0 0 [[56, 340]] 1.0 8auz Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4AFJA P49841 36 384 420.0 SJJ:1391 Type1 Active DFGin 6.937 13.715 BLAminus -130.67, 179.05 59.17, 87.64 -94.83, 20.23 280.89, 81.14 -65.73, -20.9 in-in in 8.572 Saltbr-in 2.652 HRD-in -69.53, -45.4 65.78, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.937 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.24, 160.98 APE9-dihe-na 76.37, 138.38 APE8-dihe-in -58.5, 130.27 APE8-rot-in 301.13 APE67-dihe-in -61.75, -23.96 -37.58, -52.92 APE12-dist-in 13.435 APE11-dist-in 11.681 APE10-dist-in 6.975 APE9-dist-in 3.193 None PTR216 PTR216 XRAY 1.98 0.179 0.216 A 367 344 5 0 0 0 [[56, 340]] 1.0 4afj Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4AFJB P49841 34 384 420.0 SJJ:1392 Type1 Active DFGin 6.948 14.046 BLAminus -131.53, 179.02 57.76, 85.75 -93.28, 22.08 280.88, 83.41 -64.33, -20.8 in-in in 8.525 Saltbr-in 2.743 HRD-in -67.39, -46.66 68.06, 10.89 in-in-in SNCiii in-in ActLoopNT-in 2.877 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.99, 165.35 APE9-dihe-na 75.2, 154.5 APE8-dihe-in -78.53, 128.88 APE8-rot-in 295.4 APE67-dihe-in -61.46, -24.46 -31.5, -55.04 APE12-dist-in 13.476 APE11-dist-in 11.582 APE10-dist-in 6.958 APE9-dist-in 3.146 None PTR216 PTR216 XRAY 1.98 0.179 0.216 B 367 347 4 0 0 0 [[56, 340]] 1.0 4afj Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3ZRKA P49841 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.886 13.908 BLAminus -131.68, 179.96 63.1, 79.53 -95.35, 25.37 286.53, 78.64 -74.21, -8.59 in-in in 8.474 Saltbr-in 2.75 HRD-in -67.17, -50.87 73.03, 10.45 in-in-in SNCiii in-in ActLoopNT-in 2.841 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.35, 160.84 APE9-dihe-na 74.59, 142.57 APE8-dihe-in -61.86, 136.31 APE8-rot-in 305.46 APE67-dihe-in -59.75, -23.44 -46.23, -50.56 APE12-dist-in 13.377 APE11-dist-in 11.67 APE10-dist-in 7.003 APE9-dist-in 3.16 None PTR216 PTR216 XRAY 2.37 0.201 0.243 A 371 347 2 0 0 0 [[56, 340]] 1.0 3zrk Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3ZRKB P49841 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.715 14.017 BLAminus -139.49, -177.28 57.97, 77.09 -90.4, 24.0 286.01, 81.23 -69.91, -16.36 in-in in 8.587 Saltbr-in 2.732 HRD-in -64.4, -48.95 71.37, 3.03 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.35, 163.72 APE9-dihe-na 73.35, 153.59 APE8-dihe-in -70.79, 138.65 APE8-rot-in 292.42 APE67-dihe-in -62.81, -26.76 -44.91, -48.41 APE12-dist-in 13.36 APE11-dist-in 11.482 APE10-dist-in 6.882 APE9-dist-in 3.161 None PTR216 PTR216 XRAY 2.37 0.201 0.243 B 371 349 0 0 0 0 [[56, 340]] 1.0 3zrk Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3ZRLA P49841 36 385 420.0 ZRL:1390 Type1 Active DFGin 6.976 14.145 BLAminus -134.74, 178.82 66.15, 74.2 -88.14, 21.07 285.95, 79.46 -68.66, -8.3 in-in in 8.484 Saltbr-in 2.586 HRD-in -74.36, -46.11 75.3, 2.22 in-in-in SNCiii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.36, 158.14 APE9-dihe-na 75.43, 144.25 APE8-dihe-in -61.72, 142.08 APE8-rot-in 315.78 APE67-dihe-in -63.29, -26.99 -52.04, -46.88 APE12-dist-in 13.478 APE11-dist-in 11.716 APE10-dist-in 7.157 APE9-dist-in 3.171 None PTR216 PTR216 XRAY 2.48 0.188 0.249 A 371 348 2 0 0 0 [[56, 340]] 1.0 3zrl Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3ZRLB P49841 36 384 420.0 ZRL:1390 Type1 Active DFGin 6.816 14.066 BLAminus -140.64, -176.21 56.19, 79.11 -88.83, 19.02 286.49, 80.49 -67.02, -13.2 in-in in 8.613 Saltbr-in 2.734 HRD-in -62.44, -47.89 69.81, 8.62 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.8, 160.71 APE9-dihe-na 76.77, 159.03 APE8-dihe-in -75.92, 142.27 APE8-rot-in 284.41 APE67-dihe-in -61.87, -25.02 -48.38, -50.46 APE12-dist-in 13.452 APE11-dist-in 11.697 APE10-dist-in 7.085 APE9-dist-in 3.218 None PTR216 PTR216 XRAY 2.48 0.188 0.249 B 371 349 0 0 0 0 [[56, 340]] 1.0 3zrl Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3ZRMA P49841 36 383 420.0 ZRM:1388 Type1 Active DFGin 6.934 13.954 BLAminus -132.01, -179.16 64.76, 76.89 -91.07, 16.45 285.73, 79.52 -60.99, -14.53 in-in in 8.379 Saltbr-in 2.59 HRD-in -73.17, -48.0 77.03, 4.47 in-in-in SNCiii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.45, 164.9 APE9-dihe-na 71.3, 144.2 APE8-dihe-in -61.55, 140.83 APE8-rot-in 305.4 APE67-dihe-in -61.36, -25.73 -52.92, -47.77 APE12-dist-in 13.418 APE11-dist-in 11.733 APE10-dist-in 7.034 APE9-dist-in 3.184 None PTR216 PTR216 XRAY 2.49 0.19 0.247 A 371 346 2 0 0 0 [[56, 340]] 1.0 3zrm Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3ZRMB P49841 36 384 420.0 ZRM:1389 Type1 Active DFGin 6.902 14.104 BLAminus -140.7, -177.64 59.24, 76.67 -89.43, 25.85 287.41, 78.75 -71.45, -17.33 in-in in 8.556 Saltbr-in 2.639 HRD-in -65.21, -46.92 71.38, 6.55 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.4, 163.13 APE9-dihe-na 76.6, 157.17 APE8-dihe-in -72.35, 137.17 APE8-rot-in 272.08 APE67-dihe-in -62.09, -20.43 -43.42, -53.94 APE12-dist-in 13.463 APE11-dist-in 11.697 APE10-dist-in 7.031 APE9-dist-in 3.11 None PTR216 PTR216 XRAY 2.49 0.19 0.247 B 371 349 0 0 0 0 [[56, 340]] 1.0 3zrm Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5K5NA P49841 36 382 420.0 6QH:4001 Type1 Active DFGin 6.867 13.803 BLAminus -136.97, -178.03 58.54, 81.58 -94.06, 22.59 285.28, 80.04 -66.6, -22.76 in-in in 8.685 Saltbr-in 2.763 HRD-in -65.0, -45.17 61.7, 20.55 in-in-in SNCiii in-in ActLoopNT-in 2.904 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.55, 163.97 APE9-dihe-na 70.72, 157.82 APE8-dihe-in -71.18, 131.1 APE8-rot-in 299.71 APE67-dihe-in -62.03, -24.12 -33.31, -56.32 APE12-dist-in 13.585 APE11-dist-in 11.966 APE10-dist-in 6.992 APE9-dist-in 3.201 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 A 370 332 12 0 0 0 [[56, 340]] 1.0 5k5n Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5K5NB P49841 36 384 420.0 6QH:401 Type1 Active DFGin 6.968 13.745 BLAminus -135.06, -178.44 58.85, 83.42 -94.58, 20.58 286.7, 80.8 -64.41, -22.37 in-in in 8.869 Saltbr-in 2.795 HRD-in -64.71, -45.91 63.61, 14.11 in-in-in SNCiii in-in ActLoopNT-in 2.88 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.36, 162.07 APE9-dihe-na 75.01, 147.36 APE8-dihe-in -65.41, 124.62 APE8-rot-in 290.2 APE67-dihe-in -56.35, -27.77 -26.59, -62.75 APE12-dist-in 13.372 APE11-dist-in 11.994 APE10-dist-in 6.896 APE9-dist-in 3.109 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 B 370 335 11 0 0 0 [[56, 340]] 1.0 5k5n Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1R0EA P49841 35 383 420.0 DFN:702 Type1 Active DFGin 7.211 13.978 BLAminus -134.01, -179.44 58.42, 85.11 -96.64, 20.85 278.46, 77.75 -63.57, -17.65 in-in in 8.372 Saltbr-in 2.716 HRD-in -68.9, -46.99 73.89, 15.3 in-in-in SNCiii in-in ActLoopNT-in 2.817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.99, 167.9 APE9-dihe-na 82.35, 148.07 APE8-dihe-in -104.61, 148.9 APE8-rot-in 290.93 APE67-dihe-inflip 91.63, -34.6 -37.68, 131.22 APE12-dist-in 13.098 APE11-dist-in 11.094 APE10-dist-in 6.24 APE9-dist-in 3.395 None None None XRAY 2.25 0.225 0.252 A 391 344 5 0 0 0 [[56, 340]] 1.0 1r0e Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1R0EB P49841 35 383 420.0 DFN:501 Type1 Active DFGin 7.247 14.105 BLAminus -133.07, -177.02 55.1, 85.48 -97.08, 20.86 276.04, 78.13 -65.93, -17.26 in-in in 8.445 Saltbr-in 2.91 HRD-in -68.16, -44.28 70.07, 10.75 in-in-in SNCiii in-in ActLoopNT-in 2.884 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.79, 168.13 APE9-dihe-na 84.81, 147.78 APE8-dihe-in -104.27, 148.93 APE8-rot-in 288.7 APE67-dihe-inflip 91.14, -35.24 -35.52, 130.18 APE12-dist-in 13.079 APE11-dist-in 11.011 APE10-dist-in 6.177 APE9-dist-in 3.369 None None None XRAY 2.25 0.225 0.252 B 391 344 5 0 0 0 [[56, 340]] 1.0 1r0e Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q5KA P49841 35 384 420.0 TMU:901 Type1 Active DFGin 6.988 13.863 BLAminus -136.18, -175.74 56.25, 81.9 -94.66, 24.16 283.53, 73.95 -64.32, -18.01 in-in in 8.227 Saltbr-in 2.549 HRD-in -67.21, -47.72 71.71, 7.94 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.63, 174.67 APE9-dihe-na 78.79, 134.14 APE8-dihe-in -77.03, 144.65 APE8-rot-in 302.42 APE67-dihe-inflip 99.66, -34.41 -53.93, 140.09 APE12-dist-in 12.905 APE11-dist-in 11.002 APE10-dist-in 5.832 APE9-dist-in 3.144 None None None XRAY 1.94 0.222 0.242 A 414 345 5 0 0 0 [[56, 340]] 1.0 1q5k Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q5KB P49841 35 384 420.0 TMU:902 Type1 Active DFGin 6.985 13.773 BLAminus -138.67, -177.12 58.86, 79.46 -94.38, 28.16 285.34, 70.82 -69.41, -14.87 in-in in 8.132 Saltbr-in 2.832 HRD-in -69.04, -44.01 68.27, 5.21 in-in-in SNCiii in-in ActLoopNT-in 2.916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.05, 176.86 APE9-dihe-na 75.09, 135.72 APE8-dihe-in -79.59, 144.98 APE8-rot-in 303.4 APE67-dihe-inflip 93.62, -37.01 -50.51, 145.1 APE12-dist-in 12.931 APE11-dist-in 11.072 APE10-dist-in 5.846 APE9-dist-in 3.103 None None None XRAY 1.94 0.222 0.242 B 414 344 6 0 0 0 [[56, 340]] 1.0 1q5k Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3I4BA P49841 25 385 420.0 Z48:501 Type1 Active DFGin 6.641 13.646 BLAminus -134.01, -176.44 58.71, 78.24 -93.71, 24.37 285.69, 79.56 -67.57, -20.03 in-in in 8.476 Saltbr-in 2.637 HRD-in -63.92, -46.73 77.65, -7.51 in-in-in SNCiii in-in ActLoopNT-in 2.95 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.08, 174.13 APE9-dihe-na 79.29, 137.44 APE8-dihe-in -92.27, 151.07 APE8-rot-in 303.5 APE67-dihe-inflip 83.63, -1.22 -43.52, 132.98 APE12-dist-in 13.009 APE11-dist-in 10.939 APE10-dist-in 5.839 APE9-dist-in 3.102 None None None XRAY 2.3 0.181 0.222 A 414 359 0 0 0 0 [[56, 340]] 1.0 3i4b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3I4BB P49841 36 382 420.0 Z48:501 Type1 Active DFGin 7.01 13.655 BLAminus -135.85, -175.31 58.14, 77.59 -93.89, 21.58 285.55, 84.81 -65.19, -18.79 in-in in 8.508 Saltbr-in 2.617 HRD-in -67.57, -44.79 75.92, -6.36 in-in-in SNCiii in-in ActLoopNT-in 2.941 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.93, 173.5 APE9-dihe-na 79.53, 137.7 APE8-dihe-in -93.51, 150.41 APE8-rot-in 299.4 APE67-dihe-inflip 78.16, -1.88 -37.33, 134.24 APE12-dist-in 13.043 APE11-dist-in 10.917 APE10-dist-in 5.828 APE9-dist-in 3.115 None None None XRAY 2.3 0.181 0.222 B 414 347 0 0 0 0 [[56, 340]] 1.0 3i4b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3L1SA P49841 25 384 420.0 Z92:421 Type1 Active DFGin 6.757 13.748 BLAminus -136.19, -175.27 59.75, 67.96 -82.46, 22.04 287.73, 86.13 -66.81, -21.63 in-in in 8.518 Saltbr-in 2.708 HRD-in -64.1, -46.34 73.45, -1.44 in-in-in SNCiii in-in ActLoopNT-in 2.949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 172.3 APE9-dihe-na 79.23, 137.51 APE8-dihe-in -89.89, 147.82 APE8-rot-in 303.47 APE67-dihe-inflip 83.2, -1.08 -42.22, 131.52 APE12-dist-in 13.007 APE11-dist-in 10.892 APE10-dist-in 5.894 APE9-dist-in 3.161 None None None XRAY 2.9 0.186 0.232 A 414 336 21 0 0 0 [[56, 340]] 1.0 3l1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3L1SB P49841 36 382 420.0 Z92:422 Type1 Active DFGin 6.984 13.78 BLAminus -136.63, -175.36 61.34, 59.7 -75.09, 22.69 291.46, 84.75 -66.47, -23.35 in-in in 8.551 Saltbr-in 2.737 HRD-in -65.65, -45.98 77.68, -13.89 in-in-in SNCiii in-in ActLoopNT-in 2.937 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.08, 173.03 APE9-dihe-na 76.72, 137.31 APE8-dihe-in -89.1, 148.7 APE8-rot-in 302.46 APE67-dihe-inflip 83.32, 3.78 -42.62, 131.74 APE12-dist-in 13.014 APE11-dist-in 10.916 APE10-dist-in 6.149 APE9-dist-in 3.121 None None None XRAY 2.9 0.186 0.232 B 414 330 17 0 0 0 [[56, 340]] 1.0 3l1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 2JLDA P49841 35 385 420.0 AG1:1385 Type1 Active DFGin 7.247 13.619 BLAminus -128.74, 174.0 65.55, 89.02 -101.06, 20.23 281.85, 78.64 -66.01, -16.46 in-in in 8.535 Saltbr-in 2.901 HRD-in -68.74, -48.89 74.29, 10.13 in-in-in SNCiii in-in ActLoopNT-in 2.846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -80.14, 165.31 APE9-dihe-na 82.65, 142.84 APE8-dihe-in -89.49, 145.54 APE8-rot-in 290.56 APE67-dihe-inflip 101.97, -33.31 -39.01, 124.35 APE12-dist-in 13.012 APE11-dist-in 11.005 APE10-dist-in 6.058 APE9-dist-in 3.239 None None None XRAY 2.35 0.192 0.227 A 420 349 2 0 0 0 [[56, 340]] 1.0 2jld Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 2JLDB P49841 35 384 420.0 AG1:1385 Type1 Active DFGin 7.117 13.681 BLAminus -134.8, 174.83 62.6, 85.31 -97.62, 21.89 284.88, 76.87 -65.09, -17.38 in-in in 8.458 Saltbr-in 2.725 HRD-in -67.92, -46.43 70.86, 13.33 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.11, 167.47 APE9-dihe-na 84.04, 143.71 APE8-dihe-in -89.79, 148.89 APE8-rot-in 294.08 APE67-dihe-inflip 95.31, -31.23 -37.35, 123.61 APE12-dist-in 13.044 APE11-dist-in 10.951 APE10-dist-in 5.995 APE9-dist-in 3.203 None None None XRAY 2.35 0.192 0.227 B 420 349 1 0 0 0 [[56, 340]] 1.0 2jld Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3M1SB P49841 35 384 420.0 DW1:421 Type1 Active DFGin 7.187 13.372 BLAminus -147.84, 174.37 70.86, 99.58 -120.24, 19.87 286.56, 80.37 -63.52, -14.18 in-in in 8.585 Saltbr-in 2.441 HRD-in -69.47, -49.47 71.23, 28.36 in-in-in SNCiii in-in ActLoopNT-in 3.091 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -106.87, 165.89 APE9-dihe-na 90.21, 134.65 APE8-dihe-in -74.2, 145.74 APE8-rot-in 300.21 APE67-dihe-in -72.41, -23.39 -22.57, -69.43 APE12-dist-in 12.944 APE11-dist-in 10.712 APE10-dist-in 5.899 APE9-dist-in 3.769 None None None XRAY 3.134 0.171 0.228 B 420 349 1 0 0 0 [[56, 340]] 1.0 3m1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3PUPA P49841 35 382 420.0 OS1:421 Type1 Active DFGin 6.995 13.637 BLAminus -143.74, 172.61 64.16, 94.87 -107.49, 13.61 287.44, 72.72 -52.4, -32.47 in-in in 8.443 Saltbr-in 2.807 HRD-in -86.73, -34.2 66.44, 7.86 in-in-in SNCiii in-in ActLoopNT-in 2.857 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.24, -13.27 APE9-dihe-na -89.84, 168.85 APE8-dihe-in -94.34, 159.6 APE8-rot-in 296.79 APE67-dihe-in -69.26, -2.79 -42.9, -70.67 APE12-dist-in 13.056 APE11-dist-in 10.912 APE10-dist-in 6.171 APE9-dist-in 3.486 None None None XRAY 2.99 0.206 0.249 A 420 346 2 0 0 0 [[56, 340]] 1.0 3pup Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3PUPB P49841 35 383 420.0 OS1:421 Type1 Active DFGin 6.987 13.646 BLAminus -146.61, 171.7 65.62, 100.17 -113.12, 21.06 287.13, 70.81 -60.05, -30.47 in-in in 8.479 Saltbr-in 2.972 HRD-in -88.21, -42.27 77.46, 8.13 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.13, -17.37 APE9-dihe-na -97.38, 160.84 APE8-dihe-in -100.44, 160.76 APE8-rot-in 282.35 APE67-dihe-in -75.14, -2.22 -49.84, -64.39 APE12-dist-in 13.107 APE11-dist-in 10.976 APE10-dist-in 6.5 APE9-dist-in 3.751 None None None XRAY 2.99 0.206 0.249 B 420 347 2 0 0 0 [[56, 340]] 1.0 3pup Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6B8JA P49841 37 384 420.0 65C:502 Type1 Active DFGin 6.868 13.909 BLAminus -142.04, -175.4 56.86, 72.8 -87.54, 21.75 287.01, 61.58 -69.77, -16.08 in-in in 8.507 Saltbr-in 2.318 HRD-in -66.49, -42.97 62.67, 20.6 in-in-in SNCiii in-in ActLoopNT-in 2.821 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.37, 166.1 APE9-dihe-na 69.29, 116.74 APE8-dihe-in -38.51, 137.94 APE8-rot-in 299.43 APE67-dihe-in -65.74, -24.52 -56.45, -42.14 APE12-dist-in 13.685 APE11-dist-in 11.734 APE10-dist-in 7.018 APE9-dist-in 3.326 None PTR216 PTR216 XRAY 2.595 0.215 0.247 A 420 345 3 0 0 0 [[56, 340]] 1.0 6b8j Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6H0UA P49841 36 383 420.0 FKB:501 Type1 Active DFGin 6.732 13.816 BLAminus -102.2, -173.91 62.01, 94.18 -105.02, 23.81 292.61, 84.27 -66.96, -25.5 in-in in 8.798 Saltbr-in 2.726 HRD-in -71.89, -49.13 79.92, 3.93 in-in-in SNCiii in-in ActLoopNT-in 2.966 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.85, 170.11 APE9-dihe-na 84.06, 143.45 APE8-dihe-in -90.7, 142.53 APE8-rot-in 301.69 APE67-dihe-in -73.12, -14.65 -13.27, -76.63 APE12-dist-in 12.955 APE11-dist-in 10.868 APE10-dist-in 5.76 APE9-dist-in 3.223 None None None XRAY 2.3 0.195 0.24 A 420 348 0 0 0 0 [[56, 340]] 1.0 6h0u Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6H0UB P49841 36 383 420.0 FKB:501 Type1 Active DFGin 6.648 13.973 BLAminus -111.78, 175.04 68.36, 93.29 -102.83, 22.46 286.57, 84.56 -63.31, -24.15 in-in in 8.763 Saltbr-in 2.745 HRD-in -68.5, -49.8 75.08, 1.45 in-in-in SNCiii in-in ActLoopNT-in 2.851 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.21, 171.64 APE9-dihe-na 80.61, 138.7 APE8-dihe-in -91.3, 150.17 APE8-rot-in 304.68 APE67-dihe-inflip 101.55, -29.52 -53.44, 134.06 APE12-dist-in 12.722 APE11-dist-in 10.726 APE10-dist-in 5.704 APE9-dist-in 3.163 None None None XRAY 2.3 0.195 0.24 B 420 348 0 0 0 0 [[56, 340]] 1.0 6h0u Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6V6LA P49841 37 384 420.0 QQA:501 Type1 Active DFGin 7.244 14.228 BLAminus -134.87, -179.15 59.4, 83.41 -98.99, 30.0 283.16, 72.37 -75.66, -20.38 in-in in 8.388 Saltbr-in 2.736 HRD-in -68.21, -49.19 67.93, 18.71 in-in-in SNCiii in-in ActLoopNT-in 3.016 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.84, 162.85 APE9-dihe-na 77.33, 149.16 APE8-dihe-in -69.69, 129.38 APE8-rot-in 287.88 APE67-dihe-in -58.07, -31.39 -36.48, -49.2 APE12-dist-in 13.461 APE11-dist-in 11.648 APE10-dist-in 6.953 APE9-dist-in 3.241 None PTR216 PTR216 XRAY 2.19 0.204 0.234 A 420 344 4 0 0 0 [[56, 340]] 1.0 6v6l Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3DU8A P49841 35 382 420.0 553:553 Type1 Active DFGin 6.992 13.938 BLAminus -138.88, -177.6 60.76, 81.45 -97.52, 17.85 284.1, 81.79 -60.5, -23.71 in-in in 8.713 Saltbr-in 2.686 HRD-in -70.97, -44.22 68.9, 5.64 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.61, 170.6 APE9-dihe-na 82.17, 142.06 APE8-dihe-in -90.1, 145.24 APE8-rot-in 300.29 APE67-dihe-inflip 98.68, -34.99 -51.44, 136.14 APE12-dist-in 13.036 APE11-dist-in 10.944 APE10-dist-in 5.764 APE9-dist-in 3.152 None None None XRAY 2.2 0.215 0.246 A 422 336 12 0 0 0 [[56, 340]] 1.0 3du8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3DU8B P49841 35 385 420.0 553:553 Type1 Active DFGin 7.11 14.001 BLAminus -130.0, -177.1 64.69, 78.27 -91.27, 21.46 283.91, 80.88 -65.59, -20.64 in-in in 8.742 Saltbr-in 2.702 HRD-in -71.12, -43.48 71.58, 1.27 in-in-in SNCiii in-in ActLoopNT-in 2.992 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -75.13, 166.25 APE9-dihe-na 83.98, 139.39 APE8-dihe-in -88.38, 143.61 APE8-rot-in 294.95 APE67-dihe-inflip 93.54, -38.98 -56.03, 145.75 APE12-dist-in 13.05 APE11-dist-in 11.13 APE10-dist-in 5.901 APE9-dist-in 3.176 None None None XRAY 2.2 0.215 0.246 B 422 339 12 0 0 0 [[56, 340]] 1.0 3du8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR5A P49841 25 385 420.0 A1IE8:501 Type1 Active DFGin 7.063 14.321 BLAminus -141.02, 178.57 59.76, 86.64 -101.14, 27.38 287.09, 76.28 -70.78, -13.94 in-in in 8.363 Saltbr-in 2.867 HRD-in -72.5, -48.23 71.7, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.985 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.15, 177.99 APE9-dihe-na 68.95, 145.14 APE8-dihe-in -94.16, 151.35 APE8-rot-in 288.71 APE67-dihe-inflip 90.22, -34.5 -47.82, 143.36 APE12-dist-in 13.104 APE11-dist-in 11.105 APE10-dist-in 6.167 APE9-dist-in 3.186 None None None XRAY 2.3 0.204 0.235 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR5B P49841 36 382 420.0 A1IE8:501 Type1 Active DFGin 7.068 14.397 BLAminus -143.23, 179.4 62.21, 84.47 -103.42, 28.19 287.66, 78.04 -72.31, -18.53 in-in in 8.684 Saltbr-in 2.965 HRD-in -72.41, -47.52 71.61, 14.06 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.66, -179.45 APE9-dihe-na 68.77, 147.4 APE8-dihe-in -97.67, 156.22 APE8-rot-in 283.57 APE67-dihe-inflip 84.77, -33.0 -49.59, 145.66 APE12-dist-in 13.056 APE11-dist-in 10.953 APE10-dist-in 5.986 APE9-dist-in 3.188 None None None XRAY 2.3 0.204 0.235 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR6A P49841 25 385 420.0 A1IFO:501 Type1 Active DFGin 7.074 14.161 BLAminus -136.83, -174.79 60.55, 80.3 -97.86, 24.81 287.57, 77.74 -66.69, -16.26 in-in in 8.556 Saltbr-in 2.935 HRD-in -72.59, -48.06 71.15, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.992 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.91, 171.88 APE9-dihe-na 74.24, 144.89 APE8-dihe-in -96.08, 152.09 APE8-rot-in 291.49 APE67-dihe-inflip 90.67, -36.1 -52.14, 144.18 APE12-dist-in 13.022 APE11-dist-in 11.047 APE10-dist-in 6.124 APE9-dist-in 3.24 None None None XRAY 2.3 0.2 0.232 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR6B P49841 36 382 420.0 A1IFO:501 Type1 Active DFGin 7.128 14.36 BLAminus -139.12, -179.31 63.06, 81.93 -99.98, 26.01 286.75, 75.51 -71.16, -14.75 in-in in 8.843 Saltbr-in 2.836 HRD-in -72.29, -48.89 71.91, 12.0 in-in-in SNCiii in-in ActLoopNT-in 2.917 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.4, 172.1 APE9-dihe-na 77.09, 144.87 APE8-dihe-in -98.08, 154.15 APE8-rot-in 291.27 APE67-dihe-inflip 90.37, -33.63 -52.57, 140.86 APE12-dist-in 13.071 APE11-dist-in 10.957 APE10-dist-in 5.983 APE9-dist-in 3.22 None None None XRAY 2.3 0.2 0.232 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR7A P49841 25 385 420.0 A1IFJ:501 Type1 Active DFGin 6.912 13.949 BLAminus -136.24, -176.42 58.55, 87.09 -104.67, 27.04 287.13, 78.6 -71.53, -14.0 in-in in 8.632 Saltbr-in 2.802 HRD-in -71.98, -46.0 72.36, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.987 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.42, 177.43 APE9-dihe-na 69.9, 145.82 APE8-dihe-in -94.03, 156.28 APE8-rot-in 289.17 APE67-dihe-inflip 91.05, -31.63 -52.45, 141.85 APE12-dist-in 13.108 APE11-dist-in 11.121 APE10-dist-in 6.121 APE9-dist-in 3.15 None None None XRAY 2.3 0.199 0.229 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR7B P49841 36 382 420.0 A1IFJ:501 Type1 Active DFGin 6.99 13.952 BLAminus -139.3, -178.5 61.7, 87.08 -105.92, 24.05 284.91, 80.77 -70.11, -13.68 in-in in 8.593 Saltbr-in 2.71 HRD-in -71.41, -48.43 71.41, 11.5 in-in-in SNCiii in-in ActLoopNT-in 2.94 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.82, 177.23 APE9-dihe-na 70.05, 146.13 APE8-dihe-in -96.47, 160.58 APE8-rot-in 285.27 APE67-dihe-inflip 87.67, -29.95 -51.57, 140.33 APE12-dist-in 13.008 APE11-dist-in 11.007 APE10-dist-in 6.045 APE9-dist-in 3.156 None None None XRAY 2.3 0.199 0.229 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR8A P49841 25 385 420.0 A1IE7:501 Type1 Active DFGin 6.991 14.325 BLAminus -138.39, -179.52 63.72, 81.82 -96.4, 23.65 287.29, 75.6 -66.3, -11.74 in-in in 8.553 Saltbr-in 2.906 HRD-in -71.33, -45.89 67.7, 10.94 in-in-in SNCiii in-in ActLoopNT-in 2.957 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.78, 169.84 APE9-dihe-na 80.06, 148.59 APE8-dihe-in -102.16, 146.47 APE8-rot-in 284.89 APE67-dihe-inflip 97.34, -39.62 -53.84, 140.75 APE12-dist-in 13.081 APE11-dist-in 11.083 APE10-dist-in 6.012 APE9-dist-in 3.197 None None None XRAY 2.3 0.191 0.221 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR8B P49841 36 383 420.0 A1IE7:501 Type1 Active DFGin 7.087 14.356 BLAminus -145.34, 175.42 68.0, 83.84 -100.29, 22.36 287.83, 75.27 -65.32, -15.0 in-in in 8.715 Saltbr-in 2.898 HRD-in -76.0, -49.5 72.49, 12.34 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.57, 172.15 APE9-dihe-na 78.67, 145.51 APE8-dihe-in -99.99, 146.48 APE8-rot-in 286.49 APE67-dihe-inflip 90.46, -36.44 -48.06, 141.27 APE12-dist-in 13.067 APE11-dist-in 10.852 APE10-dist-in 5.85 APE9-dist-in 3.153 None None None XRAY 2.3 0.191 0.221 B 442 348 0 0 0 0 [[56, 340]] 1.0 9fr8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR9A P49841 25 385 420.0 A1IE6:501 Type1 Active DFGin 7.037 14.325 BLAminus -140.22, -173.71 59.89, 84.2 -98.36, 22.56 286.21, 81.87 -68.06, -16.06 in-in in 8.462 Saltbr-in 2.928 HRD-in -72.09, -48.73 72.37, 5.47 in-in-in SNCiii in-in ActLoopNT-in 2.971 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.48, 176.45 APE9-dihe-na 79.51, 153.1 APE8-dihe-in -106.78, 146.27 APE8-rot-in 287.32 APE67-dihe-inflip 100.87, -37.49 -40.18, 126.82 APE12-dist-in 13.02 APE11-dist-in 11.03 APE10-dist-in 5.997 APE9-dist-in 3.173 None None None XRAY 2.55 0.197 0.234 A 442 361 0 0 0 0 [[56, 340]] 1.0 9fr9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9FR9B P49841 36 382 420.0 A1IE6:501 Type1 Active DFGin 6.97 14.413 BLAminus -146.13, 179.78 62.16, 86.8 -103.01, 25.64 284.6, 80.86 -74.54, -16.98 in-in in 8.76 Saltbr-in 3.487 HRD-in -67.74, -52.21 72.42, 13.09 in-in-in SNCiii in-in ActLoopNT-in 2.872 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.09, 170.35 APE9-dihe-na 79.85, 140.07 APE8-dihe-in -93.7, 153.67 APE8-rot-in 288.81 APE67-dihe-inflip 99.37, -31.56 -52.24, 133.09 APE12-dist-in 12.982 APE11-dist-in 10.81 APE10-dist-in 5.791 APE9-dist-in 3.181 None None None XRAY 2.55 0.197 0.234 B 442 347 0 0 0 0 [[56, 340]] 1.0 9fr9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9HUKB P49841 26 382 420.0 A1IXL:501 Type1 Active DFGin 7.463 14.062 BLAminus -139.0, -179.94 58.73, 94.97 -114.49, 25.32 285.15, 69.98 -63.61, -20.61 in-in in 8.13 Saltbr-in 3.28 HRD-in -69.2, -40.72 63.39, 20.78 in-in-in SNCiii in-in ActLoopNT-in 3.042 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.58, -178.87 APE9-dihe-na 67.27, 135.83 APE8-dihe-in -80.15, 163.62 APE8-rot-in 319.54 APE67-dihe-inflip 75.84, -27.97 -60.6, 162.6 APE12-dist-in 12.838 APE11-dist-in 10.744 APE10-dist-in 5.73 APE9-dist-in 3.212 None None None XRAY 3.5 0.219 0.25 B 442 357 0 0 0 0 [[56, 340]] 1.0 9huk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9HULA P49841 25 385 420.0 A1IXM:501 Type1 Active DFGin 7.07 13.943 BLAminus -137.8, -179.92 58.93, 93.22 -109.33, 21.24 284.01, 77.28 -66.77, -7.95 in-in in 8.344 Saltbr-in 2.923 HRD-in -67.44, -42.84 67.99, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.167 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.24, 178.29 APE9-dihe-na 68.13, 143.96 APE8-dihe-in -84.08, 162.04 APE8-rot-in 308.02 APE67-dihe-inflip 75.91, -35.84 -57.58, 161.58 APE12-dist-in 13.066 APE11-dist-in 11.024 APE10-dist-in 5.997 APE9-dist-in 3.163 None None None XRAY 2.9 0.218 0.244 A 442 361 0 0 0 0 [[56, 340]] 1.0 9hul Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9HULB P49841 26 383 420.0 A1IXM:501 Type1 Active DFGin 7.218 13.9 BLAminus -141.92, -177.61 60.57, 66.5 -86.27, 21.98 288.8, 69.64 -66.75, -12.19 in-in in 8.268 Saltbr-in 2.748 HRD-in -68.36, -43.53 65.84, 14.02 in-in-in SNCiii in-in ActLoopNT-in 3.018 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.86, 177.51 APE9-dihe-na 70.81, 136.76 APE8-dihe-in -79.57, 164.11 APE8-rot-in 