CMGC_GSK3B (Glycogen synthase kinase-3 beta)

Total number of chains: 177
Active chains: 143
Uniprot: GSK3B_HUMAN
Kinase Domain Residues: 56 - 340
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 174 98.3% AF-P49841-K1A
DFGin ABAminus 2 1.1% 6Y9SA
DFGin None 1 0.6% 8QJIA

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GSK3B 4NM5A P49841 24 383 420.0 ADP:60401 ATPlike Active DFGin 6.5502 14.0064 BLAminus -136.16, -177.73 61.88, 88.47 -108.64, 28.76 287.87, 80.78 -73.66, -15.44 in-in in 8.6187 Saltbr-in 2.6732 HRD-in -65.83, -43.73 64.82, 15.23 in-in-in SNCiii in-in ActLoopNT-in 2.8386 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.92, 173.97 APE9-dihe-na 66.26, 147.02 APE8-dihe-in -77.1, 152.8 APE8-rot-in 293.28 APE67-dihe-inflip 82.03, -25.76 -52.23, 150.7 APE12-dist-in 13.2793 APE11-dist-in 11.5989 APE10-dist-in 6.9485 APE9-dist-in 3.2377 None None None XRAY 2.3 0.185 0.232 A 377.0 360.0 0 27 27 0 [[56, 340]] 1.0 4nm5 CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4NM7A P49841 25 383 420.0 ADP:60401 ATPlike Active DFGin 6.5153 13.993 BLAminus -137.35, -178.06 62.82, 88.6 -107.3, 24.56 288.41, 80.2 -69.84, -12.63 in-in in 8.8181 Saltbr-in 2.743 HRD-in -66.5, -46.64 67.84, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.8287 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 172.54 APE9-dihe-na 68.99, 153.43 APE8-dihe-in -86.9, 151.79 APE8-rot-in 300.04 APE67-dihe-inflip 84.67, -25.93 -50.38, 146.2 APE12-dist-in 13.3553 APE11-dist-in 11.6779 APE10-dist-in 6.9055 APE9-dist-in 3.2102 None None None XRAY 2.3 0.185 0.234 A 377.0 354.0 2 27 27 0 [[56, 340]] 1.0 4nm7 CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4NM3A P49841 6 383 420.0 ADP:60409 ATPlike Active DFGin 6.4747 13.947 BLAminus -129.98, -178.05 63.17, 87.87 -103.96, 21.26 289.38, 80.04 -65.46, -16.35 in-in in 8.8058 Saltbr-in 2.7256 HRD-in -69.81, -46.77 71.59, 6.75 in-in-in SNCiii in-in ActLoopNT-in 2.7503 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.34, 169.99 APE9-dihe-na 69.15, 146.37 APE8-dihe-in -83.47, 151.55 APE8-rot-in 296.54 APE67-dihe-inflip 86.0, -31.11 -49.79, 146.79 APE12-dist-in 13.2688 APE11-dist-in 11.4837 APE10-dist-in 6.9065 APE9-dist-in 3.1117 None SEP9 SEP9 XRAY 2.1 0.197 0.242 A 389.0 357.0 2 27 27 0 [[56, 340]] 1.0 4nm3 CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1J1BA P49841 35 388 420.0 ANP:60430 ATPlike Active DFGin 6.7667 13.7876 BLAminus -136.8, -178.88 61.6, 83.12 -97.64, 25.1 286.09, 80.4 -68.7, -13.11 in-in in 8.5659 Saltbr-in 2.59 HRD-in -71.16, -45.98 70.36, 3.88 in-in-in SNCiii in-in ActLoopNT-in 3.0085 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.52, 175.26 APE9-dihe-na 75.44, 133.64 APE8-dihe-in -75.76, 147.49 APE8-rot-in 306.57 APE67-dihe-inflip 98.15, -33.72 -56.43, 141.52 APE12-dist-in 13.0562 APE11-dist-in 10.9736 APE10-dist-in 5.8926 APE9-dist-in 3.1122 None None None XRAY 1.8 0.216 0.242 A 420.0 354.0 0 27 27 0 [[56, 340]] 1.0 1j1b CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1J1BB P49841 23 386 420.0 ANP:60930 ATPlike Active DFGin 6.6091 13.6686 BLAminus -136.4, -177.03 61.49, 81.88 -98.08, 27.2 288.49, 82.07 -71.33, -13.14 in-in in 8.4573 Saltbr-in 2.713 HRD-in -67.51, -45.87 68.87, 6.43 in-in-in SNCiii in-in ActLoopNT-in 2.9624 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.88, 174.17 APE9-dihe-na 76.18, 138.08 APE8-dihe-in -76.12, 141.41 APE8-rot-in 301.11 APE67-dihe-inflip 98.0, -37.59 -54.78, 144.25 APE12-dist-in 12.9784 APE11-dist-in 11.0659 APE10-dist-in 6.0113 APE9-dist-in 3.1744 None None None XRAY 1.8 0.216 0.242 B 420.0 364.0 0 27 27 0 [[56, 340]] 1.0 1j1b CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1J1CA P49841 35 388 420.0 ADP:60430 ATPlike Active DFGin 6.8122 13.9298 BLAminus -139.24, -179.75 62.79, 82.17 -97.34, 25.19 286.68, 82.3 -65.83, -19.9 in-in in 8.6015 Saltbr-in 2.6465 HRD-in -68.65, -43.85 68.34, 7.36 in-in-in SNCiii in-in ActLoopNT-in 2.9774 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.05, 172.96 APE9-dihe-na 78.17, 130.85 APE8-dihe-in -73.54, 145.97 APE8-rot-in 310.16 APE67-dihe-inflip 99.09, -35.01 -54.43, 141.28 APE12-dist-in 13.0771 APE11-dist-in 11.0674 APE10-dist-in 5.9263 APE9-dist-in 3.1997 None None None XRAY 2.1 0.218 0.242 A 420.0 354.0 0 27 27 0 [[56, 340]] 1.0 1j1c CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1J1CB P49841 23 386 420.0 ADP:60930 ATPlike Active DFGin 6.6935 13.7094 BLAminus -138.27, -179.99 63.33, 82.68 -100.46, 28.2 289.88, 80.26 -70.45, -13.94 in-in in 8.52 Saltbr-in 2.738 HRD-in -67.92, -43.36 67.59, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.9803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.71, 170.27 APE9-dihe-na 78.71, 139.86 APE8-dihe-in -81.56, 140.05 APE8-rot-in 302.5 APE67-dihe-inflip 101.62, -36.53 -50.52, 137.44 APE12-dist-in 12.8683 APE11-dist-in 11.1277 APE10-dist-in 6.0252 APE9-dist-in 3.2076 None None None XRAY 2.1 0.218 0.242 B 420.0 364.0 0 27 27 0 [[56, 340]] 1.0 1j1c CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8XN6A P49841 35 384 420.0 ANP:501 ATPlike Active DFGin 6.682 13.8624 BLAminus -137.72, 173.39 67.73, 84.48 -99.84, 22.57 287.77, 80.54 -65.33, -24.58 in-in in 8.4632 Saltbr-in 2.6302 HRD-in -71.05, -47.88 67.82, 15.5 in-in-in SNCiii in-in ActLoopNT-in 3.0543 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.0, 164.43 APE9-dihe-na 85.44, 135.36 APE8-dihe-in -74.2, 151.55 APE8-rot-in 291.81 APE67-dihe-in -69.28, -17.83 -36.59, -67.98 APE12-dist-in 12.9066 APE11-dist-in 10.7867 APE10-dist-in 5.6801 APE9-dist-in 3.1824 None None None XRAY 2.4 0.194 0.242 A 421.0 350.0 0 27 27 0 [[56, 340]] 1.0 8xn6 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1PYXA P49841 35 386 420.0 ANP:1001 ATPlike Active DFGin 6.5838 13.6216 BLAminus -138.81, -178.07 65.18, 79.92 -98.83, 26.07 289.95, 78.27 -73.24, -7.6 in-in in 8.3727 Saltbr-in 2.7648 HRD-in -67.79, -47.84 71.28, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.9483 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.12, 170.17 APE9-dihe-na 80.64, 129.74 APE8-dihe-in -63.79, 140.05 APE8-rot-in 299.48 APE67-dihe-in -56.43, -21.61 -20.65, -80.28 APE12-dist-in 12.9032 APE11-dist-in 10.9366 APE10-dist-in 5.7841 APE9-dist-in 3.1495 None None None XRAY 2.4 0.206 0.233 A 422.0 343.0 9 27 27 0 [[56, 340]] 1.0 1pyx CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1PYXB P49841 35 383 420.0 ANP:2001 ATPlike Active DFGin 6.5927 13.7178 BLAminus -140.94, -178.47 65.26, 79.98 -98.11, 22.32 290.75, 76.51 -68.32, -7.73 in-in in 8.4877 Saltbr-in 2.6657 HRD-in -69.98, -47.18 70.83, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.9383 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.3, 169.41 APE9-dihe-na 81.27, 131.24 APE8-dihe-in -66.67, 140.79 APE8-rot-in 300.74 APE67-dihe-in -56.9, -22.2 -20.58, -79.9 APE12-dist-in 12.8382 APE11-dist-in 10.8615 APE10-dist-in 5.7183 APE9-dist-in 3.132 None None None XRAY 2.4 0.206 0.233 B 422.0 338.0 11 27 27 0 [[56, 340]] 1.0 1pyx CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B AF-P49841-K1A P49841 48 348 420.0 No_ligand No_ligand Active DFGin 6.7843 14.0695 BLAminus -132.22, 178.4 62.95, 68.76 -81.18, 15.79 285.47, 79.99 -60.59, -34.48 in-in in 8.4747 Saltbr-in 2.7102 HRD-in -72.93, -43.95 66.08, 11.33 in-in-in SNCiii in-in ActLoopNT-in 2.8921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.31, 173.16 APE9-dihe-na 65.7, 144.93 APE8-dihe-in -63.41, 136.54 APE8-rot-in 298.96 APE67-dihe-in -66.32, -15.33 -50.7, -49.59 APE12-dist-in 13.4502 APE11-dist-in 11.9889 APE10-dist-in 6.9958 APE9-dist-in 3.1274 None None None AF2 -1.0 1.0 1.0 A 301.0 301.0 0 27 27 0 [[56, 340]] 1.0 AF-P49841-K1 CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B AF-P49841-K3A P49841 48 348 420.0 No_ligand No_ligand Active DFGin 6.5244 13.8836 BLAminus -137.65, -179.24 64.43, 60.31 -74.11, 11.79 288.76, 87.67 -59.53, -33.87 in-in in 8.2321 Saltbr-in 2.6752 HRD-in -76.11, -42.33 64.92, 19.4 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, -179.86 APE9-dihe-na 61.35, 145.02 APE8-dihe-in -62.21, 135.58 APE8-rot-in 295.17 APE67-dihe-in -63.79, -15.52 -52.47, -50.54 APE12-dist-in 13.4857 APE11-dist-in 11.9949 APE10-dist-in 7.0698 APE9-dist-in 3.244 None None None AF2 -1.0 1.0 1.0 A 301.0 301.0 0 27 27 0 [[56, 340]] 1.0 AF-P49841-K3 CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1GNGA P49841 36 385 420.0 No_ligand No_ligand Active DFGin 6.8854 14.0642 BLAminus -143.26, -176.0 52.72, 77.37 -90.17, 24.13 284.09, 64.37 -57.11, -28.67 in-in in 7.9042 Saltbr-in 2.9159 HRD-in -73.29, -39.28 60.06, 11.92 in-in-in SNCiii in-in ActLoopNT-in 2.8439 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.61, 159.4 APE9-dihe-na 81.31, 139.52 APE8-dihe-in -59.26, 125.44 APE8-rot-in 312.57 APE67-dihe-in -52.62, -25.58 -28.83, -64.47 APE12-dist-in 13.5503 APE11-dist-in 11.9569 APE10-dist-in 7.016 APE9-dist-in 3.1105 None PTR216 PTR216 XRAY 2.6 0.196 0.262 A 378.0 350.0 0 27 27 0 [[56, 340]] 1.0 1gng CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1GNGB P49841 28 384 420.0 No_ligand No_ligand Active DFGin 7.075 14.1431 BLAminus -137.26, -174.12 57.41, 76.0 -92.3, 24.73 292.83, 74.1 -62.54, -16.26 in-in in 8.1028 Saltbr-in 2.801 HRD-in -56.65, -46.78 67.13, 3.53 in-in-in SNCiii in-in ActLoopNT-in 3.0528 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.46, 162.71 APE9-dihe-na 73.79, 160.3 APE8-dihe-in -71.09, 143.31 APE8-rot-in 306.45 APE67-dihe-in -62.51, -22.51 -44.24, -51.03 APE12-dist-in 13.4613 APE11-dist-in 11.7372 APE10-dist-in 7.2333 APE9-dist-in 3.2921 None PTR216 PTR216 XRAY 2.6 0.196 0.262 B 378.0 357.0 0 27 27 0 [[56, 340]] 1.0 1gng CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1H8FA P49841 35 386 420.0 No_ligand No_ligand Active DFGin 7.0053 14.4673 BLAminus -132.29, -174.92 54.46, 76.42 -91.57, 20.83 287.85, 73.58 -61.47, -17.91 in-in in 8.8115 Saltbr-in 2.6295 HRD-in -65.88, -45.02 68.7, 5.89 in-in-in SNCiii in-in ActLoopNT-in 3.0299 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.85, 172.29 APE9-dihe-na 81.77, 142.51 APE8-dihe-in -88.0, 149.96 APE8-rot-in 300.12 APE67-dihe-in -68.04, -14.11 -16.17, -79.65 APE12-dist-in 12.8766 APE11-dist-in 10.8744 APE10-dist-in 5.7937 APE9-dist-in 3.0888 None None None XRAY 2.8 0.22 0.256 A 352.0 352.0 0 27 27 0 [[56, 340]] 1.0 1h8f CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1H8FB P49841 35 384 420.0 No_ligand No_ligand Active DFGin 7.053 14.4881 BLAminus -137.11, -175.26 54.49, 79.79 -96.15, 19.99 284.33, 74.24 -61.84, -16.45 in-in in 8.7842 Saltbr-in 2.6311 HRD-in -65.99, -45.44 68.05, 7.58 in-in-in SNCiii in-in ActLoopNT-in 2.9921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.76, 172.7 APE9-dihe-na 81.11, 140.51 APE8-dihe-in -87.0, 149.5 APE8-rot-in 302.15 APE67-dihe-in -67.01, -11.3 -16.16, -82.04 APE12-dist-in 12.8754 APE11-dist-in 10.8434 APE10-dist-in 5.7606 APE9-dist-in 3.101 None None None XRAY 2.8 0.22 0.256 B 352.0 350.0 0 27 27 0 [[56, 340]] 1.0 1h8f CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1I09A P49841 25 384 420.0 No_ligand No_ligand Active DFGin 6.9144 14.1487 BLAminus -130.79, -175.77 55.31, 78.24 -94.52, 21.05 292.59, 69.56 -64.23, -6.99 in-in in 8.5205 Saltbr-in 2.7631 HRD-in -66.04, -49.2 76.06, -6.11 in-in-in SNCiii in-in ActLoopNT-in 3.0217 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.67, -13.88 APE9-dihe-na -95.25, 153.25 APE8-dihe-in -66.11, 146.74 APE8-rot-in 277.64 APE67-dihe-in -57.92, -5.44 -43.43, -74.88 APE12-dist-in 12.9676 APE11-dist-in 11.1602 APE10-dist-in 5.9721 APE9-dist-in 3.3336 None None None XRAY 2.7 0.242 0.274 A 420.0 338.0 22 27 27 0 [[56, 340]] 1.0 1i09 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U2ZA P49841 35 382 420.0 L7C:401 Type1 Active DFGin 7.0437 14.3283 BLAminus -133.1, 179.76 62.32, 79.84 -96.99, 23.84 285.42, 79.62 -65.82, -25.41 in-in in 8.5578 Saltbr-in 2.7638 HRD-in -73.49, -48.13 70.69, 16.81 in-in-in SNCiii in-in ActLoopNT-in 2.9072 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.38, 169.05 APE9-dihe-na 81.0, 139.13 APE8-dihe-in -79.34, 150.41 APE8-rot-in 288.38 APE67-dihe-inflip 98.4, -32.71 -58.44, 134.12 APE12-dist-in 13.1383 APE11-dist-in 11.05 APE10-dist-in 5.8885 APE9-dist-in 3.0925 None None None XRAY 2.21 0.248 0.266 A 348.0 345.0 3 27 27 0 [[56, 340]] 1.0 7u2z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U2ZB P49841 35 382 420.0 L7C:401 Type1 Active DFGin 7.0832 14.3162 BLAminus -133.0, 179.81 61.72, 80.12 -97.27, 23.94 285.32, 79.23 -65.78, -25.41 in-in in 8.5159 Saltbr-in 2.7654 HRD-in -73.41, -48.27 70.6, 17.33 in-in-in SNCiii in-in ActLoopNT-in 2.9123 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.19, 168.84 APE9-dihe-na 80.53, 139.96 APE8-dihe-in -79.72, 154.04 APE8-rot-in 288.98 APE67-dihe-in -82.66, -15.29 -42.95, -55.79 APE12-dist-in 13.132 APE11-dist-in 11.0815 APE10-dist-in 5.8924 APE9-dist-in 3.0994 None None None XRAY 2.21 0.248 0.266 B 348.0 348.0 0 27 27 0 [[56, 340]] 1.0 7u2z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3F7ZB P49841 35 383 420.0 34O:63000 Type1 Active DFGin 7.0223 13.8784 BLAminus -136.68, -179.55 57.9, 84.9 -98.68, 23.48 283.23, 74.81 -68.95, -21.14 in-in in 8.4241 Saltbr-in 2.704 HRD-in -69.78, -45.02 65.34, 14.6 in-in-in SNCiii in-in ActLoopNT-in 2.8686 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.88, 179.92 APE9-dihe-na 68.48, 153.11 APE8-dihe-in -69.08, 139.27 APE8-rot-in 289.99 APE67-dihe-in -60.9, -22.52 -35.36, -58.5 APE12-dist-in 13.6463 APE11-dist-in 11.9538 APE10-dist-in 6.7778 APE9-dist-in 3.2477 None PTR216 PTR216 XRAY 2.4 0.206 0.253 B 350.0 339.0 10 27 27 0 [[56, 340]] 1.0 3f7z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3SD0B P49841 35 383 420.0 TSK:400 Type1 Active DFGin 7.1882 14.0242 BLAminus -142.24, -171.3 46.91, 83.25 -91.85, 32.36 285.89, 73.19 -82.63, -8.9 in-in in 8.2345 Saltbr-in 2.887 HRD-in -76.13, -44.58 70.79, 3.58 in-in-in SNCiii in-in ActLoopNT-in 2.8942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.6, 179.93 APE9-dihe-na 74.21, 152.1 APE8-dihe-in -107.68, 155.88 APE8-rot-in 296.61 APE67-dihe-in -78.55, -3.01 -13.04, -81.61 APE12-dist-in 13.0175 APE11-dist-in 11.0989 APE10-dist-in 6.1509 APE9-dist-in 3.1559 None None None XRAY 2.7 0.179 0.254 B 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 3sd0 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6HK3B P49841 35 384 420.0 G8B:401 Type1 Active DFGin 6.7879 13.6408 BLAminus -137.2, -177.06 49.94, 95.88 -103.42, 19.32 279.02, 79.18 -69.5, -12.66 in-in in 8.1675 Saltbr-in 2.6023 HRD-in -82.47, -44.32 66.17, 21.49 in-in-in SNCiii in-in ActLoopNT-in 2.8186 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.65, -179.5 APE9-dihe-na 72.73, 150.58 APE8-dihe-in -63.57, 140.77 APE8-rot-in 271.9 APE67-dihe-in -55.77, -29.98 -51.2, -52.31 APE12-dist-in 13.4077 APE11-dist-in 11.6419 APE10-dist-in 6.3651 APE9-dist-in 3.2489 None PTR216 PTR216 XRAY 2.35 0.206 0.234 B 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6HK4A P49841 35 384 420.0 G8E:408 Type1 Active DFGin 6.9285 13.5081 BLAminus -141.9, -175.7 56.05, 83.18 -94.87, 22.99 284.64, 79.88 -61.73, -17.34 in-in in 8.3712 Saltbr-in 2.6563 HRD-in -76.65, -40.11 61.36, 16.95 in-in-in SNCiii in-in ActLoopNT-in 2.9232 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.26, 167.76 APE9-dihe-na 63.34, 157.04 APE8-dihe-in -69.05, 135.63 APE8-rot-in 300.42 APE67-dihe-in -54.24, -34.87 -29.95, -58.61 APE12-dist-in 13.2335 APE11-dist-in 11.745 APE10-dist-in 7.1618 APE9-dist-in 3.1917 None PTR216 PTR216 XRAY 2.5 0.212 0.249 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk4 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6HK4B P49841 35 384 420.0 G8E:409 Type1 Active DFGin 6.9427 13.5412 BLAminus -140.37, -179.48 60.09, 87.67 -101.02, 22.8 284.5, 76.31 -75.88, -10.96 in-in in 8.2076 Saltbr-in 2.5056 HRD-in -82.4, -45.58 68.54, 13.94 in-in-in SNCiii in-in ActLoopNT-in 2.9046 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.02, 172.84 APE9-dihe-na 63.46, 139.74 APE8-dihe-in -57.57, 136.79 APE8-rot-in 295.89 APE67-dihe-in -60.79, -29.87 -46.27, -47.23 APE12-dist-in 13.2677 APE11-dist-in 11.6783 APE10-dist-in 6.8983 APE9-dist-in 3.0744 None PTR216 PTR216 XRAY 2.5 0.212 0.249 B 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk4 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5F94A P49841 36 381 420.0 3UO:401 Type1 Active DFGin 6.9408 13.7851 BLAminus -132.23, -171.99 59.12, 80.79 -95.82, 23.07 289.16, 72.98 -56.52, -34.28 in-in in 8.4861 Saltbr-in 2.7108 HRD-in -71.8, -46.49 68.5, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.7841 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.99, 174.92 APE9-dihe-na 77.27, 148.67 APE8-dihe-in -101.45, 151.47 APE8-rot-in 289.94 APE67-dihe-inflip 89.58, -29.34 -36.24, 131.42 APE12-dist-in 12.915 APE11-dist-in 10.9124 APE10-dist-in 5.9524 APE9-dist-in 3.1086 None None None XRAY 2.51 0.191 0.226 A 350.0 346.0 0 27 27 0 [[56, 340]] 1.0 5f94 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5F94B P49841 37 385 420.0 3UO:401 Type1 Active DFGin 6.9206 13.9028 BLAminus -131.5, -174.71 60.13, 82.54 -97.18, 23.01 287.88, 72.62 -56.23, -35.38 in-in in 8.3979 Saltbr-in 2.8901 HRD-in -70.35, -45.36 66.02, 7.89 in-in-in SNCiii in-in ActLoopNT-in 2.8563 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.68, 174.32 APE9-dihe-na 79.06, 151.27 APE8-dihe-in -105.02, 147.7 APE8-rot-in 292.84 APE67-dihe-inflip 87.17, -28.31 -40.05, 137.25 APE12-dist-in 12.8868 APE11-dist-in 10.9014 APE10-dist-in 5.8663 APE9-dist-in 3.1931 None None None XRAY 2.51 0.191 0.226 B 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 5f94 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5F95A P49841 36 383 420.0 3UP:401 Type1 Active DFGin 6.8507 14.1212 BLAminus -131.03, -172.49 54.11, 85.8 -99.54, 23.42 287.04, 73.17 -58.21, -30.13 in-in in 8.4923 Saltbr-in 2.6419 HRD-in -68.05, -46.73 71.39, 6.88 in-in-in SNCiii in-in ActLoopNT-in 2.8734 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.52, 167.77 APE9-dihe-na 81.86, 152.62 APE8-dihe-in -108.33, 161.23 APE8-rot-in 296.59 APE67-dihe-in -81.75, 2.56 -4.13, -93.98 APE12-dist-in 13.0998 APE11-dist-in 11.0871 APE10-dist-in 6.3777 APE9-dist-in 3.2624 None None None XRAY 2.525 0.204 0.242 A 350.0 345.0 3 27 27 0 [[56, 340]] 1.0 5f95 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5F95B P49841 36 385 420.0 3UP:401 Type1 Active DFGin 7.0295 14.1311 BLAminus -130.15, -170.55 52.93, 82.9 -96.95, 23.47 283.9, 71.07 -57.67, -29.42 in-in in 8.5241 Saltbr-in 2.2415 HRD-in -68.94, -45.23 69.65, 6.25 in-in-in SNCiii in-in ActLoopNT-in 3.0094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.14, 169.18 APE9-dihe-na 82.46, 143.88 APE8-dihe-in -96.17, 168.5 APE8-rot-in 296.7 APE67-dihe-in -78.34, 2.06 -36.18, -73.12 APE12-dist-in 13.0212 APE11-dist-in 11.0271 APE10-dist-in 6.0921 APE9-dist-in 3.2102 None None None XRAY 2.525 0.204 0.242 B 350.0 338.0 12 27 27 0 [[56, 340]] 1.0 5f95 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U31A P49841 36 385 420.0 L7I:402 Type1 Active DFGin 7.0942 14.1832 BLAminus -142.39, 178.42 62.99, 82.78 -98.0, 19.46 288.1, 81.67 -57.1, -32.73 in-in in 8.1645 Saltbr-in 2.8395 HRD-in -76.17, -49.99 76.15, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.9293 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.54, -23.16 APE9-dihe-na -100.68, 154.06 APE8-dihe-in -79.73, 162.4 APE8-rot-in 294.75 APE67-dihe-in -75.9, -12.27 -44.4, -68.17 APE12-dist-in 13.1024 APE11-dist-in 10.9281 APE10-dist-in 5.9089 APE9-dist-in 3.4164 None None None XRAY 2.38 0.244 0.276 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 7u31 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U31B P49841 37 382 420.0 L7I:402 Type1 Active DFGin 7.0487 14.2873 BLAminus -143.88, 177.54 62.09, 82.63 -98.02, 19.8 287.95, 82.15 -57.33, -32.15 in-in in 8.3774 Saltbr-in 2.7171 HRD-in -76.73, -50.12 75.35, 8.49 in-in-in SNCiii in-in ActLoopNT-in 2.9329 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.33, 167.82 APE9-dihe-na 83.33, 132.28 APE8-dihe-in -83.68, 163.51 APE8-rot-in 292.75 APE67-dihe-in -76.54, -11.97 -40.44, -69.75 APE12-dist-in 13.1082 APE11-dist-in 10.9788 APE10-dist-in 5.927 APE9-dist-in 3.1265 None None None XRAY 2.38 0.244 0.276 B 350.0 346.0 0 27 27 0 [[56, 340]] 1.0 7u31 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7SXJA P49841 34 383 420.0 6VL:60401 Type1 Active DFGin 6.916 14.335 BLAminus -142.41, -179.99 59.67, 72.96 -86.59, 25.21 285.68, 73.81 -69.07, -21.65 in-in in 8.2686 Saltbr-in 2.692 HRD-in -74.28, -41.7 68.05, 5.57 in-in-in SNCiii in-in ActLoopNT-in 2.943 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.32, 170.09 APE9-dihe-na 72.35, 148.74 APE8-dihe-in -71.51, 141.06 APE8-rot-in 303.21 APE67-dihe-in -59.11, -26.68 -51.44, -48.71 APE12-dist-in 13.5034 APE11-dist-in 11.843 APE10-dist-in 7.0416 APE9-dist-in 3.173 None PTR216 PTR216 XRAY 1.85 0.185 0.203 A 351.0 346.0 4 27 27 0 [[56, 340]] 1.0 7sxj CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7OY5A P49841 35 385 420.0 39I:401 Type1 Active DFGin 6.9265 14.0328 BLAminus -126.76, 175.34 72.52, 92.63 -110.59, 33.29 286.05, 82.06 -75.35, -28.56 in-in in 8.6875 Saltbr-in 2.9358 HRD-in -72.48, -55.14 81.29, 7.92 in-in-in SNCiii in-in ActLoopNT-in 2.9168 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.43, 173.86 APE9-dihe-na 80.53, 146.3 APE8-dihe-in -94.81, 142.24 APE8-rot-in 295.61 APE67-dihe-inflip 101.01, -30.19 -44.76, 139.01 APE12-dist-in 12.9243 APE11-dist-in 10.9605 APE10-dist-in 5.8925 APE9-dist-in 3.2763 None None None XRAY 2.57 0.221 0.26 A 351.0 343.0 8 27 27 0 [[56, 340]] 1.0 7oy5 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7OY5B P49841 35 383 420.0 39I:401 Type1 Active DFGin 7.1149 14.145 BLAminus -131.55, -176.92 63.09, 57.6 -70.26, 11.8 285.25, 87.17 -66.04, -15.46 in-in in 8.4954 Saltbr-in 3.0267 HRD-in -75.85, -49.73 71.52, 4.36 in-in-in SNCiii in-in ActLoopNT-in 3.0392 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.28, 172.83 APE9-dihe-na 79.24, 135.47 APE8-dihe-in -76.12, 154.7 APE8-rot-in 287.59 APE67-dihe-inflip 110.96, -34.61 -67.01, 135.0 APE12-dist-in 13.0301 APE11-dist-in 10.9583 APE10-dist-in 5.9922 APE9-dist-in 3.0083 None None None XRAY 2.57 0.221 0.26 B 351.0 344.0 5 27 27 0 [[56, 340]] 1.0 7oy5 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U33A P49841 36 385 420.0 L7R:402 Type1 Active DFGin 7.0231 14.0492 BLAminus -140.49, 178.19 60.8, 84.54 -99.85, 16.49 288.62, 77.82 -50.41, -27.99 in-in in 8.5115 Saltbr-in 2.7738 HRD-in -71.53, -50.0 75.9, 8.27 in-in-in SNCiii in-in ActLoopNT-in 2.9863 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.78, -39.59 APE9-dihe-na -85.32, 160.12 APE8-dihe-in -84.45, 147.1 APE8-rot-in 286.21 APE67-dihe-inflip 87.92, -34.06 -59.31, 147.18 APE12-dist-in 13.0363 APE11-dist-in 10.9912 APE10-dist-in 6.0319 APE9-dist-in 3.2624 None None None XRAY 2.6 0.233 0.264 A 351.0 350.0 0 27 27 0 [[56, 340]] 1.0 7u33 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U33B P49841 37 382 420.0 L7R:402 Type1 Active DFGin 6.9949 14.0924 BLAminus -141.31, 178.2 60.97, 83.82 -100.06, 16.34 288.93, 78.7 -51.51, -27.59 in-in in 8.5327 Saltbr-in 2.7534 HRD-in -72.1, -49.87 75.78, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.62, 168.53 APE9-dihe-na 77.45, 140.58 APE8-dihe-in -89.54, 146.71 APE8-rot-in 285.53 APE67-dihe-in -82.12, -10.74 -0.24, -85.34 APE12-dist-in 13.0347 APE11-dist-in 10.9604 APE10-dist-in 6.0286 APE9-dist-in 3.1028 None None None XRAY 2.6 0.233 0.264 B 351.0 346.0 0 27 27 0 [[56, 340]] 1.0 7u33 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U36A P49841 36 385 420.0 L7W:402 Type1 Active DFGin 7.0548 14.0575 BLAminus -140.39, -178.87 60.34, 89.59 -105.19, 18.12 284.52, 86.52 -57.6, -32.5 in-in in 8.4531 Saltbr-in 3.0188 HRD-in -77.18, -47.14 70.51, 17.98 in-in-in SNCiii in-in ActLoopNT-in 2.9592 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.43, -45.81 APE9-dihe-na -84.57, 153.41 APE8-dihe-in -68.83, 161.86 APE8-rot-in 280.03 APE67-dihe-in -82.26, -16.89 -53.14, -56.37 APE12-dist-in 12.8704 APE11-dist-in 10.7585 APE10-dist-in 5.8125 APE9-dist-in 3.1894 None None None XRAY 2.75 0.24 0.275 A 351.0 350.0 0 27 27 0 [[56, 340]] 1.0 7u36 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7U36B