306.92 APE67-dihe-inflip 69.45, -30.71 -58.24, 165.67 APE12-dist-in 13.055 APE11-dist-in 10.975 APE10-dist-in 6.055 APE9-dist-in 3.14 None None None XRAY 2.9 0.218 0.244 B 442 358 0 0 0 0 [[56, 340]] 1.0 9hul Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9HV3A P49841 25 385 420.0 A1IXN:501 Type1 Active DFGin 7.125 13.97 BLAminus -135.63, 170.17 69.98, 84.71 -102.55, 20.46 290.46, 80.59 -69.94, -0.25 in-in in 8.537 Saltbr-in 2.868 HRD-in -69.25, -48.0 72.7, 9.47 in-in-in SNCiii in-in ActLoopNT-in 2.935 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.1, 169.69 APE9-dihe-na 79.34, 142.23 APE8-dihe-in -80.23, 146.96 APE8-rot-in 316.9 APE67-dihe-inflip 78.3, -27.2 -49.89, 154.45 APE12-dist-in 13.123 APE11-dist-in 11.12 APE10-dist-in 6.197 APE9-dist-in 3.136 None None None XRAY 2.9 0.208 0.238 A 442 361 0 0 0 0 [[56, 340]] 1.0 9hv3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9HV3B P49841 25 382 420.0 A1IXN:501 Type1 Active DFGin 7.087 13.912 BLAminus -155.32, 174.2 63.74, 86.56 -102.98, 16.67 284.3, 76.87 -64.93, -6.56 in-in in 8.597 Saltbr-in 2.606 HRD-in -75.09, -41.25 66.67, 4.87 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.85, 168.81 APE9-dihe-na 83.21, 130.42 APE8-dihe-in -66.5, 151.79 APE8-rot-in 306.21 APE67-dihe-inflip 94.47, -29.15 -64.06, 143.12 APE12-dist-in 12.974 APE11-dist-in 10.879 APE10-dist-in 5.979 APE9-dist-in 3.017 None None None XRAY 2.9 0.208 0.238 B 442 358 0 0 0 0 [[56, 340]] 1.0 9hv3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q3DA P49841 35 385 420.0 STU:451 Type1 Active DFGin 7.206 14.411 BLAminus -139.48, 178.33 63.94, 87.17 -99.43, 23.77 282.58, 69.4 -66.25, -14.58 in-in in 8.701 Saltbr-in 2.855 HRD-in -65.74, -44.7 66.01, 11.52 in-in-in SNCiii in-in ActLoopNT-in 3.036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.53, 169.72 APE9-dihe-na 81.56, 143.56 APE8-dihe-in -91.54, 154.32 APE8-rot-in 294.67 APE67-dihe-inflip 96.36, -28.56 -51.12, 132.48 APE12-dist-in 13.074 APE11-dist-in 11.108 APE10-dist-in 6.087 APE9-dist-in 3.274 None None None XRAY 2.2 0.23 0.252 A 424 339 12 0 0 0 [[56, 340]] 1.0 1q3d Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q3DB P49841 35 383 420.0 STU:452 Type1 Active DFGin 7.26 14.419 BLAminus -137.95, 177.39 64.41, 87.07 -97.99, 22.53 282.7, 70.11 -63.96, -17.29 in-in in 8.708 Saltbr-in 2.972 HRD-in -67.72, -45.35 66.86, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.75, 170.28 APE9-dihe-na 79.08, 144.81 APE8-dihe-in -89.94, 151.95 APE8-rot-in 299.26 APE67-dihe-inflip 101.61, -31.22 -54.51, 132.99 APE12-dist-in 13.085 APE11-dist-in 11.088 APE10-dist-in 6.146 APE9-dist-in 3.238 None None None XRAY 2.2 0.23 0.252 B 424 339 10 0 0 0 [[56, 340]] 1.0 1q3d Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q3WA P49841 35 386 420.0 ATU:502 Type1 Active DFGin 7.146 13.952 BLAminus -137.77, 177.61 62.94, 83.24 -96.07, 24.67 288.22, 69.87 -66.71, -10.0 in-in in 8.322 Saltbr-in 2.924 HRD-in -67.11, -47.79 71.57, 6.31 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.32, 172.63 APE9-dihe-na 77.53, 136.48 APE8-dihe-in -79.93, 143.51 APE8-rot-in 298.62 APE67-dihe-in -62.35, -17.4 -13.52, -82.56 APE12-dist-in 13.075 APE11-dist-in 11.129 APE10-dist-in 5.964 APE9-dist-in 3.143 None None None XRAY 2.3 0.225 0.248 A 424 344 8 0 0 0 [[56, 340]] 1.0 1q3w Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q3WB P49841 35 383 420.0 ATU:501 Type1 Active DFGin 7.09 14.27 BLAminus -140.46, 175.46 63.78, 84.76 -97.02, 22.89 286.31, 71.96 -64.9, -10.6 in-in in 8.547 Saltbr-in 2.792 HRD-in -67.92, -47.98 71.69, 6.95 in-in-in SNCiii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.2, 172.08 APE9-dihe-na 78.0, 136.99 APE8-dihe-in -80.5, 143.58 APE8-rot-in 301.78 APE67-dihe-in -64.47, -16.3 -12.81, -81.64 APE12-dist-in 13.069 APE11-dist-in 11.111 APE10-dist-in 5.938 APE9-dist-in 3.147 None None None XRAY 2.3 0.225 0.248 B 424 341 8 0 0 0 [[56, 340]] 1.0 1q3w Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q41A P49841 35 386 420.0 IXM:451 Type1 Active DFGin 7.096 13.742 BLAminus -140.31, 177.95 63.36, 85.31 -97.68, 24.93 285.2, 72.61 -64.62, -16.75 in-in in 8.182 Saltbr-in 2.845 HRD-in -70.03, -43.74 69.02, 2.85 in-in-in SNCiii in-in ActLoopNT-in 3.007 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.85, 173.09 APE9-dihe-na 80.34, 135.13 APE8-dihe-in -75.55, 139.31 APE8-rot-in 298.19 APE67-dihe-in -65.33, -18.78 -13.64, -78.26 APE12-dist-in 13.068 APE11-dist-in 11.057 APE10-dist-in 5.915 APE9-dist-in 3.225 None None None XRAY 2.1 0.229 0.245 A 424 339 13 0 0 0 [[56, 340]] 1.0 1q41 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q41B P49841 35 383 420.0 IXM:452 Type1 Active DFGin 7.094 13.894 BLAminus -139.75, 177.7 62.59, 85.88 -97.92, 24.85 285.3, 70.28 -63.82, -17.54 in-in in 8.388 Saltbr-in 2.83 HRD-in -70.82, -46.38 71.27, 6.28 in-in-in SNCiii in-in ActLoopNT-in 3.007 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.0, 171.76 APE9-dihe-na 82.35, 130.54 APE8-dihe-in -71.97, 140.37 APE8-rot-in 298.15 APE67-dihe-in -64.0, -13.46 -11.43, -84.5 APE12-dist-in 13.056 APE11-dist-in 11.055 APE10-dist-in 5.884 APE9-dist-in 3.236 None None None XRAY 2.1 0.229 0.245 B 424 343 6 0 0 0 [[56, 340]] 1.0 1q41 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q4LA P49841 35 386 420.0 679:451 Type1 Active DFGin 6.944 13.754 BLAminus -138.39, -176.39 57.74, 86.06 -99.56, 21.29 285.7, 72.79 -65.03, -5.34 in-in in 8.524 Saltbr-in 3.007 HRD-in -67.11, -46.06 68.04, 16.48 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -95.21, 168.86 APE9-dihe-na 81.69, 129.23 APE8-dihe-in -70.09, 146.41 APE8-rot-in 291.03 APE67-dihe-inflip 104.98, -29.32 -58.42, 137.67 APE12-dist-in 13.117 APE11-dist-in 11.352 APE10-dist-in 6.301 APE9-dist-in 3.339 None None None XRAY 2.77 0.212 0.251 A 424 342 10 0 0 0 [[56, 340]] 1.0 1q4l Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1Q4LB P49841 35 383 420.0 679:452 Type1 Active DFGin 7.169 13.649 BLAminus -140.11, -177.14 58.72, 87.12 -99.76, 20.01 285.14, 71.58 -64.5, -5.39 in-in in 8.339 Saltbr-in 2.673 HRD-in -67.89, -45.11 67.21, 17.1 in-in-in SNCiii in-in ActLoopNT-in 2.996 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.61, 167.87 APE9-dihe-na 83.04, 132.56 APE8-dihe-in -74.69, 156.93 APE8-rot-in 311.31 APE67-dihe-inflip 93.39, -29.64 -61.08, 141.61 APE12-dist-in 13.098 APE11-dist-in 11.322 APE10-dist-in 6.253 APE9-dist-in 3.349 None None None XRAY 2.77 0.212 0.251 B 424 337 12 0 0 0 [[56, 340]] 1.0 1q4l Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3Q3BA P49841 35 386 420.0 55E:421 Type1 Active DFGin 6.859 13.89 BLAminus -146.51, -174.92 60.73, 82.19 -97.34, 22.93 287.93, 77.72 -66.67, -8.01 in-in in 8.46 Saltbr-in 2.718 HRD-in -65.09, -51.43 75.32, 0.61 in-in-in SNCiii in-in ActLoopNT-in 3.024 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.28, 172.26 APE9-dihe-na 79.45, 140.83 APE8-dihe-in -87.39, 149.52 APE8-rot-in 308.45 APE67-dihe-in -68.31, -14.9 -12.45, -80.03 APE12-dist-in 13.004 APE11-dist-in 11.06 APE10-dist-in 6.186 APE9-dist-in 3.146 None None None XRAY 2.7 0.228 0.259 A 424 344 8 0 0 0 [[56, 340]] 1.0 3q3b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3Q3BB P49841 35 383 420.0 55E:421 Type1 Active DFGin 6.944 13.767 BLAminus -148.03, -175.09 60.19, 82.65 -96.08, 19.99 287.37, 77.74 -64.82, -9.3 in-in in 8.443 Saltbr-in 2.789 HRD-in -64.26, -50.5 74.85, 0.78 in-in-in SNCiii in-in ActLoopNT-in 3.048 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.17, 172.11 APE9-dihe-na 80.0, 136.06 APE8-dihe-in -78.43, 156.9 APE8-rot-in 303.64 APE67-dihe-in -69.77, -0.18 -23.17, -84.47 APE12-dist-in 12.996 APE11-dist-in 11.045 APE10-dist-in 6.179 APE9-dist-in 3.102 None None None XRAY 2.7 0.228 0.259 B 424 341 8 0 0 0 [[56, 340]] 1.0 3q3b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4J1RA P49841 36 383 420.0 I5R:502 Type1 Active DFGin 7.143 14.149 BLAminus -140.34, -172.16 50.83, 73.0 -88.1, 31.44 288.82, 75.41 -70.78, -20.52 in-in in 8.339 Saltbr-in 3.026 HRD-in -70.85, -43.96 67.49, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.918 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.66, 159.85 APE9-dihe-na 83.41, 158.3 APE8-dihe-in -70.39, 137.75 APE8-rot-in 276.14 APE67-dihe-in -62.89, -24.7 -48.3, -48.41 APE12-dist-in 13.466 APE11-dist-in 11.878 APE10-dist-in 7.006 APE9-dist-in 3.199 None PTR216 PTR216 XRAY 2.702 0.174 0.193 A 424 344 4 0 0 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4J1RB P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.16 14.132 BLAminus -138.14, -172.1 51.97, 73.85 -90.74, 32.74 288.65, 76.48 -71.96, -19.84 in-in in 8.351 Saltbr-in 3.08 HRD-in -72.6, -39.29 60.47, 16.92 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.96, 157.32 APE9-dihe-na 86.27, 160.84 APE8-dihe-in -74.2, 139.51 APE8-rot-in 270.87 APE67-dihe-in -63.78, -23.12 -48.17, -50.06 APE12-dist-in 13.461 APE11-dist-in 11.633 APE10-dist-in 6.981 APE9-dist-in 3.199 None PTR216 PTR216 XRAY 2.702 0.174 0.193 B 424 347 2 0 0 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4J1RC P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.154 14.145 BLAminus -137.53, -170.95 51.06, 74.57 -90.65, 33.09 289.21, 75.99 -73.08, -20.73 in-in in 8.344 Saltbr-in 3.009 HRD-in -71.61, -39.59 60.78, 16.42 in-in-in SNCiii in-in ActLoopNT-in 2.951 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.54, 161.15 APE9-dihe-na 82.95, 157.27 APE8-dihe-in -71.13, 139.05 APE8-rot-in 271.75 APE67-dihe-in -63.34, -23.83 -48.75, -48.68 APE12-dist-in 13.475 APE11-dist-in 11.975 APE10-dist-in 7.027 APE9-dist-in 3.219 None PTR216 PTR216 XRAY 2.702 0.174 0.193 C 424 345 4 0 0 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4J1RD P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.157 14.143 BLAminus -136.3, -170.0 51.29, 73.39 -89.98, 32.08 288.97, 75.59 -72.78, -18.14 in-in in 8.347 Saltbr-in 3.082 HRD-in -65.4, -45.24 73.44, 1.93 in-in-in SNCiii in-in ActLoopNT-in 2.929 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.81, 157.82 APE9-dihe-na 85.66, 159.76 APE8-dihe-in -71.48, 137.15 APE8-rot-in 266.3 APE67-dihe-in -62.21, -25.06 -46.41, -50.2 APE12-dist-in 13.465 APE11-dist-in 11.902 APE10-dist-in 7.024 APE9-dist-in 3.117 None PTR216 PTR216 XRAY 2.702 0.174 0.193 D 424 346 3 0 0 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5HLNA P49841 34 384 420.0 65C:501 Type1 Active DFGin 6.971 13.539 BLAminus -145.82, 177.83 61.52, 84.96 -98.63, 20.2 288.24, 74.65 -61.35, -16.22 in-in in 8.64 Saltbr-in 2.97 HRD-in -72.97, -42.53 59.11, 33.41 in-in-in SNCiii in-in ActLoopNT-in 2.966 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.08, -68.13 APE9-dihe-na -70.88, 179.27 APE8-dihe-in -73.41, 154.88 APE8-rot-in 283.39 APE67-dihe-in -59.67, -27.13 -52.94, -57.58 APE12-dist-in 13.109 APE11-dist-in 11.767 APE10-dist-in 7.214 APE9-dist-in 3.907 None PTR216 PTR216 XRAY 3.1 0.173 0.236 A 424 347 4 0 0 0 [[56, 340]] 1.0 5hln Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5HLPA P49841 36 382 420.0 65A:501 Type1 Active DFGin 7.186 14.396 BLAminus -136.58, -178.8 62.45, 78.77 -95.76, 20.37 283.01, 75.68 -68.07, -12.1 in-in in 8.146 Saltbr-in 2.605 HRD-in -72.39, -43.73 64.36, 19.61 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.83, 176.24 APE9-dihe-na 71.02, 146.23 APE8-dihe-in -63.35, 144.14 APE8-rot-in 289.42 APE67-dihe-in -64.86, -21.95 -54.37, -48.38 APE12-dist-in 13.667 APE11-dist-in 11.819 APE10-dist-in 6.644 APE9-dist-in 3.298 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 A 424 339 8 0 0 0 [[56, 340]] 1.0 5hlp Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5HLPB P49841 36 383 420.0 65A:501 Type1 Active DFGin 7.115 14.467 BLAminus -132.96, -174.02 57.79, 78.12 -94.26, 22.08 284.54, 74.66 -71.61, -17.17 in-in in 8.276 Saltbr-in 2.716 HRD-in -71.48, -47.76 70.66, 10.73 in-in-in SNCiii in-in ActLoopNT-in 2.837 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.37, 176.63 APE9-dihe-na 72.15, 149.52 APE8-dihe-in -67.13, 142.42 APE8-rot-in 293.57 APE67-dihe-in -63.1, -24.66 -49.41, -51.54 APE12-dist-in 13.356 APE11-dist-in 11.821 APE10-dist-in 6.581 APE9-dist-in 3.135 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 B 424 337 11 0 0 0 [[56, 340]] 1.0 5hlp Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5KPKA P49841 35 384 420.0 6VK:500 Type1 Active DFGin 6.912 14.508 BLAminus -138.4, -178.64 58.08, 79.3 -90.22, 19.44 284.58, 73.09 -63.35, -18.32 in-in in 8.574 Saltbr-in 2.73 HRD-in -73.46, -47.41 66.88, 21.39 in-in-in SNCiii in-in ActLoopNT-in 2.95 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.73, 163.34 APE9-dihe-na 69.65, 162.27 APE8-dihe-in -73.86, 143.79 APE8-rot-in 303.06 APE67-dihe-in -60.34, -24.86 -54.25, -52.95 APE12-dist-in 13.597 APE11-dist-in 12.156 APE10-dist-in 7.487 APE9-dist-in 3.243 None PTR216 PTR216 XRAY 2.4 0.17 0.224 A 424 347 3 0 0 0 [[56, 340]] 1.0 5kpk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5KPKB P49841 35 383 420.0 6VK:500 Type1 Active DFGin 7.028 14.524 BLAminus -138.48, -175.82 55.16, 85.06 -97.98, 23.13 277.82, 78.64 -67.65, -21.76 in-in in 8.585 Saltbr-in 2.685 HRD-in -71.19, -45.78 65.3, 13.14 in-in-in SNCiii in-in ActLoopNT-in 3.004 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.69, 168.24 APE9-dihe-na 65.31, 163.84 APE8-dihe-in -77.16, 143.7 APE8-rot-in 304.59 APE67-dihe-in -57.42, -23.92 -54.57, -50.84 APE12-dist-in 13.693 APE11-dist-in 12.164 APE10-dist-in 7.395 APE9-dist-in 3.104 None PTR216 PTR216 XRAY 2.4 0.17 0.224 B 424 345 4 0 0 0 [[56, 340]] 1.0 5kpk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5KPLA P49841 36 384 420.0 6VL:500 Type1 Active DFGin 7.044 14.253 BLAminus -136.48, 178.55 58.11, 81.69 -92.72, 18.86 289.18, 73.73 -64.85, -20.41 in-in in 8.348 Saltbr-in 2.486 HRD-in -65.11, -50.47 69.64, 19.91 in-in-in SNCiii in-in ActLoopNT-in 3.088 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.42, 168.54 APE9-dihe-na 62.76, 158.29 APE8-dihe-in -78.28, 147.71 APE8-rot-in 310.05 APE67-dihe-in -62.4, -23.75 -53.92, -48.24 APE12-dist-in 13.434 APE11-dist-in 11.879 APE10-dist-in 7.137 APE9-dist-in 3.388 None PTR216 PTR216 XRAY 2.6 0.182 0.244 A 424 340 9 0 0 0 [[56, 340]] 1.0 5kpl Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5KPLB P49841 36 383 420.0 6VL:500 Type1 Active DFGin 7.154 14.616 BLAminus -138.92, -172.41 52.88, 79.26 -88.95, 20.81 278.36, 73.5 -72.97, -16.23 in-in in 8.498 Saltbr-in 2.971 HRD-in -70.3, -40.66 56.94, 24.57 in-in-in SNCiii in-in ActLoopNT-in 2.781 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.07, 160.76 APE9-dihe-na 66.33, 169.2 APE8-dihe-in -85.14, 144.57 APE8-rot-in 313.48 APE67-dihe-in -71.14, -21.99 -47.02, -47.87 APE12-dist-in 13.645 APE11-dist-in 11.859 APE10-dist-in 7.367 APE9-dist-in 3.38 None PTR216 PTR216 XRAY 2.6 0.182 0.244 B 424 340 8 0 0 0 [[56, 340]] 1.0 5kpl Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5KPMA P49841 36 383 420.0 6VM:500 Type1 Active DFGin 7.179 14.152 BLAminus -127.54, 178.59 63.4, 85.66 -102.69, 28.41 287.99, 66.47 -62.48, -34.28 in-in in 8.406 Saltbr-in 2.669 HRD-in -73.98, -45.27 60.61, 25.04 in-in-in SNCiii in-in ActLoopNT-in 2.733 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.88, 162.98 APE9-dihe-na 64.81, 161.74 APE8-dihe-in -75.86, 141.16 APE8-rot-in 297.33 APE67-dihe-in -64.41, -17.12 -48.06, -52.48 APE12-dist-in 13.62 APE11-dist-in 11.838 APE10-dist-in 7.363 APE9-dist-in 3.261 None PTR216 PTR216 XRAY 2.69 0.178 0.24 A 424 345 3 0 0 0 [[56, 340]] 1.0 5kpm Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5KPMB P49841 36 384 420.0 6VM:500 Type1 Active DFGin 7.141 14.638 BLAminus -142.12, 178.63 60.71, 81.6 -96.16, 22.05 281.72, 76.19 -66.25, -7.91 in-in in 8.609 Saltbr-in 2.581 HRD-in -65.22, -49.2 64.23, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.993 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.34, 163.89 APE9-dihe-na 62.78, 158.8 APE8-dihe-in -77.09, 139.57 APE8-rot-in 302.93 APE67-dihe-in -64.17, -18.23 -41.12, -52.04 APE12-dist-in 13.559 APE11-dist-in 11.972 APE10-dist-in 7.47 APE9-dist-in 3.193 None PTR216 PTR216 XRAY 2.69 0.178 0.24 B 424 346 3 0 0 0 [[56, 340]] 1.0 5kpm Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4IQ6A P49841 37 382 420.0 IQ6:501 Type1 Active DFGin 7.068 14.008 BLAminus -142.1, 176.37 68.23, 72.95 -88.9, 16.75 291.61, 92.77 -55.61, -37.28 in-in in 8.574 Saltbr-in 2.841 HRD-in -66.67, -43.42 72.45, -14.35 in-in-in SNCiii in-in ActLoopNT-in 3.012 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.44, 163.79 APE9-dihe-na 84.06, 140.31 APE8-dihe-in -95.86, 141.6 APE8-rot-in 294.32 APE67-dihe-inflip 102.08, -40.06 -38.49, 130.32 APE12-dist-in 13.214 APE11-dist-in 11.007 APE10-dist-in 6.193 APE9-dist-in 3.167 None None None XRAY 3.12 0.188 0.227 A 426 324 22 0 0 0 [[56, 340]] 1.0 4iq6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3SAYA P49841 35 384 420.0 OFT:431 Type1 Active DFGin 6.924 14.208 BLAminus -134.06, -176.24 58.1, 80.75 -95.49, 24.69 285.79, 80.8 -58.99, -23.52 in-in in 8.765 Saltbr-in 2.683 HRD-in -76.77, -47.73 71.86, 15.98 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 177.68 APE9-dihe-na 70.36, 150.2 APE8-dihe-in -70.69, 142.5 APE8-rot-in 303.06 APE67-dihe-in -64.8, -21.63 -53.21, -43.25 APE12-dist-in 13.475 APE11-dist-in 11.768 APE10-dist-in 6.474 APE9-dist-in 3.141 None PTR216 PTR216 XRAY 2.231 0.202 0.23 A 430 348 2 0 0 0 [[56, 340]] 1.0 3say Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3SAYB P49841 35 382 420.0 OFT:431 Type1 Active DFGin 7.095 14.208 BLAminus -125.43, -174.49 59.4, 82.08 -94.07, 22.41 283.95, 82.11 -68.04, -11.91 in-in in 8.776 Saltbr-in 2.596 HRD-in -71.92, -46.59 68.83, 6.83 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.5, 172.68 APE9-dihe-na 72.51, 152.54 APE8-dihe-in -66.45, 133.95 APE8-rot-in 293.34 APE67-dihe-in -62.41, -25.02 -42.21, -48.58 APE12-dist-in 13.503 APE11-dist-in 11.83 APE10-dist-in 6.704 APE9-dist-in 3.093 None PTR216 PTR216 XRAY 2.231 0.202 0.23 B 430 348 0 0 0 0 [[56, 340]] 1.0 3say Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4PTCA P49841 36 381 420.0 2WE:501 Type1 Active DFGin 6.936 14.398 BLAminus -147.73, -174.11 62.98, 81.81 -100.26, 25.83 284.28, 79.03 -59.65, -43.28 in-in in 9.162 Saltbr-in 2.729 HRD-in -73.84, -45.42 69.86, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.77 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.04, 172.51 APE9-dihe-na 77.59, 144.28 APE8-dihe-in -89.54, 156.63 APE8-rot-in 297.82 APE67-dihe-inflip 95.7, -27.15 -58.15, 143.88 APE12-dist-in 13.05 APE11-dist-in 10.779 APE10-dist-in 6.004 APE9-dist-in 3.272 None None None XRAY 2.711 0.217 0.281 A 441 342 4 0 0 0 [[56, 340]] 1.0 4ptc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4PTCB P49841 35 385 420.0 2WE:501 Type1 Active DFGin 7.213 14.605 BLAminus -123.82, -167.89 50.38, 80.91 -94.33, 28.59 284.85, 71.64 -64.12, -29.45 in-in in 8.924 Saltbr-in 2.402 HRD-in -67.43, -42.31 63.02, 14.07 in-in-in SNCiii in-in ActLoopNT-in 2.936 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.89, 173.71 APE9-dihe-na 81.21, 152.66 APE8-dihe-in -112.25, 156.82 APE8-rot-in 292.56 APE67-dihe-inflip 100.85, -22.79 -44.26, 123.15 APE12-dist-in 13.083 APE11-dist-in 10.918 APE10-dist-in 5.89 APE9-dist-in 3.28 None None None XRAY 2.711 0.217 0.281 B 441 347 4 0 0 0 [[56, 340]] 1.0 4ptc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4PTEA P49841 36 382 420.0 2WF:501 Type1 Active DFGin 6.932 14.017 BLAminus -141.21, 178.04 57.99, 89.39 -100.23, 24.26 286.38, 75.9 -68.08, -19.02 in-in in 8.716 Saltbr-in 2.635 HRD-in -73.56, -44.45 69.11, 4.74 in-in-in SNCiii in-in ActLoopNT-in 2.792 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.74, 175.98 APE9-dihe-na 75.98, 148.82 APE8-dihe-in -103.79, 152.51 APE8-rot-in 295.33 APE67-dihe-inflip 95.08, -28.26 -38.95, 126.56 APE12-dist-in 12.979 APE11-dist-in 10.89 APE10-dist-in 5.883 APE9-dist-in 3.088 None None None XRAY 2.033 0.17 0.195 A 441 341 6 0 0 0 [[56, 340]] 1.0 4pte Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4PTEB P49841 36 385 420.0 2WF:501 Type1 Active DFGin 6.918 13.937 BLAminus -137.07, 179.43 58.52, 88.98 -101.38, 27.88 284.28, 76.88 -69.85, -20.65 in-in in 8.484 Saltbr-in 2.685 HRD-in -70.9, -46.61 73.05, 2.3 in-in-in SNCiii in-in ActLoopNT-in 2.887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.76, 178.59 APE9-dihe-na 72.73, 147.77 APE8-dihe-in -103.48, 150.66 APE8-rot-in 296.89 APE67-dihe-inflip 94.67, -27.57 -36.66, 125.81 APE12-dist-in 12.935 APE11-dist-in 10.88 APE10-dist-in 5.877 APE9-dist-in 3.154 None None None XRAY 2.033 0.17 0.195 B 441 347 3 0 0 0 [[56, 340]] 1.0 4pte Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4PTGA P49841 36 382 420.0 2WG:501 Type1 Active DFGin 7.003 13.916 BLAminus -132.5, 179.85 66.28, 92.0 -106.7, 26.9 285.24, 77.28 -68.07, -25.88 in-in in 8.541 Saltbr-in 2.828 HRD-in -68.57, -44.88 68.54, 10.31 in-in-in SNCiii in-in ActLoopNT-in 2.939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.39, 169.96 APE9-dihe-na 80.02, 147.16 APE8-dihe-in -96.08, 142.52 APE8-rot-in 290.31 APE67-dihe-inflip 90.23, -35.22 -45.66, 142.01 APE12-dist-in 13.056 APE11-dist-in 11.019 APE10-dist-in 6.12 APE9-dist-in 3.284 None None None XRAY 2.361 0.173 0.211 A 441 333 14 0 0 0 [[56, 340]] 1.0 4ptg Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4PTGB P49841 37 385 420.0 2WG:501 Type1 Active DFGin 6.951 13.863 BLAminus -136.28, -175.42 57.62, 87.0 -101.31, 27.32 285.42, 76.21 -67.67, -26.13 in-in in 8.437 Saltbr-in 2.705 HRD-in -71.07, -46.44 71.76, 6.12 in-in-in SNCiii in-in ActLoopNT-in 2.9 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.44, 175.88 APE9-dihe-na 76.35, 149.91 APE8-dihe-in -109.95, 151.08 APE8-rot-in 289.69 APE67-dihe-inflip 91.44, -30.76 -44.23, 136.59 APE12-dist-in 12.988 APE11-dist-in 11.009 APE10-dist-in 5.91 APE9-dist-in 3.16 None None None XRAY 2.361 0.173 0.211 B 441 332 17 0 0 0 [[56, 340]] 1.0 4ptg Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8DJCA P49841 35 382 420.0 UAU:501 Type1 Active DFGin 7.107 13.645 BLAminus -130.93, 175.08 68.46, 84.27 -99.8, 25.87 290.84, 77.95 -66.29, -22.25 in-in in 8.442 Saltbr-in 2.699 HRD-in -67.33, -44.59 69.12, 7.74 in-in-in SNCiii in-in ActLoopNT-in 2.984 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 169.18 APE9-dihe-na 83.11, 139.06 APE8-dihe-in -86.29, 148.88 APE8-rot-in 301.44 APE67-dihe-inflip 95.96, -28.78 -50.91, 136.23 APE12-dist-in 12.912 APE11-dist-in 10.831 APE10-dist-in 5.804 APE9-dist-in 3.257 None None None XRAY 2.463 0.217 0.242 A 441 331 17 0 0 0 [[56, 340]] 1.0 8djc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8DJCB P49841 35 385 420.0 UAU:501 Type1 Active DFGin 7.125 13.633 BLAminus -137.19, 179.71 59.65, 83.27 -96.94, 27.03 290.51, 79.22 -67.53, -21.56 in-in in 8.328 Saltbr-in 2.738 HRD-in -65.99, -44.91 69.53, 7.25 in-in-in SNCiii in-in ActLoopNT-in 2.986 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.05, 167.49 APE9-dihe-na 82.24, 138.29 APE8-dihe-in -85.04, 145.47 APE8-rot-in 300.63 APE67-dihe-inflip 98.12, -32.04 -46.91, 135.02 APE12-dist-in 12.942 APE11-dist-in 10.888 APE10-dist-in 5.944 APE9-dist-in 3.259 None None None XRAY 2.463 0.217 0.242 B 441 332 19 0 0 0 [[56, 340]] 1.0 8djc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8DJDA P49841 36 383 420.0 U3E:501 Type1 Active DFGin 7.183 13.878 BLAminus -134.36, -179.72 59.88, 85.28 -97.18, 26.66 285.76, 75.79 -65.91, -27.91 in-in in 8.357 Saltbr-in 2.704 HRD-in -66.89, -45.93 70.71, 8.73 in-in-in SNCiii in-in ActLoopNT-in 2.974 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -97.03, 169.31 APE9-dihe-na 77.5, 142.18 APE8-dihe-in -93.09, 155.03 APE8-rot-in 301.61 APE67-dihe-inflip 94.8, -31.52 -52.67, 137.81 APE12-dist-in 13.059 APE11-dist-in 11.039 APE10-dist-in 6.129 APE9-dist-in 3.198 None None None XRAY 2.205 0.209 0.222 A 441 338 10 0 0 0 [[56, 340]] 1.0 8djd Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8DJDB P49841 36 384 420.0 U3E:501 Type1 Active DFGin 7.129 13.919 BLAminus -133.17, 179.77 59.91, 85.17 -97.09, 26.57 285.62, 75.36 -66.56, -27.45 in-in in 8.347 Saltbr-in 2.697 HRD-in -66.65, -46.07 70.85, 8.52 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.46, 170.54 APE9-dihe-na 79.57, 140.07 APE8-dihe-in -94.46, 154.56 APE8-rot-in 301.16 APE67-dihe-inflip 94.52, -31.07 -52.58, 138.22 APE12-dist-in 13.086 APE11-dist-in 11.08 APE10-dist-in 6.077 APE9-dist-in 3.217 None None None XRAY 2.205 0.209 0.222 B 441 341 8 0 0 0 [[56, 340]] 1.0 8djd Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8DJEA P49841 36 384 420.0 U6S:501 Type1 Active DFGin 7.26 13.369 BLAminus -139.51, 175.88 67.17, 88.55 -102.31, 22.49 287.71, 78.25 -63.99, -27.99 in-in in 8.313 Saltbr-in 2.716 HRD-in -68.38, -45.52 70.24, 12.16 in-in-in SNCiii in-in ActLoopNT-in 2.893 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.85, 166.32 APE9-dihe-na 87.14, 140.36 APE8-dihe-in -88.6, 149.46 APE8-rot-in 293.07 APE67-dihe-inflip 99.13, -30.7 -44.53, 124.89 APE12-dist-in 12.957 APE11-dist-in 10.867 APE10-dist-in 6.044 APE9-dist-in 3.353 None None None XRAY 2.374 0.201 0.227 A 441 347 2 0 0 0 [[56, 340]] 1.0 8dje Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8DJEB P49841 36 385 420.0 U6S:501 Type1 Active DFGin 7.239 13.421 BLAminus -137.87, 177.52 63.92, 86.56 -101.17, 24.78 290.39, 74.84 -68.33, -25.47 in-in in 8.265 Saltbr-in 2.736 HRD-in -65.34, -46.08 68.76, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.889 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.12, 167.71 APE9-dihe-na 84.3, 145.94 APE8-dihe-in -98.8, 148.34 APE8-rot-in 293.36 APE67-dihe-inflip 97.13, -37.27 -40.76, 129.94 APE12-dist-in 12.957 APE11-dist-in 10.932 APE10-dist-in 5.908 APE9-dist-in 3.263 None None None XRAY 2.374 0.201 0.227 B 441 343 7 0 0 0 [[56, 340]] 1.0 8dje Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8FF8A P49841 36 382 420.0 XV0:501 Type1 Active DFGin 7.2 13.736 BLAminus -135.89, 175.65 65.86, 84.5 -97.83, 25.7 284.17, 77.94 -66.05, -27.44 in-in in 8.341 Saltbr-in 2.752 HRD-in -68.43, -43.4 70.29, 3.62 in-in-in SNCiii in-in ActLoopNT-in 2.842 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 167.87 APE9-dihe-na 84.02, 136.04 APE8-dihe-in -86.03, 151.96 APE8-rot-in 298.92 APE67-dihe-inflip 95.48, -31.71 -43.39, 129.41 APE12-dist-in 12.741 APE11-dist-in 10.753 APE10-dist-in 5.791 APE9-dist-in 3.211 None None None XRAY 2.33 0.198 0.217 A 441 347 0 0 0 0 [[56, 340]] 1.0 8ff8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8FF8B