P49841 37 382 420.0 L7W:402 Type1 Active DFGin 7.0561 14.0712 BLAminus -141.26, -179.45 60.58, 88.51 -105.71, 18.11 283.81, 87.44 -57.54, -31.03 in-in in 8.4984 Saltbr-in 2.9906 HRD-in -77.32, -47.05 68.98, 19.83 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -102.55, 163.3 APE9-dihe-na 90.09, 132.18 APE8-dihe-in -72.41, 162.37 APE8-rot-in 279.62 APE67-dihe-in -81.75, -17.56 -53.5, -56.42 APE12-dist-in 12.8558 APE11-dist-in 10.7783 APE10-dist-in 5.7902 APE9-dist-in 3.107 None None None XRAY 2.75 0.24 0.275 B 351.0 346.0 0 27 27 0 [[56, 340]] 1.0 7u36 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 2OW3A P49841 35 385 420.0 BIM:387 Type1 Active DFGin 6.8544 14.0885 BLAminus -145.58, -177.16 62.63, 79.7 -96.04, 38.01 299.18, 104.83 -72.62, -36.62 in-in in 8.3402 Saltbr-in 2.8377 HRD-in -75.79, -46.9 63.78, 27.01 in-in-in SNCiii in-in ActLoopNT-in 2.8813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.84, 153.8 APE9-dihe-na 77.18, 154.82 APE8-dihe-in -72.33, 143.1 APE8-rot-in 299.46 APE67-dihe-in -64.33, -22.16 -49.08, -49.27 APE12-dist-in 13.7242 APE11-dist-in 12.3631 APE10-dist-in 7.5149 APE9-dist-in 3.7839 None PTR216 PTR216 XRAY 2.8 0.248 0.295 A 352.0 347.0 4 27 27 0 [[56, 340]] 1.0 2ow3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 2OW3B P49841 35 386 420.0 BIM:387 Type1 Active DFGin 6.7681 14.5197 BLAminus -140.91, -178.82 62.87, 80.36 -94.83, 34.08 291.22, 81.94 -79.34, -15.72 in-in in 8.4802 Saltbr-in 2.7885 HRD-in -91.97, -42.45 64.4, 21.24 in-in-in SNCiii in-in ActLoopNT-in 2.8773 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.27, 157.33 APE9-dihe-na 81.52, 163.87 APE8-dihe-in -81.91, 157.75 APE8-rot-in 308.08 APE67-dihe-in -65.81, -19.16 -55.34, -61.54 APE12-dist-in 13.9045 APE11-dist-in 12.5424 APE10-dist-in 7.6276 APE9-dist-in 3.5378 None PTR216 PTR216 XRAY 2.8 0.248 0.295 B 352.0 352.0 0 27 27 0 [[56, 340]] 1.0 2ow3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3GB2A P49841 35 383 420.0 G3B:999 Type1 Active DFGin 7.0809 13.5025 BLAminus -136.77, -176.86 57.81, 94.36 -109.09, 24.06 290.54, 74.85 -73.21, 4.88 in-in in 8.4499 Saltbr-in 2.8117 HRD-in -66.76, -55.55 72.33, 20.67 in-in-in SNCiii in-in ActLoopNT-in 2.8594 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.38, -175.57 APE9-dihe-na 67.46, 160.91 APE8-dihe-in -72.68, 139.68 APE8-rot-in 245.03 APE67-dihe-in -60.68, -25.16 -49.04, -51.42 APE12-dist-in 13.505 APE11-dist-in 11.9733 APE10-dist-in 7.0043 APE9-dist-in 3.2866 None PTR216 PTR216 XRAY 2.4 0.225 0.289 A 353.0 341.0 8 27 27 0 [[56, 340]] 1.0 3gb2 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6TCUA P49841 35 384 420.0 N1Q:401 Type1 Active DFGin 7.2707 14.1909 BLAminus -132.13, 178.03 59.16, 82.25 -93.13, 22.32 285.63, 78.52 -60.3, -31.7 in-in in 8.3524 Saltbr-in 2.9119 HRD-in -72.47, -46.38 65.88, 22.79 in-in-in SNCiii in-in ActLoopNT-in 2.8967 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.64, 162.18 APE9-dihe-na 73.42, 158.65 APE8-dihe-in -78.26, 138.24 APE8-rot-in 295.07 APE67-dihe-in -60.71, -25.87 -50.61, -49.17 APE12-dist-in 13.5559 APE11-dist-in 11.9425 APE10-dist-in 7.1969 APE9-dist-in 3.2398 None PTR216 PTR216 XRAY 2.14 0.204 0.24 A 355.0 350.0 0 27 27 0 [[56, 340]] 1.0 6tcu CMGC_GSK3B_HUMAN CMGC 1.9e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5T31A P49841 35 381 420.0 6VL:501 Type1 Active DFGin 7.0002 14.6002 BLAminus -146.5, -178.72 58.09, 85.8 -94.81, 34.39 283.96, 70.89 -72.9, -29.06 in-in in 8.1833 Saltbr-in 2.8228 HRD-in -85.27, -37.65 59.13, 22.16 in-in-in SNCiii in-in ActLoopNT-in 2.9632 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.45, 179.68 APE9-dihe-na 63.71, 158.01 APE8-dihe-in -85.57, 141.47 APE8-rot-in 304.73 APE67-dihe-in -68.11, -24.88 -45.34, -45.1 APE12-dist-in 13.218 APE11-dist-in 11.5452 APE10-dist-in 6.5643 APE9-dist-in 3.195 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 A 420.0 335.0 12 27 27 0 [[56, 340]] 1.0 5t31 CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5T31B P49841 36 382 420.0 6VL:501 Type1 Active DFGin 7.2086 14.6047 BLAminus -147.12, 178.9 61.54, 81.68 -96.09, 32.98 286.61, 73.16 -76.82, -18.6 in-in in 8.229 Saltbr-in 2.5809 HRD-in -64.89, -47.6 63.02, 19.09 in-in-in SNCiii in-in ActLoopNT-in 3.0176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.39, 179.54 APE9-dihe-na 63.77, 153.96 APE8-dihe-in -75.26, 136.0 APE8-rot-in 291.41 APE67-dihe-in -61.67, -31.85 -41.28, -53.13 APE12-dist-in 13.3814 APE11-dist-in 11.678 APE10-dist-in 6.473 APE9-dist-in 3.2366 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 B 420.0 334.0 13 27 27 0 [[56, 340]] 1.0 5t31 CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7Z1GA P49841 27 383 420.0 3NG:60401 Type1 Active DFGin 7.2716 14.699 BLAminus -137.45, -179.93 52.32, 81.51 -93.1, 20.22 282.75, 78.65 -65.74, -16.48 in-in in 8.9685 Saltbr-in 2.7705 HRD-in -67.62, -47.44 74.98, 2.45 in-in-in SNCiii in-in ActLoopNT-in 2.9264 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.67, 177.94 APE9-dihe-na 70.81, 142.84 APE8-dihe-in -95.23, 170.55 APE8-rot-in 305.08 APE67-dihe-inflip 72.5, -37.64 -53.01, 158.1 APE12-dist-in 12.7846 APE11-dist-in 10.8474 APE10-dist-in 5.858 APE9-dist-in 2.9838 None None None XRAY 2.85 0.204 0.228 A 364.0 355.0 2 27 27 0 [[56, 340]] 1.0 7z1g CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7B6FA P49841 36 382 420.0 SZW:401 Type1 Active DFGin 6.7876 14.0024 BLAminus -139.5, -179.55 63.73, 84.52 -97.59, 24.1 286.83, 79.42 -64.99, -20.21 in-in in 8.3187 Saltbr-in 2.5726 HRD-in -72.27, -45.59 68.3, 15.73 in-in-in SNCiii in-in ActLoopNT-in 2.8606 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.61, 164.26 APE9-dihe-na 74.41, 146.1 APE8-dihe-in -66.85, 137.72 APE8-rot-in 301.31 APE67-dihe-in -60.67, -24.91 -43.57, -54.9 APE12-dist-in 13.468 APE11-dist-in 11.6748 APE10-dist-in 7.0867 APE9-dist-in 3.2029 None PTR216 PTR216 XRAY 2.05 0.176 0.209 A 365.0 347.0 0 27 27 0 [[56, 340]] 1.0 7b6f CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8AUZA P49841 27 381 420.0 O9C:402 Type1 Active DFGin 7.0282 13.8218 BLAminus -150.9, 179.1 54.07, 83.84 -94.84, 28.62 288.95, 81.72 -71.58, -10.75 in-in in 8.4971 Saltbr-in 2.7343 HRD-in -57.37, -52.37 73.76, 8.1 in-in-in SNCiii in-in ActLoopNT-in 3.1547 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.43, 171.72 APE9-dihe-na 68.38, 153.94 APE8-dihe-in -73.1, 142.46 APE8-rot-in 305.9 APE67-dihe-in -60.73, -30.47 -42.52, -61.25 APE12-dist-in 13.255 APE11-dist-in 11.714 APE10-dist-in 7.0252 APE9-dist-in 3.0553 None PTR216 PTR216 XRAY 2.66 0.172 0.229 A 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8auz CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8AUZB P49841 27 381 420.0 O9C:402 Type1 Active DFGin 7.0993 13.9066 BLAminus -145.47, 175.75 60.6, 82.78 -92.91, 28.92 286.05, 79.75 -73.75, -11.85 in-in in 8.5865 Saltbr-in 2.6974 HRD-in -55.14, -51.91 71.49, 10.11 in-in-in SNCiii in-in ActLoopNT-in 3.1386 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.91, 170.34 APE9-dihe-na 66.33, 153.39 APE8-dihe-in -70.91, 144.03 APE8-rot-in 280.02 APE67-dihe-in -59.87, -32.25 -43.58, -60.53 APE12-dist-in 13.1722 APE11-dist-in 11.6615 APE10-dist-in 6.9239 APE9-dist-in 3.0036 None PTR216 PTR216 XRAY 2.66 0.172 0.229 B 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8auz CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4AFJA P49841 36 384 420.0 SJJ:1391 Type1 Active DFGin 6.9374 13.7151 BLAminus -130.67, 179.05 59.17, 87.64 -94.83, 20.23 280.89, 81.14 -65.73, -20.9 in-in in 8.572 Saltbr-in 2.6523 HRD-in -69.53, -45.4 65.78, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.9368 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.24, 160.98 APE9-dihe-na 76.37, 138.38 APE8-dihe-in -58.5, 130.27 APE8-rot-in 301.13 APE67-dihe-in -61.75, -23.96 -37.58, -52.92 APE12-dist-in 13.4348 APE11-dist-in 11.6806 APE10-dist-in 6.9749 APE9-dist-in 3.1929 None PTR216 PTR216 XRAY 1.98 0.179 0.216 A 367.0 344.0 5 27 27 0 [[56, 340]] 1.0 4afj CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4AFJB P49841 34 384 420.0 SJJ:1392 Type1 Active DFGin 6.9478 14.0458 BLAminus -131.53, 179.02 57.76, 85.75 -93.28, 22.08 280.88, 83.41 -64.33, -20.8 in-in in 8.5255 Saltbr-in 2.7428 HRD-in -67.39, -46.66 68.06, 10.89 in-in-in SNCiii in-in ActLoopNT-in 2.8765 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.99, 165.35 APE9-dihe-na 75.2, 154.5 APE8-dihe-in -78.53, 128.88 APE8-rot-in 295.4 APE67-dihe-in -61.46, -24.46 -31.5, -55.04 APE12-dist-in 13.4761 APE11-dist-in 11.5819 APE10-dist-in 6.9584 APE9-dist-in 3.1461 None PTR216 PTR216 XRAY 1.98 0.179 0.216 B 367.0 347.0 4 27 27 0 [[56, 340]] 1.0 4afj CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3ZRKA P49841 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.8856 13.908 BLAminus -131.68, 179.96 63.1, 79.53 -95.35, 25.37 286.53, 78.64 -74.21, -8.59 in-in in 8.4741 Saltbr-in 2.7497 HRD-in -67.17, -50.87 73.03, 10.45 in-in-in SNCiii in-in ActLoopNT-in 2.8412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.35, 160.84 APE9-dihe-na 74.59, 142.57 APE8-dihe-in -61.86, 136.31 APE8-rot-in 305.46 APE67-dihe-in -59.75, -23.44 -46.23, -50.56 APE12-dist-in 13.3769 APE11-dist-in 11.6698 APE10-dist-in 7.0029 APE9-dist-in 3.1599 None PTR216 PTR216 XRAY 2.37 0.201 0.243 A 371.0 347.0 2 27 27 0 [[56, 340]] 1.0 3zrk CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3ZRKB P49841 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.7154 14.0168 BLAminus -139.49, -177.28 57.97, 77.09 -90.4, 24.0 286.01, 81.23 -69.91, -16.36 in-in in 8.587 Saltbr-in 2.7319 HRD-in -64.4, -48.95 71.37, 3.03 in-in-in SNCiii in-in ActLoopNT-in 2.8439 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.35, 163.72 APE9-dihe-na 73.35, 153.59 APE8-dihe-in -70.79, 138.65 APE8-rot-in 292.42 APE67-dihe-in -62.81, -26.76 -44.91, -48.41 APE12-dist-in 13.3599 APE11-dist-in 11.4817 APE10-dist-in 6.8819 APE9-dist-in 3.1614 None PTR216 PTR216 XRAY 2.37 0.201 0.243 B 371.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zrk CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3ZRLA P49841 36 385 420.0 ZRL:1390 Type1 Active DFGin 6.9762 14.1446 BLAminus -134.74, 178.82 66.15, 74.2 -88.14, 21.07 285.95, 79.46 -68.66, -8.3 in-in in 8.4844 Saltbr-in 2.5864 HRD-in -74.36, -46.11 75.3, 2.22 in-in-in SNCiii in-in ActLoopNT-in 2.8884 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.36, 158.14 APE9-dihe-na 75.43, 144.25 APE8-dihe-in -61.72, 142.08 APE8-rot-in 315.78 APE67-dihe-in -63.29, -26.99 -52.04, -46.88 APE12-dist-in 13.4779 APE11-dist-in 11.7165 APE10-dist-in 7.1567 APE9-dist-in 3.1714 None PTR216 PTR216 XRAY 2.48 0.188 0.249 A 371.0 348.0 2 27 27 0 [[56, 340]] 1.0 3zrl CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3ZRLB P49841 36 384 420.0 ZRL:1390 Type1 Active DFGin 6.8163 14.0659 BLAminus -140.64, -176.21 56.19, 79.11 -88.83, 19.02 286.49, 80.49 -67.02, -13.2 in-in in 8.6131 Saltbr-in 2.7337 HRD-in -62.44, -47.89 69.81, 8.62 in-in-in SNCiii in-in ActLoopNT-in 2.8941 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.8, 160.71 APE9-dihe-na 76.77, 159.03 APE8-dihe-in -75.92, 142.27 APE8-rot-in 284.41 APE67-dihe-in -61.87, -25.02 -48.38, -50.46 APE12-dist-in 13.4519 APE11-dist-in 11.6967 APE10-dist-in 7.0855 APE9-dist-in 3.2183 None PTR216 PTR216 XRAY 2.48 0.188 0.249 B 371.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zrl CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3ZRMA P49841 36 383 420.0 ZRM:1388 Type1 Active DFGin 6.9338 13.9541 BLAminus -132.01, -179.16 64.76, 76.89 -91.07, 16.45 285.73, 79.52 -60.99, -14.53 in-in in 8.3792 Saltbr-in 2.5899 HRD-in -73.17, -48.0 77.03, 4.47 in-in-in SNCiii in-in ActLoopNT-in 2.8649 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.45, 164.9 APE9-dihe-na 71.3, 144.2 APE8-dihe-in -61.55, 140.83 APE8-rot-in 305.4 APE67-dihe-in -61.36, -25.73 -52.92, -47.77 APE12-dist-in 13.4177 APE11-dist-in 11.7327 APE10-dist-in 7.034 APE9-dist-in 3.1836 None PTR216 PTR216 XRAY 2.49 0.19 0.247 A 371.0 346.0 2 27 27 0 [[56, 340]] 1.0 3zrm CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3ZRMB P49841 36 384 420.0 ZRM:1389 Type1 Active DFGin 6.9018 14.1037 BLAminus -140.7, -177.64 59.24, 76.67 -89.43, 25.85 287.41, 78.75 -71.45, -17.33 in-in in 8.556 Saltbr-in 2.6387 HRD-in -65.21, -46.92 71.38, 6.55 in-in-in SNCiii in-in ActLoopNT-in 2.8965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.4, 163.13 APE9-dihe-na 76.6, 157.17 APE8-dihe-in -72.35, 137.17 APE8-rot-in 272.08 APE67-dihe-in -62.09, -20.43 -43.42, -53.94 APE12-dist-in 13.4635 APE11-dist-in 11.6966 APE10-dist-in 7.0308 APE9-dist-in 3.1098 None PTR216 PTR216 XRAY 2.49 0.19 0.247 B 371.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zrm CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5K5NA P49841 36 382 420.0 6QH:4001 Type1 Active DFGin 6.8671 13.8031 BLAminus -136.97, -178.03 58.54, 81.58 -94.06, 22.59 285.28, 80.04 -66.6, -22.76 in-in in 8.6849 Saltbr-in 2.7627 HRD-in -65.0, -45.17 61.7, 20.55 in-in-in SNCiii in-in ActLoopNT-in 2.9036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.55, 163.97 APE9-dihe-na 70.72, 157.82 APE8-dihe-in -71.18, 131.1 APE8-rot-in 299.71 APE67-dihe-in -62.03, -24.12 -33.31, -56.32 APE12-dist-in 13.5851 APE11-dist-in 11.9664 APE10-dist-in 6.9925 APE9-dist-in 3.2009 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 A 370.0 332.0 12 27 27 0 [[56, 340]] 1.0 5k5n CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5K5NB P49841 36 384 420.0 6QH:401 Type1 Active DFGin 6.9681 13.7452 BLAminus -135.06, -178.44 58.85, 83.42 -94.58, 20.58 286.7, 80.8 -64.41, -22.37 in-in in 8.8691 Saltbr-in 2.795 HRD-in -64.71, -45.91 63.61, 14.11 in-in-in SNCiii in-in ActLoopNT-in 2.8804 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.36, 162.07 APE9-dihe-na 75.01, 147.36 APE8-dihe-in -65.41, 124.62 APE8-rot-in 290.2 APE67-dihe-in -56.35, -27.77 -26.59, -62.75 APE12-dist-in 13.3721 APE11-dist-in 11.9936 APE10-dist-in 6.8964 APE9-dist-in 3.1086 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 B 370.0 335.0 11 27 27 0 [[56, 340]] 1.0 5k5n CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1R0EA P49841 35 383 420.0 DFN:702 Type1 Active DFGin 7.2106 13.9782 BLAminus -134.01, -179.44 58.42, 85.11 -96.64, 20.85 278.46, 77.75 -63.57, -17.65 in-in in 8.3722 Saltbr-in 2.7157 HRD-in -68.9, -46.99 73.89, 15.3 in-in-in SNCiii in-in ActLoopNT-in 2.8169 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.99, 167.9 APE9-dihe-na 82.35, 148.07 APE8-dihe-in -104.61, 148.9 APE8-rot-in 290.93 APE67-dihe-inflip 91.63, -34.6 -37.68, 131.22 APE12-dist-in 13.0977 APE11-dist-in 11.0936 APE10-dist-in 6.2403 APE9-dist-in 3.3951 None None None XRAY 2.25 0.225 0.252 A 391.0 344.0 5 27 27 0 [[56, 340]] 1.0 1r0e CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1R0EB P49841 35 383 420.0 DFN:501 Type1 Active DFGin 7.2465 14.1047 BLAminus -133.07, -177.02 55.1, 85.48 -97.08, 20.86 276.04, 78.13 -65.93, -17.26 in-in in 8.4454 Saltbr-in 2.9103 HRD-in -68.16, -44.28 70.07, 10.75 in-in-in SNCiii in-in ActLoopNT-in 2.8839 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.79, 168.13 APE9-dihe-na 84.81, 147.78 APE8-dihe-in -104.27, 148.93 APE8-rot-in 288.7 APE67-dihe-inflip 91.14, -35.24 -35.52, 130.18 APE12-dist-in 13.0787 APE11-dist-in 11.0114 APE10-dist-in 6.1772 APE9-dist-in 3.3688 None None None XRAY 2.25 0.225 0.252 B 391.0 344.0 5 27 27 0 [[56, 340]] 1.0 1r0e CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q5KA P49841 35 384 420.0 TMU:901 Type1 Active DFGin 6.9883 13.8632 BLAminus -136.18, -175.74 56.25, 81.9 -94.66, 24.16 283.53, 73.95 -64.32, -18.01 in-in in 8.2268 Saltbr-in 2.5487 HRD-in -67.21, -47.72 71.71, 7.94 in-in-in SNCiii in-in ActLoopNT-in 2.9814 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.63, 174.67 APE9-dihe-na 78.79, 134.14 APE8-dihe-in -77.03, 144.65 APE8-rot-in 302.42 APE67-dihe-inflip 99.66, -34.41 -53.93, 140.09 APE12-dist-in 12.9051 APE11-dist-in 11.0016 APE10-dist-in 5.832 APE9-dist-in 3.1437 None None None XRAY 1.94 0.222 0.242 A 414.0 345.0 5 27 27 0 [[56, 340]] 1.0 1q5k CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q5KB P49841 35 384 420.0 TMU:902 Type1 Active DFGin 6.9852 13.7726 BLAminus -138.67, -177.12 58.86, 79.46 -94.38, 28.16 285.34, 70.82 -69.41, -14.87 in-in in 8.1321 Saltbr-in 2.8315 HRD-in -69.04, -44.01 68.27, 5.21 in-in-in SNCiii in-in ActLoopNT-in 2.9161 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.05, 176.86 APE9-dihe-na 75.09, 135.72 APE8-dihe-in -79.59, 144.98 APE8-rot-in 303.4 APE67-dihe-inflip 93.62, -37.01 -50.51, 145.1 APE12-dist-in 12.9305 APE11-dist-in 11.072 APE10-dist-in 5.8459 APE9-dist-in 3.1034 None None None XRAY 1.94 0.222 0.242 B 414.0 344.0 6 27 27 0 [[56, 340]] 1.0 1q5k CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3I4BA P49841 25 385 420.0 Z48:501 Type1 Active DFGin 6.6409 13.6459 BLAminus -134.01, -176.44 58.71, 78.24 -93.71, 24.37 285.69, 79.56 -67.57, -20.03 in-in in 8.4755 Saltbr-in 2.6366 HRD-in -63.92, -46.73 77.65, -7.51 in-in-in SNCiii in-in ActLoopNT-in 2.9496 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.08, 174.13 APE9-dihe-na 79.29, 137.44 APE8-dihe-in -92.27, 151.07 APE8-rot-in 303.5 APE67-dihe-inflip 83.63, -1.22 -43.52, 132.98 APE12-dist-in 13.0087 APE11-dist-in 10.9391 APE10-dist-in 5.839 APE9-dist-in 3.1024 None None None XRAY 2.3 0.181 0.222 A 414.0 359.0 0 27 27 0 [[56, 340]] 1.0 3i4b CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3I4BB P49841 36 382 420.0 Z48:501 Type1 Active DFGin 7.0103 13.6549 BLAminus -135.85, -175.31 58.14, 77.59 -93.89, 21.58 285.55, 84.81 -65.19, -18.79 in-in in 8.5085 Saltbr-in 2.617 HRD-in -67.57, -44.79 75.92, -6.36 in-in-in SNCiii in-in ActLoopNT-in 2.941 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.93, 173.5 APE9-dihe-na 79.53, 137.7 APE8-dihe-in -93.51, 150.41 APE8-rot-in 299.4 APE67-dihe-inflip 78.16, -1.88 -37.33, 134.24 APE12-dist-in 13.0428 APE11-dist-in 10.917 APE10-dist-in 5.8278 APE9-dist-in 3.1154 None None None XRAY 2.3 0.181 0.222 B 414.0 347.0 0 27 27 0 [[56, 340]] 1.0 3i4b CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3L1SA P49841 25 384 420.0 Z92:421 Type1 Active DFGin 6.7571 13.7476 BLAminus -136.19, -175.27 59.75, 67.96 -82.46, 22.04 287.73, 86.13 -66.81, -21.63 in-in in 8.5179 Saltbr-in 2.7076 HRD-in -64.1, -46.34 73.45, -1.44 in-in-in SNCiii in-in ActLoopNT-in 2.949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 172.3 APE9-dihe-na 79.23, 137.51 APE8-dihe-in -89.89, 147.82 APE8-rot-in 303.47 APE67-dihe-inflip 83.2, -1.08 -42.22, 131.52 APE12-dist-in 13.0072 APE11-dist-in 10.8922 APE10-dist-in 5.8943 APE9-dist-in 3.1607 None None None XRAY 2.9 0.186 0.232 A 414.0 336.0 21 27 27 0 [[56, 340]] 1.0 3l1s CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3L1SB P49841 36 382 420.0 Z92:422 Type1 Active DFGin 6.9841 13.7797 BLAminus -136.63, -175.36 61.34, 59.7 -75.09, 22.69 291.46, 84.75 -66.47, -23.35 in-in in 8.551 Saltbr-in 2.7367 HRD-in -65.65, -45.98 77.68, -13.89 in-in-in SNCiii in-in ActLoopNT-in 2.9365 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.08, 173.03 APE9-dihe-na 76.72, 137.31 APE8-dihe-in -89.1, 148.7 APE8-rot-in 302.46 APE67-dihe-inflip 83.32, 3.78 -42.62, 131.74 APE12-dist-in 13.0142 APE11-dist-in 10.916 APE10-dist-in 6.1494 APE9-dist-in 3.1214 None None None XRAY 2.9 0.186 0.232 B 414.0 330.0 17 27 27 0 [[56, 340]] 1.0 3l1s CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 2JLDA P49841 35 385 420.0 AG1:1385 Type1 Active DFGin 7.2466 13.6191 BLAminus -128.74, 174.0 65.55, 89.02 -101.06, 20.23 281.85, 78.64 -66.01, -16.46 in-in in 8.5348 Saltbr-in 2.9005 HRD-in -68.74, -48.89 74.29, 10.13 in-in-in SNCiii in-in ActLoopNT-in 2.8459 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -80.14, 165.31 APE9-dihe-na 82.65, 142.84 APE8-dihe-in -89.49, 145.54 APE8-rot-in 290.56 APE67-dihe-inflip 101.97, -33.31 -39.01, 124.35 APE12-dist-in 13.012 APE11-dist-in 11.0047 APE10-dist-in 6.0583 APE9-dist-in 3.2394 None None None XRAY 2.35 0.192 0.227 A 420.0 349.0 2 27 27 0 [[56, 340]] 1.0 2jld CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 2JLDB P49841 35 384 420.0 AG1:1385 Type1 Active DFGin 7.1172 13.6811 BLAminus -134.8, 174.83 62.6, 85.31 -97.62, 21.89 284.88, 76.87 -65.09, -17.38 in-in in 8.458 Saltbr-in 2.7255 HRD-in -67.92, -46.43 70.86, 13.33 in-in-in SNCiii in-in ActLoopNT-in 2.9206 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.11, 167.47 APE9-dihe-na 84.04, 143.71 APE8-dihe-in -89.79, 148.89 APE8-rot-in 294.08 APE67-dihe-inflip 95.31, -31.23 -37.35, 123.61 APE12-dist-in 13.0443 APE11-dist-in 10.9507 APE10-dist-in 5.9948 APE9-dist-in 3.2028 None None None XRAY 2.35 0.192 0.227 B 420.0 349.0 1 27 27 0 [[56, 340]] 1.0 2jld CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3M1SB P49841 35 384 420.0 DW1:421 Type1 Active DFGin 7.1866 13.372 BLAminus -147.84, 174.37 70.86, 99.58 -120.24, 19.87 286.56, 80.37 -63.52, -14.18 in-in in 8.5847 Saltbr-in 2.4408 HRD-in -69.47, -49.47 71.23, 28.36 in-in-in SNCiii in-in ActLoopNT-in 3.0905 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -106.87, 165.89 APE9-dihe-na 90.21, 134.65 APE8-dihe-in -74.2, 145.74 APE8-rot-in 300.21 APE67-dihe-in -72.41, -23.39 -22.57, -69.43 APE12-dist-in 12.9441 APE11-dist-in 10.7117 APE10-dist-in 5.8988 APE9-dist-in 3.769 None None None XRAY 3.134 0.171 0.228 B 420.0 349.0 1 27 27 0 [[56, 340]] 1.0 3m1s CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3PUPA P49841 35 382 420.0 OS1:421 Type1 Active DFGin 6.9952 13.6372 BLAminus -143.74, 172.61 64.16, 94.87 -107.49, 13.61 287.44, 72.72 -52.4, -32.47 in-in in 8.4428 Saltbr-in 2.8069 HRD-in -86.73, -34.2 66.44, 7.86 in-in-in SNCiii in-in ActLoopNT-in 2.8568 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.24, -13.27 APE9-dihe-na -89.84, 168.85 APE8-dihe-in -94.34, 159.6 APE8-rot-in 296.79 APE67-dihe-in -69.26, -2.79 -42.9, -70.67 APE12-dist-in 13.0555 APE11-dist-in 10.9122 APE10-dist-in 6.171 APE9-dist-in 3.4857 None None None XRAY 2.99 0.206 0.249 A 420.0 346.0 2 27 27 0 [[56, 340]] 1.0 3pup CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3PUPB P49841 35 383 420.0 OS1:421 Type1 Active DFGin 6.9868 13.6463 BLAminus -146.61, 171.7 65.62, 100.17 -113.12, 21.06 287.13, 70.81 -60.05, -30.47 in-in in 8.4793 Saltbr-in 2.972 HRD-in -88.21, -42.27 77.46, 8.13 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.13, -17.37 APE9-dihe-na -97.38, 160.84 APE8-dihe-in -100.44, 160.76 APE8-rot-in 282.35 APE67-dihe-in -75.14, -2.22 -49.84, -64.39 APE12-dist-in 13.1068 APE11-dist-in 10.9755 APE10-dist-in 6.4999 APE9-dist-in 3.7505 None None None XRAY 2.99 0.206 0.249 B 420.0 347.0 2 27 27 0 [[56, 340]] 1.0 3pup CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6B8JA P49841 37 384 420.0 65C:502 Type1 Active DFGin 6.8683 13.9089 BLAminus -142.04, -175.4 56.86, 72.8 -87.54, 21.75 287.01, 61.58 -69.77, -16.08 in-in in 8.5074 Saltbr-in 2.3182 HRD-in -66.49, -42.97 62.67, 20.6 in-in-in SNCiii in-in ActLoopNT-in 2.8209 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.37, 166.1 APE9-dihe-na 69.29, 116.74 APE8-dihe-in -38.51, 137.94 APE8-rot-in 299.43 APE67-dihe-in -65.74, -24.52 -56.45, -42.14 APE12-dist-in 13.6847 APE11-dist-in 11.734 APE10-dist-in 7.0179 APE9-dist-in 3.3258 None PTR216 PTR216 XRAY 2.595 0.215 0.247 A 420.0 345.0 3 27 27 0 [[56, 340]] 1.0 6b8j CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6H0UA P49841 36 383 420.0 FKB:501 Type1 Active DFGin 6.7319 13.816 BLAminus -102.2, -173.91 62.01, 94.18 -105.02, 23.81 292.61, 84.27 -66.96, -25.5 in-in in 8.7982 Saltbr-in 2.7262 HRD-in -71.89, -49.13 79.92, 3.93 in-in-in SNCiii in-in ActLoopNT-in 2.9659 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.85, 170.11 APE9-dihe-na 84.06, 143.45 APE8-dihe-in -90.7, 142.53 APE8-rot-in 301.69 APE67-dihe-in -73.12, -14.65 -13.27, -76.63 APE12-dist-in 12.9549 APE11-dist-in 10.8677 APE10-dist-in 5.7603 APE9-dist-in 3.2229 None None None XRAY 2.3 0.195 0.24 A 420.0 348.0 0 27 27 0 [[56, 340]] 1.0 6h0u CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6H0UB P49841 36 383 420.0 FKB:501 Type1 Active DFGin 6.6481 13.9725 BLAminus -111.78, 175.04 68.36, 93.29 -102.83, 22.46 286.57, 84.56 -63.31, -24.15 in-in in 8.7633 Saltbr-in 2.7449 HRD-in -68.5, -49.8 75.08, 