P49841 36 385 420.0 XV0:501 Type1 Active DFGin 7.2 13.811 BLAminus -130.19, -175.53 57.72, 85.5 -98.92, 25.25 283.55, 78.69 -65.7, -29.77 in-in in 8.339 Saltbr-in 2.746 HRD-in -67.11, -43.98 70.41, 3.15 in-in-in SNCiii in-in ActLoopNT-in 2.825 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.86, 169.83 APE9-dihe-na 81.04, 142.01 APE8-dihe-in -96.19, 150.13 APE8-rot-in 300.46 APE67-dihe-inflip 95.56, -32.32 -40.34, 130.68 APE12-dist-in 12.779 APE11-dist-in 10.784 APE10-dist-in 5.825 APE9-dist-in 3.218 None None None XRAY 2.33 0.198 0.217 B 441 346 4 0 0 0 [[56, 340]] 1.0 8ff8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3F88A P49841 35 383 420.0 3HT:999 Type1 Active DFGin 7.247 13.73 BLAminus -137.96, -171.11 53.2, 96.02 -109.46, 31.55 277.23, 77.74 -85.58, 3.2 in-in in 8.62 Saltbr-in 2.516 HRD-in -66.41, -48.84 71.78, 26.38 in-in-in SNCiii in-in ActLoopNT-in 3.141 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.98, 165.73 APE9-dihe-na 69.33, 171.05 APE8-dihe-in -86.85, 130.82 APE8-rot-in 314.66 APE67-dihe-in -71.94, -20.16 -24.55, -52.13 APE12-dist-in 13.547 APE11-dist-in 12.041 APE10-dist-in 7.341 APE9-dist-in 3.599 None PTR216 PTR216 XRAY 2.6 0.204 0.281 A 349 341 8 0 0 0 [[56, 340]] 1.0 3f88 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3F88B P49841 35 383 420.0 3HT:999 Type1 Active DFGin 7.0 13.651 BLAminus -143.93, 176.87 66.18, 95.41 -113.06, 21.86 281.61, 81.82 -72.47, -7.16 in-in in 8.765 Saltbr-in 2.671 HRD-in -64.13, -56.14 79.67, 28.55 in-in-in SNCiii in-in ActLoopNT-in 3.176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.92, 167.15 APE9-dihe-na 65.97, 165.61 APE8-dihe-in -80.57, 145.62 APE8-rot-in 308.56 APE67-dihe-in -71.31, -21.5 -44.75, -45.4 APE12-dist-in 13.509 APE11-dist-in 11.967 APE10-dist-in 7.257 APE9-dist-in 3.406 None PTR216 PTR216 XRAY 2.6 0.204 0.281 B 349 341 8 0 0 0 [[56, 340]] 1.0 3f88 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACCA P49841 35 385 420.0 7YG:1387 Type1 Active DFGin 7.183 13.581 BLAminus -136.28, 179.66 61.59, 88.25 -100.04, 20.56 281.3, 79.98 -65.9, -21.03 in-in in 8.347 Saltbr-in 2.762 HRD-in -66.74, -44.81 68.93, 1.06 in-in-in SNCiii in-in ActLoopNT-in 2.897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.14, 170.6 APE9-dihe-na 77.6, 138.09 APE8-dihe-in -85.62, 145.43 APE8-rot-in 296.7 APE67-dihe-inflip 94.96, -30.16 -47.88, 136.19 APE12-dist-in 13.034 APE11-dist-in 10.957 APE10-dist-in 5.889 APE9-dist-in 3.171 None None None XRAY 2.21 0.191 0.219 A 465 351 0 0 0 0 [[56, 340]] 1.0 4acc Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACCB P49841 35 385 420.0 7YG:1386 Type1 Active DFGin 7.228 13.524 BLAminus -136.66, 179.59 61.79, 88.29 -99.73, 21.22 281.91, 80.18 -66.08, -22.29 in-in in 8.245 Saltbr-in 2.871 HRD-in -66.61, -45.06 69.24, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.27, 172.02 APE9-dihe-na 75.79, 137.96 APE8-dihe-in -86.62, 146.41 APE8-rot-in 295.61 APE67-dihe-inflip 93.46, -30.62 -49.23, 136.97 APE12-dist-in 13.056 APE11-dist-in 11.009 APE10-dist-in 5.912 APE9-dist-in 3.182 None None None XRAY 2.21 0.191 0.219 B 465 351 0 0 0 0 [[56, 340]] 1.0 4acc Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACDA P49841 35 385 420.0 GR9:1385 Type1 Active DFGin 7.186 13.357 BLAminus -142.44, 176.49 66.05, 88.14 -100.25, 16.93 286.04, 81.9 -64.04, -24.03 in-in in 8.306 Saltbr-in 2.937 HRD-in -63.25, -48.42 73.67, 5.76 in-in-in SNCiii in-in ActLoopNT-in 2.883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.94, 167.01 APE9-dihe-na 78.77, 128.64 APE8-dihe-in -74.85, 143.25 APE8-rot-in 302.95 APE67-dihe-inflip 99.55, -31.6 -49.31, 132.99 APE12-dist-in 12.877 APE11-dist-in 10.868 APE10-dist-in 5.91 APE9-dist-in 3.21 None None None XRAY 2.6 0.18 0.226 A 465 351 0 0 0 0 [[56, 340]] 1.0 4acd Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACDB P49841 35 385 420.0 GR9:1385 Type1 Active DFGin 7.141 13.377 BLAminus -142.06, 177.81 64.05, 89.32 -100.31, 16.47 285.95, 82.89 -62.46, -26.08 in-in in 8.223 Saltbr-in 2.941 HRD-in -62.52, -48.15 72.88, 6.33 in-in-in SNCiii in-in ActLoopNT-in 2.892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.53, 167.96 APE9-dihe-na 77.33, 127.92 APE8-dihe-in -74.4, 143.25 APE8-rot-in 302.61 APE67-dihe-inflip 99.75, -32.16 -47.58, 132.33 APE12-dist-in 12.928 APE11-dist-in 10.947 APE10-dist-in 5.956 APE9-dist-in 3.211 None None None XRAY 2.6 0.18 0.226 B 465 351 0 0 0 0 [[56, 340]] 1.0 4acd Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACGA P49841 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.003 13.717 BLAminus -136.29, 179.17 66.16, 92.5 -104.82, 26.85 285.89, 83.54 -71.26, -31.7 in-in in 8.275 Saltbr-in 2.866 HRD-in -62.3, -47.68 71.35, 0.06 in-in-in SNCiii in-in ActLoopNT-in 2.99 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.26, 169.3 APE9-dihe-na 82.24, 136.71 APE8-dihe-in -91.92, 145.05 APE8-rot-in 294.1 APE67-dihe-inflip 97.4, -31.68 -47.8, 134.4 APE12-dist-in 12.946 APE11-dist-in 10.981 APE10-dist-in 5.928 APE9-dist-in 3.292 None None None XRAY 2.6 0.177 0.225 A 465 351 0 0 0 0 [[56, 340]] 1.0 4acg Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACGB P49841 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.06 13.61 BLAminus -135.89, 178.4 67.23, 92.34 -105.78, 27.09 285.23, 82.98 -71.05, -30.43 in-in in 8.379 Saltbr-in 2.98 HRD-in -63.74, -47.68 70.98, 1.15 in-in-in SNCiii in-in ActLoopNT-in 2.973 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.69, 168.91 APE9-dihe-na 83.12, 137.88 APE8-dihe-in -91.66, 145.04 APE8-rot-in 292.39 APE67-dihe-inflip 98.28, -31.78 -48.39, 133.48 APE12-dist-in 12.918 APE11-dist-in 10.934 APE10-dist-in 5.917 APE9-dist-in 3.29 None None None XRAY 2.6 0.177 0.225 B 465 351 0 0 0 0 [[56, 340]] 1.0 4acg Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACHA P49841 35 385 420.0 KDI:1386 Type1 Active DFGin 7.131 13.843 BLAminus -136.87, 179.55 65.58, 91.16 -104.2, 25.64 286.28, 84.07 -69.39, -35.2 in-in in 8.234 Saltbr-in 2.935 HRD-in -61.5, -48.36 72.42, -0.28 in-in-in SNCiii in-in ActLoopNT-in 2.982 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.62, 166.44 APE9-dihe-na 83.56, 135.36 APE8-dihe-in -86.16, 143.31 APE8-rot-in 295.11 APE67-dihe-inflip 98.78, -32.06 -48.27, 133.26 APE12-dist-in 12.998 APE11-dist-in 11.059 APE10-dist-in 5.983 APE9-dist-in 3.322 None None None XRAY 2.6 0.231 0.252 A 465 351 0 0 0 0 [[56, 340]] 1.0 4ach Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4ACHB P49841 35 385 420.0 KDI:1386 Type1 Active DFGin 7.081 13.716 BLAminus -136.91, 178.72 65.4, 91.31 -104.6, 25.63 285.26, 83.9 -68.47, -34.59 in-in in 8.36 Saltbr-in 2.938 HRD-in -60.93, -48.9 72.19, 0.38 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.1, 166.35 APE9-dihe-na 83.22, 136.77 APE8-dihe-in -87.16, 144.14 APE8-rot-in 294.96 APE67-dihe-inflip 98.6, -31.77 -49.65, 133.73 APE12-dist-in 12.935 APE11-dist-in 10.985 APE10-dist-in 5.938 APE9-dist-in 3.29 None None None XRAY 2.6 0.231 0.252 B 465 351 0 0 0 0 [[56, 340]] 1.0 4ach Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5OY4A P49841 36 385 420.0 B4K:504 Type1.5_Back Active DFGin 6.999 13.822 BLAminus -130.87, 178.64 57.91, 86.19 -95.47, 21.04 282.05, 81.42 -63.36, -27.5 in-in in 8.088 Saltbr-in 2.722 HRD-in -68.24, -44.36 63.28, 15.03 in-in-in SNCiii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.23, 157.34 APE9-dihe-na 87.05, 159.63 APE8-dihe-in -83.83, 115.67 APE8-rot-in 295.36 APE67-dihe-in -60.03, -25.52 -23.01, -56.29 APE12-dist-in 13.558 APE11-dist-in 11.689 APE10-dist-in 7.058 APE9-dist-in 3.446 None PTR216 PTR216 XRAY 3.2 0.196 0.229 A 420 350 0 0 0 0 [[56, 340]] 1.0 5oy4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4IQ6B P49841 37 382 420.0 IQ6:501 Type1.5_Back Active DFGin 7.065 14.057 BLAminus -142.54, 175.49 69.06, 72.09 -88.69, 16.42 291.37, 92.47 -54.24, -38.91 in-in in 8.609 Saltbr-in 2.85 HRD-in -66.96, -42.68 72.42, -15.31 in-in-in SNCiii in-in ActLoopNT-in 3.009 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.08, 167.69 APE9-dihe-na 81.68, 134.42 APE8-dihe-in -80.06, 146.43 APE8-rot-in 285.37 APE67-dihe-inflip 104.71, -27.8 -48.51, 126.71 APE12-dist-in 13.148 APE11-dist-in 10.908 APE10-dist-in 6.244 APE9-dist-in 3.115 None None None XRAY 3.12 0.188 0.227 B 426 332 14 0 0 0 [[56, 340]] 1.0 4iq6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6Y9SA P49841 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.759 13.615 ABAminus -144.68, -36.37 -95.25, 102.78 -104.54, 22.52 286.7, 80.89 -71.31, -22.3 in-in in 8.469 Saltbr-in 2.731 HRD-in -69.96, -46.79 66.16, 22.69 in-in-out SNCiio in-out ActLoopNT-in 2.869 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.41, 160.13 APE9-dihe-na 78.21, 163.56 APE8-dihe-in -74.57, 133.14 APE8-rot-out 174.03 APE67-dihe-in -60.25, -21.67 -45.31, -52.5 APE12-dist-in 13.391 APE11-dist-in 11.634 APE10-dist-in 6.815 APE9-dist-in 3.217 None PTR216 PTR216 XRAY 2.03 0.204 0.249 A 350 344 5 0 0 0 [[56, 340]] 1.0 6y9s Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6Y9SB P49841 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.466 13.644 ABAminus -142.08, -29.11 -101.71, 107.32 -109.34, 26.02 290.64, 79.47 -70.13, -24.37 in-in in 8.627 Saltbr-in 2.626 HRD-in -62.98, -47.75 66.63, 19.7 in-in-out SNCiio in-out ActLoopNT-in 2.871 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -149.54, 160.17 APE9-dihe-na 74.78, 156.26 APE8-dihe-in -72.21, 136.72 APE8-rot-out 179.96 APE67-dihe-in -63.91, -18.81 -47.88, -49.22 APE12-dist-in 13.498 APE11-dist-in 11.696 APE10-dist-in 6.94 APE9-dist-in 3.172 None PTR216 PTR216 XRAY 2.03 0.204 0.249 B 350 340 9 0 0 0 [[56, 340]] 1.0 6y9s Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4NM0A P49841 26 383 420.0 ADP:60408 ATPlike Inactive DFGin 6.641 14.213 BLAminus -133.4, -174.33 56.9, 85.51 -105.72, 27.83 287.31, 80.39 -76.48, -2.57 in-in in 8.774 Saltbr-in 3.094 HRD-in -69.87, -45.12 67.03, 14.87 in-in-out SNCiio in-out ActLoopNT-in 2.927 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -71.29, 168.54 APE9-dihe-na 70.19, 144.11 APE8-dihe-in -96.47, 160.21 APE8-rot-out 64.82 APE67-dihe-inflip 78.46, -27.02 -43.67, 149.07 APE12-dist-in 13.091 APE11-dist-in 10.885 APE10-dist-in 6.571 APE9-dist-in 3.135 None None None XRAY 2.5 0.193 0.239 A 389 355 0 0 0 0 [[56, 340]] 1.0 4nm0 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8XN6B P49841 26 386 420.0 ANP:501 ATPlike Inactive DFGin 6.538 13.65 BLAminus -128.79, 173.26 73.68, 79.74 -95.9, 22.51 291.63, 80.46 -68.54, -21.83 in-in in 8.329 Saltbr-in 2.823 HRD-in -66.59, -53.03 79.09, 5.6 in-in-out SNCiio in-out ActLoopNT-in 2.951 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -88.32, 165.9 APE9-dihe-na 83.63, 132.42 APE8-dihe-in -59.67, 147.17 APE8-rot-out 189.94 APE67-dihe-in -64.51, -21.68 -60.38, -49.59 APE12-dist-in 13.024 APE11-dist-in 10.97 APE10-dist-in 5.846 APE9-dist-in 3.081 None None None XRAY 2.4 0.194 0.242 B 421 359 2 0 0 0 [[56, 340]] 1.0 8xn6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9X2VA P49841 35 383 420.0 PG6:502 Allosteric Inactive DFGin 6.894 14.046 BLAminus -136.47, 179.58 67.71, 81.15 -94.13, 21.93 285.02, 80.61 -69.61, -16.35 in-in in 8.707 Saltbr-in 2.796 HRD-in -72.8, -46.17 70.48, 11.06 in-in-out SNCiio in-out ActLoopNT-in 2.929 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_iiii APE10-dihe-na -102.48, 5.03 APE9-dihe-na -128.33, 167.55 APE8-dihe-out 50.5, 42.65 APE8-rot-in 319.92 APE67-dihe-in -79.33, -58.3 -90.94, -21.28 APE12-dist-in 10.275 APE11-dist-in 11.184 APE10-dist-in 7.71 APE9-dist-in 4.04 None None None XRAY 1.39 0.179 0.195 A 359 347 2 0 0 0 [[56, 340]] 1.0 9x2v Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1I09B P49841 37 382 420.0 No_ligand No_ligand Inactive DFGin 6.861 14.025 BLAminus -135.93, 178.35 61.75, 84.0 -100.67, 24.72 288.55, 74.93 -64.65, -15.56 in-in in 8.483 Saltbr-in 2.711 HRD-in -62.69, -41.62 66.11, 9.61 in-in-out SNCiio in-out ActLoopNT-in 2.953 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.33, -45.22 APE9-dihe-na -71.78, 167.71 APE8-dihe-in -94.58, 171.33 APE8-rot-out 74.32 APE67-dihe-in -65.52, -17.17 -44.16, -80.97 APE12-dist-in 12.764 APE11-dist-in 11.113 APE10-dist-in 6.221 APE9-dist-in 3.37 None None None XRAY 2.7 0.242 0.274 B 420 341 5 0 0 0 [[56, 340]] 1.0 1i09 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6HK7A P49841 36 382 420.0 G8N:403 Type1 Inactive DFGin 7.181 13.926 BLAminus -137.45, -171.56 51.7, 92.53 -104.06, 22.16 271.05, 85.97 -65.5, -26.28 in-in in 8.435 Saltbr-in 2.767 HRD-in -53.21, -66.83 89.97, 19.54 in-in-out SNCiio in-out ActLoopNT-in 2.957 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -85.73, 172.92 APE9-dihe-na 79.4, 146.18 APE8-dihe-in -92.07, 85.52 APE8-rot-in 243.21 APE67-dihe-out 35.1, -40.06 22.07, -158.21 APE12-dist-in 13.29 APE11-dist-in 11.446 APE10-dist-in 6.781 APE9-dist-in 3.32 None PTR216 PTR216 XRAY 3.2 0.204 0.286 A 347 347 0 0 0 0 [[56, 340]] 1.0 6hk7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7SXHA P49841 37 383 420.0 D1E:501 Type1 Inactive DFGin 6.65 13.944 BLAminus -139.68, -175.41 60.2, 74.18 -88.43, 22.79 288.62, 86.11 -74.83, -15.81 in-in in 8.167 Saltbr-in 2.858 HRD-in -67.33, -47.27 70.7, 6.58 in-in-out SNCiio in-out ActLoopNT-in 2.863 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -126.8, 168.99 APE9-dihe-na 70.82, 157.42 APE8-dihe-in -70.74, 147.57 APE8-rot-out 190.63 APE67-dihe-in -58.92, -21.73 -57.82, -47.78 APE12-dist-in 13.771 APE11-dist-in 11.975 APE10-dist-in 7.371 APE9-dist-in 3.432 None PTR216 PTR216 XRAY 2.09 0.216 0.255 A 347 341 6 0 0 0 [[56, 340]] 1.0 7sxh Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3F7ZA P49841 35 383 420.0 34O:63000 Type1 Inactive DFGin 7.116 13.818 BLAminus -134.47, 172.11 69.02, 81.68 -97.3, 19.46 284.39, 70.02 -68.92, -10.86 in-in in 8.485 Saltbr-in 2.575 HRD-in -62.81, -48.18 67.57, 12.21 in-in-out SNCiio in-out ActLoopNT-in 2.95 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -139.18, 179.1 APE9-dihe-na 69.89, 157.17 APE8-dihe-in -75.28, 142.37 APE8-rot-out 185.5 APE67-dihe-in -55.86, -28.19 -45.56, -57.07 APE12-dist-in 13.5 APE11-dist-in 12.029 APE10-dist-in 6.815 APE9-dist-in 3.314 None PTR216 PTR216 XRAY 2.4 0.206 0.253 A 350 339 10 0 0 0 [[56, 340]] 1.0 3f7z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3SD0A P49841 35 384 420.0 TSK:400 Type1 Inactive DFGin 6.893 13.678 BLAminus -139.29, -172.59 62.67, 82.92 -94.93, 18.52 283.9, 73.87 -68.11, -17.74 in-in in 8.419 Saltbr-in 2.824 HRD-in -68.02, -47.17 76.6, 11.56 in-in-out SNCiio in-out ActLoopNT-in 2.8 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -82.28, 176.65 APE9-dihe-na 71.42, 130.7 APE8-dihe-in -100.53, 166.25 APE8-rot-out 29.1 APE67-dihe-inflip 91.12, -25.82 -31.67, 128.67 APE12-dist-in 12.91 APE11-dist-in 10.81 APE10-dist-in 5.779 APE9-dist-in 3.042 None None None XRAY 2.7 0.179 0.254 A 350 350 0 0 0 0 [[56, 340]] 1.0 3sd0 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3ZDIA P49841 36 384 420.0 UGJ:61386 Type1 Inactive DFGin 7.09 14.011 BLAminus -139.08, 169.73 59.85, 93.36 -102.57, 31.03 284.51, 75.61 -74.44, -6.01 in-in in 8.719 Saltbr-in 2.774 HRD-in -66.47, -49.36 70.61, -12.05 in-in-out SNCiio in-out ActLoopNT-in 2.874 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.6, -176.4 APE9-dihe-na 57.27, -141.25 APE8-dihe-in -136.89, 135.85 APE8-rot-out 188.96 APE67-dihe-in -60.18, -28.67 -48.24, -43.31 APE12-dist-in 13.777 APE11-dist-in 12.116 APE10-dist-in 7.549 APE9-dist-in 3.094 None PTR216 PTR216 XRAY 2.645 0.204 0.242 A 350 349 0 0 0 0 [[56, 340]] 1.0 3zdi Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4B7TA P49841 35 384 420.0 CWT:1385 Type1 Inactive DFGin 6.733 14.135 BLAminus -139.29, -173.55 55.51, 80.28 -97.98, 26.2 284.11, 78.64 -70.02, -22.23 in-in in 8.826 Saltbr-in 2.732 HRD-in -65.66, -45.08 68.98, -4.07 in-in-out SNCiio in-out ActLoopNT-in 3.022 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -80.96, 174.72 APE9-dihe-na 79.02, 153.66 APE8-dihe-in -90.72, 141.08 APE8-rot-out 219.61 APE67-dihe-inflip 82.28, -25.01 -65.77, 158.92 APE12-dist-in 13.15 APE11-dist-in 11.315 APE10-dist-in 6.552 APE9-dist-in 3.122 None None None XRAY 2.772 0.197 0.235 A 350 350 0 0 0 0 [[56, 340]] 1.0 4b7t Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6HK3A P49841 35 384 420.0 G8B:401 Type1 Inactive DFGin 6.919 13.749 BLAminus -140.26, -177.42 53.43, 89.98 -101.44, 26.95 281.28, 77.81 -71.94, -4.92 in-in in 8.265 Saltbr-in 2.52 HRD-in -65.54, -43.12 59.71, 15.8 in-in-out SNCiio in-out ActLoopNT-in 2.931 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -120.05, -174.23 APE9-dihe-na 65.54, 142.28 APE8-dihe-in -62.37, 137.73 APE8-rot-out 183.0 APE67-dihe-in -57.53, -32.37 -39.19, -57.21 APE12-dist-in 13.389 APE11-dist-in 11.762 APE10-dist-in 6.421 APE9-dist-in 3.218 None PTR216 PTR216 XRAY 2.35 0.206 0.234 A 350 350 0 0 0 0 [[56, 340]] 1.0 6hk3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6Y9RA P49841 35 384 420.0 OH8:401 Type1 Inactive DFGin 7.213 13.956 BLAminus -128.7, 177.14 64.74, 83.75 -99.31, 22.7 285.39, 75.74 -67.18, -22.12 in-in in 8.387 Saltbr-in 2.76 HRD-in -68.2, -47.94 70.12, 17.05 in-in-out SNCiio in-out ActLoopNT-in 2.97 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -147.41, 164.13 APE9-dihe-na 71.55, 162.91 APE8-dihe-in -81.0, 136.61 APE8-rot-out 173.09 APE67-dihe-in -62.95, -25.51 -45.24, -50.14 APE12-dist-in 13.684 APE11-dist-in 12.039 APE10-dist-in 7.353 APE9-dist-in 3.295 None PTR216 PTR216 XRAY 2.08 0.191 0.226 A 350 350 0 0 0 0 [[56, 340]] 1.0 6y9r Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1O9UA P49841 35 384 420.0 ADZ:1386 Type1 Inactive DFGin 6.69 14.409 BLAminus -135.58, -170.77 57.68, 80.28 -97.17, 18.56 286.56, 73.24 -63.89, -4.57 in-in in 8.918 Saltbr-in 3.252 HRD-in -60.54, -48.22 66.04, 11.65 in-in-out SNCiio in-out ActLoopNT-in 2.965 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.51, 167.48 APE9-dihe-na 74.14, -178.83 APE8-dihe-in -103.59, 140.85 APE8-rot-out 179.41 APE67-dihe-in -52.99, -22.64 -16.1, -87.79 APE12-dist-in 13.762 APE11-dist-in 11.706 APE10-dist-in 7.362 APE9-dist-in 2.862 None PTR216 PTR216 XRAY 2.4 0.233 0.26 A 350 350 0 0 0 0 [[56, 340]] 1.0 1o9u Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-69 240.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9PE9A P49841 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.072 14.229 BLAminus -128.7, -179.96 59.31, 84.1 -97.11, 26.91 283.64, 74.63 -73.69, -18.15 in-in in 8.351 Saltbr-in 2.725 HRD-in -68.62, -45.57 65.7, 16.55 in-in-out SNCiio in-out ActLoopNT-in 2.925 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.94, 165.33 APE9-dihe-na 76.34, 152.28 APE8-dihe-in -69.82, 130.62 APE8-rot-out 176.66 APE67-dihe-in -58.68, -26.71 -39.69, -56.4 APE12-dist-in 13.28 APE11-dist-in 11.758 APE10-dist-in 7.093 APE9-dist-in 3.155 None PTR216 PTR216 XRAY 2.11 0.221 0.247 A 359 332 13 0 0 0 [[56, 340]] 1.0 9pe9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9PE9B P49841 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.058 14.218 BLAminus -128.76, -179.81 59.6, 84.42 -97.78, 27.09 283.79, 74.38 -73.25, -17.71 in-in in 8.353 Saltbr-in 2.713 HRD-in -68.49, -44.82 64.55, 18.32 in-in-out SNCiio in-out ActLoopNT-in 2.94 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.27, 163.74 APE9-dihe-na 77.64, 152.05 APE8-dihe-in -69.14, 130.82 APE8-rot-out 177.12 APE67-dihe-in -58.92, -26.81 -39.96, -55.88 APE12-dist-in 13.36 APE11-dist-in 11.824 APE10-dist-in 7.161 APE9-dist-in 3.172 None PTR216 PTR216 XRAY 2.11 0.221 0.247 B 359 332 13 0 0 0 [[56, 340]] 1.0 9pe9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7Z1FA P49841 28 383 420.0 3NG:60401 Type1 Inactive DFGin 7.172 14.387 BLAminus -140.61, -172.17 56.83, 67.31 -90.44, 24.59 283.96, 78.9 -70.58, -34.2 in-in in 8.589 Saltbr-in 2.706 HRD-in -70.71, -48.08 68.23, 20.67 in-in-out SNCiio in-out ActLoopNT-in 2.877 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -121.77, -56.1 APE9-dihe-na -73.95, 173.6 APE8-dihe-in -71.54, 133.95 APE8-rot-out 205.24 APE67-dihe-in -54.78, -22.55 -52.86, -47.6 APE12-dist-in 13.711 APE11-dist-in 11.921 APE10-dist-in 7.257 APE9-dist-in 3.478 None PTR216 PTR216 XRAY 3.0 0.224 0.249 A 364 354 2 0 0 0 [[56, 340]] 1.0 7z1f Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 7Z1FB P49841 38 382 420.0 3NG:60401 Type1 Inactive DFGin 6.87 14.469 BLAminus -141.12, -171.82 52.8, 73.11 -90.49, 20.89 285.47, 81.84 -62.59, -35.1 in-in in 9.025 Saltbr-in 2.763 HRD-in -68.41, -52.97 70.54, 14.05 in-in-out SNCiio in-out ActLoopNT-in 3.039 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.34, -53.99 APE9-dihe-na -75.88, 165.71 APE8-dihe-in -64.92, 136.76 APE8-rot-out 179.7 APE67-dihe-in -58.44, -19.64 -54.95, -47.33 APE12-dist-in 13.527 APE11-dist-in 11.859 APE10-dist-in 7.154 APE9-dist-in 3.558 None PTR216 PTR216 XRAY 3.0 0.224 0.249 B 364 321 24 0 0 0 [[56, 340]] 1.0 7z1f Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8AV1A P49841 27 381 420.0 O9L:406 Type1 Inactive DFGin 7.005 13.802 BLAminus -134.83, 176.12 61.29, 85.31 -97.92, 27.58 284.57, 74.39 -70.18, -20.31 in-in in 8.42 Saltbr-in 2.659 HRD-in -72.82, -53.06 75.09, 11.93 in-in-out SNCiio in-out ActLoopNT-in 2.811 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -162.3, 153.55 APE9-dihe-na 79.71, 140.85 APE8-dihe-in -55.94, 133.71 APE8-rot-out 187.25 APE67-dihe-in -61.14, -25.49 -46.06, -52.45 APE12-dist-in 13.268 APE11-dist-in 11.413 APE10-dist-in 6.884 APE9-dist-in 3.061 None PTR216 PTR216 XRAY 2.15 0.18 0.21 A 365 351 4 0 0 0 [[56, 340]] 1.0 8av1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8AV1B P49841 27 381 420.0 O9L:405 Type1 Inactive DFGin 7.041 13.818 BLAminus -134.53, 176.17 61.15, 83.84 -96.42, 28.03 285.62, 75.68 -72.4, -19.61 in-in in 8.351 Saltbr-in 2.648 HRD-in -70.84, -52.05 73.58, 16.86 in-in-out SNCiio in-out ActLoopNT-in 2.809 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.36, 152.7 APE9-dihe-na 82.35, 142.4 APE8-dihe-in -57.42, 133.83 APE8-rot-out 184.71 APE67-dihe-in -59.68, -24.96 -48.86, -51.78 APE12-dist-in 13.26 APE11-dist-in 11.441 APE10-dist-in 6.85 APE9-dist-in 3.06 None PTR216 PTR216 XRAY 2.15 0.18 0.21 B 365 351 4 0 0 0 [[56, 340]] 1.0 8av1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6GN1A P49841 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.94 14.335 BLAminus -135.29, 179.1 59.47, 89.49 -98.73, 29.98 286.18, 72.49 -75.74, -10.8 in-in in 8.608 Saltbr-in 3.04 HRD-in -74.24, -44.22 64.59, 22.98 in-in-out SNCiio in-out ActLoopNT-in 2.94 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -143.03, -18.16 APE9-dihe-na -103.04, 175.18 APE8-dihe-in -67.81, 136.03 APE8-rot-out 187.31 APE67-dihe-in -61.67, -27.65 -44.51, -52.79 APE12-dist-out 14.01 APE11-dist-in 12.355 APE10-dist-in 7.387 APE9-dist-in 3.587 None PTR216 PTR216 XRAY 2.6 0.224 0.259 A 368 340 8 0 0 0 [[56, 340]] 1.0 6gn1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6GN1B P49841 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.944 14.317 BLAminus -135.3, 179.27 59.56, 89.49 -98.78, 30.1 286.37, 73.15 -75.82, -10.91 in-in in 8.622 Saltbr-in 3.034 HRD-in -74.17, -44.23 64.47, 22.86 in-in-out SNCiio in-out ActLoopNT-in 2.946 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -129.39, -14.9 APE9-dihe-na -108.68, -179.33 APE8-dihe-in -68.02, 134.54 APE8-rot-out 210.75 APE67-dihe-in -62.25, -27.68 -44.3, -51.95 APE12-dist-out 14.024 APE11-dist-in 12.183 APE10-dist-in 7.403 APE9-dist-in 3.7 None PTR216 PTR216 XRAY 2.6 0.224 0.259 B 368 340 8 0 0 0 [[56, 340]] 1.0 6gn1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 2O5KA P49841 35 384 420.0 HBM:0 Type1 Inactive DFGin 6.721 13.939 BLAminus -127.34, -179.9 54.97, 85.31 -97.88, 27.22 279.56, 72.26 -63.78, -54.26 in-in in 8.352 Saltbr-in 3.376 HRD-in -66.17, -47.55 59.21, 39.45 in-in-out SNCiio in-out ActLoopNT-in 2.946 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_iiii APE10-dihe-na 170.93, -156.16 APE9-dihe-na 30.47, -152.36 APE8-dihe-out -134.5, -176.14 APE8-rot-in 306.82 APE67-dihe-in -73.05, -7.32 -59.58, -80.34 APE12-dist-in 12.679 APE11-dist-in 9.181 APE10-dist-in 5.885 APE9-dist-in 3.037 None None None XRAY 3.2 0.251 0.309 A 372 350 0 0 0 0 [[56, 340]] 1.0 2o5k Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 1UV5A P49841 35 383 420.0 BRW:1383 Type1 Inactive DFGin 6.902 14.079 BLAminus -144.35, -177.14 59.35, 81.04 -94.26, 27.94 286.0, 72.94 -59.18, -36.48 in-in in 8.299 Saltbr-in 2.561 HRD-in -65.61, -42.55 70.5, 0.98 in-in-out SNCiio in-out ActLoopNT-in 2.884 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -98.47, 172.31 APE9-dihe-na 85.56, 133.89 APE8-dihe-in -66.16, 126.55 APE8-rot-out 191.14 APE67-dihe-in -61.71, -20.34 -21.78, -65.88 APE12-dist-in 12.763 APE11-dist-in 10.989 APE10-dist-in 5.715 APE9-dist-in 3.236 None None None XRAY 2.8 0.193 0.226 A 350 349 0 0 0 0 [[56, 340]] 1.0 1uv5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 7.4e-70 241.