1.45 in-in-in SNCiii in-in ActLoopNT-in 2.8506 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.21, 171.64 APE9-dihe-na 80.61, 138.7 APE8-dihe-in -91.3, 150.17 APE8-rot-in 304.68 APE67-dihe-inflip 101.55, -29.52 -53.44, 134.06 APE12-dist-in 12.722 APE11-dist-in 10.7262 APE10-dist-in 5.7037 APE9-dist-in 3.1629 None None None XRAY 2.3 0.195 0.24 B 420.0 348.0 0 27 27 0 [[56, 340]] 1.0 6h0u CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6V6LA P49841 37 384 420.0 QQA:501 Type1 Active DFGin 7.2439 14.2279 BLAminus -134.87, -179.15 59.4, 83.41 -98.99, 30.0 283.16, 72.37 -75.66, -20.38 in-in in 8.3879 Saltbr-in 2.7358 HRD-in -68.21, -49.19 67.93, 18.71 in-in-in SNCiii in-in ActLoopNT-in 3.016 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.84, 162.85 APE9-dihe-na 77.33, 149.16 APE8-dihe-in -69.69, 129.38 APE8-rot-in 287.88 APE67-dihe-in -58.07, -31.39 -36.48, -49.2 APE12-dist-in 13.4611 APE11-dist-in 11.6477 APE10-dist-in 6.9528 APE9-dist-in 3.241 None PTR216 PTR216 XRAY 2.19 0.204 0.234 A 420.0 344.0 4 27 27 0 [[56, 340]] 1.0 6v6l CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3DU8A P49841 35 382 420.0 553:553 Type1 Active DFGin 6.9922 13.9377 BLAminus -138.88, -177.6 60.76, 81.45 -97.52, 17.85 284.1, 81.79 -60.5, -23.71 in-in in 8.7135 Saltbr-in 2.6861 HRD-in -70.97, -44.22 68.9, 5.64 in-in-in SNCiii in-in ActLoopNT-in 2.9768 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.61, 170.6 APE9-dihe-na 82.17, 142.06 APE8-dihe-in -90.1, 145.24 APE8-rot-in 300.29 APE67-dihe-inflip 98.68, -34.99 -51.44, 136.14 APE12-dist-in 13.0356 APE11-dist-in 10.9436 APE10-dist-in 5.7637 APE9-dist-in 3.1519 None None None XRAY 2.2 0.215 0.246 A 422.0 336.0 12 27 27 0 [[56, 340]] 1.0 3du8 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3DU8B P49841 35 385 420.0 553:553 Type1 Active DFGin 7.1097 14.0005 BLAminus -130.0, -177.1 64.69, 78.27 -91.27, 21.46 283.91, 80.88 -65.59, -20.64 in-in in 8.7421 Saltbr-in 2.7016 HRD-in -71.12, -43.48 71.58, 1.27 in-in-in SNCiii in-in ActLoopNT-in 2.9923 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -75.13, 166.25 APE9-dihe-na 83.98, 139.39 APE8-dihe-in -88.38, 143.61 APE8-rot-in 294.95 APE67-dihe-inflip 93.54, -38.98 -56.03, 145.75 APE12-dist-in 13.0504 APE11-dist-in 11.1301 APE10-dist-in 5.901 APE9-dist-in 3.1759 None None None XRAY 2.2 0.215 0.246 B 422.0 339.0 12 27 27 0 [[56, 340]] 1.0 3du8 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR5A P49841 25 385 420.0 A1IE8:501 Type1 Active DFGin 7.0632 14.321 BLAminus -141.02, 178.57 59.76, 86.64 -101.14, 27.38 287.09, 76.28 -70.78, -13.94 in-in in 8.3627 Saltbr-in 2.8669 HRD-in -72.5, -48.23 71.7, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.9846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.15, 177.99 APE9-dihe-na 68.95, 145.14 APE8-dihe-in -94.16, 151.35 APE8-rot-in 288.71 APE67-dihe-inflip 90.22, -34.5 -47.82, 143.36 APE12-dist-in 13.1043 APE11-dist-in 11.1055 APE10-dist-in 6.1672 APE9-dist-in 3.1855 None None None XRAY 2.3 0.204 0.235 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr5 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR5B P49841 36 382 420.0 A1IE8:501 Type1 Active DFGin 7.0679 14.3968 BLAminus -143.23, 179.4 62.21, 84.47 -103.42, 28.19 287.66, 78.04 -72.31, -18.53 in-in in 8.6835 Saltbr-in 2.9648 HRD-in -72.41, -47.52 71.61, 14.06 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.66, -179.45 APE9-dihe-na 68.77, 147.4 APE8-dihe-in -97.67, 156.22 APE8-rot-in 283.57 APE67-dihe-inflip 84.77, -33.0 -49.59, 145.66 APE12-dist-in 13.0555 APE11-dist-in 10.9532 APE10-dist-in 5.9863 APE9-dist-in 3.1875 None None None XRAY 2.3 0.204 0.235 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr5 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR6A P49841 25 385 420.0 A1IFO:501 Type1 Active DFGin 7.0735 14.1612 BLAminus -136.83, -174.79 60.55, 80.3 -97.86, 24.81 287.57, 77.74 -66.69, -16.26 in-in in 8.5559 Saltbr-in 2.9354 HRD-in -72.59, -48.06 71.15, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.9919 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.91, 171.88 APE9-dihe-na 74.24, 144.89 APE8-dihe-in -96.08, 152.09 APE8-rot-in 291.49 APE67-dihe-inflip 90.67, -36.1 -52.14, 144.18 APE12-dist-in 13.0224 APE11-dist-in 11.047 APE10-dist-in 6.1241 APE9-dist-in 3.2396 None None None XRAY 2.3 0.2 0.232 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr6 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR6B P49841 36 382 420.0 A1IFO:501 Type1 Active DFGin 7.1281 14.3598 BLAminus -139.12, -179.31 63.06, 81.93 -99.98, 26.01 286.75, 75.51 -71.16, -14.75 in-in in 8.8431 Saltbr-in 2.8359 HRD-in -72.29, -48.89 71.91, 12.0 in-in-in SNCiii in-in ActLoopNT-in 2.9172 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.4, 172.1 APE9-dihe-na 77.09, 144.87 APE8-dihe-in -98.08, 154.15 APE8-rot-in 291.27 APE67-dihe-inflip 90.37, -33.63 -52.57, 140.86 APE12-dist-in 13.0706 APE11-dist-in 10.9572 APE10-dist-in 5.9828 APE9-dist-in 3.2201 None None None XRAY 2.3 0.2 0.232 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr6 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR7A P49841 25 385 420.0 A1IFJ:501 Type1 Active DFGin 6.912 13.9494 BLAminus -136.24, -176.42 58.55, 87.09 -104.67, 27.04 287.13, 78.6 -71.53, -14.0 in-in in 8.6316 Saltbr-in 2.8018 HRD-in -71.98, -46.0 72.36, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.9869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.42, 177.43 APE9-dihe-na 69.9, 145.82 APE8-dihe-in -94.03, 156.28 APE8-rot-in 289.17 APE67-dihe-inflip 91.05, -31.63 -52.45, 141.85 APE12-dist-in 13.1081 APE11-dist-in 11.1214 APE10-dist-in 6.1207 APE9-dist-in 3.1495 None None None XRAY 2.3 0.199 0.229 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr7 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR7B P49841 36 382 420.0 A1IFJ:501 Type1 Active DFGin 6.9902 13.9524 BLAminus -139.3, -178.5 61.7, 87.08 -105.92, 24.05 284.91, 80.77 -70.11, -13.68 in-in in 8.5932 Saltbr-in 2.7099 HRD-in -71.41, -48.43 71.41, 11.5 in-in-in SNCiii in-in ActLoopNT-in 2.9398 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.82, 177.23 APE9-dihe-na 70.05, 146.13 APE8-dihe-in -96.47, 160.58 APE8-rot-in 285.27 APE67-dihe-inflip 87.67, -29.95 -51.57, 140.33 APE12-dist-in 13.0082 APE11-dist-in 11.0074 APE10-dist-in 6.0448 APE9-dist-in 3.156 None None None XRAY 2.3 0.199 0.229 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr7 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR8A P49841 25 385 420.0 A1IE7:501 Type1 Active DFGin 6.991 14.3251 BLAminus -138.39, -179.52 63.72, 81.82 -96.4, 23.65 287.29, 75.6 -66.3, -11.74 in-in in 8.5529 Saltbr-in 2.9059 HRD-in -71.33, -45.89 67.7, 10.94 in-in-in SNCiii in-in ActLoopNT-in 2.9571 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.78, 169.84 APE9-dihe-na 80.06, 148.59 APE8-dihe-in -102.16, 146.47 APE8-rot-in 284.89 APE67-dihe-inflip 97.34, -39.62 -53.84, 140.75 APE12-dist-in 13.0812 APE11-dist-in 11.083 APE10-dist-in 6.0117 APE9-dist-in 3.1971 None None None XRAY 2.3 0.191 0.221 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr8 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR8B P49841 36 383 420.0 A1IE7:501 Type1 Active DFGin 7.087 14.3561 BLAminus -145.34, 175.42 68.0, 83.84 -100.29, 22.36 287.83, 75.27 -65.32, -15.0 in-in in 8.7153 Saltbr-in 2.8977 HRD-in -76.0, -49.5 72.49, 12.34 in-in-in SNCiii in-in ActLoopNT-in 2.9624 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.57, 172.15 APE9-dihe-na 78.67, 145.51 APE8-dihe-in -99.99, 146.48 APE8-rot-in 286.49 APE67-dihe-inflip 90.46, -36.44 -48.06, 141.27 APE12-dist-in 13.0668 APE11-dist-in 10.8517 APE10-dist-in 5.8498 APE9-dist-in 3.1528 None None None XRAY 2.3 0.191 0.221 B 442.0 348.0 0 27 27 0 [[56, 340]] 1.0 9fr8 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR9A P49841 25 385 420.0 A1IE6:501 Type1 Active DFGin 7.0374 14.3248 BLAminus -140.22, -173.71 59.89, 84.2 -98.36, 22.56 286.21, 81.87 -68.06, -16.06 in-in in 8.4621 Saltbr-in 2.928 HRD-in -72.09, -48.73 72.37, 5.47 in-in-in SNCiii in-in ActLoopNT-in 2.9713 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.48, 176.45 APE9-dihe-na 79.51, 153.1 APE8-dihe-in -106.78, 146.27 APE8-rot-in 287.32 APE67-dihe-inflip 100.87, -37.49 -40.18, 126.82 APE12-dist-in 13.0195 APE11-dist-in 11.0304 APE10-dist-in 5.997 APE9-dist-in 3.1732 None None None XRAY 2.55 0.197 0.234 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr9 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9FR9B P49841 36 382 420.0 A1IE6:501 Type1 Active DFGin 6.9697 14.4133 BLAminus -146.13, 179.78 62.16, 86.8 -103.01, 25.64 284.6, 80.86 -74.54, -16.98 in-in in 8.7597 Saltbr-in 3.487 HRD-in -67.74, -52.21 72.42, 13.09 in-in-in SNCiii in-in ActLoopNT-in 2.8715 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.09, 170.35 APE9-dihe-na 79.85, 140.07 APE8-dihe-in -93.7, 153.67 APE8-rot-in 288.81 APE67-dihe-inflip 99.37, -31.56 -52.24, 133.09 APE12-dist-in 12.9815 APE11-dist-in 10.8097 APE10-dist-in 5.7912 APE9-dist-in 3.1814 None None None XRAY 2.55 0.197 0.234 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr9 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9HUKB P49841 26 382 420.0 A1IXL:501 Type1 Active DFGin 7.4628 14.0621 BLAminus -139.0, -179.94 58.73, 94.97 -114.49, 25.32 285.15, 69.98 -63.61, -20.61 in-in in 8.1298 Saltbr-in 3.2803 HRD-in -69.2, -40.72 63.39, 20.78 in-in-in SNCiii in-in ActLoopNT-in 3.0415 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.58, -178.87 APE9-dihe-na 67.27, 135.83 APE8-dihe-in -80.15, 163.62 APE8-rot-in 319.54 APE67-dihe-inflip 75.84, -27.97 -60.6, 162.6 APE12-dist-in 12.8383 APE11-dist-in 10.7437 APE10-dist-in 5.7296 APE9-dist-in 3.2115 None None None XRAY 3.5 0.219 0.25 B 442.0 357.0 0 27 27 0 [[56, 340]] 1.0 9huk CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9HULA P49841 25 385 420.0 A1IXM:501 Type1 Active DFGin 7.0701 13.9429 BLAminus -137.8, -179.92 58.93, 93.22 -109.33, 21.24 284.01, 77.28 -66.77, -7.95 in-in in 8.3439 Saltbr-in 2.9227 HRD-in -67.44, -42.84 67.99, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.1667 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.24, 178.29 APE9-dihe-na 68.13, 143.96 APE8-dihe-in -84.08, 162.04 APE8-rot-in 308.02 APE67-dihe-inflip 75.91, -35.84 -57.58, 161.58 APE12-dist-in 13.0659 APE11-dist-in 11.0236 APE10-dist-in 5.9969 APE9-dist-in 3.1634 None None None XRAY 2.9 0.218 0.244 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9hul CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9HULB P49841 26 383 420.0 A1IXM:501 Type1 Active DFGin 7.2175 13.8998 BLAminus -141.92, -177.61 60.57, 66.5 -86.27, 21.98 288.8, 69.64 -66.75, -12.19 in-in in 8.2676 Saltbr-in 2.7477 HRD-in -68.36, -43.53 65.84, 14.02 in-in-in SNCiii in-in ActLoopNT-in 3.0185 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.86, 177.51 APE9-dihe-na 70.81, 136.76 APE8-dihe-in -79.57, 164.11 APE8-rot-in 306.92 APE67-dihe-inflip 69.45, -30.71 -58.24, 165.67 APE12-dist-in 13.0545 APE11-dist-in 10.9752 APE10-dist-in 6.0547 APE9-dist-in 3.14 None None None XRAY 2.9 0.218 0.244 B 442.0 358.0 0 27 27 0 [[56, 340]] 1.0 9hul CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9HV3A P49841 25 385 420.0 A1IXN:501 Type1 Active DFGin 7.1249 13.9703 BLAminus -135.63, 170.17 69.98, 84.71 -102.55, 20.46 290.46, 80.59 -69.94, -0.25 in-in in 8.5374 Saltbr-in 2.8684 HRD-in -69.25, -48.0 72.7, 9.47 in-in-in SNCiii in-in ActLoopNT-in 2.9354 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.1, 169.69 APE9-dihe-na 79.34, 142.23 APE8-dihe-in -80.23, 146.96 APE8-rot-in 316.9 APE67-dihe-inflip 78.3, -27.2 -49.89, 154.45 APE12-dist-in 13.1231 APE11-dist-in 11.1203 APE10-dist-in 6.1972 APE9-dist-in 3.1364 None None None XRAY 2.9 0.208 0.238 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9hv3 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9HV3B P49841 25 382 420.0 A1IXN:501 Type1 Active DFGin 7.0874 13.9122 BLAminus -155.32, 174.2 63.74, 86.56 -102.98, 16.67 284.3, 76.87 -64.93, -6.56 in-in in 8.5969 Saltbr-in 2.6055 HRD-in -75.09, -41.25 66.67, 4.87 in-in-in SNCiii in-in ActLoopNT-in 2.9817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.85, 168.81 APE9-dihe-na 83.21, 130.42 APE8-dihe-in -66.5, 151.79 APE8-rot-in 306.21 APE67-dihe-inflip 94.47, -29.15 -64.06, 143.12 APE12-dist-in 12.9743 APE11-dist-in 10.8793 APE10-dist-in 5.979 APE9-dist-in 3.017 None None None XRAY 2.9 0.208 0.238 B 442.0 358.0 0 27 27 0 [[56, 340]] 1.0 9hv3 CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q3DA P49841 35 385 420.0 STU:451 Type1 Active DFGin 7.2063 14.4113 BLAminus -139.48, 178.33 63.94, 87.17 -99.43, 23.77 282.58, 69.4 -66.25, -14.58 in-in in 8.701 Saltbr-in 2.8552 HRD-in -65.74, -44.7 66.01, 11.52 in-in-in SNCiii in-in ActLoopNT-in 3.0363 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.53, 169.72 APE9-dihe-na 81.56, 143.56 APE8-dihe-in -91.54, 154.32 APE8-rot-in 294.67 APE67-dihe-inflip 96.36, -28.56 -51.12, 132.48 APE12-dist-in 13.0736 APE11-dist-in 11.1082 APE10-dist-in 6.0869 APE9-dist-in 3.274 None None None XRAY 2.2 0.23 0.252 A 424.0 339.0 12 27 27 0 [[56, 340]] 1.0 1q3d CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q3DB P49841 35 383 420.0 STU:452 Type1 Active DFGin 7.26 14.4195 BLAminus -137.95, 177.39 64.41, 87.07 -97.99, 22.53 282.7, 70.11 -63.96, -17.29 in-in in 8.7081 Saltbr-in 2.9721 HRD-in -67.72, -45.35 66.86, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.0238 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.75, 170.28 APE9-dihe-na 79.08, 144.81 APE8-dihe-in -89.94, 151.95 APE8-rot-in 299.26 APE67-dihe-inflip 101.61, -31.22 -54.51, 132.99 APE12-dist-in 13.0847 APE11-dist-in 11.0881 APE10-dist-in 6.1457 APE9-dist-in 3.2379 None None None XRAY 2.2 0.23 0.252 B 424.0 339.0 10 27 27 0 [[56, 340]] 1.0 1q3d CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q3WA P49841 35 386 420.0 ATU:502 Type1 Active DFGin 7.1464 13.9518 BLAminus -137.77, 177.61 62.94, 83.24 -96.07, 24.67 288.22, 69.87 -66.71, -10.0 in-in in 8.3223 Saltbr-in 2.9235 HRD-in -67.11, -47.79 71.57, 6.31 in-in-in SNCiii in-in ActLoopNT-in 3.0225 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.32, 172.63 APE9-dihe-na 77.53, 136.48 APE8-dihe-in -79.93, 143.51 APE8-rot-in 298.62 APE67-dihe-in -62.35, -17.4 -13.52, -82.56 APE12-dist-in 13.0749 APE11-dist-in 11.129 APE10-dist-in 5.9641 APE9-dist-in 3.1434 None None None XRAY 2.3 0.225 0.248 A 424.0 344.0 8 27 27 0 [[56, 340]] 1.0 1q3w CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q3WB P49841 35 383 420.0 ATU:501 Type1 Active DFGin 7.0895 14.2696 BLAminus -140.46, 175.46 63.78, 84.76 -97.02, 22.89 286.31, 71.96 -64.9, -10.6 in-in in 8.5467 Saltbr-in 2.7917 HRD-in -67.92, -47.98 71.69, 6.95 in-in-in SNCiii in-in ActLoopNT-in 3.0188 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.2, 172.08 APE9-dihe-na 78.0, 136.99 APE8-dihe-in -80.5, 143.58 APE8-rot-in 301.78 APE67-dihe-in -64.47, -16.3 -12.81, -81.64 APE12-dist-in 13.0688 APE11-dist-in 11.1114 APE10-dist-in 5.9384 APE9-dist-in 3.1466 None None None XRAY 2.3 0.225 0.248 B 424.0 341.0 8 27 27 0 [[56, 340]] 1.0 1q3w CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q41A P49841 35 386 420.0 IXM:451 Type1 Active DFGin 7.0961 13.7419 BLAminus -140.31, 177.95 63.36, 85.31 -97.68, 24.93 285.2, 72.61 -64.62, -16.75 in-in in 8.1819 Saltbr-in 2.8445 HRD-in -70.03, -43.74 69.02, 2.85 in-in-in SNCiii in-in ActLoopNT-in 3.0075 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.85, 173.09 APE9-dihe-na 80.34, 135.13 APE8-dihe-in -75.55, 139.31 APE8-rot-in 298.19 APE67-dihe-in -65.33, -18.78 -13.64, -78.26 APE12-dist-in 13.068 APE11-dist-in 11.0572 APE10-dist-in 5.9147 APE9-dist-in 3.2247 None None None XRAY 2.1 0.229 0.245 A 424.0 339.0 13 27 27 0 [[56, 340]] 1.0 1q41 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q41B P49841 35 383 420.0 IXM:452 Type1 Active DFGin 7.0941 13.8936 BLAminus -139.75, 177.7 62.59, 85.88 -97.92, 24.85 285.3, 70.28 -63.82, -17.54 in-in in 8.3883 Saltbr-in 2.83 HRD-in -70.82, -46.38 71.27, 6.28 in-in-in SNCiii in-in ActLoopNT-in 3.0071 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.0, 171.76 APE9-dihe-na 82.35, 130.54 APE8-dihe-in -71.97, 140.37 APE8-rot-in 298.15 APE67-dihe-in -64.0, -13.46 -11.43, -84.5 APE12-dist-in 13.0562 APE11-dist-in 11.0548 APE10-dist-in 5.884 APE9-dist-in 3.2357 None None None XRAY 2.1 0.229 0.245 B 424.0 343.0 6 27 27 0 [[56, 340]] 1.0 1q41 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q4LA P49841 35 386 420.0 679:451 Type1 Active DFGin 6.9437 13.7544 BLAminus -138.39, -176.39 57.74, 86.06 -99.56, 21.29 285.7, 72.79 -65.03, -5.34 in-in in 8.5237 Saltbr-in 3.0069 HRD-in -67.11, -46.06 68.04, 16.48 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -95.21, 168.86 APE9-dihe-na 81.69, 129.23 APE8-dihe-in -70.09, 146.41 APE8-rot-in 291.03 APE67-dihe-inflip 104.98, -29.32 -58.42, 137.67 APE12-dist-in 13.1169 APE11-dist-in 11.3523 APE10-dist-in 6.3007 APE9-dist-in 3.3388 None None None XRAY 2.77 0.212 0.251 A 424.0 342.0 10 27 27 0 [[56, 340]] 1.0 1q4l CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1Q4LB P49841 35 383 420.0 679:452 Type1 Active DFGin 7.1687 13.6494 BLAminus -140.11, -177.14 58.72, 87.12 -99.76, 20.01 285.14, 71.58 -64.5, -5.39 in-in in 8.3387 Saltbr-in 2.6728 HRD-in -67.89, -45.11 67.21, 17.1 in-in-in SNCiii in-in ActLoopNT-in 2.9961 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.61, 167.87 APE9-dihe-na 83.04, 132.56 APE8-dihe-in -74.69, 156.93 APE8-rot-in 311.31 APE67-dihe-inflip 93.39, -29.64 -61.08, 141.61 APE12-dist-in 13.0983 APE11-dist-in 11.3225 APE10-dist-in 6.2525 APE9-dist-in 3.3488 None None None XRAY 2.77 0.212 0.251 B 424.0 337.0 12 27 27 0 [[56, 340]] 1.0 1q4l CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3Q3BA P49841 35 386 420.0 55E:421 Type1 Active DFGin 6.8592 13.8905 BLAminus -146.51, -174.92 60.73, 82.19 -97.34, 22.93 287.93, 77.72 -66.67, -8.01 in-in in 8.4603 Saltbr-in 2.7177 HRD-in -65.09, -51.43 75.32, 0.61 in-in-in SNCiii in-in ActLoopNT-in 3.0239 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.28, 172.26 APE9-dihe-na 79.45, 140.83 APE8-dihe-in -87.39, 149.52 APE8-rot-in 308.45 APE67-dihe-in -68.31, -14.9 -12.45, -80.03 APE12-dist-in 13.0041 APE11-dist-in 11.0599 APE10-dist-in 6.1861 APE9-dist-in 3.1458 None None None XRAY 2.7 0.228 0.259 A 424.0 344.0 8 27 27 0 [[56, 340]] 1.0 3q3b CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3Q3BB P49841 35 383 420.0 55E:421 Type1 Active DFGin 6.9437 13.7668 BLAminus -148.03, -175.09 60.19, 82.65 -96.08, 19.99 287.37, 77.74 -64.82, -9.3 in-in in 8.4427 Saltbr-in 2.7893 HRD-in -64.26, -50.5 74.85, 0.78 in-in-in SNCiii in-in ActLoopNT-in 3.0481 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.17, 172.11 APE9-dihe-na 80.0, 136.06 APE8-dihe-in -78.43, 156.9 APE8-rot-in 303.64 APE67-dihe-in -69.77, -0.18 -23.17, -84.47 APE12-dist-in 12.9964 APE11-dist-in 11.0446 APE10-dist-in 6.1791 APE9-dist-in 3.1016 None None None XRAY 2.7 0.228 0.259 B 424.0 341.0 8 27 27 0 [[56, 340]] 1.0 3q3b CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4J1RA P49841 36 383 420.0 I5R:502 Type1 Active DFGin 7.1431 14.149 BLAminus -140.34, -172.16 50.83, 73.0 -88.1, 31.44 288.82, 75.41 -70.78, -20.52 in-in in 8.3393 Saltbr-in 3.0257 HRD-in -70.85, -43.96 67.49, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.9176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.66, 159.85 APE9-dihe-na 83.41, 158.3 APE8-dihe-in -70.39, 137.75 APE8-rot-in 276.14 APE67-dihe-in -62.89, -24.7 -48.3, -48.41 APE12-dist-in 13.4658 APE11-dist-in 11.8784 APE10-dist-in 7.0059 APE9-dist-in 3.199 None PTR216 PTR216 XRAY 2.702 0.174 0.193 A 424.0 344.0 4 27 27 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4J1RB P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.1595 14.1324 BLAminus -138.14, -172.1 51.97, 73.85 -90.74, 32.74 288.65, 76.48 -71.96, -19.84 in-in in 8.3512 Saltbr-in 3.0798 HRD-in -72.6, -39.29 60.47, 16.92 in-in-in SNCiii in-in ActLoopNT-in 2.8744 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.96, 157.32 APE9-dihe-na 86.27, 160.84 APE8-dihe-in -74.2, 139.51 APE8-rot-in 270.87 APE67-dihe-in -63.78, -23.12 -48.17, -50.06 APE12-dist-in 13.4606 APE11-dist-in 11.6326 APE10-dist-in 6.9809 APE9-dist-in 3.1987 None PTR216 PTR216 XRAY 2.702 0.174 0.193 B 424.0 347.0 2 27 27 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4J1RC P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.1535 14.1448 BLAminus -137.53, -170.95 51.06, 74.57 -90.65, 33.09 289.21, 75.99 -73.08, -20.73 in-in in 8.3436 Saltbr-in 3.0086 HRD-in -71.61, -39.59 60.78, 16.42 in-in-in SNCiii in-in ActLoopNT-in 2.9513 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.54, 161.15 APE9-dihe-na 82.95, 157.27 APE8-dihe-in -71.13, 139.05 APE8-rot-in 271.75 APE67-dihe-in -63.34, -23.83 -48.75, -48.68 APE12-dist-in 13.4752 APE11-dist-in 11.9746 APE10-dist-in 7.0273 APE9-dist-in 3.2194 None PTR216 PTR216 XRAY 2.702 0.174 0.193 C 424.0 345.0 4 27 27 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4J1RD P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.1575 14.143 BLAminus -136.3, -170.0 51.29, 73.39 -89.98, 32.08 288.97, 75.59 -72.78, -18.14 in-in in 8.3472 Saltbr-in 3.0818 HRD-in -65.4, -45.24 73.44, 1.93 in-in-in SNCiii in-in ActLoopNT-in 2.9291 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.81, 157.82 APE9-dihe-na 85.66, 159.76 APE8-dihe-in -71.48, 137.15 APE8-rot-in 266.3 APE67-dihe-in -62.21, -25.06 -46.41, -50.2 APE12-dist-in 13.4651 APE11-dist-in 11.9016 APE10-dist-in 7.0243 APE9-dist-in 3.1172 None PTR216 PTR216 XRAY 2.702 0.174 0.193 D 424.0 346.0 3 27 27 0 [[56, 340]] 1.0 4j1r CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5HLNA P49841 34 384 420.0 65C:501 Type1 Active DFGin 6.9714 13.5391 BLAminus -145.82, 177.83 61.52, 84.96 -98.63, 20.2 288.24, 74.65 -61.35, -16.22 in-in in 8.64 Saltbr-in 2.9698 HRD-in -72.97, -42.53 59.11, 33.41 in-in-in SNCiii in-in ActLoopNT-in 2.9659 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.08, -68.13 APE9-dihe-na -70.88, 179.27 APE8-dihe-in -73.41, 154.88 APE8-rot-in 283.39 APE67-dihe-in -59.67, -27.13 -52.94, -57.58 APE12-dist-in 13.1086 APE11-dist-in 11.7674 APE10-dist-in 7.2143 APE9-dist-in 3.907 None PTR216 PTR216 XRAY 3.1 0.173 0.236 A 424.0 347.0 4 27 27 0 [[56, 340]] 1.0 5hln CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5HLPA P49841 36 382 420.0 65A:501 Type1 Active DFGin 7.1863 14.396 BLAminus -136.58, -178.8 62.45, 78.77 -95.76, 20.37 283.01, 75.68 -68.07, -12.1 in-in in 8.1462 Saltbr-in 2.605 HRD-in -72.39, -43.73 64.36, 19.61 in-in-in SNCiii in-in ActLoopNT-in 2.8712 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.83, 176.24 APE9-dihe-na 71.02, 146.23 APE8-dihe-in -63.35, 144.14 APE8-rot-in 289.42 APE67-dihe-in -64.86, -21.95 -54.37, -48.38 APE12-dist-in 13.6671 APE11-dist-in 11.8195 APE10-dist-in 6.6439 APE9-dist-in 3.2984 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 A 424.0 339.0 8 27 27 0 [[56, 340]] 1.0 5hlp CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5HLPB P49841 36 383 420.0 65A:501 Type1 Active DFGin 7.1151 14.4669 BLAminus -132.96, -174.02 57.79, 78.12 -94.26, 22.08 284.54, 74.66 -71.61, -17.17 in-in in 8.276 Saltbr-in 2.7164 HRD-in -71.48, -47.76 70.66, 10.73 in-in-in SNCiii in-in ActLoopNT-in 2.8371 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.37, 176.63 APE9-dihe-na 72.15, 149.52 APE8-dihe-in -67.13, 142.42 APE8-rot-in 293.57 APE67-dihe-in -63.1, -24.66 -49.41, -51.54 APE12-dist-in 13.356 APE11-dist-in 11.8213 APE10-dist-in 6.5807 APE9-dist-in 3.1348 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 B 424.0 337.0 11 27 27 0 [[56, 340]] 1.0 5hlp CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5KPKA P49841 35 384 420.0 6VK:500 Type1 Active DFGin 6.9115 14.5084 BLAminus -138.4, -178.64 58.08, 79.3 -90.22, 19.44 284.58, 73.09 -63.35, -18.32 in-in in 8.5736 Saltbr-in 2.7304 HRD-in -73.46, -47.41 66.88, 21.39 in-in-in SNCiii in-in ActLoopNT-in 2.9498 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.73, 163.34 APE9-dihe-na 69.65, 162.27 APE8-dihe-in -73.86, 143.79 APE8-rot-in 303.06 APE67-dihe-in -60.34, -24.86 -54.25, -52.95 APE12-dist-in 13.597 APE11-dist-in 12.1565 APE10-dist-in 7.487 APE9-dist-in 3.2434 None PTR216 PTR216 XRAY 2.4 0.17 0.224 A 424.0 347.0 3 27 27 0 [[56, 340]] 1.0 5kpk CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5KPKB P49841 35 383 420.0 6VK:500 Type1 Active DFGin 7.0281 14.5236 BLAminus -138.48, -175.82 55.16, 85.06 -97.98, 23.13 277.82, 78.64 -67.65, -21.76 in-in in 8.5853 Saltbr-in 2.685 HRD-in -71.19, -45.78 65.3, 13.14 in-in-in SNCiii in-in ActLoopNT-in 3.0036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.69, 168.24 APE9-dihe-na 65.31, 163.84 APE8-dihe-in -77.16, 143.7 APE8-rot-in 304.59 APE67-dihe-in -57.42, -23.92 -54.57, -50.84 APE12-dist-in 13.6928 APE11-dist-in 12.1642 APE10-dist-in 7.3948 APE9-dist-in 3.1039 None PTR216 PTR216 XRAY 2.4 0.17 0.224 B 424.0 345.0 4 27 27 0 [[56, 340]] 1.0 5kpk CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5KPLA P49841 36 384 420.0 6VL:500 Type1 Active DFGin 7.044 14.2531 BLAminus -136.48, 178.55 58.11, 81.69 -92.72, 18.86 289.18, 73.73 -64.85, -20.41 in-in in 8.3485 Saltbr-in 2.4859 HRD-in -65.11, -50.47 69.64, 19.91 in-in-in SNCiii in-in ActLoopNT-in 3.0876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.42, 168.54 APE9-dihe-na 62.76, 158.29 APE8-dihe-in -78.28, 147.71 APE8-rot-in 310.05 APE67-dihe-in -62.4, -23.75 -53.92, -48.24 APE12-dist-in 13.4339 APE11-dist-in 11.8787 APE10-dist-in 7.1366 APE9-dist-in 3.3883 None PTR216 PTR216 XRAY 2.6 0.182 0.244 A 424.0 340.0 9 27 27 0 [[56, 340]] 1.0 5kpl CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5KPLB P49841 36 383 420.0 6VL:500 Type1 Active DFGin 7.1545 14.6155 BLAminus -138.92, -172.41 52.88, 79.26 -88.95, 20.81 278.36, 73.5 -72.97, -16.23 in-in in 8.4978 Saltbr-in 2.9713 HRD-in -70.3, -40.66 56.94, 24.57 in-in-in SNCiii in-in ActLoopNT-in 2.7814 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.07, 160.76 APE9-dihe-na 66.33, 169.2 APE8-dihe-in -85.14, 144.57 APE8-rot-in 313.48 APE67-dihe-in -71.14, -21.99 -47.02, -47.87 APE12-dist-in 13.6449 APE11-dist-in 11.8586 APE10-dist-in 7.3669 APE9-dist-in 3.3795 None PTR216 PTR216 XRAY 2.6 0.182 0.244 B 424.0 340.0 8 27 27 0 [[56, 340]] 1.0 5kpl CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5KPMA P49841 36 383 420.0 6VM:500 Type1 Active DFGin 7.1795 14.1524 BLAminus -127.54, 178.59 63.4, 85.66 -102.69, 28.41 287.99, 66.47 -62.48, -34.28 in-in in 8.4058 Saltbr-in 2.6694 HRD-in -73.98, -45.27 60.61, 25.04 in-in-in SNCiii in-in ActLoopNT-in 2.7332 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.88, 162.98 APE9-dihe-na 64.81, 161.74 APE8-dihe-in -75.86, 141.16 APE8-rot-in 297.33 APE67-dihe-in -64.41, -17.12 -48.06, -52.48 APE12-dist-in 13.62 APE11-dist-in 11.8384 APE10-dist-in 7.3632 APE9-dist-in 3.2615 None PTR216 PTR216 XRAY 2.69 0.178 0.24 A 424.0 345.0 3 27 27 0 [[56, 340]] 1.0 5kpm CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5KPMB P49841 36 384 420.0 6VM:500 Type1 Active DFGin 7.1408 14.6384 BLAminus -142.12, 178.63 60.71, 81.6 -96.16, 22.05 281.72, 76.19 -66.25, -7.91 in-in in 8.6086 Saltbr-in 2.5806 HRD-in -65.22, -49.2 64.23, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.9931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.34, 163.89 APE9-dihe-na 62.78, 158.8 APE8-dihe-in -77.09, 139.57 APE8-rot-in 302.93 APE67-dihe-in -64.17, -18.23 -41.12, -52.04 APE12-dist-in 13.5592 APE11-dist-in 11.9721 APE10-dist-in 7.4703 APE9-dist-in 3.1928 None PTR216 PTR216 XRAY 2.69 0.178 0.24 B 424.0 346.0 3 27 27 0 [[56, 340]] 1.0 5kpm CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4IQ6A P49841 37 382 420.0 IQ6:501 Type1 Active DFGin 7.0678 14.0082 BLAminus -142.1, 176.37 68.23, 72.95 -88.9, 16.75 291.61, 92.77 -55.61, -37.28 in-in in 8.5737 Saltbr-in 2.8412 HRD-in -66.67, -43.42 72.45, -14.35 in-in-in SNCiii in-in ActLoopNT-in 3.0118 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.44, 163.79 APE9-dihe-na 84.06, 140.31 APE8-dihe-in -95.86, 141.6 APE8-rot-in 294.32 APE67-dihe-inflip 102.08, -40.06 -38.49, 130.32 APE12-dist-in 13.2141 APE11-dist-in 11.0068 APE10-dist-in 6.1934 APE9-dist-in 3.1668 None None None XRAY 3.12 0.188 0.227 A 426.0 324.0 22 27 27 0 [[56, 340]] 1.0 4iq6 CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3SAYA P49841 35 384 420.0 OFT:431 Type1 Active DFGin 6.9238 14.2084 BLAminus -134.06, -176.24 58.1, 80.75 -95.49, 24.69 285.79, 80.8 -58.99, -23.52 in-in in 8.7646 Saltbr-in 2.6835 HRD-in -76.77, -47.73 71.86, 15.98 in-in-in SNCiii in-in ActLoopNT-in 2.8872 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 177.68 APE9-dihe-na 70.36, 150.2 APE8-dihe-in -70.69, 142.5 APE8-rot-in 303.06 APE67-dihe-in -64.8, -21.63 -53.21, -43.25 APE12-dist-in 13.4747 APE11-dist-in 11.7676 APE10-dist-in 6.4744 APE9-dist-in 3.1409 None PTR216 PTR216 XRAY 2.231 0.202 0.23 A 430.0 348.0 2 27 27 0 [[56, 340]] 1.0 3say CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3SAYB P49841 35 382 420.0 OFT:431 Type1 Active DFGin 7.0946 14.2081 BLAminus -125.43, -174.49 59.4, 82.08 -94.07, 22.41 283.95, 82.11 -68.04, -11.91 in-in in 8.7759 Saltbr-in 2.5965 HRD-in -71.92, -46.59 68.83, 6.83 in-in-in SNCiii in-in ActLoopNT-in 2.9773 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.5, 172.68 APE9-dihe-na 72.51, 152.54 APE8-dihe-in -66.45, 133.95 APE8-rot-in 293.34 APE67-dihe-in -62.41, -25.02 -42.21, -48.58 APE12-dist-in 13.5034 APE11-dist-in 11.8296 APE10-dist-in 6.7035 APE9-dist-in 3.0926 None PTR216 PTR216 XRAY 2.231 0.202 0.23 B 430.0 348.0 0 27 27 0 [[56, 340]] 1.0 3say CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4PTCA P49841 36 381 420.0 2WE:501 Type1 Active DFGin 6.9363 14.3975 BLAminus -147.73, -174.11 62.98, 81.81 -100.26, 25.83 284.28, 79.03 -59.65, -43.28 in-in in 9.1619 Saltbr-in 2.729 HRD-in -73.84, -45.42 69.86, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.77 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.04, 172.51 APE9-dihe-na 77.59, 144.28 APE8-dihe-in -89.54, 156.63 APE8-rot-in 297.82 APE67-dihe-inflip 95.7, -27.15 -58.15, 143.88 APE12-dist-in 13.0497 APE11-dist-in 10.7791 APE10-dist-in 6.0041 APE9-dist-in 3.2718 None None None XRAY 2.711 0.217 0.281 A 441.0 342.0 4 27 27 0 [[56, 340]] 1.0 4ptc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4PTCB P49841 35 385 420.0 2WE:501 Type1 Active DFGin 7.2125 14.6055 BLAminus -123.82, -167.89 50.38, 80.91 -94.33, 28.59 284.85, 71.64 -64.12, -29.45 in-in in 8.9235 Saltbr-in 2.4023 HRD-in -67.43, -42.31 63.02, 14.07 in-in-in SNCiii in-in ActLoopNT-in 2.9358 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.89, 173.71 APE9-dihe-na 81.21, 152.66 APE8-dihe-in -112.25, 156.82 APE8-rot-in 292.56 APE67-dihe-inflip 100.85, -22.79 -44.26, 123.15 APE12-dist-in 13.0829 APE11-dist-in 10.9184 APE10-dist-in 5.8898 APE9-dist-in 3.2799 None None None XRAY 2.711 0.217 0.281 B 441.0 347.0 4 27 27 0 [[56, 340]] 1.0 4ptc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4PTEA P49841 36 382 420.0 2WF:501 Type1 Active DFGin 6.9317 14.0172 BLAminus -141.21, 178.04 57.99, 89.39 -100.23, 24.26 286.38, 75.9 -68.08, -19.02 in-in in 8.7161 Saltbr-in 2.6354 HRD-in -73.56, -44.45 69.11, 4.74 in-in-in SNCiii in-in ActLoopNT-in 2.7924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.74, 175.98 APE9-dihe-na 75.98, 148.82 APE8-dihe-in -103.79, 152.51 APE8-rot-in 295.33 APE67-dihe-inflip 95.08, -28.26 -38.95, 126.56 APE12-dist-in 12.9786 APE11-dist-in 10.8902 APE10-dist-in 5.8826 APE9-dist-in 3.0881 None None None XRAY 2.033 0.17 0.195 A 441.0 341.0 6 27 27 0 [[56, 340]] 1.0 4pte CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4PTEB P49841 36 385 420.0 2WF:501 Type1 Active DFGin 6.9181 13.9369 BLAminus -137.07, 179.43 58.52, 88.98 -101.38, 27.88 284.28, 76.88 -69.85, -20.65 in-in in 8.4836 Saltbr-in 2.6854 HRD-in -70.9, -46.61 73.05, 2.3 in-in-in SNCiii in-in ActLoopNT-in 2.8872 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.76, 178.59 APE9-dihe-na 72.73, 147.77 APE8-dihe-in -103.48, 150.66 APE8-rot-in 296.89 APE67-dihe-inflip 94.67, -27.57 -36.66, 125.81 APE12-dist-in 12.9354 APE11-dist-in 10.8805 APE10-dist-in 5.8765 APE9-dist-in 3.1539 None None None XRAY 2.033 0.17 0.195 B 441.0 347.0 3 27 27 0 [[56, 340]] 1.0 4pte CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4PTGA P49841 36 382 420.0 2WG:501 Type1 Active DFGin 7.0033 13.9163 BLAminus -132.5, 179.85 66.28, 92.0 -106.7, 26.9 285.24, 77.28 -68.07, -25.88 in-in in 8.5408 Saltbr-in 2.8279 HRD-in -68.57, -44.88 68.54, 10.31 in-in-in SNCiii in-in ActLoopNT-in 2.939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.39, 169.96 APE9-dihe-na 80.02, 147.16 APE8-dihe-in -96.08, 142.52 APE8-rot-in 290.31 APE67-dihe-inflip 90.23, -35.22 -45.66, 142.01 APE12-dist-in 13.0565 APE11-dist-in 11.0186 APE10-dist-in 6.1199 APE9-dist-in 3.284 None None None XRAY 2.361 0.173 0.211 A 441.0 333.0 14 27 27 0 [[56, 340]] 1.0 4ptg CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4PTGB P49841 37 385 420.0 2WG:501 Type1 Active DFGin 6.9512 13.863 BLAminus -136.28, -175.42 57.62, 87.0 -101.31, 27.32 285.42, 76.21 -67.67, -26.13 in-in in 8.437 Saltbr-in 2.705 HRD-in -71.07, -46.44 71.76, 6.12 in-in-in SNCiii in-in ActLoopNT-in 2.8995 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.44, 175.88 APE9-dihe-na 76.35, 149.91 APE8-dihe-in -109.95, 151.08 APE8-rot-in 289.69 APE67-dihe-inflip 91.44, -30.76 -44.23, 136.59 APE12-dist-in 12.9878 APE11-dist-in 11.0088 APE10-dist-in 5.9105 APE9-dist-in 3.1601 None None None XRAY 2.361 0.173 0.211 B 441.0 332.0 17 27 27 0 [[56, 340]] 1.0 4ptg CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8DJCA P49841 35 382 420.0 UAU:501 Type1 Active DFGin 7.1066 13.6454 BLAminus -130.93, 175.08 68.46, 84.27 -99.8, 25.87 290.84, 77.95 -66.29, -22.25 in-in in 8.4422 Saltbr-in 2.6994 HRD-in -67.33, -44.59 69.12, 7.74 in-in-in SNCiii in-in ActLoopNT-in 2.984 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 169.18 APE9-dihe-na 83.11, 139.06 APE8-dihe-in -86.29, 148.88 APE8-rot-in 301.44 APE67-dihe-inflip 95.96, -28.78 -50.91, 136.23 APE12-dist-in 12.9117 APE11-dist-in 10.8312 APE10-dist-in 5.8045 APE9-dist-in 3.2569 None None None XRAY 2.463 0.217 0.242 A 441.0 331.0 17 27 27 0 [[56, 340]] 1.0 8djc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8DJCB P49841 35 385 420.0 UAU:501 Type1 Active DFGin 7.1252 13.6329 BLAminus -137.19, 179.71 59.65, 83.27 -96.94, 27.03 290.51, 79.22 -67.53, -21.56 in-in in 8.3277 Saltbr-in 2.738 HRD-in -65.99, -44.91 69.53, 7.25 in-in-in SNCiii in-in ActLoopNT-in 2.9859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.05, 167.49 APE9-dihe-na 82.24, 138.29 APE8-dihe-in -85.04, 145.47 APE8-rot-in 300.63 APE67-dihe-inflip 98.12, -32.04 -46.91, 135.02 APE12-dist-in 12.9423 APE11-dist-in 10.8879 APE10-dist-in 5.9441 APE9-dist-in 3.2585 None None None XRAY 2.463 0.217 0.242 B 441.0 332.0 19 27 27 0 [[56, 340]] 1.0 8djc CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8DJDA P49841 36 383 420.0 U3E:501 Type1 Active DFGin 7.1826 13.8782 BLAminus -134.36, -179.72 59.88, 85.28 -97.18, 26.66 285.76, 75.79 -65.91, -27.91 in-in in 8.3565 Saltbr-in 2.7038 HRD-in -66.89, -45.93 70.71, 8.73 in-in-in SNCiii in-in ActLoopNT-in 2.9738 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -97.03, 169.31 APE9-dihe-na 77.5, 142.18 APE8-dihe-in -93.09, 155.03 APE8-rot-in 301.61 APE67-dihe-inflip 94.8, -31.52 -52.67, 137.81 APE12-dist-in 13.0595 APE11-dist-in 11.0394 APE10-dist-in 6.1287 APE9-dist-in 3.198 None None None XRAY 2.205 0.209 0.222 A 441.0 338.0 10 27 27 0 [[56, 340]] 1.0 8djd CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8DJDB P49841 36 384 420.0 U3E:501 Type1 Active DFGin 7.129 13.9195 BLAminus -133.17, 179.77 59.91, 85.17 -97.09, 26.57 285.62, 75.36 -66.56, -27.45 in-in in 8.3472 Saltbr-in 2.6969 HRD-in -66.65, -46.07 70.85, 8.52 in-in-in SNCiii in-in ActLoopNT-in 2.9199 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.46, 170.54 APE9-dihe-na 79.57, 140.07 APE8-dihe-in -94.46, 154.56 APE8-rot-in 301.16 APE67-dihe-inflip 94.52, -31.07 -52.58, 138.22 APE12-dist-in 13.0861 APE11-dist-in 11.08 APE10-dist-in 6.0775 APE9-dist-in 3.2169 None None None XRAY 2.205 0.209 0.222 B 441.0 341.0 8 27 27 0 [[56, 340]] 1.0 8djd CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8DJEA P49841 36 384 420.0 U6S:501 Type1 Active DFGin 7.2598 13.3694 BLAminus -139.51, 175.88 67.17, 88.55 -102.31, 22.49 287.71, 78.25 -63.99, -27.99 in-in in 8.3126 Saltbr-in 2.7163 HRD-in -68.38, -45.52 70.24, 12.16 in-in-in SNCiii in-in ActLoopNT-in 2.8928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.85, 166.32 APE9-dihe-na 87.14, 140.36 APE8-dihe-in -88.6, 149.46 APE8-rot-in 293.07 APE67-dihe-inflip 99.13, -30.7 -44.53, 124.89 APE12-dist-in 12.957 APE11-dist-in 10.8666 APE10-dist-in 6.0436 APE9-dist-in 3.3533 None None None XRAY 2.374 0.201 0.227 A 441.0 347.0 2 27 27 0 [[56, 340]] 1.0 8dje CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8DJEB P49841 36 385 420.0 U6S:501 Type1 Active DFGin 7.2394 13.4205 BLAminus -137.87, 177.52 63.92, 86.56 -101.17, 24.78 290.39, 74.84 -68.33, -25.47 in-in in 8.2646 Saltbr-in 2.7355 HRD-in -65.34, -46.08 68.76, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.8895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.12, 167.71 APE9-dihe-na 84.3, 145.94 APE8-dihe-in -98.8, 148.34 APE8-rot-in 293.36 APE67-dihe-inflip 97.13, -37.27 -40.76, 129.94 APE12-dist-in 12.9575 APE11-dist-in 10.9317 APE10-dist-in 5.908 APE9-dist-in 3.263 None None None XRAY 2.374 0.201 0.227 B 441.0 343.0 7 27 27 0 [[56, 340]] 1.0 8dje CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8FF8A P49841 36 382 420.0 XV0:501 Type1 Active DFGin 7.2002 13.7357 BLAminus -135.89, 175.65 65.86, 84.5 -97.83, 25.7 284.17, 77.94 -66.05, -27.44 in-in in 8.341 Saltbr-in 2.7523 HRD-in -68.43, -43.4 70.29, 3.62 in-in-in SNCiii in-in ActLoopNT-in 2.8419 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 167.87 APE9-dihe-na 84.02, 136.04 APE8-dihe-in -86.03, 151.96 APE8-rot-in 298.92 APE67-dihe-inflip 95.48, -31.71 -43.39, 129.41 APE12-dist-in 12.7414 APE11-dist-in 10.7529 APE10-dist-in 5.7907 APE9-dist-in 3.2113 None None None XRAY 2.33 0.198 0.217 A 441.0 347.0 0 27 27 0 [[56, 340]] 1.0 8ff8 CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8FF8B P49841 36 385 420.0 XV0:501 Type1 Active DFGin 7.2005 13.8111 BLAminus -130.19, -175.53 57.72, 85.5 -98.92, 25.25 283.55, 78.69 -65.7, -29.77 in-in in 8.3387 Saltbr-in 2.7464 HRD-in -67.11, -43.98 70.41, 3.15 in-in-in SNCiii in-in ActLoopNT-in 2.825 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.86, 169.83 APE9-dihe-na 81.04, 142.01 APE8-dihe-in -96.19, 150.13 APE8-rot-in 300.46 APE67-dihe-inflip 95.56, -32.32 -40.34, 130.68 APE12-dist-in 12.779 APE11-dist-in 10.7843 APE10-dist-in 5.8246 APE9-dist-in 3.2182 None None None XRAY 2.33 0.198 0.217 B 441.0 346.0 4 27 27 0 [[56, 340]] 1.0 8ff8 CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3F88A P49841 35 383 420.0 3HT:999 Type1 Active DFGin 7.2474 13.7299 BLAminus -137.96, -171.11 53.2, 96.02 -109.46, 31.55 277.23, 77.74 -85.58, 3.2 in-in in 8.6202 Saltbr-in 2.5161 HRD-in -66.41, -48.84 71.78, 26.38 in-in-in SNCiii in-in ActLoopNT-in 3.1406 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.98, 165.73 APE9-dihe-na 69.33, 171.05 APE8-dihe-in -86.85, 130.82 APE8-rot-in 314.66 APE67-dihe-in -71.94, -20.16 -24.55, -52.13 APE12-dist-in 13.5473 APE11-dist-in 12.041 APE10-dist-in 7.3411 APE9-dist-in 3.5985 None PTR216 PTR216 XRAY 2.6 0.204 0.281 A 349.0 341.0 8 27 27 0 [[56, 340]] 1.0 3f88 CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3F88B P49841 35 383 420.0 3HT:999 Type1 Active DFGin 6.9996 13.6509 BLAminus -143.93, 176.87 66.18, 95.41 -113.06, 21.86 281.61, 81.82 -72.47, -7.16 in-in in 8.7652 Saltbr-in 2.6705 HRD-in -64.13, -56.14 79.67, 28.55 in-in-in SNCiii in-in ActLoopNT-in 3.1764 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.92, 167.15 APE9-dihe-na 65.97, 165.61 APE8-dihe-in -80.57, 145.62 APE8-rot-in 308.56 APE67-dihe-in -71.31, -21.5 -44.75, -45.4 APE12-dist-in 13.509 APE11-dist-in 11.9668 APE10-dist-in 7.2567 APE9-dist-in 3.4061 None PTR216 PTR216 XRAY 2.6 0.204 0.281 B 349.0 341.0 8 27 27 0 [[56, 340]] 1.0 3f88 CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACCA P49841 35 385 420.0 7YG:1387 Type1 Active DFGin 7.1831 13.5808 BLAminus -136.28, 179.66 61.59, 88.25 -100.04, 20.56 281.3, 79.98 -65.9, -21.03 in-in in 8.3469 Saltbr-in 2.7616 HRD-in -66.74, -44.81 68.93, 1.06 in-in-in SNCiii in-in ActLoopNT-in 2.8975 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.14, 170.6 APE9-dihe-na 77.6, 138.09 APE8-dihe-in -85.62, 145.43 APE8-rot-in 296.7 APE67-dihe-inflip 94.96, -30.16 -47.88, 136.19 APE12-dist-in 13.0341 APE11-dist-in 10.957 APE10-dist-in 5.8889 APE9-dist-in 3.171 None None None XRAY 2.21 0.191 0.219 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acc CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACCB P49841 35 385 420.0 7YG:1386 Type1 Active DFGin 7.2279 13.5244 BLAminus -136.66, 179.59 61.79, 88.29 -99.73, 21.22 281.91, 80.18 -66.08, -22.29 in-in in 8.2447 Saltbr-in 2.8714 HRD-in -66.61, -45.06 69.24, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.8922 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.27, 172.02 APE9-dihe-na 75.79, 137.96 APE8-dihe-in -86.62, 146.41 APE8-rot-in 295.61 APE67-dihe-inflip 93.46, -30.62 -49.23, 136.97 APE12-dist-in 13.056 APE11-dist-in 11.009 APE10-dist-in 5.9124 APE9-dist-in 3.1824 None None None XRAY 2.21 0.191 0.219 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acc CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACDA P49841 35 385 420.0 GR9:1385 Type1 Active DFGin 7.1862 13.3568 BLAminus -142.44, 176.49 66.05, 88.14 -100.25, 16.93 286.04, 81.9 -64.04, -24.03 in-in in 8.3063 Saltbr-in 2.9365 HRD-in -63.25, -48.42 73.67, 5.76 in-in-in SNCiii in-in ActLoopNT-in 2.8831 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.94, 167.01 APE9-dihe-na 78.77, 128.64 APE8-dihe-in -74.85, 143.25 APE8-rot-in 302.95 APE67-dihe-inflip 99.55, -31.6 -49.31, 132.99 APE12-dist-in 12.8767 APE11-dist-in 10.8678 APE10-dist-in 5.9097 APE9-dist-in 3.2101 None None None XRAY 2.6 0.18 0.226 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acd CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACDB P49841 35 385 420.0 GR9:1385 Type1 Active DFGin 7.1414 13.3767 BLAminus -142.06, 177.81 64.05, 89.32 -100.31, 16.47 285.95, 82.89 -62.46, -26.08 in-in in 8.2225 Saltbr-in 2.9412 HRD-in -62.52, -48.15 72.88, 6.33 in-in-in SNCiii in-in ActLoopNT-in 2.8916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.53, 167.96 APE9-dihe-na 77.33, 127.92 APE8-dihe-in -74.4, 143.25 APE8-rot-in 302.61 APE67-dihe-inflip 99.75, -32.16 -47.58, 132.33 APE12-dist-in 12.9284 APE11-dist-in 10.9465 APE10-dist-in 5.956 APE9-dist-in 3.211 None None None XRAY 2.6 0.18 0.226 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acd CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACGA P49841 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.0033 13.7172 BLAminus -136.29, 179.17 66.16, 92.5 -104.82, 26.85 285.89, 83.54 -71.26, -31.7 in-in in 8.2753 Saltbr-in 2.8663 HRD-in -62.3, -47.68 71.35, 0.06 in-in-in SNCiii in-in ActLoopNT-in 2.9897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.26, 169.3 APE9-dihe-na 82.24, 136.71 APE8-dihe-in -91.92, 145.05 APE8-rot-in 294.1 APE67-dihe-inflip 97.4, -31.68 -47.8, 134.4 APE12-dist-in 12.9461 APE11-dist-in 10.9812 APE10-dist-in 5.9282 APE9-dist-in 3.2924 None None None XRAY 2.6 0.177 0.225 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acg CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACGB P49841 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.0603 13.6101 BLAminus -135.89, 178.4 67.23, 92.34 -105.78, 27.09 285.23, 82.98 -71.05, -30.43 in-in in 8.3794 Saltbr-in 2.9801 HRD-in -63.74, -47.68 70.98, 1.15 in-in-in SNCiii in-in ActLoopNT-in 2.9729 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.69, 168.91 APE9-dihe-na 83.12, 137.88 APE8-dihe-in -91.66, 145.04 APE8-rot-in 292.39 APE67-dihe-inflip 98.28, -31.78 -48.39, 133.48 APE12-dist-in 12.9182 APE11-dist-in 10.9335 APE10-dist-in 5.917 APE9-dist-in 3.2904 None None None XRAY 2.6 0.177 0.225 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acg CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACHA P49841 35 385 420.0 KDI:1386 Type1 Active DFGin 7.1308 13.8433 BLAminus -136.87, 179.55 65.58, 91.16 -104.2, 25.64 286.28, 84.07 -69.39, -35.2 in-in in 8.2337 Saltbr-in 2.9352 HRD-in -61.5, -48.36 72.42, -0.28 in-in-in SNCiii in-in ActLoopNT-in 2.9817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.62, 166.44 APE9-dihe-na 83.56, 135.36 APE8-dihe-in -86.16, 143.31 APE8-rot-in 295.11 APE67-dihe-inflip 98.78, -32.06 -48.27, 133.26 APE12-dist-in 12.998 APE11-dist-in 11.0588 APE10-dist-in 5.9833 APE9-dist-in 3.3216 None None None XRAY 2.6 0.231 0.252 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4ach CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4ACHB P49841 35 385 420.0 KDI:1386 Type1 Active DFGin 7.0809 13.7158 BLAminus -136.91, 178.72 65.4, 91.31 -104.6, 25.63 285.26, 83.9 -68.47, -34.59 in-in in 8.3598 Saltbr-in 2.9378 HRD-in -60.93, -48.9 72.19, 0.38 in-in-in SNCiii in-in ActLoopNT-in 2.9768 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.1, 166.35 APE9-dihe-na 83.22, 136.77 APE8-dihe-in -87.16, 144.14 APE8-rot-in 294.96 APE67-dihe-inflip 98.6, -31.77 -49.65, 133.73 APE12-dist-in 12.9349 APE11-dist-in 10.9849 APE10-dist-in 5.9381 APE9-dist-in 3.2896 None None None XRAY 2.6 0.231 0.252 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4ach CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5OY4A P49841 36 385 420.0 B4K:504 Type1.5_Back Active DFGin 6.9988 13.8215 BLAminus -130.87, 178.64 57.91, 86.19 -95.47, 21.04 282.05, 81.42 -63.36, -27.5 in-in in 8.0884 Saltbr-in 2.722 HRD-in -68.24, -44.36 63.28, 15.03 in-in-in SNCiii in-in ActLoopNT-in 2.8882 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.23, 157.34 APE9-dihe-na 87.05, 159.63 APE8-dihe-in -83.83, 115.67 APE8-rot-in 295.36 APE67-dihe-in -60.03, -25.52 -23.01, -56.29 APE12-dist-in 13.5581 APE11-dist-in 11.6893 APE10-dist-in 7.0579 APE9-dist-in 3.4463 None PTR216 PTR216 XRAY 3.2 0.196 0.229 A 420.0 350.0 0 27 27 0 [[56, 340]] 1.0 5oy4 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4IQ6B P49841 37 382 420.0 IQ6:501 Type1.5_Back Active DFGin 7.0646 14.0574 BLAminus -142.54, 175.49 69.06, 72.09 -88.69, 16.42 291.37, 92.47 -54.24, -38.91 in-in in 8.6089 Saltbr-in 2.85 HRD-in -66.96, -42.68 72.42, -15.31 in-in-in SNCiii in-in ActLoopNT-in 3.0094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.08, 167.69 APE9-dihe-na 81.68, 134.42 APE8-dihe-in -80.06, 146.43 APE8-rot-in 285.37 APE67-dihe-inflip 104.71, -27.8 -48.51, 126.71 APE12-dist-in 13.1481 APE11-dist-in 10.9082 APE10-dist-in 6.2442 APE9-dist-in 3.1149 None None None XRAY 3.12 0.188 0.227 B 426.0 332.0 14 27 27 0 [[56, 340]] 1.0 4iq6 CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6Y9SA P49841 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.7588 13.6151 ABAminus -144.68, -36.37 -95.25, 102.78 -104.54, 22.52 286.7, 80.89 -71.31, -22.3 in-in in 8.4688 Saltbr-in 2.731 HRD-in -69.96, -46.79 66.16, 22.69 in-in-out SNCiio in-out ActLoopNT-in 2.8691 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.41, 160.13 APE9-dihe-na 78.21, 163.56 APE8-dihe-in -74.57, 133.14 APE8-rot-out 174.03 APE67-dihe-in -60.25, -21.67 -45.31, -52.5 APE12-dist-in 13.3908 APE11-dist-in 11.6341 APE10-dist-in 6.8152 APE9-dist-in 3.2172 None PTR216 PTR216 XRAY 2.03 0.204 0.249 A 350.0 344.0 5 27 27 0 [[56, 340]] 1.0 6y9s CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6Y9SB P49841 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.4656 13.6443 ABAminus -142.08, -29.11 -101.71, 107.32 -109.34, 26.02 290.64, 79.47 -70.13, -24.37 in-in in 8.6267 Saltbr-in 2.6258 HRD-in -62.98, -47.75 66.63, 19.7 in-in-out SNCiio in-out ActLoopNT-in 2.8706 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -149.54, 160.17 APE9-dihe-na 74.78, 156.26 APE8-dihe-in -72.21, 136.72 APE8-rot-out 179.96 APE67-dihe-in -63.91, -18.81 -47.88, -49.22 APE12-dist-in 13.498 APE11-dist-in 11.6964 APE10-dist-in 6.9402 APE9-dist-in 3.1721 None PTR216 PTR216 XRAY 2.03 0.204 0.249 B 350.0 340.0 9 27 27 0 [[56, 340]] 1.0 6y9s CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4NM0A P49841 26 383 420.0 ADP:60408 ATPlike Inactive DFGin 6.641 14.2129 BLAminus -133.4, -174.33 56.9, 85.51 -105.72, 27.83 287.31, 80.39 -76.48, -2.57 in-in in 8.774 Saltbr-in 3.0941 HRD-in -69.87, -45.12 67.03, 14.87 in-in-out SNCiio in-out ActLoopNT-in 2.9268 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -71.29, 168.54 APE9-dihe-na 70.19, 144.11 APE8-dihe-in -96.47, 160.21 APE8-rot-out 64.82 APE67-dihe-inflip 78.46, -27.02 -43.67, 149.07 APE12-dist-in 13.0905 APE11-dist-in 10.885 APE10-dist-in 6.5705 APE9-dist-in 3.1347 None None None XRAY 2.5 0.193 0.239 A 389.0 355.0 0 27 27 0 [[56, 340]] 1.0 4nm0 CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8XN6B P49841 26 386 420.0 ANP:501 ATPlike Inactive DFGin 6.5384 13.6503 BLAminus -128.79, 173.26 73.68, 79.74 -95.9, 22.51 291.63, 80.46 -68.54, -21.83 in-in in 8.3292 Saltbr-in 2.8234 HRD-in -66.59, -53.03 79.09, 5.6 in-in-out SNCiio in-out ActLoopNT-in 2.9512 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -88.32, 165.9 APE9-dihe-na 83.63, 132.42 APE8-dihe-in -59.67, 147.17 APE8-rot-out 189.94 APE67-dihe-in -64.51, -21.68 -60.38, -49.59 APE12-dist-in 13.0235 APE11-dist-in 10.9696 APE10-dist-in 5.846 APE9-dist-in 3.0807 None None None XRAY 2.4 0.194 0.242 B 421.0 359.0 2 27 27 0 [[56, 340]] 1.0 8xn6 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1I09B P49841 37 382 420.0 No_ligand No_ligand Inactive DFGin 6.8606 14.0248 BLAminus -135.93, 178.35 61.75, 84.0 -100.67, 24.72 288.55, 74.93 -64.65, -15.56 in-in in 8.4828 Saltbr-in 2.7113 HRD-in -62.69, -41.62 66.11, 9.61 in-in-out SNCiio in-out ActLoopNT-in 2.9529 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.33, -45.22 APE9-dihe-na -71.78, 167.71 APE8-dihe-in -94.58, 171.33 APE8-rot-out 74.32 APE67-dihe-in -65.52, -17.17 -44.16, -80.97 APE12-dist-in 12.7638 APE11-dist-in 11.113 APE10-dist-in 6.2214 APE9-dist-in 3.37 None None None XRAY 2.7 0.242 0.274 B 420.0 341.0 5 27 27 0 [[56, 340]] 1.0 1i09 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6HK7A P49841 36 382 420.0 G8N:403 Type1 Inactive DFGin 7.1812 13.9264 BLAminus -137.45, -171.56 51.7, 92.53 -104.06, 22.16 271.05, 85.97 -65.5, -26.28 in-in in 8.435 Saltbr-in 2.7671 HRD-in -53.21, -66.83 89.97, 19.54 in-in-out SNCiio in-out ActLoopNT-in 2.957 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -85.73, 172.92 APE9-dihe-na 79.4, 146.18 APE8-dihe-in -92.07, 85.52 APE8-rot-in 243.21 APE67-dihe-out 35.1, -40.06 22.07, -158.21 APE12-dist-in 13.2898 APE11-dist-in 11.4463 APE10-dist-in 6.7807 APE9-dist-in 3.3203 None PTR216 PTR216 XRAY 3.2 0.204 0.286 A 347.0 347.0 0 27 27 0 [[56, 340]] 1.0 6hk7 CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7SXHA P49841 37 383 420.0 D1E:501 Type1 Inactive DFGin 6.6502 13.9439 BLAminus -139.68, -175.41 60.2, 74.18 -88.43, 22.79 288.62, 86.11 -74.83, -15.81 in-in in 8.1673 Saltbr-in 2.8585 HRD-in -67.33, -47.27 70.7, 6.58 in-in-out SNCiio in-out ActLoopNT-in 2.863 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -126.8, 168.99 APE9-dihe-na 70.82, 157.42 APE8-dihe-in -70.74, 147.57 APE8-rot-out 190.63 APE67-dihe-in -58.92, -21.73 -57.82, -47.78 APE12-dist-in 13.7709 APE11-dist-in 11.9746 APE10-dist-in 7.3712 APE9-dist-in 3.4319 None PTR216 PTR216 XRAY 2.09 0.216 0.255 A 347.0 341.0 6 27 27 0 [[56, 340]] 1.0 7sxh CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3F7ZA P49841 35 383 420.0 34O:63000 Type1 Inactive DFGin 7.116 13.8181 BLAminus -134.47, 172.11 69.02, 81.68 -97.3, 19.46 284.39, 70.02 -68.92, -10.86 in-in in 8.4854 Saltbr-in 2.5753 HRD-in -62.81, -48.18 67.57, 12.21 in-in-out SNCiio in-out ActLoopNT-in 2.9498 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -139.18, 179.1 APE9-dihe-na 69.89, 157.17 APE8-dihe-in -75.28, 142.37 APE8-rot-out 185.5 APE67-dihe-in -55.86, -28.19 -45.56, -57.07 APE12-dist-in 13.5001 APE11-dist-in 12.029 APE10-dist-in 6.8149 APE9-dist-in 3.3141 None PTR216 PTR216 XRAY 2.4 0.206 0.253 A 350.0 339.0 10 27 27 0 [[56, 340]] 1.0 3f7z CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3SD0A P49841 35 384 420.0 TSK:400 Type1 Inactive DFGin 6.8934 13.6777 BLAminus -139.29, -172.59 62.67, 82.92 -94.93, 18.52 283.9, 73.87 -68.11, -17.74 in-in in 8.4187 Saltbr-in 2.8235 HRD-in -68.02, -47.17 76.6, 11.56 in-in-out SNCiio in-out ActLoopNT-in 2.7996 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -82.28, 176.65 APE9-dihe-na 71.42, 130.7 APE8-dihe-in -100.53, 166.25 APE8-rot-out 29.1 APE67-dihe-inflip 91.12, -25.82 -31.67, 128.67 APE12-dist-in 12.9104 APE11-dist-in 10.8103 APE10-dist-in 5.7793 APE9-dist-in 3.0415 None None None XRAY 2.7 0.179 0.254 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 3sd0 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3ZDIA P49841 36 384 420.0 UGJ:61386 Type1 Inactive DFGin 7.0898 14.0106 BLAminus -139.08, 169.73 59.85, 93.36 -102.57, 31.03 284.51, 75.61 -74.44, -6.01 in-in in 8.7186 Saltbr-in 2.7736 HRD-in -66.47, -49.36 70.61, -12.05 in-in-out SNCiio in-out ActLoopNT-in 2.8737 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.6, -176.4 APE9-dihe-na 57.27, -141.25 APE8-dihe-in -136.89, 135.85 APE8-rot-out 188.96 APE67-dihe-in -60.18, -28.67 -48.24, -43.31 APE12-dist-in 13.7771 APE11-dist-in 12.1156 APE10-dist-in 7.549 APE9-dist-in 3.0939 None PTR216 PTR216 XRAY 2.645 0.204 0.242 A 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zdi CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4B7TA P49841 35 384 420.0 CWT:1385 Type1 Inactive DFGin 6.733 14.135 BLAminus -139.29, -173.55 55.51, 80.28 -97.98, 26.2 284.11, 78.64 -70.02, -22.23 in-in in 8.8256 Saltbr-in 2.732 HRD-in -65.66, -45.08 68.98, -4.07 in-in-out SNCiio in-out ActLoopNT-in 3.0218 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -80.96, 174.72 APE9-dihe-na 79.02, 153.66 APE8-dihe-in -90.72, 141.08 APE8-rot-out 219.61 APE67-dihe-inflip 82.28, -25.01 -65.77, 158.92 APE12-dist-in 13.1502 APE11-dist-in 11.3146 APE10-dist-in 6.5521 APE9-dist-in 3.1216 None None None XRAY 2.772 0.197 0.235 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 4b7t CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6HK3A P49841 35 384 420.0 G8B:401 Type1 Inactive DFGin 6.9186 13.7488 BLAminus -140.26, -177.42 53.43, 89.98 -101.44, 26.95 281.28, 77.81 -71.94, -4.92 in-in in 8.2647 Saltbr-in 2.5202 HRD-in -65.54, -43.12 59.71, 15.8 in-in-out SNCiio in-out ActLoopNT-in 2.9314 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -120.05, -174.23 APE9-dihe-na 65.54, 142.28 APE8-dihe-in -62.37, 137.73 APE8-rot-out 183.0 APE67-dihe-in -57.53, -32.37 -39.19, -57.21 APE12-dist-in 13.3885 APE11-dist-in 11.7623 APE10-dist-in 6.4209 APE9-dist-in 3.2183 None PTR216 PTR216 XRAY 2.35 0.206 0.234 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk3 CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6Y9RA P49841 35 384 420.0 OH8:401 Type1 Inactive DFGin 7.2128 13.9564 BLAminus -128.7, 177.14 64.74, 83.75 -99.31, 22.7 285.39, 75.74 -67.18, -22.12 in-in in 8.3866 Saltbr-in 2.7599 HRD-in -68.2, -47.94 70.12, 17.05 in-in-out SNCiio in-out ActLoopNT-in 2.9695 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -147.41, 164.13 APE9-dihe-na 71.55, 162.91 APE8-dihe-in -81.0, 136.61 APE8-rot-out 173.09 APE67-dihe-in -62.95, -25.51 -45.24, -50.14 APE12-dist-in 13.6836 APE11-dist-in 12.0385 APE10-dist-in 7.353 APE9-dist-in 3.2948 None PTR216 PTR216 XRAY 2.08 0.191 0.226 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6y9r CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1O9UA P49841 35 384 420.0 ADZ:1386 Type1 Inactive DFGin 6.69 14.4088 BLAminus -135.58, -170.77 57.68, 80.28 -97.17, 18.56 286.56, 73.24 -63.89, -4.57 in-in in 8.9184 Saltbr-in 3.2524 HRD-in -60.54, -48.22 66.04, 11.65 in-in-out SNCiio in-out ActLoopNT-in 2.9648 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.51, 167.48 APE9-dihe-na 74.14, -178.83 APE8-dihe-in -103.59, 140.85 APE8-rot-out 179.41 APE67-dihe-in -52.99, -22.64 -16.1, -87.79 APE12-dist-in 13.762 APE11-dist-in 11.7056 APE10-dist-in 7.3617 APE9-dist-in 2.8623 None PTR216 PTR216 XRAY 2.4 0.233 0.26 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 1o9u CMGC_GSK3B_HUMAN CMGC 2.1e-69 240.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9PE9A P49841 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.0716 14.2287 BLAminus -128.7, -179.96 59.31, 84.1 -97.11, 26.91 283.64, 74.63 -73.69, -18.15 in-in in 8.351 Saltbr-in 2.7255 HRD-in -68.62, -45.57 65.7, 16.55 in-in-out SNCiio in-out ActLoopNT-in 2.9248 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.94, 165.33 APE9-dihe-na 76.34, 152.28 APE8-dihe-in -69.82, 130.62 APE8-rot-out 176.66 APE67-dihe-in -58.68, -26.71 -39.69, -56.4 APE12-dist-in 13.2799 APE11-dist-in 11.7578 APE10-dist-in 7.0929 APE9-dist-in 3.1547 None PTR216 PTR216 XRAY 2.11 0.221 0.247 A 359.0 332.0 13 27 27 0 [[56, 340]] 1.0 9pe9 CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9PE9B P49841 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.0575 14.2183 BLAminus -128.76, -179.81 59.6, 84.42 -97.78, 27.09 283.79, 74.38 -73.25, -17.71 in-in in 8.3532 Saltbr-in 2.7132 HRD-in -68.49, -44.82 64.55, 18.32 in-in-out SNCiio in-out ActLoopNT-in 2.9402 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.27, 163.74 APE9-dihe-na 77.64, 152.05 APE8-dihe-in -69.14, 130.82 APE8-rot-out 177.12 APE67-dihe-in -58.92, -26.81 -39.96, -55.88 APE12-dist-in 13.3604 APE11-dist-in 11.8241 APE10-dist-in 7.1609 APE9-dist-in 3.1723 None PTR216 PTR216 XRAY 2.11 0.221 0.247 B 359.0 332.0 13 27 27 0 [[56, 340]] 1.0 9pe9 CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7Z1FA P49841 28 383 420.0 3NG:60401 Type1 Inactive DFGin 7.1722 14.3874 BLAminus -140.61, -172.17 56.83, 67.31 -90.44, 24.59 283.96, 78.9 -70.58, -34.2 in-in in 8.5891 Saltbr-in 2.7064 HRD-in -70.71, -48.08 68.23, 20.67 in-in-out SNCiio in-out ActLoopNT-in 2.8765 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -121.77, -56.1 APE9-dihe-na -73.95, 173.6 APE8-dihe-in -71.54, 133.95 APE8-rot-out 205.24 APE67-dihe-in -54.78, -22.55 -52.86, -47.6 APE12-dist-in 13.7113 APE11-dist-in 11.9213 APE10-dist-in 7.2574 APE9-dist-in 3.4781 None PTR216 PTR216 XRAY 3.0 0.224 0.249 A 364.0 354.0 2 27 27 0 [[56, 340]] 1.0 7z1f CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 7Z1FB P49841 38 382 420.0 3NG:60401 Type1 Inactive DFGin 6.8696 14.4685 BLAminus -141.12, -171.82 52.8, 73.11 -90.49, 20.89 285.47, 81.84 -62.59, -35.1 in-in in 9.0255 Saltbr-in 2.7633 HRD-in -68.41, -52.97 70.54, 14.05 in-in-out SNCiio in-out ActLoopNT-in 3.0394 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.34, -53.99 APE9-dihe-na -75.88, 165.71 APE8-dihe-in -64.92, 136.76 APE8-rot-out 179.7 APE67-dihe-in -58.44, -19.64 -54.95, -47.33 APE12-dist-in 13.527 APE11-dist-in 11.8588 APE10-dist-in 7.1538 APE9-dist-in 3.5583 None PTR216 PTR216 XRAY 3.0 0.224 0.249 B 364.0 321.0 24 27 27 0 [[56, 340]] 1.0 7z1f CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8AV1A P49841 27 381 420.0 O9L:406 Type1 Inactive DFGin 7.0048 13.8018 BLAminus -134.83, 176.12 61.29, 85.31 -97.92, 27.58 284.57, 74.39 -70.18, -20.31 in-in in 8.4199 Saltbr-in 2.6588 HRD-in -72.82, -53.06 75.09, 11.93 in-in-out SNCiio in-out ActLoopNT-in 2.8108 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -162.3, 153.55 APE9-dihe-na 79.71, 140.85 APE8-dihe-in -55.94, 133.71 APE8-rot-out 187.25 APE67-dihe-in -61.14, -25.49 -46.06, -52.45 APE12-dist-in 13.2676 APE11-dist-in 11.4128 APE10-dist-in 6.8843 APE9-dist-in 3.0607 None PTR216 PTR216 XRAY 2.15 0.18 0.21 A 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8av1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8AV1B P49841 27 381 420.0 O9L:405 Type1 Inactive DFGin 7.0411 13.8178 BLAminus -134.53, 176.17 61.15, 83.84 -96.42, 28.03 285.62, 75.68 -72.4, -19.61 in-in in 8.3507 Saltbr-in 2.6481 HRD-in -70.84, -52.05 73.58, 16.86 in-in-out SNCiio in-out ActLoopNT-in 2.809 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.36, 152.7 APE9-dihe-na 82.35, 142.4 APE8-dihe-in -57.42, 133.83 APE8-rot-out 184.71 APE67-dihe-in -59.68, -24.96 -48.86, -51.78 APE12-dist-in 13.2597 APE11-dist-in 11.441 APE10-dist-in 6.8498 APE9-dist-in 3.0597 None PTR216 PTR216 XRAY 2.15 0.18 0.21 B 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8av1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6GN1A P49841 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.9399 14.3347 BLAminus -135.29, 179.1 59.47, 89.49 -98.73, 29.98 286.18, 72.49 -75.74, -10.8 in-in in 8.608 Saltbr-in 3.0396 HRD-in -74.24, -44.22 64.59, 22.98 in-in-out SNCiio in-out ActLoopNT-in 2.9401 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -143.03, -18.16 APE9-dihe-na -103.04, 175.18 APE8-dihe-in -67.81, 136.03 APE8-rot-out 187.31 APE67-dihe-in -61.67, -27.65 -44.51, -52.79 APE12-dist-out 14.0101 APE11-dist-in 12.3553 APE10-dist-in 7.3869 APE9-dist-in 3.5875 None PTR216 PTR216 XRAY 2.6 0.224 0.259 A 368.0 340.0 8 27 27 0 [[56, 340]] 1.0 6gn1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6GN1B P49841 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.9439 14.317 BLAminus -135.3, 179.27 59.56, 89.49 -98.78, 30.1 286.37, 73.15 -75.82, -10.91 in-in in 8.6216 Saltbr-in 3.0339 HRD-in -74.17, -44.23 64.47, 22.86 in-in-out SNCiio in-out ActLoopNT-in 2.9462 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -129.39, -14.9 APE9-dihe-na -108.68, -179.33 APE8-dihe-in -68.02, 134.54 APE8-rot-out 210.75 APE67-dihe-in -62.25, -27.68 -44.3, -51.95 APE12-dist-out 14.0238 APE11-dist-in 12.1834 APE10-dist-in 7.4033 APE9-dist-in 3.6999 None PTR216 PTR216 XRAY 2.6 0.224 0.259 B 368.0 340.0 8 27 27 0 [[56, 340]] 1.0 6gn1 CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 2O5KA P49841 35 384 420.0 HBM:0 Type1 Inactive DFGin 6.7209 13.939 BLAminus -127.34, -179.9 54.97, 85.31 -97.88, 27.22 279.56, 72.26 -63.78, -54.26 in-in in 8.3524 Saltbr-in 3.3761 HRD-in -66.17, -47.55 59.21, 39.45 in-in-out SNCiio in-out ActLoopNT-in 2.9464 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_iiii APE10-dihe-na 170.93, -156.16 APE9-dihe-na 30.47, -152.36 APE8-dihe-out -134.5, -176.14 APE8-rot-in 306.82 APE67-dihe-in -73.05, -7.32 -59.58, -80.34 APE12-dist-in 12.6788 APE11-dist-in 9.1805 APE10-dist-in 5.885 APE9-dist-in 3.0373 None None None XRAY 3.2 0.251 0.309 A 372.0 350.0 0 27 27 0 [[56, 340]] 1.0 2o5k CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 1UV5A P49841 35 383 420.0 BRW:1383 Type1 Inactive DFGin 6.9015 14.0788 BLAminus -144.35, -177.14 59.35, 81.04 -94.26, 27.94 286.0, 72.94 -59.18, -36.48 in-in in 8.299 Saltbr-in 2.5611 HRD-in -65.61, -42.55 70.5, 0.98 in-in-out SNCiio in-out ActLoopNT-in 2.8842 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -98.47, 172.31 APE9-dihe-na 85.56, 133.89 APE8-dihe-in -66.16, 126.55 APE8-rot-out 191.14 APE67-dihe-in -61.71, -20.34 -21.78, -65.88 APE12-dist-in 12.7631 APE11-dist-in 10.9893 APE10-dist-in 5.7154 APE9-dist-in 3.2357 None None None XRAY 2.8 0.193 0.226 A 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 1uv5 CMGC_GSK3B_HUMAN CMGC 7.4e-70 241.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6GJOA P49841 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.1764 14.254 BLAminus -136.61, 169.82 63.4, 86.22 -103.46, 25.41 276.6, 83.48 -69.91, -39.25 in-in in 8.6359 Saltbr-in 2.8102 HRD-in -57.84, -41.83 58.98, 16.97 in-in-out SNCiio in-out ActLoopNT-in 3.0119 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.92, 162.15 APE9-dihe-na 71.93, 161.47 APE8-dihe-in -78.01, 132.19 APE8-rot-out 37.25 APE67-dihe-in -62.57, -18.8 -29.28, -56.31 APE12-dist-in 13.62 APE11-dist-in 11.8617 APE10-dist-in 6.9452 APE9-dist-in 3.4449 None None None XRAY 2.91 0.218 0.237 A 414.0 349.0 0 27 27 0 [[56, 340]] 1.0 6gjo CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 6GJOB P49841 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.4783 14.2513 BLAminus -136.82, 170.18 63.9, 83.46 -101.86, 22.92 278.62, 83.32 -68.81, -38.47 in-in in 8.4049 Saltbr-in 3.0839 HRD-in -57.78, -41.9 58.99, 17.22 in-in-out SNCiio in-out ActLoopNT-in 3.0124 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.67, 163.61 APE9-dihe-na 73.76, 161.78 APE8-dihe-in -77.57, 137.96 APE8-rot-out 184.23 APE67-dihe-in -62.17, -20.4 -36.29, -55.68 APE12-dist-in 13.4495 APE11-dist-in 11.7843 APE10-dist-in 6.8542 APE9-dist-in 3.4366 None None None XRAY 2.91 0.218 0.237 B 414.0 343.0 6 27 27 0 [[56, 340]] 1.0 6gjo CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 3M1SA P49841 35 385 420.0 DW1:421 Type1 Inactive DFGin 7.021 13.7099 BLAminus -149.21, -179.05 55.83, 87.87 -101.26, 23.04 292.92, 65.81 -62.39, -0.11 in-in in 8.7264 Saltbr-in 2.9756 HRD-in -71.98, -44.05 63.65, 18.92 in-in-out SNCiio in-out ActLoopNT-in 3.0324 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -100.39, 171.9 APE9-dihe-na 82.48, 144.37 APE8-dihe-in -94.3, 96.58 APE8-rot-in 285.71 APE67-dihe-out 116.42, -45.78 9.38, 103.41 APE12-dist-in 13.6493 APE11-dist-in 11.7091 APE10-dist-in 6.707 APE9-dist-in 3.4451 None None None XRAY 3.134 0.171 0.228 A 420.0 348.0 3 27 27 0 [[56, 340]] 1.0 3m1s CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 9HUKA P49841 25 385 420.0 A1IXL:501 Type1 Inactive DFGin 7.0533 14.0777 BLAminus -135.25, -177.02 57.0, 94.14 -110.6, 20.82 285.12, 72.82 -66.1, -13.46 in-out in 8.1101 Saltbr-out 3.6586 HRD-in -70.91, -39.46 63.28, 18.66 out-in-in SNCoii in-in ActLoopNT-in 3.1574 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 179.26 APE9-dihe-na 68.03, 135.17 APE8-dihe-in -69.47, 168.34 APE8-rot-in 295.64 APE67-dihe-inflip 67.51, -44.25 -66.67, 175.58 APE12-dist-in 13.1194 APE11-dist-in 10.9456 APE10-dist-in 5.924 APE9-dist-in 3.2016 None None None XRAY 3.5 0.219 0.25 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9huk CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4J71A P49841 36 383 420.0 1JX:501 Type1 Inactive DFGin 6.9292 14.0341 BLAminus -134.37, 178.91 60.63, 80.22 -96.96, 24.92 284.72, 75.18 -68.29, -15.66 in-in in 8.4479 Saltbr-in 3.0956 HRD-in -74.9, -47.0 72.06, 4.98 in-in-out SNCiio in-out ActLoopNT-in 2.7141 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.32, 163.35 APE9-dihe-na 76.45, 151.25 APE8-dihe-in -65.19, 140.55 APE8-rot-out 188.84 APE67-dihe-in -55.99, -28.06 -50.85, -54.43 APE12-dist-in 13.3964 APE11-dist-in 11.8958 APE10-dist-in 7.1633 APE9-dist-in 2.9983 None PTR216 PTR216 XRAY 2.31 0.191 0.234 A 424.0 348.0 0 27 27 0 [[56, 340]] 1.0 4j71 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4J71B P49841 36 383 420.0 1JX:501 Type1 Inactive DFGin 7.043 13.8316 BLAminus -140.62, 179.7 59.87, 90.62 -104.73, 25.33 288.76, 76.25 -66.71, -17.33 in-in in 8.3305 Saltbr-in 2.8961 HRD-in -77.92, -46.29 72.36, 3.7 in-in-out SNCiio in-out ActLoopNT-in 2.834 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.74, 169.96 APE9-dihe-na 69.52, 149.79 APE8-dihe-in -68.04, 134.18 APE8-rot-out 173.06 APE67-dihe-in -53.62, -29.43 -43.81, -55.09 APE12-dist-in 13.2129 APE11-dist-in 11.9572 APE10-dist-in 7.1265 APE9-dist-in 2.9738 None PTR216 PTR216 XRAY 2.31 0.191 0.234 B 424.0 348.0 0 27 27 0 [[56, 340]] 1.0 4j71 CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5HLNB P49841 37 383 420.0 65C:501 Type1 Inactive DFGin 6.8475 13.3316 BLAminus -143.06, -174.61 53.09, 90.34 -103.45, 33.01 288.97, 83.64 -74.69, -34.84 in-in in 8.9958 Saltbr-in 2.6044 HRD-in -68.15, -40.04 65.1, 19.28 in-in-out SNCiio in-out ActLoopNT-in 2.9629 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -137.65, -62.86 APE9-dihe-na -78.36, 171.11 APE8-dihe-in -56.52, 151.93 APE8-rot-out 161.85 APE67-dihe-in -56.43, -28.42 -72.24, -45.62 APE12-dist-in 13.5983 APE11-dist-in 11.8341 APE10-dist-in 7.3737 APE9-dist-in 3.4156 None PTR216 PTR216 XRAY 3.1 0.173 0.236 B 424.0 347.0 0 27 27 0 [[56, 340]] 1.0 5hln CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 5OY4B P49841 30 384 420.0 B4K:502 Type1.5_Back Inactive DFGin 7.0077 13.7409 BLAminus -131.51, 177.88 58.43, 85.84 -94.85, 21.53 281.4, 81.96 -63.5, -26.63 in-in in 7.965 Saltbr-in 2.7509 HRD-in -68.43, -44.24 63.59, 14.9 in-in-out SNCiio in-out ActLoopNT-in 2.8689 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -145.82, 158.71 APE9-dihe-na 86.22, 156.23 APE8-dihe-in -75.92, 122.37 APE8-rot-out 226.12 APE67-dihe-in -60.14, -24.48 -28.85, -54.97 APE12-dist-in 13.5037 APE11-dist-in 11.6211 APE10-dist-in 7.0093 APE9-dist-in 3.404 None PTR216 PTR216 XRAY 3.2 0.196 0.229 B 420.0 354.0 1 27 27 0 [[56, 340]] 1.0 5oy4 CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 8QJIA P49841 36 381 420.0 VNG:401 Type1 Inactive DFGin 6.9495 14.1959 None -92.57, -90.5 -72.82, 155.73 -144.36, 17.02 276.05, 102.26 -73.85, -19.5 in-in in 8.3845 Saltbr-in 2.6943 HRD-in -65.27, -43.08 63.67, 22.78 in-in-out SNCiio in-out ActLoopNT-in 3.34 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -115.54, 179.17 APE9-dihe-na 65.4, 161.24 APE8-dihe-in -68.89, 150.02 APE8-rot-out 175.4 APE67-dihe-in -64.21, -18.12 -58.7, -47.99 APE12-dist-in 13.3857 APE11-dist-in 12.0024 APE10-dist-in 7.07 APE9-dist-in 3.4473 None PTR216 PTR216 XRAY 3.02 0.253 0.289 A 364.0 340.0 6 27 27 0 [[56, 340]] 1.0 8qji CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B 4DITA P49841 35 387 420.0 0KD:501 Type1 None DFGin 6.8051 13.9479 BLAminus -145.37, 179.76 65.92, 81.37 -105.97, 22.54 288.96, 82.14 -68.29, -17.95 in-in in 8.8255 Saltbr-in 2.717 HRD-in -69.87, -50.6 73.87, 5.2 in-in-none SNCiin in-none ActLoopNT-in 2.9388 ActLoopCT-none nonTYR APEdihe_aannn APEdist_iinn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 14.5 999.0, 999.0 APE12-dist-in 13.4889 APE11-dist-in 10.3847 APE10-dist-none 999.0 APE9-dist-none 999.0 None PTR216 PTR216 XRAY 2.6 0.243 0.304 A 382.0 329.0 24 27 23 4 [[56, 340]] 1.0 4dit CMGC_GSK3B_HUMAN CMGC 2.4e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta

CMGC_GSK3B (Glycogen synthase kinase-3 beta)

Total number of chains: 193
Active chains: 149
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 189 97.9% AF-P49841-K1A
DFGin ABAminus 3 1.6% 5AIRA
DFGin None 1 0.5% 8QJIA

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GSK3B GSK3B_HUMAN 4NM5A P49841 24 383 420.0 ADP:60401 ATPlike Active DFGin 6.5502 14.0064 BLAminus -136.16, -177.73 61.88, 88.47 -108.64, 28.76 287.87, 80.78 -73.66, -15.44 in-in in 8.6187 Saltbr-in 2.6732 HRD-in -65.83, -43.73 64.82, 15.23 in-in-in SNCiii in-in ActLoopNT-in 2.8386 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.92, 173.97 APE9-dihe-na 66.26, 147.02 APE8-dihe-in -77.1, 152.8 APE8-rot-in 293.28 APE67-dihe-inflip 82.03, -25.76 -52.23, 150.7 APE12-dist-in 13.2793 APE11-dist-in 11.5989 APE10-dist-in 6.9485 APE9-dist-in 3.2377 None None None XRAY 2.3 0.185 0.232 A 377.0 360.0 0 27 27 0 [[56, 340]] 1.0 4nm5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4NM7A P49841 25 383 420.0 ADP:60401 ATPlike Active DFGin 6.5153 13.993 BLAminus -137.35, -178.06 62.82, 88.6 -107.3, 24.56 288.41, 80.2 -69.84, -12.63 in-in in 8.8181 Saltbr-in 2.743 HRD-in -66.5, -46.64 67.84, 11.79 in-in-in SNCiii in-in ActLoopNT-in 2.8287 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.92, 172.54 APE9-dihe-na 68.99, 153.43 APE8-dihe-in -86.9, 151.79 APE8-rot-in 300.04 APE67-dihe-inflip 84.67, -25.93 -50.38, 146.2 APE12-dist-in 13.3553 APE11-dist-in 11.6779 APE10-dist-in 6.9055 APE9-dist-in 3.2102 None None None XRAY 2.3 0.185 0.234 A 377.0 354.0 2 27 27 0 [[56, 340]] 1.0 4nm7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4NM3A P49841 6 383 420.0 ADP:60409 ATPlike Active DFGin 6.4747 13.947 BLAminus -129.98, -178.05 63.17, 87.87 -103.96, 21.26 289.38, 80.04 -65.46, -16.35 in-in in 8.8058 Saltbr-in 2.7256 HRD-in -69.81, -46.77 71.59, 6.75 in-in-in SNCiii in-in ActLoopNT-in 2.7503 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.34, 169.99 APE9-dihe-na 69.15, 146.37 APE8-dihe-in -83.47, 151.55 APE8-rot-in 296.54 APE67-dihe-inflip 86.0, -31.11 -49.79, 146.79 APE12-dist-in 13.2688 APE11-dist-in 11.4837 APE10-dist-in 6.9065 APE9-dist-in 3.1117 None SEP9 SEP9 XRAY 2.1 0.197 0.242 A 389.0 357.0 2 27 27 0 [[56, 340]] 1.0 4nm3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1J1BA P49841 35 388 420.0 ANP:60430 ATPlike Active DFGin 6.7667 13.7876 BLAminus -136.8, -178.88 61.6, 83.12 -97.64, 25.1 286.09, 80.4 -68.7, -13.11 in-in in 8.5659 Saltbr-in 2.59 HRD-in -71.16, -45.98 70.36, 3.88 in-in-in SNCiii in-in ActLoopNT-in 3.0085 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.52, 175.26 APE9-dihe-na 75.44, 133.64 APE8-dihe-in -75.76, 147.49 APE8-rot-in 306.57 APE67-dihe-inflip 98.15, -33.72 -56.43, 141.52 APE12-dist-in 13.0562 APE11-dist-in 10.9736 APE10-dist-in 5.8926 APE9-dist-in 3.1122 None None None XRAY 1.8 0.216 0.242 A 420.0 354.0 0 27 27 0 [[56, 340]] 1.0 1j1b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1J1BB P49841 23 386 420.0 ANP:60930 ATPlike Active DFGin 6.6091 13.6686 BLAminus -136.4, -177.03 61.49, 81.88 -98.08, 27.2 288.49, 82.07 -71.33, -13.14 in-in in 8.4573 Saltbr-in 2.713 HRD-in -67.51, -45.87 68.87, 6.43 in-in-in SNCiii in-in ActLoopNT-in 2.9624 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.88, 174.17 APE9-dihe-na 76.18, 138.08 APE8-dihe-in -76.12, 141.41 APE8-rot-in 301.11 APE67-dihe-inflip 98.0, -37.59 -54.78, 144.25 APE12-dist-in 12.9784 APE11-dist-in 11.0659 APE10-dist-in 6.0113 APE9-dist-in 3.1744 None None None XRAY 1.8 0.216 0.242 B 420.0 364.0 0 27 27 0 [[56, 340]] 1.0 1j1b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1J1CA P49841 35 388 420.0 ADP:60430 ATPlike Active DFGin 6.8122 13.9298 BLAminus -139.24, -179.75 62.79, 82.17 -97.34, 25.19 286.68, 82.3 -65.83, -19.9 in-in in 8.6015 Saltbr-in 2.6465 HRD-in -68.65, -43.85 68.34, 7.36 in-in-in SNCiii in-in ActLoopNT-in 2.9774 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.05, 172.96 APE9-dihe-na 78.17, 130.85 APE8-dihe-in -73.54, 145.97 APE8-rot-in 310.16 APE67-dihe-inflip 99.09, -35.01 -54.43, 141.28 APE12-dist-in 13.0771 APE11-dist-in 11.0674 APE10-dist-in 5.9263 APE9-dist-in 3.1997 None None None XRAY 2.1 0.218 0.242 A 420.0 354.0 0 27 27 0 [[56, 340]] 1.0 1j1c Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1J1CB P49841 23 386 420.0 ADP:60930 ATPlike Active DFGin 6.6935 13.7094 BLAminus -138.27, -179.99 63.33, 82.68 -100.46, 28.2 289.88, 80.26 -70.45, -13.94 in-in in 8.52 Saltbr-in 2.738 HRD-in -67.92, -43.36 67.59, 5.86 in-in-in SNCiii in-in ActLoopNT-in 2.9803 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.71, 170.27 APE9-dihe-na 78.71, 139.86 APE8-dihe-in -81.56, 140.05 APE8-rot-in 302.5 APE67-dihe-inflip 101.62, -36.53 -50.52, 137.44 APE12-dist-in 12.8683 APE11-dist-in 11.1277 APE10-dist-in 6.0252 APE9-dist-in 3.2076 None None None XRAY 2.1 0.218 0.242 B 420.0 364.0 0 27 27 0 [[56, 340]] 1.0 1j1c Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8XN6A P49841 35 384 420.0 ANP:501 ATPlike Active DFGin 6.682 13.8624 BLAminus -137.72, 173.39 67.73, 84.48 -99.84, 22.57 287.77, 80.54 -65.33, -24.58 in-in in 8.4632 Saltbr-in 2.6302 HRD-in -71.05, -47.88 67.82, 15.5 in-in-in SNCiii in-in ActLoopNT-in 3.0543 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.0, 164.43 APE9-dihe-na 85.44, 135.36 APE8-dihe-in -74.2, 151.55 APE8-rot-in 291.81 APE67-dihe-in -69.28, -17.83 -36.59, -67.98 APE12-dist-in 12.9066 APE11-dist-in 10.7867 APE10-dist-in 5.6801 APE9-dist-in 3.1824 None None None XRAY 2.4 0.194 0.242 A 421.0 350.0 0 27 27 0 [[56, 340]] 1.0 8xn6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1PYXA P49841 35 386 420.0 ANP:1001 ATPlike Active DFGin 6.5838 13.6216 BLAminus -138.81, -178.07 65.18, 79.92 -98.83, 26.07 289.95, 78.27 -73.24, -7.6 in-in in 8.3727 Saltbr-in 2.7648 HRD-in -67.79, -47.84 71.28, 6.53 in-in-in SNCiii in-in ActLoopNT-in 2.9483 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.12, 170.17 APE9-dihe-na 80.64, 129.74 APE8-dihe-in -63.79, 140.05 APE8-rot-in 299.48 APE67-dihe-in -56.43, -21.61 -20.65, -80.28 APE12-dist-in 12.9032 APE11-dist-in 10.9366 APE10-dist-in 5.7841 APE9-dist-in 3.1495 None None None XRAY 2.4 0.206 0.233 A 422.0 343.0 9 27 27 0 [[56, 340]] 1.0 1pyx Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1PYXB P49841 35 383 420.0 ANP:2001 ATPlike Active DFGin 6.5927 13.7178 BLAminus -140.94, -178.47 65.26, 79.98 -98.11, 22.32 290.75, 76.51 -68.32, -7.73 in-in in 8.4877 Saltbr-in 2.6657 HRD-in -69.98, -47.18 70.83, 5.6 in-in-in SNCiii in-in ActLoopNT-in 2.9383 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.3, 169.41 APE9-dihe-na 81.27, 131.24 APE8-dihe-in -66.67, 140.79 APE8-rot-in 300.74 APE67-dihe-in -56.9, -22.2 -20.58, -79.9 APE12-dist-in 12.8382 APE11-dist-in 10.8615 APE10-dist-in 5.7183 APE9-dist-in 3.132 None None None XRAY 2.4 0.206 0.233 B 422.0 338.0 11 27 27 0 [[56, 340]] 1.0 1pyx Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN AF-P49841-K1A P49841 48 348 420.0 No_ligand No_ligand Active DFGin 6.7843 14.0695 BLAminus -132.22, 178.4 62.95, 68.76 -81.18, 15.79 285.47, 79.99 -60.59, -34.48 in-in in 8.4747 Saltbr-in 2.7102 HRD-in -72.93, -43.95 66.08, 11.33 in-in-in SNCiii in-in ActLoopNT-in 2.8921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.31, 173.16 APE9-dihe-na 65.7, 144.93 APE8-dihe-in -63.41, 136.54 APE8-rot-in 298.96 APE67-dihe-in -66.32, -15.33 -50.7, -49.59 APE12-dist-in 13.4502 APE11-dist-in 11.9889 APE10-dist-in 6.9958 APE9-dist-in 3.1274 None None None AF2 -1.0 1.0 1.0 A 301.0 301.0 0 27 27 0 [[56, 340]] 1.0 AF-P49841-K1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN AF-P49841-K3A P49841 48 348 420.0 No_ligand No_ligand Active DFGin 6.5244 13.8836 BLAminus -137.65, -179.24 64.43, 60.31 -74.11, 11.79 288.76, 87.67 -59.53, -33.87 in-in in 8.2321 Saltbr-in 2.6752 HRD-in -76.11, -42.33 64.92, 19.4 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, -179.86 APE9-dihe-na 61.35, 145.02 APE8-dihe-in -62.21, 135.58 APE8-rot-in 295.17 APE67-dihe-in -63.79, -15.52 -52.47, -50.54 APE12-dist-in 13.4857 APE11-dist-in 11.9949 APE10-dist-in 7.0698 APE9-dist-in 3.244 None None None AF2 -1.0 1.0 1.0 A 301.0 301.0 0 27 27 0 [[56, 340]] 1.0 AF-P49841-K3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1e-70 244.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1GNGA P49841 36 385 420.0 No_ligand No_ligand Active DFGin 6.8854 14.0642 BLAminus -143.26, -176.0 52.72, 77.37 -90.17, 24.13 284.09, 64.37 -57.11, -28.67 in-in in 7.9042 Saltbr-in 2.9159 HRD-in -73.29, -39.28 60.06, 11.92 in-in-in SNCiii in-in ActLoopNT-in 2.8439 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.61, 159.4 APE9-dihe-na 81.31, 139.52 APE8-dihe-in -59.26, 125.44 APE8-rot-in 312.57 APE67-dihe-in -52.62, -25.58 -28.83, -64.47 APE12-dist-in 13.5503 APE11-dist-in 11.9569 APE10-dist-in 7.016 APE9-dist-in 3.1105 None PTR216 PTR216 XRAY 2.6 0.196 0.262 A 378.0 350.0 0 27 27 0 [[56, 340]] 1.0 1gng Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1GNGB P49841 28 384 420.0 No_ligand No_ligand Active DFGin 7.075 14.1431 BLAminus -137.26, -174.12 57.41, 76.0 -92.3, 24.73 292.83, 74.1 -62.54, -16.26 in-in in 8.1028 Saltbr-in 2.801 HRD-in -56.65, -46.78 67.13, 3.53 in-in-in SNCiii in-in ActLoopNT-in 3.0528 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.46, 162.71 APE9-dihe-na 73.79, 160.3 APE8-dihe-in -71.09, 143.31 APE8-rot-in 306.45 APE67-dihe-in -62.51, -22.51 -44.24, -51.03 APE12-dist-in 13.4613 APE11-dist-in 11.7372 APE10-dist-in 7.2333 APE9-dist-in 3.2921 None PTR216 PTR216 XRAY 2.6 0.196 0.262 B 378.0 357.0 0 27 27 0 [[56, 340]] 1.0 1gng Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.3e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1H8FA P49841 35 386 420.0 No_ligand No_ligand Active DFGin 7.0053 14.4673 BLAminus -132.29, -174.92 54.46, 76.42 -91.57, 20.83 287.85, 73.58 -61.47, -17.91 in-in in 8.8115 Saltbr-in 2.6295 HRD-in -65.88, -45.02 68.7, 5.89 in-in-in SNCiii in-in ActLoopNT-in 3.0299 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.85, 172.29 APE9-dihe-na 81.77, 142.51 APE8-dihe-in -88.0, 149.96 APE8-rot-in 300.12 APE67-dihe-in -68.04, -14.11 -16.17, -79.65 APE12-dist-in 12.8766 APE11-dist-in 10.8744 APE10-dist-in 5.7937 APE9-dist-in 3.0888 None None None XRAY 2.8 0.22 0.256 A 352.0 352.0 0 27 27 0 [[56, 340]] 1.0 1h8f Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1H8FB P49841 35 384 420.0 No_ligand No_ligand Active DFGin 7.053 14.4881 BLAminus -137.11, -175.26 54.49, 79.79 -96.15, 19.99 284.33, 74.24 -61.84, -16.45 in-in in 8.7842 Saltbr-in 2.6311 HRD-in -65.99, -45.44 68.05, 7.58 in-in-in SNCiii in-in ActLoopNT-in 2.9921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.76, 172.7 APE9-dihe-na 81.11, 140.51 APE8-dihe-in -87.0, 149.5 APE8-rot-in 302.15 APE67-dihe-in -67.01, -11.3 -16.16, -82.04 APE12-dist-in 12.8754 APE11-dist-in 10.8434 APE10-dist-in 5.7606 APE9-dist-in 3.101 None None None XRAY 2.8 0.22 0.256 B 352.0 350.0 0 27 27 0 [[56, 340]] 1.0 1h8f Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.6e-69 240.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1I09A P49841 25 384 420.0 No_ligand No_ligand Active DFGin 6.9144 14.1487 BLAminus -130.79, -175.77 55.31, 78.24 -94.52, 21.05 292.59, 69.56 -64.23, -6.99 in-in in 8.5205 Saltbr-in 2.7631 HRD-in -66.04, -49.2 76.06, -6.11 in-in-in SNCiii in-in ActLoopNT-in 3.0217 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.67, -13.88 APE9-dihe-na -95.25, 153.25 APE8-dihe-in -66.11, 146.74 APE8-rot-in 277.64 APE67-dihe-in -57.92, -5.44 -43.43, -74.88 APE12-dist-in 12.9676 APE11-dist-in 11.1602 APE10-dist-in 5.9721 APE9-dist-in 3.3336 None None None XRAY 2.7 0.242 0.274 A 420.0 338.0 22 27 27 0 [[56, 340]] 1.0 1i09 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U2ZA P49841 35 382 420.0 L7C:401 Type1 Active DFGin 7.0437 14.3283 BLAminus -133.1, 179.76 62.32, 79.84 -96.99, 23.84 285.42, 79.62 -65.82, -25.41 in-in in 8.5578 Saltbr-in 2.7638 HRD-in -73.49, -48.13 70.69, 16.81 in-in-in SNCiii in-in ActLoopNT-in 2.9072 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.38, 169.05 APE9-dihe-na 81.0, 139.13 APE8-dihe-in -79.34, 150.41 APE8-rot-in 288.38 APE67-dihe-inflip 98.4, -32.71 -58.44, 134.12 APE12-dist-in 13.1383 APE11-dist-in 11.05 APE10-dist-in 5.8885 APE9-dist-in 3.0925 None None None XRAY 2.21 0.248 0.266 A 348.0 345.0 3 27 27 0 [[56, 340]] 1.0 7u2z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U2ZB P49841 35 382 420.0 L7C:401 Type1 Active DFGin 7.0832 14.3162 BLAminus -133.0, 179.81 61.72, 80.12 -97.27, 23.94 285.32, 79.23 -65.78, -25.41 in-in in 8.5159 Saltbr-in 2.7654 HRD-in -73.41, -48.27 70.6, 17.33 in-in-in SNCiii in-in ActLoopNT-in 2.9123 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.19, 168.84 APE9-dihe-na 80.53, 139.96 APE8-dihe-in -79.72, 154.04 APE8-rot-in 288.98 APE67-dihe-in -82.66, -15.29 -42.95, -55.79 APE12-dist-in 13.132 APE11-dist-in 11.0815 APE10-dist-in 5.8924 APE9-dist-in 3.0994 None None None XRAY 2.21 0.248 0.266 B 348.0 348.0 0 27 27 0 [[56, 340]] 1.0 7u2z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3F7ZB P49841 35 383 420.0 34O:63000 Type1 Active DFGin 7.0223 13.8784 BLAminus -136.68, -179.55 57.9, 84.9 -98.68, 23.48 283.23, 74.81 -68.95, -21.14 in-in in 8.4241 Saltbr-in 2.704 HRD-in -69.78, -45.02 65.34, 14.6 in-in-in SNCiii in-in ActLoopNT-in 2.8686 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.88, 179.92 APE9-dihe-na 68.48, 153.11 APE8-dihe-in -69.08, 139.27 APE8-rot-in 289.99 APE67-dihe-in -60.9, -22.52 -35.36, -58.5 APE12-dist-in 13.6463 APE11-dist-in 11.9538 APE10-dist-in 6.7778 APE9-dist-in 3.2477 None PTR216 PTR216 XRAY 2.4 0.206 0.253 B 350.0 339.0 10 27 27 0 [[56, 340]] 1.0 3f7z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3SD0B P49841 35 383 420.0 TSK:400 Type1 Active DFGin 7.1882 14.0242 BLAminus -142.24, -171.3 46.91, 83.25 -91.85, 32.36 285.89, 73.19 -82.63, -8.9 in-in in 8.2345 Saltbr-in 2.887 HRD-in -76.13, -44.58 70.79, 3.58 in-in-in SNCiii in-in ActLoopNT-in 2.8942 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.6, 179.93 APE9-dihe-na 74.21, 152.1 APE8-dihe-in -107.68, 155.88 APE8-rot-in 296.61 APE67-dihe-in -78.55, -3.01 -13.04, -81.61 APE12-dist-in 13.0175 APE11-dist-in 11.0989 APE10-dist-in 6.1509 APE9-dist-in 3.1559 None None None XRAY 2.7 0.179 0.254 B 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 3sd0 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6HK3B P49841 35 384 420.0 G8B:401 Type1 Active DFGin 6.7879 13.6408 BLAminus -137.2, -177.06 49.94, 95.88 -103.42, 19.32 279.02, 79.18 -69.5, -12.66 in-in in 8.1675 Saltbr-in 2.6023 HRD-in -82.47, -44.32 66.17, 21.49 in-in-in SNCiii in-in ActLoopNT-in 2.8186 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -116.65, -179.5 APE9-dihe-na 72.73, 150.58 APE8-dihe-in -63.57, 140.77 APE8-rot-in 271.9 APE67-dihe-in -55.77, -29.98 -51.2, -52.31 APE12-dist-in 13.4077 APE11-dist-in 11.6419 APE10-dist-in 6.3651 APE9-dist-in 3.2489 None PTR216 PTR216 XRAY 2.35 0.206 0.234 B 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6HK4A P49841 35 384 420.0 G8E:408 Type1 Active DFGin 6.9285 13.5081 BLAminus -141.9, -175.7 56.05, 83.18 -94.87, 22.99 284.64, 79.88 -61.73, -17.34 in-in in 8.3712 Saltbr-in 2.6563 HRD-in -76.65, -40.11 61.36, 16.95 in-in-in SNCiii in-in ActLoopNT-in 2.9232 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.26, 167.76 APE9-dihe-na 63.34, 157.04 APE8-dihe-in -69.05, 135.63 APE8-rot-in 300.42 APE67-dihe-in -54.24, -34.87 -29.95, -58.61 APE12-dist-in 13.2335 APE11-dist-in 11.745 APE10-dist-in 7.1618 APE9-dist-in 3.1917 None PTR216 PTR216 XRAY 2.5 0.212 0.249 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6HK4B P49841 35 384 420.0 G8E:409 Type1 Active DFGin 6.9427 13.5412 BLAminus -140.37, -179.48 60.09, 87.67 -101.02, 22.8 284.5, 76.31 -75.88, -10.96 in-in in 8.2076 Saltbr-in 2.5056 HRD-in -82.4, -45.58 68.54, 13.94 in-in-in SNCiii in-in ActLoopNT-in 2.9046 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.02, 172.84 APE9-dihe-na 63.46, 139.74 APE8-dihe-in -57.57, 136.79 APE8-rot-in 295.89 APE67-dihe-in -60.79, -29.87 -46.27, -47.23 APE12-dist-in 13.2677 APE11-dist-in 11.6783 APE10-dist-in 6.8983 APE9-dist-in 3.0744 None PTR216 PTR216 XRAY 2.5 0.212 0.249 B 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5F94A P49841 36 381 420.0 3UO:401 Type1 Active DFGin 6.9408 13.7851 BLAminus -132.23, -171.99 59.12, 80.79 -95.82, 23.07 289.16, 72.98 -56.52, -34.28 in-in in 8.4861 Saltbr-in 2.7108 HRD-in -71.8, -46.49 68.5, 7.3 in-in-in SNCiii in-in ActLoopNT-in 2.7841 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.99, 174.92 APE9-dihe-na 77.27, 148.67 APE8-dihe-in -101.45, 151.47 APE8-rot-in 289.94 APE67-dihe-inflip 89.58, -29.34 -36.24, 131.42 APE12-dist-in 12.915 APE11-dist-in 10.9124 APE10-dist-in 5.9524 APE9-dist-in 3.1086 None None None XRAY 2.51 0.191 0.226 A 350.0 346.0 0 27 27 0 [[56, 340]] 1.0 5f94 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5F94B P49841 37 385 420.0 3UO:401 Type1 Active DFGin 6.9206 13.9028 BLAminus -131.5, -174.71 60.13, 82.54 -97.18, 23.01 287.88, 72.62 -56.23, -35.38 in-in in 8.3979 Saltbr-in 2.8901 HRD-in -70.35, -45.36 66.02, 7.89 in-in-in SNCiii in-in ActLoopNT-in 2.8563 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.68, 174.32 APE9-dihe-na 79.06, 151.27 APE8-dihe-in -105.02, 147.7 APE8-rot-in 292.84 APE67-dihe-inflip 87.17, -28.31 -40.05, 137.25 APE12-dist-in 12.8868 APE11-dist-in 10.9014 APE10-dist-in 5.8663 APE9-dist-in 3.1931 None None None XRAY 2.51 0.191 0.226 B 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 5f94 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5F95A P49841 36 383 420.0 3UP:401 Type1 Active DFGin 6.8507 14.1212 BLAminus -131.03, -172.49 54.11, 85.8 -99.54, 23.42 287.04, 73.17 -58.21, -30.13 in-in in 8.4923 Saltbr-in 2.6419 HRD-in -68.05, -46.73 71.39, 6.88 in-in-in SNCiii in-in ActLoopNT-in 2.8734 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.52, 167.77 APE9-dihe-na 81.86, 152.62 APE8-dihe-in -108.33, 161.23 APE8-rot-in 296.59 APE67-dihe-in -81.75, 2.56 -4.13, -93.98 APE12-dist-in 13.0998 APE11-dist-in 11.0871 APE10-dist-in 6.3777 APE9-dist-in 3.2624 None None None XRAY 2.525 0.204 0.242 A 350.0 345.0 3 27 27 0 [[56, 340]] 1.0 5f95 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5F95B P49841 36 385 420.0 3UP:401 Type1 Active DFGin 7.0295 14.1311 BLAminus -130.15, -170.55 52.93, 82.9 -96.95, 23.47 283.9, 71.07 -57.67, -29.42 in-in in 8.5241 Saltbr-in 2.2415 HRD-in -68.94, -45.23 69.65, 6.25 in-in-in SNCiii in-in ActLoopNT-in 3.0094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.14, 169.18 APE9-dihe-na 82.46, 143.88 APE8-dihe-in -96.17, 168.5 APE8-rot-in 296.7 APE67-dihe-in -78.34, 2.06 -36.18, -73.12 APE12-dist-in 13.0212 APE11-dist-in 11.0271 APE10-dist-in 6.0921 APE9-dist-in 3.2102 None None None XRAY 2.525 0.204 0.242 B 350.0 338.0 12 27 27 0 [[56, 340]] 1.0 5f95 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U31A P49841 36 385 420.0 L7I:402 Type1 Active DFGin 7.0942 14.1832 BLAminus -142.39, 178.42 62.99, 82.78 -98.0, 19.46 288.1, 81.67 -57.1, -32.73 in-in in 8.1645 Saltbr-in 2.8395 HRD-in -76.17, -49.99 76.15, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.9293 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.54, -23.16 APE9-dihe-na -100.68, 154.06 APE8-dihe-in -79.73, 162.4 APE8-rot-in 294.75 APE67-dihe-in -75.9, -12.27 -44.4, -68.17 APE12-dist-in 13.1024 APE11-dist-in 10.9281 APE10-dist-in 5.9089 APE9-dist-in 3.4164 None None None XRAY 2.38 0.244 0.276 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 7u31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U31B P49841 37 382 420.0 L7I:402 Type1 Active DFGin 7.0487 14.2873 BLAminus -143.88, 177.54 62.09, 82.63 -98.02, 19.8 287.95, 82.15 -57.33, -32.15 in-in in 8.3774 Saltbr-in 2.7171 HRD-in -76.73, -50.12 75.35, 8.49 in-in-in SNCiii in-in ActLoopNT-in 2.9329 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.33, 167.82 APE9-dihe-na 83.33, 132.28 APE8-dihe-in -83.68, 163.51 APE8-rot-in 292.75 APE67-dihe-in -76.54, -11.97 -40.44, -69.75 APE12-dist-in 13.1082 APE11-dist-in 10.9788 APE10-dist-in 5.927 APE9-dist-in 3.1265 None None None XRAY 2.38 0.244 0.276 B 350.0 346.0 0 27 27 0 [[56, 340]] 1.0 7u31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7SXJA P49841 34 383 420.0 6VL:60401 Type1 Active DFGin 6.916 14.335 BLAminus -142.41, -179.99 59.67, 72.96 -86.59, 25.21 285.68, 73.81 -69.07, -21.65 in-in in 8.2686 Saltbr-in 2.692 HRD-in -74.28, -41.7 68.05, 5.57 in-in-in SNCiii in-in ActLoopNT-in 2.943 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.32, 170.09 APE9-dihe-na 72.35, 148.74 APE8-dihe-in -71.51, 141.06 APE8-rot-in 303.21 APE67-dihe-in -59.11, -26.68 -51.44, -48.71 APE12-dist-in 13.5034 APE11-dist-in 11.843 APE10-dist-in 7.0416 APE9-dist-in 3.173 None PTR216 PTR216 XRAY 1.85 0.185 0.203 A 351.0 346.0 4 27 27 0 [[56, 340]] 1.0 7sxj Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7OY5A P49841 35 385 420.0 39I:401 Type1 Active DFGin 6.9265 14.0328 BLAminus -126.76, 175.34 72.52, 92.63 -110.59, 33.29 286.05, 82.06 -75.35, -28.56 in-in in 8.6875 Saltbr-in 2.9358 HRD-in -72.48, -55.14 81.29, 7.92 in-in-in SNCiii in-in ActLoopNT-in 2.9168 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.43, 173.86 APE9-dihe-na 80.53, 146.3 APE8-dihe-in -94.81, 142.24 APE8-rot-in 295.61 APE67-dihe-inflip 101.01, -30.19 -44.76, 139.01 APE12-dist-in 12.9243 APE11-dist-in 10.9605 APE10-dist-in 5.8925 APE9-dist-in 3.2763 None None None XRAY 2.57 0.221 0.26 A 351.0 343.0 8 27 27 0 [[56, 340]] 1.0 7oy5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7OY5B P49841 35 383 420.0 39I:401 Type1 Active DFGin 7.1149 14.145 BLAminus -131.55, -176.92 63.09, 57.6 -70.26, 11.8 285.25, 87.17 -66.04, -15.46 in-in in 8.4954 Saltbr-in 3.0267 HRD-in -75.85, -49.73 71.52, 4.36 in-in-in SNCiii in-in ActLoopNT-in 3.0392 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.28, 172.83 APE9-dihe-na 79.24, 135.47 APE8-dihe-in -76.12, 154.7 APE8-rot-in 287.59 APE67-dihe-inflip 110.96, -34.61 -67.01, 135.0 APE12-dist-in 13.0301 APE11-dist-in 10.9583 APE10-dist-in 5.9922 APE9-dist-in 3.0083 None None None XRAY 2.57 0.221 0.26 B 351.0 344.0 5 27 27 0 [[56, 340]] 1.0 7oy5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U33A P49841 36 385 420.0 L7R:402 Type1 Active DFGin 7.0231 14.0492 BLAminus -140.49, 178.19 60.8, 84.54 -99.85, 16.49 288.62, 77.82 -50.41, -27.99 in-in in 8.5115 Saltbr-in 2.7738 HRD-in -71.53, -50.0 75.9, 8.27 in-in-in SNCiii in-in ActLoopNT-in 2.9863 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.78, -39.59 APE9-dihe-na -85.32, 160.12 APE8-dihe-in -84.45, 147.1 APE8-rot-in 286.21 APE67-dihe-inflip 87.92, -34.06 -59.31, 147.18 APE12-dist-in 13.0363 APE11-dist-in 10.9912 APE10-dist-in 6.0319 APE9-dist-in 3.2624 None None None XRAY 2.6 0.233 0.264 A 351.0 350.0 0 27 27 0 [[56, 340]] 1.0 7u33 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U33B P49841 37 382 420.0 L7R:402 Type1 Active DFGin 6.9949 14.0924 BLAminus -141.31, 178.2 60.97, 83.82 -100.06, 16.34 288.93, 78.7 -51.51, -27.59 in-in in 8.5327 Saltbr-in 2.7534 HRD-in -72.1, -49.87 75.78, 7.85 in-in-in SNCiii in-in ActLoopNT-in 2.989 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.62, 168.53 APE9-dihe-na 77.45, 140.58 APE8-dihe-in -89.54, 146.71 APE8-rot-in 285.53 APE67-dihe-in -82.12, -10.74 -0.24, -85.34 APE12-dist-in 13.0347 APE11-dist-in 10.9604 APE10-dist-in 6.0286 APE9-dist-in 3.1028 None None None XRAY 2.6 0.233 0.264 B 351.0 346.0 0 27 27 0 [[56, 340]] 1.0 7u33 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U36A P49841 36 385 420.0 L7W:402 Type1 Active DFGin 7.0548 14.0575 BLAminus -140.39, -178.87 60.34, 89.59 -105.19, 18.12 284.52, 86.52 -57.6, -32.5 in-in in 8.4531 Saltbr-in 3.0188 HRD-in -77.18, -47.14 70.51, 17.98 in-in-in SNCiii in-in ActLoopNT-in 2.9592 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.43, -45.81 APE9-dihe-na -84.57, 153.41 APE8-dihe-in -68.83, 161.86 APE8-rot-in 280.03 APE67-dihe-in -82.26, -16.89 -53.14, -56.37 APE12-dist-in 12.8704 APE11-dist-in 10.7585 APE10-dist-in 5.8125 APE9-dist-in 3.1894 None None None XRAY 2.75 0.24 0.275 A 351.0 350.0 0 27 27 0 [[56, 340]] 1.0 7u36 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7U36B P49841 37 382 420.0 L7W:402 Type1 Active DFGin 7.0561 14.0712 BLAminus -141.26, -179.45 60.58, 88.51 -105.71, 18.11 283.81, 87.44 -57.54, -31.03 in-in in 8.4984 Saltbr-in 2.9906 HRD-in -77.32, -47.05 68.98, 19.83 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -102.55, 163.3 APE9-dihe-na 90.09, 132.18 APE8-dihe-in -72.41, 162.37 APE8-rot-in 279.62 APE67-dihe-in -81.75, -17.56 -53.5, -56.42 APE12-dist-in 12.8558 APE11-dist-in 10.7783 APE10-dist-in 5.7902 APE9-dist-in 3.107 None None None XRAY 2.75 0.24 0.275 B 351.0 346.0 0 27 27 0 [[56, 340]] 1.0 7u36 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 2OW3A P49841 35 385 420.0 BIM:387 Type1 Active DFGin 6.8544 14.0885 BLAminus -145.58, -177.16 62.63, 79.7 -96.04, 38.01 299.18, 104.83 -72.62, -36.62 in-in in 8.3402 Saltbr-in 2.8377 HRD-in -75.79, -46.9 63.78, 27.01 in-in-in SNCiii in-in ActLoopNT-in 2.8813 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -159.84, 153.8 APE9-dihe-na 77.18, 154.82 APE8-dihe-in -72.33, 143.1 APE8-rot-in 299.46 APE67-dihe-in -64.33, -22.16 -49.08, -49.27 APE12-dist-in 13.7242 APE11-dist-in 12.3631 APE10-dist-in 7.5149 APE9-dist-in 3.7839 None PTR216 PTR216 XRAY 2.8 0.248 0.295 A 352.0 347.0 4 27 27 0 [[56, 340]] 1.0 2ow3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 2OW3B P49841 35 386 420.0 BIM:387 Type1 Active DFGin 6.7681 14.5197 BLAminus -140.91, -178.82 62.87, 80.36 -94.83, 34.08 291.22, 81.94 -79.34, -15.72 in-in in 8.4802 Saltbr-in 2.7885 HRD-in -91.97, -42.45 64.4, 21.24 in-in-in SNCiii in-in ActLoopNT-in 2.8773 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.27, 157.33 APE9-dihe-na 81.52, 163.87 APE8-dihe-in -81.91, 157.75 APE8-rot-in 308.08 APE67-dihe-in -65.81, -19.16 -55.34, -61.54 APE12-dist-in 13.9045 APE11-dist-in 12.5424 APE10-dist-in 7.6276 APE9-dist-in 3.5378 None PTR216 PTR216 XRAY 2.8 0.248 0.295 B 352.0 352.0 0 27 27 0 [[56, 340]] 1.0 2ow3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3GB2A P49841 35 383 420.0 G3B:999 Type1 Active DFGin 7.0809 13.5025 BLAminus -136.77, -176.86 57.81, 94.36 -109.09, 24.06 290.54, 74.85 -73.21, 4.88 in-in in 8.4499 Saltbr-in 2.8117 HRD-in -66.76, -55.55 72.33, 20.67 in-in-in SNCiii in-in ActLoopNT-in 2.8594 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.38, -175.57 APE9-dihe-na 67.46, 160.91 APE8-dihe-in -72.68, 139.68 APE8-rot-in 245.03 APE67-dihe-in -60.68, -25.16 -49.04, -51.42 APE12-dist-in 13.505 APE11-dist-in 11.9733 APE10-dist-in 7.0043 APE9-dist-in 3.2866 None PTR216 PTR216 XRAY 2.4 0.225 0.289 A 353.0 341.0 8 27 27 0 [[56, 340]] 1.0 3gb2 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6TCUA P49841 35 384 420.0 N1Q:401 Type1 Active DFGin 7.2707 14.1909 BLAminus -132.13, 178.03 59.16, 82.25 -93.13, 22.32 285.63, 78.52 -60.3, -31.7 in-in in 8.3524 Saltbr-in 2.9119 HRD-in -72.47, -46.38 65.88, 22.79 in-in-in SNCiii in-in ActLoopNT-in 2.8967 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.64, 162.18 APE9-dihe-na 73.42, 158.65 APE8-dihe-in -78.26, 138.24 APE8-rot-in 295.07 APE67-dihe-in -60.71, -25.87 -50.61, -49.17 APE12-dist-in 13.5559 APE11-dist-in 11.9425 APE10-dist-in 7.1969 APE9-dist-in 3.2398 None PTR216 PTR216 XRAY 2.14 0.204 0.24 A 355.0 350.0 0 27 27 0 [[56, 340]] 1.0 6tcu Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.9e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5T31A P49841 35 381 420.0 6VL:501 Type1 Active DFGin 7.0002 14.6002 BLAminus -146.5, -178.72 58.09, 85.8 -94.81, 34.39 283.96, 70.89 -72.9, -29.06 in-in in 8.1833 Saltbr-in 2.8228 HRD-in -85.27, -37.65 59.13, 22.16 in-in-in SNCiii in-in ActLoopNT-in 2.9632 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.45, 179.68 APE9-dihe-na 63.71, 158.01 APE8-dihe-in -85.57, 141.47 APE8-rot-in 304.73 APE67-dihe-in -68.11, -24.88 -45.34, -45.1 APE12-dist-in 13.218 APE11-dist-in 11.5452 APE10-dist-in 6.5643 APE9-dist-in 3.195 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 A 420.0 335.0 12 27 27 0 [[56, 340]] 1.0 5t31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5T31B P49841 36 382 420.0 6VL:501 Type1 Active DFGin 7.2086 14.6047 BLAminus -147.12, 178.9 61.54, 81.68 -96.09, 32.98 286.61, 73.16 -76.82, -18.6 in-in in 8.229 Saltbr-in 2.5809 HRD-in -64.89, -47.6 63.02, 19.09 in-in-in SNCiii in-in ActLoopNT-in 3.0176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.39, 179.54 APE9-dihe-na 63.77, 153.96 APE8-dihe-in -75.26, 136.0 APE8-rot-in 291.41 APE67-dihe-in -61.67, -31.85 -41.28, -53.13 APE12-dist-in 13.3814 APE11-dist-in 11.678 APE10-dist-in 6.473 APE9-dist-in 3.2366 D133E PTR216 PTR216 XRAY 2.85 0.2 0.268 B 420.0 334.0 13 27 27 0 [[56, 340]] 1.0 5t31 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.2e-70 244.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7Z1GA P49841 27 383 420.0 3NG:60401 Type1 Active DFGin 7.2716 14.699 BLAminus -137.45, -179.93 52.32, 81.51 -93.1, 20.22 282.75, 78.65 -65.74, -16.48 in-in in 8.9685 Saltbr-in 2.7705 HRD-in -67.62, -47.44 74.98, 2.45 in-in-in SNCiii in-in ActLoopNT-in 2.9264 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.67, 177.94 APE9-dihe-na 70.81, 142.84 APE8-dihe-in -95.23, 170.55 APE8-rot-in 305.08 APE67-dihe-inflip 72.5, -37.64 -53.01, 158.1 APE12-dist-in 12.7846 APE11-dist-in 10.8474 APE10-dist-in 5.858 APE9-dist-in 2.9838 None None None XRAY 2.85 0.204 0.228 A 364.0 355.0 2 27 27 0 [[56, 340]] 1.0 7z1g Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7B6FA P49841 36 382 420.0 SZW:401 Type1 Active DFGin 6.7876 14.0024 BLAminus -139.5, -179.55 63.73, 84.52 -97.59, 24.1 286.83, 79.42 -64.99, -20.21 in-in in 8.3187 Saltbr-in 2.5726 HRD-in -72.27, -45.59 68.3, 15.73 in-in-in SNCiii in-in ActLoopNT-in 2.8606 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.61, 164.26 APE9-dihe-na 74.41, 146.1 APE8-dihe-in -66.85, 137.72 APE8-rot-in 301.31 APE67-dihe-in -60.67, -24.91 -43.57, -54.9 APE12-dist-in 13.468 APE11-dist-in 11.6748 APE10-dist-in 7.0867 APE9-dist-in 3.2029 None PTR216 PTR216 XRAY 2.05 0.176 0.209 A 365.0 347.0 0 27 27 0 [[56, 340]] 1.0 7b6f Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8AUZA P49841 27 381 420.0 O9C:402 Type1 Active DFGin 7.0282 13.8218 BLAminus -150.9, 179.1 54.07, 83.84 -94.84, 28.62 288.95, 81.72 -71.58, -10.75 in-in in 8.4971 Saltbr-in 2.7343 HRD-in -57.37, -52.37 73.76, 8.1 in-in-in SNCiii in-in ActLoopNT-in 3.1547 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.43, 171.72 APE9-dihe-na 68.38, 153.94 APE8-dihe-in -73.1, 142.46 APE8-rot-in 305.9 APE67-dihe-in -60.73, -30.47 -42.52, -61.25 APE12-dist-in 13.255 APE11-dist-in 11.714 APE10-dist-in 7.0252 APE9-dist-in 3.0553 None PTR216 PTR216 XRAY 2.66 0.172 0.229 A 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8auz Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8AUZB P49841 27 381 420.0 O9C:402 Type1 Active DFGin 7.0993 13.9066 BLAminus -145.47, 175.75 60.6, 82.78 -92.91, 28.92 286.05, 79.75 -73.75, -11.85 in-in in 8.5865 Saltbr-in 2.6974 HRD-in -55.14, -51.91 71.49, 10.11 in-in-in SNCiii in-in ActLoopNT-in 3.1386 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.91, 170.34 APE9-dihe-na 66.33, 153.39 APE8-dihe-in -70.91, 144.03 APE8-rot-in 280.02 APE67-dihe-in -59.87, -32.25 -43.58, -60.53 APE12-dist-in 13.1722 APE11-dist-in 11.6615 APE10-dist-in 6.9239 APE9-dist-in 3.0036 None PTR216 PTR216 XRAY 2.66 0.172 0.229 B 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8auz Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4AFJA P49841 36 384 420.0 SJJ:1391 Type1 Active DFGin 6.9374 13.7151 BLAminus -130.67, 179.05 59.17, 87.64 -94.83, 20.23 280.89, 81.14 -65.73, -20.9 in-in in 8.572 Saltbr-in 2.6523 HRD-in -69.53, -45.4 65.78, 13.52 in-in-in SNCiii in-in ActLoopNT-in 2.9368 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.24, 160.98 APE9-dihe-na 76.37, 138.38 APE8-dihe-in -58.5, 130.27 APE8-rot-in 301.13 APE67-dihe-in -61.75, -23.96 -37.58, -52.92 APE12-dist-in 13.4348 APE11-dist-in 11.6806 APE10-dist-in 6.9749 APE9-dist-in 3.1929 None PTR216 PTR216 XRAY 1.98 0.179 0.216 A 367.0 344.0 5 27 27 0 [[56, 340]] 1.0 4afj Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4AFJB P49841 34 384 420.0 SJJ:1392 Type1 Active DFGin 6.9478 14.0458 BLAminus -131.53, 179.02 57.76, 85.75 -93.28, 22.08 280.88, 83.41 -64.33, -20.8 in-in in 8.5255 Saltbr-in 2.7428 HRD-in -67.39, -46.66 68.06, 10.89 in-in-in SNCiii in-in ActLoopNT-in 2.8765 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -147.99, 165.35 APE9-dihe-na 75.2, 154.5 APE8-dihe-in -78.53, 128.88 APE8-rot-in 295.4 APE67-dihe-in -61.46, -24.46 -31.5, -55.04 APE12-dist-in 13.4761 APE11-dist-in 11.5819 APE10-dist-in 6.9584 APE9-dist-in 3.1461 None PTR216 PTR216 XRAY 1.98 0.179 0.216 B 367.0 347.0 4 27 27 0 [[56, 340]] 1.0 4afj Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3ZRKA P49841 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.8856 13.908 BLAminus -131.68, 179.96 63.1, 79.53 -95.35, 25.37 286.53, 78.64 -74.21, -8.59 in-in in 8.4741 Saltbr-in 2.7497 HRD-in -67.17, -50.87 73.03, 10.45 in-in-in SNCiii in-in ActLoopNT-in 2.8412 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.35, 160.84 APE9-dihe-na 74.59, 142.57 APE8-dihe-in -61.86, 136.31 APE8-rot-in 305.46 APE67-dihe-in -59.75, -23.44 -46.23, -50.56 APE12-dist-in 13.3769 APE11-dist-in 11.6698 APE10-dist-in 7.0029 APE9-dist-in 3.1599 None PTR216 PTR216 XRAY 2.37 0.201 0.243 A 371.0 347.0 2 27 27 0 [[56, 340]] 1.0 3zrk Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3ZRKB P49841 36 384 420.0 ZRK:1400 Type1 Active DFGin 6.7154 14.0168 BLAminus -139.49, -177.28 57.97, 77.09 -90.4, 24.0 286.01, 81.23 -69.91, -16.36 in-in in 8.587 Saltbr-in 2.7319 HRD-in -64.4, -48.95 71.37, 3.03 in-in-in SNCiii in-in ActLoopNT-in 2.8439 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.35, 163.72 APE9-dihe-na 73.35, 153.59 APE8-dihe-in -70.79, 138.65 APE8-rot-in 292.42 APE67-dihe-in -62.81, -26.76 -44.91, -48.41 APE12-dist-in 13.3599 APE11-dist-in 11.4817 APE10-dist-in 6.8819 APE9-dist-in 3.1614 None PTR216 PTR216 XRAY 2.37 0.201 0.243 B 371.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zrk Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3ZRLA P49841 36 385 420.0 ZRL:1390 Type1 Active DFGin 6.9762 14.1446 BLAminus -134.74, 178.82 66.15, 74.2 -88.14, 21.07 285.95, 79.46 -68.66, -8.3 in-in in 8.4844 Saltbr-in 2.5864 HRD-in -74.36, -46.11 75.3, 2.22 in-in-in SNCiii in-in ActLoopNT-in 2.8884 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.36, 158.14 APE9-dihe-na 75.43, 144.25 APE8-dihe-in -61.72, 142.08 APE8-rot-in 315.78 APE67-dihe-in -63.29, -26.99 -52.04, -46.88 APE12-dist-in 13.4779 APE11-dist-in 11.7165 APE10-dist-in 7.1567 APE9-dist-in 3.1714 None PTR216 PTR216 XRAY 2.48 0.188 0.249 A 371.0 348.0 2 27 27 0 [[56, 340]] 1.0 3zrl Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3ZRLB P49841 36 384 420.0 ZRL:1390 Type1 Active DFGin 6.8163 14.0659 BLAminus -140.64, -176.21 56.19, 79.11 -88.83, 19.02 286.49, 80.49 -67.02, -13.2 in-in in 8.6131 Saltbr-in 2.7337 HRD-in -62.44, -47.89 69.81, 8.62 in-in-in SNCiii in-in ActLoopNT-in 2.8941 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.8, 160.71 APE9-dihe-na 76.77, 159.03 APE8-dihe-in -75.92, 142.27 APE8-rot-in 284.41 APE67-dihe-in -61.87, -25.02 -48.38, -50.46 APE12-dist-in 13.4519 APE11-dist-in 11.6967 APE10-dist-in 7.0855 APE9-dist-in 3.2183 None PTR216 PTR216 XRAY 2.48 0.188 0.249 B 371.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zrl Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3ZRMA P49841 36 383 420.0 ZRM:1388 Type1 Active DFGin 6.9338 13.9541 BLAminus -132.01, -179.16 64.76, 76.89 -91.07, 16.45 285.73, 79.52 -60.99, -14.53 in-in in 8.3792 Saltbr-in 2.5899 HRD-in -73.17, -48.0 77.03, 4.47 in-in-in SNCiii in-in ActLoopNT-in 2.8649 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.45, 164.9 APE9-dihe-na 71.3, 144.2 APE8-dihe-in -61.55, 140.83 APE8-rot-in 305.4 APE67-dihe-in -61.36, -25.73 -52.92, -47.77 APE12-dist-in 13.4177 APE11-dist-in 11.7327 APE10-dist-in 7.034 APE9-dist-in 3.1836 None PTR216 PTR216 XRAY 2.49 0.19 0.247 A 371.0 346.0 2 27 27 0 [[56, 340]] 1.0 3zrm Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3ZRMB P49841 36 384 420.0 ZRM:1389 Type1 Active DFGin 6.9018 14.1037 BLAminus -140.7, -177.64 59.24, 76.67 -89.43, 25.85 287.41, 78.75 -71.45, -17.33 in-in in 8.556 Saltbr-in 2.6387 HRD-in -65.21, -46.92 71.38, 6.55 in-in-in SNCiii in-in ActLoopNT-in 2.8965 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.4, 163.13 APE9-dihe-na 76.6, 157.17 APE8-dihe-in -72.35, 137.17 APE8-rot-in 272.08 APE67-dihe-in -62.09, -20.43 -43.42, -53.94 APE12-dist-in 13.4635 APE11-dist-in 11.6966 APE10-dist-in 7.0308 APE9-dist-in 3.1098 None PTR216 PTR216 XRAY 2.49 0.19 0.247 B 371.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zrm Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5K5NA P49841 36 382 420.0 6QH:4001 Type1 Active DFGin 6.8671 13.8031 BLAminus -136.97, -178.03 58.54, 81.58 -94.06, 22.59 285.28, 80.04 -66.6, -22.76 in-in in 8.6849 Saltbr-in 2.7627 HRD-in -65.0, -45.17 61.7, 20.55 in-in-in SNCiii in-in ActLoopNT-in 2.9036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.55, 163.97 APE9-dihe-na 70.72, 157.82 APE8-dihe-in -71.18, 131.1 APE8-rot-in 299.71 APE67-dihe-in -62.03, -24.12 -33.31, -56.32 APE12-dist-in 13.5851 APE11-dist-in 11.9664 APE10-dist-in 6.9925 APE9-dist-in 3.2009 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 A 370.0 332.0 12 27 27 0 [[56, 340]] 1.0 5k5n Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5K5NB P49841 36 384 420.0 6QH:401 Type1 Active DFGin 6.9681 13.7452 BLAminus -135.06, -178.44 58.85, 83.42 -94.58, 20.58 286.7, 80.8 -64.41, -22.37 in-in in 8.8691 Saltbr-in 2.795 HRD-in -64.71, -45.91 63.61, 14.11 in-in-in SNCiii in-in ActLoopNT-in 2.8804 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.36, 162.07 APE9-dihe-na 75.01, 147.36 APE8-dihe-in -65.41, 124.62 APE8-rot-in 290.2 APE67-dihe-in -56.35, -27.77 -26.59, -62.75 APE12-dist-in 13.3721 APE11-dist-in 11.9936 APE10-dist-in 6.8964 APE9-dist-in 3.1086 V28G PTR216 PTR216 XRAY 2.2 0.205 0.229 B 370.0 335.0 11 27 27 0 [[56, 340]] 1.0 5k5n Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1R0EA P49841 35 383 420.0 DFN:702 Type1 Active DFGin 7.2106 13.9782 BLAminus -134.01, -179.44 58.42, 85.11 -96.64, 20.85 278.46, 77.75 -63.57, -17.65 in-in in 8.3722 Saltbr-in 2.7157 HRD-in -68.9, -46.99 73.89, 15.3 in-in-in SNCiii in-in ActLoopNT-in 2.8169 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.99, 167.9 APE9-dihe-na 82.35, 148.07 APE8-dihe-in -104.61, 148.9 APE8-rot-in 290.93 APE67-dihe-inflip 91.63, -34.6 -37.68, 131.22 APE12-dist-in 13.0977 APE11-dist-in 11.0936 APE10-dist-in 6.2403 APE9-dist-in 3.3951 None None None XRAY 2.25 0.225 0.252 A 391.0 344.0 5 27 27 0 [[56, 340]] 1.0 1r0e Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1R0EB P49841 35 383 420.0 DFN:501 Type1 Active DFGin 7.2465 14.1047 BLAminus -133.07, -177.02 55.1, 85.48 -97.08, 20.86 276.04, 78.13 -65.93, -17.26 in-in in 8.4454 Saltbr-in 2.9103 HRD-in -68.16, -44.28 70.07, 10.75 in-in-in SNCiii in-in ActLoopNT-in 2.8839 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.79, 168.13 APE9-dihe-na 84.81, 147.78 APE8-dihe-in -104.27, 148.93 APE8-rot-in 288.7 APE67-dihe-inflip 91.14, -35.24 -35.52, 130.18 APE12-dist-in 13.0787 APE11-dist-in 11.0114 APE10-dist-in 6.1772 APE9-dist-in 3.3688 None None None XRAY 2.25 0.225 0.252 B 391.0 344.0 5 27 27 0 [[56, 340]] 1.0 1r0e Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.6e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q5KA P49841 35 384 420.0 TMU:901 Type1 Active DFGin 6.9883 13.8632 BLAminus -136.18, -175.74 56.25, 81.9 -94.66, 24.16 283.53, 73.95 -64.32, -18.01 in-in in 8.2268 Saltbr-in 2.5487 HRD-in -67.21, -47.72 71.71, 7.94 in-in-in SNCiii in-in ActLoopNT-in 2.9814 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.63, 174.67 APE9-dihe-na 78.79, 134.14 APE8-dihe-in -77.03, 144.65 APE8-rot-in 302.42 APE67-dihe-inflip 99.66, -34.41 -53.93, 140.09 APE12-dist-in 12.9051 APE11-dist-in 11.0016 APE10-dist-in 5.832 APE9-dist-in 3.1437 None None None XRAY 1.94 0.222 0.242 A 414.0 345.0 5 27 27 0 [[56, 340]] 1.0 1q5k Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q5KB P49841 35 384 420.0 TMU:902 Type1 Active DFGin 6.9852 13.7726 BLAminus -138.67, -177.12 58.86, 79.46 -94.38, 28.16 285.34, 70.82 -69.41, -14.87 in-in in 8.1321 Saltbr-in 2.8315 HRD-in -69.04, -44.01 68.27, 5.21 in-in-in SNCiii in-in ActLoopNT-in 2.9161 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.05, 176.86 APE9-dihe-na 75.09, 135.72 APE8-dihe-in -79.59, 144.98 APE8-rot-in 303.4 APE67-dihe-inflip 93.62, -37.01 -50.51, 145.1 APE12-dist-in 12.9305 APE11-dist-in 11.072 APE10-dist-in 5.8459 APE9-dist-in 3.1034 None None None XRAY 1.94 0.222 0.242 B 414.0 344.0 6 27 27 0 [[56, 340]] 1.0 1q5k Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3I4BA P49841 25 385 420.0 Z48:501 Type1 Active DFGin 6.6409 13.6459 BLAminus -134.01, -176.44 58.71, 78.24 -93.71, 24.37 285.69, 79.56 -67.57, -20.03 in-in in 8.4755 Saltbr-in 2.6366 HRD-in -63.92, -46.73 77.65, -7.51 in-in-in SNCiii in-in ActLoopNT-in 2.9496 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.08, 174.13 APE9-dihe-na 79.29, 137.44 APE8-dihe-in -92.27, 151.07 APE8-rot-in 303.5 APE67-dihe-inflip 83.63, -1.22 -43.52, 132.98 APE12-dist-in 13.0087 APE11-dist-in 10.9391 APE10-dist-in 5.839 APE9-dist-in 3.1024 None None None XRAY 2.3 0.181 0.222 A 414.0 359.0 0 27 27 0 [[56, 340]] 1.0 3i4b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3I4BB P49841 36 382 420.0 Z48:501 Type1 Active DFGin 7.0103 13.6549 BLAminus -135.85, -175.31 58.14, 77.59 -93.89, 21.58 285.55, 84.81 -65.19, -18.79 in-in in 8.5085 Saltbr-in 2.617 HRD-in -67.57, -44.79 75.92, -6.36 in-in-in SNCiii in-in ActLoopNT-in 2.941 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.93, 173.5 APE9-dihe-na 79.53, 137.7 APE8-dihe-in -93.51, 150.41 APE8-rot-in 299.4 APE67-dihe-inflip 78.16, -1.88 -37.33, 134.24 APE12-dist-in 13.0428 APE11-dist-in 10.917 APE10-dist-in 5.8278 APE9-dist-in 3.1154 None None None XRAY 2.3 0.181 0.222 B 414.0 347.0 0 27 27 0 [[56, 340]] 1.0 3i4b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3L1SA P49841 25 384 420.0 Z92:421 Type1 Active DFGin 6.7571 13.7476 BLAminus -136.19, -175.27 59.75, 67.96 -82.46, 22.04 287.73, 86.13 -66.81, -21.63 in-in in 8.5179 Saltbr-in 2.7076 HRD-in -64.1, -46.34 73.45, -1.44 in-in-in SNCiii in-in ActLoopNT-in 2.949 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 172.3 APE9-dihe-na 79.23, 137.51 APE8-dihe-in -89.89, 147.82 APE8-rot-in 303.47 APE67-dihe-inflip 83.2, -1.08 -42.22, 131.52 APE12-dist-in 13.0072 APE11-dist-in 10.8922 APE10-dist-in 5.8943 APE9-dist-in 3.1607 None None None XRAY 2.9 0.186 0.232 A 414.0 336.0 21 27 27 0 [[56, 340]] 1.0 3l1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3L1SB P49841 36 382 420.0 Z92:422 Type1 Active DFGin 6.9841 13.7797 BLAminus -136.63, -175.36 61.34, 59.7 -75.09, 22.69 291.46, 84.75 -66.47, -23.35 in-in in 8.551 Saltbr-in 2.7367 HRD-in -65.65, -45.98 77.68, -13.89 in-in-in SNCiii in-in ActLoopNT-in 2.9365 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.08, 173.03 APE9-dihe-na 76.72, 137.31 APE8-dihe-in -89.1, 148.7 APE8-rot-in 302.46 APE67-dihe-inflip 83.32, 3.78 -42.62, 131.74 APE12-dist-in 13.0142 APE11-dist-in 10.916 APE10-dist-in 6.1494 APE9-dist-in 3.1214 None None None XRAY 2.9 0.186 0.232 B 414.0 330.0 17 27 27 0 [[56, 340]] 1.0 3l1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 2JLDA P49841 35 385 420.0 AG1:1385 Type1 Active DFGin 7.2466 13.6191 BLAminus -128.74, 174.0 65.55, 89.02 -101.06, 20.23 281.85, 78.64 -66.01, -16.46 in-in in 8.5348 Saltbr-in 2.9005 HRD-in -68.74, -48.89 74.29, 10.13 in-in-in SNCiii in-in ActLoopNT-in 2.8459 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -80.14, 165.31 APE9-dihe-na 82.65, 142.84 APE8-dihe-in -89.49, 145.54 APE8-rot-in 290.56 APE67-dihe-inflip 101.97, -33.31 -39.01, 124.35 APE12-dist-in 13.012 APE11-dist-in 11.0047 APE10-dist-in 6.0583 APE9-dist-in 3.2394 None None None XRAY 2.35 0.192 0.227 A 420.0 349.0 2 27 27 0 [[56, 340]] 1.0 2jld Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 2JLDB P49841 35 384 420.0 AG1:1385 Type1 Active DFGin 7.1172 13.6811 BLAminus -134.8, 174.83 62.6, 85.31 -97.62, 21.89 284.88, 76.87 -65.09, -17.38 in-in in 8.458 Saltbr-in 2.7255 HRD-in -67.92, -46.43 70.86, 13.33 in-in-in SNCiii in-in ActLoopNT-in 2.9206 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.11, 167.47 APE9-dihe-na 84.04, 143.71 APE8-dihe-in -89.79, 148.89 APE8-rot-in 294.08 APE67-dihe-inflip 95.31, -31.23 -37.35, 123.61 APE12-dist-in 13.0443 APE11-dist-in 10.9507 APE10-dist-in 5.9948 APE9-dist-in 3.2028 None None None XRAY 2.35 0.192 0.227 B 420.0 349.0 1 27 27 0 [[56, 340]] 1.0 2jld Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3M1SB P49841 35 384 420.0 DW1:421 Type1 Active DFGin 7.1866 13.372 BLAminus -147.84, 174.37 70.86, 99.58 -120.24, 19.87 286.56, 80.37 -63.52, -14.18 in-in in 8.5847 Saltbr-in 2.4408 HRD-in -69.47, -49.47 71.23, 28.36 in-in-in SNCiii in-in ActLoopNT-in 3.0905 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -106.87, 165.89 APE9-dihe-na 90.21, 134.65 APE8-dihe-in -74.2, 145.74 APE8-rot-in 300.21 APE67-dihe-in -72.41, -23.39 -22.57, -69.43 APE12-dist-in 12.9441 APE11-dist-in 10.7117 APE10-dist-in 5.8988 APE9-dist-in 3.769 None None None XRAY 3.134 0.171 0.228 B 420.0 349.0 1 27 27 0 [[56, 340]] 1.0 3m1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3PUPA P49841 35 382 420.0 OS1:421 Type1 Active DFGin 6.9952 13.6372 BLAminus -143.74, 172.61 64.16, 94.87 -107.49, 13.61 287.44, 72.72 -52.4, -32.47 in-in in 8.4428 Saltbr-in 2.8069 HRD-in -86.73, -34.2 66.44, 7.86 in-in-in SNCiii in-in ActLoopNT-in 2.8568 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -111.24, -13.27 APE9-dihe-na -89.84, 168.85 APE8-dihe-in -94.34, 159.6 APE8-rot-in 296.79 APE67-dihe-in -69.26, -2.79 -42.9, -70.67 APE12-dist-in 13.0555 APE11-dist-in 10.9122 APE10-dist-in 6.171 APE9-dist-in 3.4857 None None None XRAY 2.99 0.206 0.249 A 420.0 346.0 2 27 27 0 [[56, 340]] 1.0 3pup Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3PUPB P49841 35 383 420.0 OS1:421 Type1 Active DFGin 6.9868 13.6463 BLAminus -146.61, 171.7 65.62, 100.17 -113.12, 21.06 287.13, 70.81 -60.05, -30.47 in-in in 8.4793 Saltbr-in 2.972 HRD-in -88.21, -42.27 77.46, 8.13 in-in-in SNCiii in-in ActLoopNT-in 2.812 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -103.13, -17.37 APE9-dihe-na -97.38, 160.84 APE8-dihe-in -100.44, 160.76 APE8-rot-in 282.35 APE67-dihe-in -75.14, -2.22 -49.84, -64.39 APE12-dist-in 13.1068 APE11-dist-in 10.9755 APE10-dist-in 6.4999 APE9-dist-in 3.7505 None None None XRAY 2.99 0.206 0.249 B 420.0 347.0 2 27 27 0 [[56, 340]] 1.0 3pup Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6B8JA P49841 37 384 420.0 65C:502 Type1 Active DFGin 6.8683 13.9089 BLAminus -142.04, -175.4 56.86, 72.8 -87.54, 21.75 287.01, 61.58 -69.77, -16.08 in-in in 8.5074 Saltbr-in 2.3182 HRD-in -66.49, -42.97 62.67, 20.6 in-in-in SNCiii in-in ActLoopNT-in 2.8209 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.37, 166.1 APE9-dihe-na 69.29, 116.74 APE8-dihe-in -38.51, 137.94 APE8-rot-in 299.43 APE67-dihe-in -65.74, -24.52 -56.45, -42.14 APE12-dist-in 13.6847 APE11-dist-in 11.734 APE10-dist-in 7.0179 APE9-dist-in 3.3258 None PTR216 PTR216 XRAY 2.595 0.215 0.247 A 420.0 345.0 3 27 27 0 [[56, 340]] 1.0 6b8j Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6H0UA P49841 36 383 420.0 FKB:501 Type1 Active DFGin 6.7319 13.816 BLAminus -102.2, -173.91 62.01, 94.18 -105.02, 23.81 292.61, 84.27 -66.96, -25.5 in-in in 8.7982 Saltbr-in 2.7262 HRD-in -71.89, -49.13 79.92, 3.93 in-in-in SNCiii in-in ActLoopNT-in 2.9659 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.85, 170.11 APE9-dihe-na 84.06, 143.45 APE8-dihe-in -90.7, 142.53 APE8-rot-in 301.69 APE67-dihe-in -73.12, -14.65 -13.27, -76.63 APE12-dist-in 12.9549 APE11-dist-in 10.8677 APE10-dist-in 5.7603 APE9-dist-in 3.2229 None None None XRAY 2.3 0.195 0.24 A 420.0 348.0 0 27 27 0 [[56, 340]] 1.0 6h0u Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6H0UB P49841 36 383 420.0 FKB:501 Type1 Active DFGin 6.6481 13.9725 BLAminus -111.78, 175.04 68.36, 93.29 -102.83, 22.46 286.57, 84.56 -63.31, -24.15 in-in in 8.7633 Saltbr-in 2.7449 HRD-in -68.5, -49.8 75.08, 1.45 in-in-in SNCiii in-in ActLoopNT-in 2.8506 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.21, 171.64 APE9-dihe-na 80.61, 138.7 APE8-dihe-in -91.3, 150.17 APE8-rot-in 304.68 APE67-dihe-inflip 101.55, -29.52 -53.44, 134.06 APE12-dist-in 12.722 APE11-dist-in 10.7262 APE10-dist-in 5.7037 APE9-dist-in 3.1629 None None None XRAY 2.3 0.195 0.24 B 420.0 348.0 0 27 27 0 [[56, 340]] 1.0 6h0u Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6V6LA P49841 37 384 420.0 QQA:501 Type1 Active DFGin 7.2439 14.2279 BLAminus -134.87, -179.15 59.4, 83.41 -98.99, 30.0 283.16, 72.37 -75.66, -20.38 in-in in 8.3879 Saltbr-in 2.7358 HRD-in -68.21, -49.19 67.93, 18.71 in-in-in SNCiii in-in ActLoopNT-in 3.016 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.84, 162.85 APE9-dihe-na 77.33, 149.16 APE8-dihe-in -69.69, 129.38 APE8-rot-in 287.88 APE67-dihe-in -58.07, -31.39 -36.48, -49.2 APE12-dist-in 13.4611 APE11-dist-in 11.6477 APE10-dist-in 6.9528 APE9-dist-in 3.241 None PTR216 PTR216 XRAY 2.19 0.204 0.234 A 420.0 344.0 4 27 27 0 [[56, 340]] 1.0 6v6l Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3DU8A P49841 35 382 420.0 553:553 Type1 Active DFGin 6.9922 13.9377 BLAminus -138.88, -177.6 60.76, 81.45 -97.52, 17.85 284.1, 81.79 -60.5, -23.71 in-in in 8.7135 Saltbr-in 2.6861 HRD-in -70.97, -44.22 68.9, 5.64 in-in-in SNCiii in-in ActLoopNT-in 2.9768 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.61, 170.6 APE9-dihe-na 82.17, 142.06 APE8-dihe-in -90.1, 145.24 APE8-rot-in 300.29 APE67-dihe-inflip 98.68, -34.99 -51.44, 136.14 APE12-dist-in 13.0356 APE11-dist-in 10.9436 APE10-dist-in 5.7637 APE9-dist-in 3.1519 None None None XRAY 2.2 0.215 0.246 A 422.0 336.0 12 27 27 0 [[56, 340]] 1.0 3du8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3DU8B P49841 35 385 420.0 553:553 Type1 Active DFGin 7.1097 14.0005 BLAminus -130.0, -177.1 64.69, 78.27 -91.27, 21.46 283.91, 80.88 -65.59, -20.64 in-in in 8.7421 Saltbr-in 2.7016 HRD-in -71.12, -43.48 71.58, 1.27 in-in-in SNCiii in-in ActLoopNT-in 2.9923 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -75.13, 166.25 APE9-dihe-na 83.98, 139.39 APE8-dihe-in -88.38, 143.61 APE8-rot-in 294.95 APE67-dihe-inflip 93.54, -38.98 -56.03, 145.75 APE12-dist-in 13.0504 APE11-dist-in 11.1301 APE10-dist-in 5.901 APE9-dist-in 3.1759 None None None XRAY 2.2 0.215 0.246 B 422.0 339.0 12 27 27 0 [[56, 340]] 1.0 3du8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR5A P49841 25 385 420.0 A1IE8:501 Type1 Active DFGin 7.0632 14.321 BLAminus -141.02, 178.57 59.76, 86.64 -101.14, 27.38 287.09, 76.28 -70.78, -13.94 in-in in 8.3627 Saltbr-in 2.8669 HRD-in -72.5, -48.23 71.7, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.9846 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.15, 177.99 APE9-dihe-na 68.95, 145.14 APE8-dihe-in -94.16, 151.35 APE8-rot-in 288.71 APE67-dihe-inflip 90.22, -34.5 -47.82, 143.36 APE12-dist-in 13.1043 APE11-dist-in 11.1055 APE10-dist-in 6.1672 APE9-dist-in 3.1855 None None None XRAY 2.3 0.204 0.235 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR5B P49841 36 382 420.0 A1IE8:501 Type1 Active DFGin 7.0679 14.3968 BLAminus -143.23, 179.4 62.21, 84.47 -103.42, 28.19 287.66, 78.04 -72.31, -18.53 in-in in 8.6835 Saltbr-in 2.9648 HRD-in -72.41, -47.52 71.61, 14.06 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.66, -179.45 APE9-dihe-na 68.77, 147.4 APE8-dihe-in -97.67, 156.22 APE8-rot-in 283.57 APE67-dihe-inflip 84.77, -33.0 -49.59, 145.66 APE12-dist-in 13.0555 APE11-dist-in 10.9532 APE10-dist-in 5.9863 APE9-dist-in 3.1875 None None None XRAY 2.3 0.204 0.235 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR6A P49841 25 385 420.0 A1IFO:501 Type1 Active DFGin 7.0735 14.1612 BLAminus -136.83, -174.79 60.55, 80.3 -97.86, 24.81 287.57, 77.74 -66.69, -16.26 in-in in 8.5559 Saltbr-in 2.9354 HRD-in -72.59, -48.06 71.15, 12.43 in-in-in SNCiii in-in ActLoopNT-in 2.9919 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.91, 171.88 APE9-dihe-na 74.24, 144.89 APE8-dihe-in -96.08, 152.09 APE8-rot-in 291.49 APE67-dihe-inflip 90.67, -36.1 -52.14, 144.18 APE12-dist-in 13.0224 APE11-dist-in 11.047 APE10-dist-in 6.1241 APE9-dist-in 3.2396 None None None XRAY 2.3 0.2 0.232 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR6B P49841 36 382 420.0 A1IFO:501 Type1 Active DFGin 7.1281 14.3598 BLAminus -139.12, -179.31 63.06, 81.93 -99.98, 26.01 286.75, 75.51 -71.16, -14.75 in-in in 8.8431 Saltbr-in 2.8359 HRD-in -72.29, -48.89 71.91, 12.0 in-in-in SNCiii in-in ActLoopNT-in 2.9172 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.4, 172.1 APE9-dihe-na 77.09, 144.87 APE8-dihe-in -98.08, 154.15 APE8-rot-in 291.27 APE67-dihe-inflip 90.37, -33.63 -52.57, 140.86 APE12-dist-in 13.0706 APE11-dist-in 10.9572 APE10-dist-in 5.9828 APE9-dist-in 3.2201 None None None XRAY 2.3 0.2 0.232 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR7A P49841 25 385 420.0 A1IFJ:501 Type1 Active DFGin 6.912 13.9494 BLAminus -136.24, -176.42 58.55, 87.09 -104.67, 27.04 287.13, 78.6 -71.53, -14.0 in-in in 8.6316 Saltbr-in 2.8018 HRD-in -71.98, -46.0 72.36, 9.7 in-in-in SNCiii in-in ActLoopNT-in 2.9869 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.42, 177.43 APE9-dihe-na 69.9, 145.82 APE8-dihe-in -94.03, 156.28 APE8-rot-in 289.17 APE67-dihe-inflip 91.05, -31.63 -52.45, 141.85 APE12-dist-in 13.1081 APE11-dist-in 11.1214 APE10-dist-in 6.1207 APE9-dist-in 3.1495 None None None XRAY 2.3 0.199 0.229 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR7B P49841 36 382 420.0 A1IFJ:501 Type1 Active DFGin 6.9902 13.9524 BLAminus -139.3, -178.5 61.7, 87.08 -105.92, 24.05 284.91, 80.77 -70.11, -13.68 in-in in 8.5932 Saltbr-in 2.7099 HRD-in -71.41, -48.43 71.41, 11.5 in-in-in SNCiii in-in ActLoopNT-in 2.9398 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.82, 177.23 APE9-dihe-na 70.05, 146.13 APE8-dihe-in -96.47, 160.58 APE8-rot-in 285.27 APE67-dihe-inflip 87.67, -29.95 -51.57, 140.33 APE12-dist-in 13.0082 APE11-dist-in 11.0074 APE10-dist-in 6.0448 APE9-dist-in 3.156 None None None XRAY 2.3 0.199 0.229 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR8A P49841 25 385 420.0 A1IE7:501 Type1 Active DFGin 6.991 14.3251 BLAminus -138.39, -179.52 63.72, 81.82 -96.4, 23.65 287.29, 75.6 -66.3, -11.74 in-in in 8.5529 Saltbr-in 2.9059 HRD-in -71.33, -45.89 67.7, 10.94 in-in-in SNCiii in-in ActLoopNT-in 2.9571 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.78, 169.84 APE9-dihe-na 80.06, 148.59 APE8-dihe-in -102.16, 146.47 APE8-rot-in 284.89 APE67-dihe-inflip 97.34, -39.62 -53.84, 140.75 APE12-dist-in 13.0812 APE11-dist-in 11.083 APE10-dist-in 6.0117 APE9-dist-in 3.1971 None None None XRAY 2.3 0.191 0.221 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR8B P49841 36 383 420.0 A1IE7:501 Type1 Active DFGin 7.087 14.3561 BLAminus -145.34, 175.42 68.0, 83.84 -100.29, 22.36 287.83, 75.27 -65.32, -15.0 in-in in 8.7153 Saltbr-in 2.8977 HRD-in -76.0, -49.5 72.49, 12.34 in-in-in SNCiii in-in ActLoopNT-in 2.9624 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.57, 172.15 APE9-dihe-na 78.67, 145.51 APE8-dihe-in -99.99, 146.48 APE8-rot-in 286.49 APE67-dihe-inflip 90.46, -36.44 -48.06, 141.27 APE12-dist-in 13.0668 APE11-dist-in 10.8517 APE10-dist-in 5.8498 APE9-dist-in 3.1528 None None None XRAY 2.3 0.191 0.221 B 442.0 348.0 0 27 27 0 [[56, 340]] 1.0 9fr8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR9A P49841 25 385 420.0 A1IE6:501 Type1 Active DFGin 7.0374 14.3248 BLAminus -140.22, -173.71 59.89, 84.2 -98.36, 22.56 286.21, 81.87 -68.06, -16.06 in-in in 8.4621 Saltbr-in 2.928 HRD-in -72.09, -48.73 72.37, 5.47 in-in-in SNCiii in-in ActLoopNT-in 2.9713 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.48, 176.45 APE9-dihe-na 79.51, 153.1 APE8-dihe-in -106.78, 146.27 APE8-rot-in 287.32 APE67-dihe-inflip 100.87, -37.49 -40.18, 126.82 APE12-dist-in 13.0195 APE11-dist-in 11.0304 APE10-dist-in 5.997 APE9-dist-in 3.1732 None None None XRAY 2.55 0.197 0.234 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9fr9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9FR9B P49841 36 382 420.0 A1IE6:501 Type1 Active DFGin 6.9697 14.4133 BLAminus -146.13, 179.78 62.16, 86.8 -103.01, 25.64 284.6, 80.86 -74.54, -16.98 in-in in 8.7597 Saltbr-in 3.487 HRD-in -67.74, -52.21 72.42, 13.09 in-in-in SNCiii in-in ActLoopNT-in 2.8715 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.09, 170.35 APE9-dihe-na 79.85, 140.07 APE8-dihe-in -93.7, 153.67 APE8-rot-in 288.81 APE67-dihe-inflip 99.37, -31.56 -52.24, 133.09 APE12-dist-in 12.9815 APE11-dist-in 10.8097 APE10-dist-in 5.7912 APE9-dist-in 3.1814 None None None XRAY 2.55 0.197 0.234 B 442.0 347.0 0 27 27 0 [[56, 340]] 1.0 9fr9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9HUKB P49841 26 382 420.0 A1IXL:501 Type1 Active DFGin 7.4628 14.0621 BLAminus -139.0, -179.94 58.73, 94.97 -114.49, 25.32 285.15, 69.98 -63.61, -20.61 in-in in 8.1298 Saltbr-in 3.2803 HRD-in -69.2, -40.72 63.39, 20.78 in-in-in SNCiii in-in ActLoopNT-in 3.0415 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.58, -178.87 APE9-dihe-na 67.27, 135.83 APE8-dihe-in -80.15, 163.62 APE8-rot-in 319.54 APE67-dihe-inflip 75.84, -27.97 -60.6, 162.6 APE12-dist-in 12.8383 APE11-dist-in 10.7437 APE10-dist-in 5.7296 APE9-dist-in 3.2115 None None None XRAY 3.5 0.219 0.25 B 442.0 357.0 0 27 27 0 [[56, 340]] 1.0 9huk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9HULA P49841 25 385 420.0 A1IXM:501 Type1 Active DFGin 7.0701 13.9429 BLAminus -137.8, -179.92 58.93, 93.22 -109.33, 21.24 284.01, 77.28 -66.77, -7.95 in-in in 8.3439 Saltbr-in 2.9227 HRD-in -67.44, -42.84 67.99, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.1667 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.24, 178.29 APE9-dihe-na 68.13, 143.96 APE8-dihe-in -84.08, 162.04 APE8-rot-in 308.02 APE67-dihe-inflip 75.91, -35.84 -57.58, 161.58 APE12-dist-in 13.0659 APE11-dist-in 11.0236 APE10-dist-in 5.9969 APE9-dist-in 3.1634 None None None XRAY 2.9 0.218 0.244 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9hul Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9HULB P49841 26 383 420.0 A1IXM:501 Type1 Active DFGin 7.2175 13.8998 BLAminus -141.92, -177.61 60.57, 66.5 -86.27, 21.98 288.8, 69.64 -66.75, -12.19 in-in in 8.2676 Saltbr-in 2.7477 HRD-in -68.36, -43.53 65.84, 14.02 in-in-in SNCiii in-in ActLoopNT-in 3.0185 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.86, 177.51 APE9-dihe-na 70.81, 136.76 APE8-dihe-in -79.57, 164.11 APE8-rot-in 306.92 APE67-dihe-inflip 69.45, -30.71 -58.24, 165.67 APE12-dist-in 13.0545 APE11-dist-in 10.9752 APE10-dist-in 6.0547 APE9-dist-in 3.14 None None None XRAY 2.9 0.218 0.244 B 442.0 358.0 0 27 27 0 [[56, 340]] 1.0 9hul Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9HV3A P49841 25 385 420.0 A1IXN:501 Type1 Active DFGin 7.1249 13.9703 BLAminus -135.63, 170.17 69.98, 84.71 -102.55, 20.46 290.46, 80.59 -69.94, -0.25 in-in in 8.5374 Saltbr-in 2.8684 HRD-in -69.25, -48.0 72.7, 9.47 in-in-in SNCiii in-in ActLoopNT-in 2.9354 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -88.1, 169.69 APE9-dihe-na 79.34, 142.23 APE8-dihe-in -80.23, 146.96 APE8-rot-in 316.9 APE67-dihe-inflip 78.3, -27.2 -49.89, 154.45 APE12-dist-in 13.1231 APE11-dist-in 11.1203 APE10-dist-in 6.1972 APE9-dist-in 3.1364 None None None XRAY 2.9 0.208 0.238 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9hv3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9HV3B P49841 25 382 420.0 A1IXN:501 Type1 Active DFGin 7.0874 13.9122 BLAminus -155.32, 174.2 63.74, 86.56 -102.98, 16.67 284.3, 76.87 -64.93, -6.56 in-in in 8.5969 Saltbr-in 2.6055 HRD-in -75.09, -41.25 66.67, 4.87 in-in-in SNCiii in-in ActLoopNT-in 2.9817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.85, 168.81 APE9-dihe-na 83.21, 130.42 APE8-dihe-in -66.5, 151.79 APE8-rot-in 306.21 APE67-dihe-inflip 94.47, -29.15 -64.06, 143.12 APE12-dist-in 12.9743 APE11-dist-in 10.8793 APE10-dist-in 5.979 APE9-dist-in 3.017 None None None XRAY 2.9 0.208 0.238 B 442.0 358.0 0 27 27 0 [[56, 340]] 1.0 9hv3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q3DA P49841 35 385 420.0 STU:451 Type1 Active DFGin 7.2063 14.4113 BLAminus -139.48, 178.33 63.94, 87.17 -99.43, 23.77 282.58, 69.4 -66.25, -14.58 in-in in 8.701 Saltbr-in 2.8552 HRD-in -65.74, -44.7 66.01, 11.52 in-in-in SNCiii in-in ActLoopNT-in 3.0363 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.53, 169.72 APE9-dihe-na 81.56, 143.56 APE8-dihe-in -91.54, 154.32 APE8-rot-in 294.67 APE67-dihe-inflip 96.36, -28.56 -51.12, 132.48 APE12-dist-in 13.0736 APE11-dist-in 11.1082 APE10-dist-in 6.0869 APE9-dist-in 3.274 None None None XRAY 2.2 0.23 0.252 A 424.0 339.0 12 27 27 0 [[56, 340]] 1.0 1q3d Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q3DB P49841 35 383 420.0 STU:452 Type1 Active DFGin 7.26 14.4195 BLAminus -137.95, 177.39 64.41, 87.07 -97.99, 22.53 282.7, 70.11 -63.96, -17.29 in-in in 8.7081 Saltbr-in 2.9721 HRD-in -67.72, -45.35 66.86, 12.1 in-in-in SNCiii in-in ActLoopNT-in 3.0238 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.75, 170.28 APE9-dihe-na 79.08, 144.81 APE8-dihe-in -89.94, 151.95 APE8-rot-in 299.26 APE67-dihe-inflip 101.61, -31.22 -54.51, 132.99 APE12-dist-in 13.0847 APE11-dist-in 11.0881 APE10-dist-in 6.1457 APE9-dist-in 3.2379 None None None XRAY 2.2 0.23 0.252 B 424.0 339.0 10 27 27 0 [[56, 340]] 1.0 1q3d Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q3WA P49841 35 386 420.0 ATU:502 Type1 Active DFGin 7.1464 13.9518 BLAminus -137.77, 177.61 62.94, 83.24 -96.07, 24.67 288.22, 69.87 -66.71, -10.0 in-in in 8.3223 Saltbr-in 2.9235 HRD-in -67.11, -47.79 71.57, 6.31 in-in-in SNCiii in-in ActLoopNT-in 3.0225 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.32, 172.63 APE9-dihe-na 77.53, 136.48 APE8-dihe-in -79.93, 143.51 APE8-rot-in 298.62 APE67-dihe-in -62.35, -17.4 -13.52, -82.56 APE12-dist-in 13.0749 APE11-dist-in 11.129 APE10-dist-in 5.9641 APE9-dist-in 3.1434 None None None XRAY 2.3 0.225 0.248 A 424.0 344.0 8 27 27 0 [[56, 340]] 1.0 1q3w Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q3WB P49841 35 383 420.0 ATU:501 Type1 Active DFGin 7.0895 14.2696 BLAminus -140.46, 175.46 63.78, 84.76 -97.02, 22.89 286.31, 71.96 -64.9, -10.6 in-in in 8.5467 Saltbr-in 2.7917 HRD-in -67.92, -47.98 71.69, 6.95 in-in-in SNCiii in-in ActLoopNT-in 3.0188 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.2, 172.08 APE9-dihe-na 78.0, 136.99 APE8-dihe-in -80.5, 143.58 APE8-rot-in 301.78 APE67-dihe-in -64.47, -16.3 -12.81, -81.64 APE12-dist-in 13.0688 APE11-dist-in 11.1114 APE10-dist-in 5.9384 APE9-dist-in 3.1466 None None None XRAY 2.3 0.225 0.248 B 424.0 341.0 8 27 27 0 [[56, 340]] 1.0 1q3w Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q41A P49841 35 386 420.0 IXM:451 Type1 Active DFGin 7.0961 13.7419 BLAminus -140.31, 177.95 63.36, 85.31 -97.68, 24.93 285.2, 72.61 -64.62, -16.75 in-in in 8.1819 Saltbr-in 2.8445 HRD-in -70.03, -43.74 69.02, 2.85 in-in-in SNCiii in-in ActLoopNT-in 3.0075 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.85, 173.09 APE9-dihe-na 80.34, 135.13 APE8-dihe-in -75.55, 139.31 APE8-rot-in 298.19 APE67-dihe-in -65.33, -18.78 -13.64, -78.26 APE12-dist-in 13.068 APE11-dist-in 11.0572 APE10-dist-in 5.9147 APE9-dist-in 3.2247 None None None XRAY 2.1 0.229 0.245 A 424.0 339.0 13 27 27 0 [[56, 340]] 1.0 1q41 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q41B P49841 35 383 420.0 IXM:452 Type1 Active DFGin 7.0941 13.8936 BLAminus -139.75, 177.7 62.59, 85.88 -97.92, 24.85 285.3, 70.28 -63.82, -17.54 in-in in 8.3883 Saltbr-in 2.83 HRD-in -70.82, -46.38 71.27, 6.28 in-in-in SNCiii in-in ActLoopNT-in 3.0071 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.0, 171.76 APE9-dihe-na 82.35, 130.54 APE8-dihe-in -71.97, 140.37 APE8-rot-in 298.15 APE67-dihe-in -64.0, -13.46 -11.43, -84.5 APE12-dist-in 13.0562 APE11-dist-in 11.0548 APE10-dist-in 5.884 APE9-dist-in 3.2357 None None None XRAY 2.1 0.229 0.245 B 424.0 343.0 6 27 27 0 [[56, 340]] 1.0 1q41 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q4LA P49841 35 386 420.0 679:451 Type1 Active DFGin 6.9437 13.7544 BLAminus -138.39, -176.39 57.74, 86.06 -99.56, 21.29 285.7, 72.79 -65.03, -5.34 in-in in 8.5237 Saltbr-in 3.0069 HRD-in -67.11, -46.06 68.04, 16.48 in-in-in SNCiii in-in ActLoopNT-in 2.962 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -95.21, 168.86 APE9-dihe-na 81.69, 129.23 APE8-dihe-in -70.09, 146.41 APE8-rot-in 291.03 APE67-dihe-inflip 104.98, -29.32 -58.42, 137.67 APE12-dist-in 13.1169 APE11-dist-in 11.3523 APE10-dist-in 6.3007 APE9-dist-in 3.3388 None None None XRAY 2.77 0.212 0.251 A 424.0 342.0 10 27 27 0 [[56, 340]] 1.0 1q4l Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1Q4LB P49841 35 383 420.0 679:452 Type1 Active DFGin 7.1687 13.6494 BLAminus -140.11, -177.14 58.72, 87.12 -99.76, 20.01 285.14, 71.58 -64.5, -5.39 in-in in 8.3387 Saltbr-in 2.6728 HRD-in -67.89, -45.11 67.21, 17.1 in-in-in SNCiii in-in ActLoopNT-in 2.9961 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.61, 167.87 APE9-dihe-na 83.04, 132.56 APE8-dihe-in -74.69, 156.93 APE8-rot-in 311.31 APE67-dihe-inflip 93.39, -29.64 -61.08, 141.61 APE12-dist-in 13.0983 APE11-dist-in 11.3225 APE10-dist-in 6.2525 APE9-dist-in 3.3488 None None None XRAY 2.77 0.212 0.251 B 424.0 337.0 12 27 27 0 [[56, 340]] 1.0 1q4l Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3Q3BA P49841 35 386 420.0 55E:421 Type1 Active DFGin 6.8592 13.8905 BLAminus -146.51, -174.92 60.73, 82.19 -97.34, 22.93 287.93, 77.72 -66.67, -8.01 in-in in 8.4603 Saltbr-in 2.7177 HRD-in -65.09, -51.43 75.32, 0.61 in-in-in SNCiii in-in ActLoopNT-in 3.0239 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -93.28, 172.26 APE9-dihe-na 79.45, 140.83 APE8-dihe-in -87.39, 149.52 APE8-rot-in 308.45 APE67-dihe-in -68.31, -14.9 -12.45, -80.03 APE12-dist-in 13.0041 APE11-dist-in 11.0599 APE10-dist-in 6.1861 APE9-dist-in 3.1458 None None None XRAY 2.7 0.228 0.259 A 424.0 344.0 8 27 27 0 [[56, 340]] 1.0 3q3b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3Q3BB P49841 35 383 420.0 55E:421 Type1 Active DFGin 6.9437 13.7668 BLAminus -148.03, -175.09 60.19, 82.65 -96.08, 19.99 287.37, 77.74 -64.82, -9.3 in-in in 8.4427 Saltbr-in 2.7893 HRD-in -64.26, -50.5 74.85, 0.78 in-in-in SNCiii in-in ActLoopNT-in 3.0481 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.17, 172.11 APE9-dihe-na 80.0, 136.06 APE8-dihe-in -78.43, 156.9 APE8-rot-in 303.64 APE67-dihe-in -69.77, -0.18 -23.17, -84.47 APE12-dist-in 12.9964 APE11-dist-in 11.0446 APE10-dist-in 6.1791 APE9-dist-in 3.1016 None None None XRAY 2.7 0.228 0.259 B 424.0 341.0 8 27 27 0 [[56, 340]] 1.0 3q3b Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4J1RA P49841 36 383 420.0 I5R:502 Type1 Active DFGin 7.1431 14.149 BLAminus -140.34, -172.16 50.83, 73.0 -88.1, 31.44 288.82, 75.41 -70.78, -20.52 in-in in 8.3393 Saltbr-in 3.0257 HRD-in -70.85, -43.96 67.49, 12.65 in-in-in SNCiii in-in ActLoopNT-in 2.9176 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.66, 159.85 APE9-dihe-na 83.41, 158.3 APE8-dihe-in -70.39, 137.75 APE8-rot-in 276.14 APE67-dihe-in -62.89, -24.7 -48.3, -48.41 APE12-dist-in 13.4658 APE11-dist-in 11.8784 APE10-dist-in 7.0059 APE9-dist-in 3.199 None PTR216 PTR216 XRAY 2.702 0.174 0.193 A 424.0 344.0 4 27 27 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4J1RB P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.1595 14.1324 BLAminus -138.14, -172.1 51.97, 73.85 -90.74, 32.74 288.65, 76.48 -71.96, -19.84 in-in in 8.3512 Saltbr-in 3.0798 HRD-in -72.6, -39.29 60.47, 16.92 in-in-in SNCiii in-in ActLoopNT-in 2.8744 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.96, 157.32 APE9-dihe-na 86.27, 160.84 APE8-dihe-in -74.2, 139.51 APE8-rot-in 270.87 APE67-dihe-in -63.78, -23.12 -48.17, -50.06 APE12-dist-in 13.4606 APE11-dist-in 11.6326 APE10-dist-in 6.9809 APE9-dist-in 3.1987 None PTR216 PTR216 XRAY 2.702 0.174 0.193 B 424.0 347.0 2 27 27 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4J1RC P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.1535 14.1448 BLAminus -137.53, -170.95 51.06, 74.57 -90.65, 33.09 289.21, 75.99 -73.08, -20.73 in-in in 8.3436 Saltbr-in 3.0086 HRD-in -71.61, -39.59 60.78, 16.42 in-in-in SNCiii in-in ActLoopNT-in 2.9513 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.54, 161.15 APE9-dihe-na 82.95, 157.27 APE8-dihe-in -71.13, 139.05 APE8-rot-in 271.75 APE67-dihe-in -63.34, -23.83 -48.75, -48.68 APE12-dist-in 13.4752 APE11-dist-in 11.9746 APE10-dist-in 7.0273 APE9-dist-in 3.2194 None PTR216 PTR216 XRAY 2.702 0.174 0.193 C 424.0 345.0 4 27 27 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4J1RD P49841 36 384 420.0 I5R:502 Type1 Active DFGin 7.1575 14.143 BLAminus -136.3, -170.0 51.29, 73.39 -89.98, 32.08 288.97, 75.59 -72.78, -18.14 in-in in 8.3472 Saltbr-in 3.0818 HRD-in -65.4, -45.24 73.44, 1.93 in-in-in SNCiii in-in ActLoopNT-in 2.9291 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.81, 157.82 APE9-dihe-na 85.66, 159.76 APE8-dihe-in -71.48, 137.15 APE8-rot-in 266.3 APE67-dihe-in -62.21, -25.06 -46.41, -50.2 APE12-dist-in 13.4651 APE11-dist-in 11.9016 APE10-dist-in 7.0243 APE9-dist-in 3.1172 None PTR216 PTR216 XRAY 2.702 0.174 0.193 D 424.0 346.0 3 27 27 0 [[56, 340]] 1.0 4j1r Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5HLNA P49841 34 384 420.0 65C:501 Type1 Active DFGin 6.9714 13.5391 BLAminus -145.82, 177.83 61.52, 84.96 -98.63, 20.2 288.24, 74.65 -61.35, -16.22 in-in in 8.64 Saltbr-in 2.9698 HRD-in -72.97, -42.53 59.11, 33.41 in-in-in SNCiii in-in ActLoopNT-in 2.9659 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.08, -68.13 APE9-dihe-na -70.88, 179.27 APE8-dihe-in -73.41, 154.88 APE8-rot-in 283.39 APE67-dihe-in -59.67, -27.13 -52.94, -57.58 APE12-dist-in 13.1086 APE11-dist-in 11.7674 APE10-dist-in 7.2143 APE9-dist-in 3.907 None PTR216 PTR216 XRAY 3.1 0.173 0.236 A 424.0 347.0 4 27 27 0 [[56, 340]] 1.0 5hln Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5HLPA P49841 36 382 420.0 65A:501 Type1 Active DFGin 7.1863 14.396 BLAminus -136.58, -178.8 62.45, 78.77 -95.76, 20.37 283.01, 75.68 -68.07, -12.1 in-in in 8.1462 Saltbr-in 2.605 HRD-in -72.39, -43.73 64.36, 19.61 in-in-in SNCiii in-in ActLoopNT-in 2.8712 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.83, 176.24 APE9-dihe-na 71.02, 146.23 APE8-dihe-in -63.35, 144.14 APE8-rot-in 289.42 APE67-dihe-in -64.86, -21.95 -54.37, -48.38 APE12-dist-in 13.6671 APE11-dist-in 11.8195 APE10-dist-in 6.6439 APE9-dist-in 3.2984 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 A 424.0 339.0 8 27 27 0 [[56, 340]] 1.0 5hlp Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5HLPB P49841 36 383 420.0 65A:501 Type1 Active DFGin 7.1151 14.4669 BLAminus -132.96, -174.02 57.79, 78.12 -94.26, 22.08 284.54, 74.66 -71.61, -17.17 in-in in 8.276 Saltbr-in 2.7164 HRD-in -71.48, -47.76 70.66, 10.73 in-in-in SNCiii in-in ActLoopNT-in 2.8371 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.37, 176.63 APE9-dihe-na 72.15, 149.52 APE8-dihe-in -67.13, 142.42 APE8-rot-in 293.57 APE67-dihe-in -63.1, -24.66 -49.41, -51.54 APE12-dist-in 13.356 APE11-dist-in 11.8213 APE10-dist-in 6.5807 APE9-dist-in 3.1348 None PTR216,TPO277 PTR216,TPO277 XRAY 2.45 0.19 0.24 B 424.0 337.0 11 27 27 0 [[56, 340]] 1.0 5hlp Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5KPKA P49841 35 384 420.0 6VK:500 Type1 Active DFGin 6.9115 14.5084 BLAminus -138.4, -178.64 58.08, 79.3 -90.22, 19.44 284.58, 73.09 -63.35, -18.32 in-in in 8.5736 Saltbr-in 2.7304 HRD-in -73.46, -47.41 66.88, 21.39 in-in-in SNCiii in-in ActLoopNT-in 2.9498 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.73, 163.34 APE9-dihe-na 69.65, 162.27 APE8-dihe-in -73.86, 143.79 APE8-rot-in 303.06 APE67-dihe-in -60.34, -24.86 -54.25, -52.95 APE12-dist-in 13.597 APE11-dist-in 12.1565 APE10-dist-in 7.487 APE9-dist-in 3.2434 None PTR216 PTR216 XRAY 2.4 0.17 0.224 A 424.0 347.0 3 27 27 0 [[56, 340]] 1.0 5kpk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5KPKB P49841 35 383 420.0 6VK:500 Type1 Active DFGin 7.0281 14.5236 BLAminus -138.48, -175.82 55.16, 85.06 -97.98, 23.13 277.82, 78.64 -67.65, -21.76 in-in in 8.5853 Saltbr-in 2.685 HRD-in -71.19, -45.78 65.3, 13.14 in-in-in SNCiii in-in ActLoopNT-in 3.0036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.69, 168.24 APE9-dihe-na 65.31, 163.84 APE8-dihe-in -77.16, 143.7 APE8-rot-in 304.59 APE67-dihe-in -57.42, -23.92 -54.57, -50.84 APE12-dist-in 13.6928 APE11-dist-in 12.1642 APE10-dist-in 7.3948 APE9-dist-in 3.1039 None PTR216 PTR216 XRAY 2.4 0.17 0.224 B 424.0 345.0 4 27 27 0 [[56, 340]] 1.0 5kpk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5KPLA P49841 36 384 420.0 6VL:500 Type1 Active DFGin 7.044 14.2531 BLAminus -136.48, 178.55 58.11, 81.69 -92.72, 18.86 289.18, 73.73 -64.85, -20.41 in-in in 8.3485 Saltbr-in 2.4859 HRD-in -65.11, -50.47 69.64, 19.91 in-in-in SNCiii in-in ActLoopNT-in 3.0876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.42, 168.54 APE9-dihe-na 62.76, 158.29 APE8-dihe-in -78.28, 147.71 APE8-rot-in 310.05 APE67-dihe-in -62.4, -23.75 -53.92, -48.24 APE12-dist-in 13.4339 APE11-dist-in 11.8787 APE10-dist-in 7.1366 APE9-dist-in 3.3883 None PTR216 PTR216 XRAY 2.6 0.182 0.244 A 424.0 340.0 9 27 27 0 [[56, 340]] 1.0 5kpl Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5KPLB P49841 36 383 420.0 6VL:500 Type1 Active DFGin 7.1545 14.6155 BLAminus -138.92, -172.41 52.88, 79.26 -88.95, 20.81 278.36, 73.5 -72.97, -16.23 in-in in 8.4978 Saltbr-in 2.9713 HRD-in -70.3, -40.66 56.94, 24.57 in-in-in SNCiii in-in ActLoopNT-in 2.7814 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.07, 160.76 APE9-dihe-na 66.33, 169.2 APE8-dihe-in -85.14, 144.57 APE8-rot-in 313.48 APE67-dihe-in -71.14, -21.99 -47.02, -47.87 APE12-dist-in 13.6449 APE11-dist-in 11.8586 APE10-dist-in 7.3669 APE9-dist-in 3.3795 None PTR216 PTR216 XRAY 2.6 0.182 0.244 B 424.0 340.0 8 27 27 0 [[56, 340]] 1.0 5kpl Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5KPMA P49841 36 383 420.0 6VM:500 Type1 Active DFGin 7.1795 14.1524 BLAminus -127.54, 178.59 63.4, 85.66 -102.69, 28.41 287.99, 66.47 -62.48, -34.28 in-in in 8.4058 Saltbr-in 2.6694 HRD-in -73.98, -45.27 60.61, 25.04 in-in-in SNCiii in-in ActLoopNT-in 2.7332 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.88, 162.98 APE9-dihe-na 64.81, 161.74 APE8-dihe-in -75.86, 141.16 APE8-rot-in 297.33 APE67-dihe-in -64.41, -17.12 -48.06, -52.48 APE12-dist-in 13.62 APE11-dist-in 11.8384 APE10-dist-in 7.3632 APE9-dist-in 3.2615 None PTR216 PTR216 XRAY 2.69 0.178 0.24 A 424.0 345.0 3 27 27 0 [[56, 340]] 1.0 5kpm Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5KPMB P49841 36 384 420.0