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6GJOA P49841 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.176 14.254 BLAminus -136.61, 169.82 63.4, 86.22 -103.46, 25.41 276.6, 83.48 -69.91, -39.25 in-in in 8.636 Saltbr-in 2.81 HRD-in -57.84, -41.83 58.98, 16.97 in-in-out SNCiio in-out ActLoopNT-in 3.012 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.92, 162.15 APE9-dihe-na 71.93, 161.47 APE8-dihe-in -78.01, 132.19 APE8-rot-out 37.25 APE67-dihe-in -62.57, -18.8 -29.28, -56.31 APE12-dist-in 13.62 APE11-dist-in 11.862 APE10-dist-in 6.945 APE9-dist-in 3.445 None None None XRAY 2.91 0.218 0.237 A 414 349 0 0 0 0 [[56, 340]] 1.0 6gjo Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 6GJOB P49841 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.478 14.251 BLAminus -136.82, 170.18 63.9, 83.46 -101.86, 22.92 278.62, 83.32 -68.81, -38.47 in-in in 8.405 Saltbr-in 3.084 HRD-in -57.78, -41.9 58.99, 17.22 in-in-out SNCiio in-out ActLoopNT-in 3.012 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.67, 163.61 APE9-dihe-na 73.76, 161.78 APE8-dihe-in -77.57, 137.96 APE8-rot-out 184.23 APE67-dihe-in -62.17, -20.4 -36.29, -55.68 APE12-dist-in 13.45 APE11-dist-in 11.784 APE10-dist-in 6.854 APE9-dist-in 3.437 None None None XRAY 2.91 0.218 0.237 B 414 343 6 0 0 0 [[56, 340]] 1.0 6gjo Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 3M1SA P49841 35 385 420.0 DW1:421 Type1 Inactive DFGin 7.021 13.71 BLAminus -149.21, -179.05 55.83, 87.87 -101.26, 23.04 292.92, 65.81 -62.39, -0.11 in-in in 8.726 Saltbr-in 2.976 HRD-in -71.98, -44.05 63.65, 18.92 in-in-out SNCiio in-out ActLoopNT-in 3.032 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -100.39, 171.9 APE9-dihe-na 82.48, 144.37 APE8-dihe-in -94.3, 96.58 APE8-rot-in 285.71 APE67-dihe-out 116.42, -45.78 9.38, 103.41 APE12-dist-in 13.649 APE11-dist-in 11.709 APE10-dist-in 6.707 APE9-dist-in 3.445 None None None XRAY 3.134 0.171 0.228 A 420 348 3 0 0 0 [[56, 340]] 1.0 3m1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 9HUKA P49841 25 385 420.0 A1IXL:501 Type1 Inactive DFGin 7.053 14.078 BLAminus -135.25, -177.02 57.0, 94.14 -110.6, 20.82 285.12, 72.82 -66.1, -13.46 in-out in 8.11 Saltbr-out 3.659 HRD-in -70.91, -39.46 63.28, 18.66 out-in-in SNCoii in-in ActLoopNT-in 3.157 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 179.26 APE9-dihe-na 68.03, 135.17 APE8-dihe-in -69.47, 168.34 APE8-rot-in 295.64 APE67-dihe-inflip 67.51, -44.25 -66.67, 175.58 APE12-dist-in 13.119 APE11-dist-in 10.946 APE10-dist-in 5.924 APE9-dist-in 3.202 None None None XRAY 3.5 0.219 0.25 A 442 361 0 0 0 0 [[56, 340]] 1.0 9huk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4J71A P49841 36 383 420.0 1JX:501 Type1 Inactive DFGin 6.929 14.034 BLAminus -134.37, 178.91 60.63, 80.22 -96.96, 24.92 284.72, 75.18 -68.29, -15.66 in-in in 8.448 Saltbr-in 3.096 HRD-in -74.9, -47.0 72.06, 4.98 in-in-out SNCiio in-out ActLoopNT-in 2.714 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.32, 163.35 APE9-dihe-na 76.45, 151.25 APE8-dihe-in -65.19, 140.55 APE8-rot-out 188.84 APE67-dihe-in -55.99, -28.06 -50.85, -54.43 APE12-dist-in 13.396 APE11-dist-in 11.896 APE10-dist-in 7.163 APE9-dist-in 2.998 None PTR216 PTR216 XRAY 2.31 0.191 0.234 A 424 348 0 0 0 0 [[56, 340]] 1.0 4j71 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4J71B P49841 36 383 420.0 1JX:501 Type1 Inactive DFGin 7.043 13.832 BLAminus -140.62, 179.7 59.87, 90.62 -104.73, 25.33 288.76, 76.25 -66.71, -17.33 in-in in 8.331 Saltbr-in 2.896 HRD-in -77.92, -46.29 72.36, 3.7 in-in-out SNCiio in-out ActLoopNT-in 2.834 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.74, 169.96 APE9-dihe-na 69.52, 149.79 APE8-dihe-in -68.04, 134.18 APE8-rot-out 173.06 APE67-dihe-in -53.62, -29.43 -43.81, -55.09 APE12-dist-in 13.213 APE11-dist-in 11.957 APE10-dist-in 7.127 APE9-dist-in 2.974 None PTR216 PTR216 XRAY 2.31 0.191 0.234 B 424 348 0 0 0 0 [[56, 340]] 1.0 4j71 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5HLNB P49841 37 383 420.0 65C:501 Type1 Inactive DFGin 6.848 13.332 BLAminus -143.06, -174.61 53.09, 90.34 -103.45, 33.01 288.97, 83.64 -74.69, -34.84 in-in in 8.996 Saltbr-in 2.604 HRD-in -68.15, -40.04 65.1, 19.28 in-in-out SNCiio in-out ActLoopNT-in 2.963 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -137.65, -62.86 APE9-dihe-na -78.36, 171.11 APE8-dihe-in -56.52, 151.93 APE8-rot-out 161.85 APE67-dihe-in -56.43, -28.42 -72.24, -45.62 APE12-dist-in 13.598 APE11-dist-in 11.834 APE10-dist-in 7.374 APE9-dist-in 3.416 None PTR216 PTR216 XRAY 3.1 0.173 0.236 B 424 347 0 0 0 0 [[56, 340]] 1.0 5hln Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 5OY4B P49841 30 384 420.0 B4K:502 Type1.5_Back Inactive DFGin 7.008 13.741 BLAminus -131.51, 177.88 58.43, 85.84 -94.85, 21.53 281.4, 81.96 -63.5, -26.63 in-in in 7.965 Saltbr-in 2.751 HRD-in -68.43, -44.24 63.59, 14.9 in-in-out SNCiio in-out ActLoopNT-in 2.869 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -145.82, 158.71 APE9-dihe-na 86.22, 156.23 APE8-dihe-in -75.92, 122.37 APE8-rot-out 226.12 APE67-dihe-in -60.14, -24.48 -28.85, -54.97 APE12-dist-in 13.504 APE11-dist-in 11.621 APE10-dist-in 7.009 APE9-dist-in 3.404 None PTR216 PTR216 XRAY 3.2 0.196 0.229 B 420 354 1 0 0 0 [[56, 340]] 1.0 5oy4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 8QJIA P49841 36 381 420.0 VNG:401 Type1 Inactive DFGin 6.949 14.196 None -92.57, -90.5 -72.82, 155.73 -144.36, 17.02 276.05, 102.26 -73.85, -19.5 in-in in 8.384 Saltbr-in 2.694 HRD-in -65.27, -43.08 63.67, 22.78 in-in-out SNCiio in-out ActLoopNT-in 3.34 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -115.54, 179.17 APE9-dihe-na 65.4, 161.24 APE8-dihe-in -68.89, 150.02 APE8-rot-out 175.4 APE67-dihe-in -64.21, -18.12 -58.7, -47.99 APE12-dist-in 13.386 APE11-dist-in 12.002 APE10-dist-in 7.07 APE9-dist-in 3.447 None PTR216 PTR216 XRAY 3.02 0.253 0.289 A 364 340 6 0 0 0 [[56, 340]] 1.0 8qji Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_HUMAN 4DITA P49841 35 387 420.0 0KD:501 Type1 None DFGin 6.805 13.948 BLAminus -145.37, 179.76 65.92, 81.37 -105.97, 22.54 288.96, 82.14 -68.29, -17.95 in-in in 8.825 Saltbr-in 2.717 HRD-in -69.87, -50.6 73.87, 5.2 in-in-none SNCiin in-none ActLoopNT-in 2.939 ActLoopCT-none nonTYR APEdihe_aannn APEdist_iinn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 14.5 999.0, 999.0 APE12-dist-in 13.489 APE11-dist-in 10.385 APE10-dist-none 999.0 APE9-dist-none 999.0 None PTR216 PTR216 XRAY 2.6 0.243 0.304 A 382 329 24 0 0 4 [[56, 340]] 1.0 4dit Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.4e-70 243.3 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 8VMFA Q9WV60 27 383 420.0 ADP:60504 ATPlike Active DFGin 6.612 14.1 BLAminus -148.4, -167.57 58.53, 66.72 -90.57, 24.21 287.49, 78.37 -75.04, -7.89 in-in in 8.66 Saltbr-in 2.678 HRD-in -67.34, -47.3 70.6, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.84 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.01, -20.74 APE9-dihe-na -93.16, -168.14 APE8-dihe-in -112.8, 164.36 APE8-rot-in 304.6 APE67-dihe-inflip 78.98, -8.38 -56.8, 140.56 APE12-dist-in 13.183 APE11-dist-in 10.949 APE10-dist-in 6.514 APE9-dist-in 3.308 None None None XRAY 2.5 0.21 0.251 A 364 354 0 0 0 0 [[56, 340]] 1.0 8vmf Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 8VMGA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 7.0 13.999 BLAminus -139.67, -176.86 60.44, 73.06 -89.27, 27.07 283.1, 81.19 -73.23, -12.63 in-in in 8.478 Saltbr-in 2.688 HRD-in -67.64, -48.38 72.75, 3.36 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.26, 164.63 APE9-dihe-na 72.45, 142.8 APE8-dihe-in -66.41, 146.08 APE8-rot-in 307.07 APE67-dihe-in -64.3, -22.81 -57.43, -46.54 APE12-dist-in 13.278 APE11-dist-in 11.627 APE10-dist-in 6.941 APE9-dist-in 2.984 None None None XRAY 2.45 0.195 0.23 A 364 358 0 0 0 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 8VMEA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 6.469 13.844 BLAminus -131.0, -171.33 63.41, 73.0 -92.56, 22.88 289.27, 83.61 -79.03, -1.02 in-in in 8.753 Saltbr-in 2.78 HRD-in -67.9, -47.67 70.4, 7.52 in-in-in SNCiii in-in ActLoopNT-in 2.731 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.18, 168.01 APE9-dihe-na 68.83, 161.19 APE8-dihe-in -90.7, 152.54 APE8-rot-in 290.93 APE67-dihe-inflip 82.32, -22.26 -51.38, 150.9 APE12-dist-in 13.288 APE11-dist-in 12.071 APE10-dist-in 6.934 APE9-dist-in 3.292 None None None XRAY 2.3 0.183 0.23 A 365 355 0 0 0 0 [[56, 340]] 1.0 8vme Mus musculus CMGC_GSK3B_MOUSE CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 4NU1A Q9WV60 6 383 420.0 ADP:405 ATPlike Active DFGin 6.109 13.677 BLAminus -140.27, -172.8 60.29, 88.19 -108.14, 24.39 289.57, 88.21 -68.01, -14.99 in-in in 8.691 Saltbr-in 2.793 HRD-in -66.76, -45.51 62.96, 19.85 in-in-in SNCiii in-in ActLoopNT-in 2.682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.38, 172.68 APE9-dihe-na 66.76, 153.81 APE8-dihe-in -82.08, 156.46 APE8-rot-in 299.93 APE67-dihe-inflip 76.53, -25.22 -54.39, 158.45 APE12-dist-in 13.51 APE11-dist-in 11.621 APE10-dist-in 7.126 APE9-dist-in 3.15 None SEP9 SEP9 XRAY 2.5 0.194 0.245 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nu1 Mus musculus CMGC_GSK3B_MOUSE CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3D Q9WV60 36 382 420.0 No_ligand No_ligand Active DFGin 6.846 14.395 BLAminus -141.83, -176.77 60.2, 77.49 -89.39, 22.71 281.69, 81.03 -67.16, -17.62 in-in in 8.597 Saltbr-in 2.92 HRD-in -66.38, -49.02 71.39, 7.08 in-in-in SNCiii in-in ActLoopNT-in 3.026 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.65, -50.64 APE9-dihe-na -86.99, 177.5 APE8-dihe-in -52.77, 135.95 APE8-rot-in 241.34 APE67-dihe-in -60.13, -26.01 -56.25, -47.64 APE12-dist-in 13.537 APE11-dist-in 11.767 APE10-dist-in 7.278 APE9-dist-in 3.256 None PTR216 PTR216 XRAY 2.14 0.192 0.226 D 420 333 13 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 5AIRB Q9WV60 22 384 420.0 No_ligand No_ligand Active DFGin 7.213 14.683 BLAminus -135.77, 173.37 62.69, 75.87 -94.37, 22.65 282.98, 71.43 -62.58, -24.12 in-in in 8.743 Saltbr-in 3.194 HRD-in -72.7, -48.08 74.63, 8.38 in-in-in SNCiii in-in ActLoopNT-in 3.078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.78, -34.05 APE9-dihe-na -91.23, 159.66 APE8-dihe-in -80.14, 164.39 APE8-rot-in 286.43 APE67-dihe-in -76.71, -12.41 -69.97, -37.36 APE12-dist-in 12.725 APE11-dist-in 10.771 APE10-dist-in 5.798 APE9-dist-in 3.28 None None None XRAY 2.53 0.215 0.26 B 430 361 2 0 0 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 5AIRA Q9WV60 26 383 420.0 No_ligand No_ligand Inactive DFGin 6.987 14.337 ABAminus -142.69, -19.87 -113.16, 97.17 -94.15, 12.11 276.77, 85.56 -67.43, -12.28 in-in in 8.78 Saltbr-in 2.843 HRD-in -76.77, -43.42 72.44, 6.11 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.55, -31.48 APE9-dihe-na -99.45, 158.56 APE8-dihe-in -79.74, 161.48 APE8-rot-in 283.68 APE67-dihe-in -67.71, -13.15 -61.56, -52.85 APE12-dist-in 12.745 APE11-dist-in 10.563 APE10-dist-in 5.802 APE9-dist-in 3.216 None None None XRAY 2.53 0.215 0.26 A 430 353 2 0 0 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 8VMGB Q9WV60 35 383 420.0 No_ligand No_ligand Inactive DFGin 7.035 14.105 BLAminus -148.77, -175.26 61.58, 69.86 -88.49, 24.73 286.58, 81.46 -68.41, -21.39 in-in in 8.506 Saltbr-in 2.822 HRD-in -64.17, -52.24 74.94, 4.57 in-in-out SNCiio in-out ActLoopNT-in 2.751 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -148.65, 168.87 APE9-dihe-na 71.82, 140.54 APE8-dihe-in -63.28, 148.93 APE8-rot-out 168.42 APE67-dihe-in -62.52, -22.04 -64.28, -46.93 APE12-dist-in 13.497 APE11-dist-in 11.807 APE10-dist-in 7.007 APE9-dist-in 3.01 None None None XRAY 2.45 0.195 0.23 B 364 349 0 0 0 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3C Q9WV60 37 383 420.0 No_ligand No_ligand Inactive DFGin 7.085 14.246 BLAminus -138.84, 177.7 70.47, 68.34 -81.63, 23.64 278.71, 79.84 -68.29, -26.67 in-in in 8.543 Saltbr-in 3.1 HRD-in -63.75, -49.26 68.09, 4.78 in-in-out SNCiio in-out ActLoopNT-in 2.931 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.25, -51.04 APE9-dihe-na -75.73, 169.64 APE8-dihe-in -64.7, 134.47 APE8-rot-out 205.91 APE67-dihe-in -59.9, -28.79 -47.43, -50.42 APE12-dist-in 13.357 APE11-dist-in 11.82 APE10-dist-in 6.617 APE9-dist-in 3.416 None PTR216 PTR216 XRAY 2.14 0.192 0.226 C 420 332 14 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3A Q9WV60 36 387 420.0 MRI:501 Type1 Inactive DFGin 6.894 14.102 BLAminus -136.0, 177.47 66.33, 76.64 -88.44, 20.33 285.85, 84.43 -66.44, -23.98 in-in in 8.877 Saltbr-in 2.954 HRD-in -71.52, -49.56 71.35, 12.25 in-in-out SNCiio in-out ActLoopNT-in 3.032 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.99, -47.87 APE9-dihe-na -84.23, -172.24 APE8-dihe-in -75.59, 135.74 APE8-rot-out 167.98 APE67-dihe-in -65.02, -21.79 -52.52, -47.78 APE12-dist-in 13.692 APE11-dist-in 12.024 APE10-dist-in 7.314 APE9-dist-in 3.334 None PTR216 PTR216 XRAY 2.14 0.192 0.226 A 420 348 4 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3B Q9WV60 36 384 420.0 MRI:501 Type1 Inactive DFGin 6.739 14.09 BLAminus -133.31, 179.77 64.96, 75.18 -85.96, 22.4 281.26, 80.21 -65.67, -27.09 in-in in 8.98 Saltbr-in 3.019 HRD-in -70.11, -50.99 71.74, 15.55 in-in-out SNCiio in-out ActLoopNT-in 2.922 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.24, -38.47 APE9-dihe-na -87.03, 178.23 APE8-dihe-in -68.15, 134.76 APE8-rot-out 177.54 APE67-dihe-in -64.59, -23.54 -47.57, -47.97 APE12-dist-in 13.626 APE11-dist-in 11.908 APE10-dist-in 6.694 APE9-dist-in 3.414 None PTR216 PTR216 XRAY 2.14 0.192 0.226 B 420 344 5 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
A0A125YY75_TOXGG 9HVXA A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.812 13.739 BLAminus -151.79, -170.99 58.28, 71.83 -90.67, 23.31 282.96, 81.43 -68.24, -23.58 in-in in 7.973 Saltbr-in 2.67 HRD-in -79.27, -44.62 69.75, 6.05 in-in-out SNCiio in-out ActLoopNT-in 2.916 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -133.04, -39.68 APE9-dihe-na -85.38, 168.26 APE8-dihe-in -65.75, 139.05 APE8-rot-out 179.82 APE67-dihe-in -62.31, -27.06 -57.82, -44.69 APE12-dist-in 13.505 APE11-dist-in 11.868 APE10-dist-in 7.371 APE9-dist-in 3.499 None PTR211 PTR211 XRAY 2.1 0.203 0.25 A 350 323 16 0 0 0 [[47, 344]] 1.0 9hvx Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 6.4e-71 244.9 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6A A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.554 13.514 BLAminus -159.29, -172.81 63.26, 75.9 -98.23, 18.12 289.64, 83.03 -60.9, -17.5 in-in in 8.248 Saltbr-in 2.913 HRD-in -74.22, -42.3 70.91, -2.75 in-in-out SNCiio in-out ActLoopNT-in 2.779 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -107.29, 145.01 APE9-dihe-na -102.07, 19.34 APE8-dihe-in -80.82, 138.15 APE8-rot-out 53.99 APE67-dihe-in -80.29, -18.75 -104.8, -54.34 APE12-dist-none 999.0 APE11-dist-in 10.111 APE10-dist-in 7.183 APE9-dist-out 8.805 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 A 373 332 7 0 0 3 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6B A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.969 13.759 BLAminus -158.71, -175.52 61.04, 75.48 -97.8, 20.68 289.3, 83.48 -61.51, -18.44 in-in in 8.34 Saltbr-in 2.533 HRD-in -73.25, -38.58 70.21, -4.6 in-in-out SNCiio in-out ActLoopNT-in 2.957 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnio APE10-dihe-na 999.0, 137.93 APE9-dihe-na -128.88, -94.97 APE8-dihe-out 8.76, 102.73 APE8-rot-out 52.93 APE67-dihe-in -72.89, -15.66 -99.47, -15.26 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 6.673 APE9-dist-out 7.874 None PTR211 PTR211 XRAY 2.9 0.207 0.26 B 373 332 7 0 0 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6D A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.752 13.545 BLAminus -157.98, -176.25 63.15, 72.4 -94.88, 18.71 288.21, 86.06 -60.77, -17.66 in-in in 8.448 Saltbr-in 3.001 HRD-in -74.85, -41.94 71.3, -1.92 in-in-out SNCiio in-out ActLoopNT-in 2.853 ActLoopCT-out nonTYR APEdihe_aaooo APEdist_nnio APE10-dihe-na 999.0, -28.71 APE9-dihe-na 70.23, 60.42 APE8-dihe-out -136.17, -56.82 APE8-rot-out 132.32 APE67-dihe-out -77.45, -28.23 69.46, -39.41 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 7.077 APE9-dist-out 8.582 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 D 373 327 12 0 0 9 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6F A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.98 13.82 BLAminus -156.62, -174.56 59.51, 71.39 -97.24, 16.48 288.27, 84.06 -60.16, -18.79 in-in in 8.206 Saltbr-in 2.735 HRD-in -76.38, -41.74 71.66, -4.7 in-in-out SNCiio in-out ActLoopNT-in 2.744 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -146.52, 154.45 APE9-dihe-na -92.11, 49.24 APE8-dihe-in -83.14, 134.37 APE8-rot-out 54.49 APE67-dihe-in -77.45, -15.85 -109.34, -69.31 APE12-dist-none 999.0 APE11-dist-in 9.936 APE10-dist-in 6.674 APE9-dist-out 9.042 None PTR211 PTR211 XRAY 2.9 0.207 0.26 F 373 325 14 0 0 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK

CMGC_GSK3B (Glycogen synthase kinase-3 beta)

Total number of chains: 16
Active chains: 6
Family: CMGC
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 15 93.8% 8VMEA
DFGin ABAminus 1 6.2% 5AIRA

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GSK3B_MOUSE 8VMFA Q9WV60 27 383 420.0 ADP:60504 ATPlike Active DFGin 6.612 14.1 BLAminus -148.4, -167.57 58.53, 66.72 -90.57, 24.21 287.49, 78.37 -75.04, -7.89 in-in in 8.66 Saltbr-in 2.678 HRD-in -67.34, -47.3 70.6, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.84 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.01, -20.74 APE9-dihe-na -93.16, -168.14 APE8-dihe-in -112.8, 164.36 APE8-rot-in 304.6 APE67-dihe-inflip 78.98, -8.38 -56.8, 140.56 APE12-dist-in 13.183 APE11-dist-in 10.949 APE10-dist-in 6.514 APE9-dist-in 3.308 None None None XRAY 2.5 0.21 0.251 A 364 354 0 0 0 0 [[56, 340]] 1.0 8vmf Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 8VMGA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 7.0 13.999 BLAminus -139.67, -176.86 60.44, 73.06 -89.27, 27.07 283.1, 81.19 -73.23, -12.63 in-in in 8.478 Saltbr-in 2.688 HRD-in -67.64, -48.38 72.75, 3.36 in-in-in SNCiii in-in ActLoopNT-in 2.844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.26, 164.63 APE9-dihe-na 72.45, 142.8 APE8-dihe-in -66.41, 146.08 APE8-rot-in 307.07 APE67-dihe-in -64.3, -22.81 -57.43, -46.54 APE12-dist-in 13.278 APE11-dist-in 11.627 APE10-dist-in 6.941 APE9-dist-in 2.984 None None None XRAY 2.45 0.195 0.23 A 364 358 0 0 0 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 8VMEA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 6.469 13.844 BLAminus -131.0, -171.33 63.41, 73.0 -92.56, 22.88 289.27, 83.61 -79.03, -1.02 in-in in 8.753 Saltbr-in 2.78 HRD-in -67.9, -47.67 70.4, 7.52 in-in-in SNCiii in-in ActLoopNT-in 2.731 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.18, 168.01 APE9-dihe-na 68.83, 161.19 APE8-dihe-in -90.7, 152.54 APE8-rot-in 290.93 APE67-dihe-inflip 82.32, -22.26 -51.38, 150.9 APE12-dist-in 13.288 APE11-dist-in 12.071 APE10-dist-in 6.934 APE9-dist-in 3.292 None None None XRAY 2.3 0.183 0.23 A 365 355 0 0 0 0 [[56, 340]] 1.0 8vme Mus musculus CMGC_GSK3B_MOUSE CMGC 2.1e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 4NU1A Q9WV60 6 383 420.0 ADP:405 ATPlike Active DFGin 6.109 13.677 BLAminus -140.27, -172.8 60.29, 88.19 -108.14, 24.39 289.57, 88.21 -68.01, -14.99 in-in in 8.691 Saltbr-in 2.793 HRD-in -66.76, -45.51 62.96, 19.85 in-in-in SNCiii in-in ActLoopNT-in 2.682 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.38, 172.68 APE9-dihe-na 66.76, 153.81 APE8-dihe-in -82.08, 156.46 APE8-rot-in 299.93 APE67-dihe-inflip 76.53, -25.22 -54.39, 158.45 APE12-dist-in 13.51 APE11-dist-in 11.621 APE10-dist-in 7.126 APE9-dist-in 3.15 None SEP9 SEP9 XRAY 2.5 0.194 0.245 A 389 357 2 0 0 0 [[56, 340]] 1.0 4nu1 Mus musculus CMGC_GSK3B_MOUSE CMGC 2.5e-70 243.2 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3D Q9WV60 36 382 420.0 No_ligand No_ligand Active DFGin 6.846 14.395 BLAminus -141.83, -176.77 60.2, 77.49 -89.39, 22.71 281.69, 81.03 -67.16, -17.62 in-in in 8.597 Saltbr-in 2.92 HRD-in -66.38, -49.02 71.39, 7.08 in-in-in SNCiii in-in ActLoopNT-in 3.026 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.65, -50.64 APE9-dihe-na -86.99, 177.5 APE8-dihe-in -52.77, 135.95 APE8-rot-in 241.34 APE67-dihe-in -60.13, -26.01 -56.25, -47.64 APE12-dist-in 13.537 APE11-dist-in 11.767 APE10-dist-in 7.278 APE9-dist-in 3.256 None PTR216 PTR216 XRAY 2.14 0.192 0.226 D 420 333 13 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 5AIRB Q9WV60 22 384 420.0 No_ligand No_ligand Active DFGin 7.213 14.683 BLAminus -135.77, 173.37 62.69, 75.87 -94.37, 22.65 282.98, 71.43 -62.58, -24.12 in-in in 8.743 Saltbr-in 3.194 HRD-in -72.7, -48.08 74.63, 8.38 in-in-in SNCiii in-in ActLoopNT-in 3.078 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.78, -34.05 APE9-dihe-na -91.23, 159.66 APE8-dihe-in -80.14, 164.39 APE8-rot-in 286.43 APE67-dihe-in -76.71, -12.41 -69.97, -37.36 APE12-dist-in 12.725 APE11-dist-in 10.771 APE10-dist-in 5.798 APE9-dist-in 3.28 None None None XRAY 2.53 0.215 0.26 B 430 361 2 0 0 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 5AIRA Q9WV60 26 383 420.0 No_ligand No_ligand Inactive DFGin 6.987 14.337 ABAminus -142.69, -19.87 -113.16, 97.17 -94.15, 12.11 276.77, 85.56 -67.43, -12.28 in-in in 8.78 Saltbr-in 2.843 HRD-in -76.77, -43.42 72.44, 6.11 in-in-in SNCiii in-in ActLoopNT-in 2.92 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.55, -31.48 APE9-dihe-na -99.45, 158.56 APE8-dihe-in -79.74, 161.48 APE8-rot-in 283.68 APE67-dihe-in -67.71, -13.15 -61.56, -52.85 APE12-dist-in 12.745 APE11-dist-in 10.563 APE10-dist-in 5.802 APE9-dist-in 3.216 None None None XRAY 2.53 0.215 0.26 A 430 353 2 0 0 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 8VMGB Q9WV60 35 383 420.0 No_ligand No_ligand Inactive DFGin 7.035 14.105 BLAminus -148.77, -175.26 61.58, 69.86 -88.49, 24.73 286.58, 81.46 -68.41, -21.39 in-in in 8.506 Saltbr-in 2.822 HRD-in -64.17, -52.24 74.94, 4.57 in-in-out SNCiio in-out ActLoopNT-in 2.751 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -148.65, 168.87 APE9-dihe-na 71.82, 140.54 APE8-dihe-in -63.28, 148.93 APE8-rot-out 168.42 APE67-dihe-in -62.52, -22.04 -64.28, -46.93 APE12-dist-in 13.497 APE11-dist-in 11.807 APE10-dist-in 7.007 APE9-dist-in 3.01 None None None XRAY 2.45 0.195 0.23 B 364 349 0 0 0 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3C Q9WV60 37 383 420.0 No_ligand No_ligand Inactive DFGin 7.085 14.246 BLAminus -138.84, 177.7 70.47, 68.34 -81.63, 23.64 278.71, 79.84 -68.29, -26.67 in-in in 8.543 Saltbr-in 3.1 HRD-in -63.75, -49.26 68.09, 4.78 in-in-out SNCiio in-out ActLoopNT-in 2.931 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.25, -51.04 APE9-dihe-na -75.73, 169.64 APE8-dihe-in -64.7, 134.47 APE8-rot-out 205.91 APE67-dihe-in -59.9, -28.79 -47.43, -50.42 APE12-dist-in 13.357 APE11-dist-in 11.82 APE10-dist-in 6.617 APE9-dist-in 3.416 None PTR216 PTR216 XRAY 2.14 0.192 0.226 C 420 332 14 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3A Q9WV60 36 387 420.0 MRI:501 Type1 Inactive DFGin 6.894 14.102 BLAminus -136.0, 177.47 66.33, 76.64 -88.44, 20.33 285.85, 84.43 -66.44, -23.98 in-in in 8.877 Saltbr-in 2.954 HRD-in -71.52, -49.56 71.35, 12.25 in-in-out SNCiio in-out ActLoopNT-in 3.032 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.99, -47.87 APE9-dihe-na -84.23, -172.24 APE8-dihe-in -75.59, 135.74 APE8-rot-out 167.98 APE67-dihe-in -65.02, -21.79 -52.52, -47.78 APE12-dist-in 13.692 APE11-dist-in 12.024 APE10-dist-in 7.314 APE9-dist-in 3.334 None PTR216 PTR216 XRAY 2.14 0.192 0.226 A 420 348 4 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B_MOUSE 6AE3B Q9WV60 36 384 420.0 MRI:501 Type1 Inactive DFGin 6.739 14.09 BLAminus -133.31, 179.77 64.96, 75.18 -85.96, 22.4 281.26, 80.21 -65.67, -27.09 in-in in 8.98 Saltbr-in 3.019 HRD-in -70.11, -50.99 71.74, 15.55 in-in-out SNCiio in-out ActLoopNT-in 2.922 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.24, -38.47 APE9-dihe-na -87.03, 178.23 APE8-dihe-in -68.15, 134.76 APE8-rot-out 177.54 APE67-dihe-in -64.59, -23.54 -47.57, -47.97 APE12-dist-in 13.626 APE11-dist-in 11.908 APE10-dist-in 6.694 APE9-dist-in 3.414 None PTR216 PTR216 XRAY 2.14 0.192 0.226 B 420 344 5 0 0 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1 301 301 199 200 201 203 205 85 97 101 178 180 179 181 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
A0A125YY75_TOXGG 9HVXA A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.812 13.739 BLAminus -151.79, -170.99 58.28, 71.83 -90.67, 23.31 282.96, 81.43 -68.24, -23.58 in-in in 7.973 Saltbr-in 2.67 HRD-in -79.27, -44.62 69.75, 6.05 in-in-out SNCiio in-out ActLoopNT-in 2.916 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -133.04, -39.68 APE9-dihe-na -85.38, 168.26 APE8-dihe-in -65.75, 139.05 APE8-rot-out 179.82 APE67-dihe-in -62.31, -27.06 -57.82, -44.69 APE12-dist-in 13.505 APE11-dist-in 11.868 APE10-dist-in 7.371 APE9-dist-in 3.499 None PTR211 PTR211 XRAY 2.1 0.203 0.25 A 350 323 16 0 0 0 [[47, 344]] 1.0 9hvx Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 6.4e-71 244.9 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6A A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.554 13.514 BLAminus -159.29, -172.81 63.26, 75.9 -98.23, 18.12 289.64, 83.03 -60.9, -17.5 in-in in 8.248 Saltbr-in 2.913 HRD-in -74.22, -42.3 70.91, -2.75 in-in-out SNCiio in-out ActLoopNT-in 2.779 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -107.29, 145.01 APE9-dihe-na -102.07, 19.34 APE8-dihe-in -80.82, 138.15 APE8-rot-out 53.99 APE67-dihe-in -80.29, -18.75 -104.8, -54.34 APE12-dist-none 999.0 APE11-dist-in 10.111 APE10-dist-in 7.183 APE9-dist-out 8.805 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 A 373 332 7 0 0 3 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6B A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.969 13.759 BLAminus -158.71, -175.52 61.04, 75.48 -97.8, 20.68 289.3, 83.48 -61.51, -18.44 in-in in 8.34 Saltbr-in 2.533 HRD-in -73.25, -38.58 70.21, -4.6 in-in-out SNCiio in-out ActLoopNT-in 2.957 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnio APE10-dihe-na 999.0, 137.93 APE9-dihe-na -128.88, -94.97 APE8-dihe-out 8.76, 102.73 APE8-rot-out 52.93 APE67-dihe-in -72.89, -15.66 -99.47, -15.26 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 6.673 APE9-dist-out 7.874 None PTR211 PTR211 XRAY 2.9 0.207 0.26 B 373 332 7 0 0 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6D A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.752 13.545 BLAminus -157.98, -176.25 63.15, 72.4 -94.88, 18.71 288.21, 86.06 -60.77, -17.66 in-in in 8.448 Saltbr-in 3.001 HRD-in -74.85, -41.94 71.3, -1.92 in-in-out SNCiio in-out ActLoopNT-in 2.853 ActLoopCT-out nonTYR APEdihe_aaooo APEdist_nnio APE10-dihe-na 999.0, -28.71 APE9-dihe-na 70.23, 60.42 APE8-dihe-out -136.17, -56.82 APE8-rot-out 132.32 APE67-dihe-out -77.45, -28.23 69.46, -39.41 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 7.077 APE9-dist-out 8.582 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 D 373 327 12 0 0 9 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
A0A125YY75_TOXGG 9HW6F A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.98 13.82 BLAminus -156.62, -174.56 59.51, 71.39 -97.24, 16.48 288.27, 84.06 -60.16, -18.79 in-in in 8.206 Saltbr-in 2.735 HRD-in -76.38, -41.74 71.66, -4.7 in-in-out SNCiio in-out ActLoopNT-in 2.744 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -146.52, 154.45 APE9-dihe-na -92.11, 49.24 APE8-dihe-in -83.14, 134.37 APE8-rot-out 54.49 APE67-dihe-in -77.45, -15.85 -109.34, -69.31 APE12-dist-none 999.0 APE11-dist-in 9.936 APE10-dist-in 6.674 APE9-dist-out 9.042 None PTR211 PTR211 XRAY 2.9 0.207 0.26 F 373 325 14 0 0 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1 301 301 194 195 196 198 200 76 88 92 173 175 174 176 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK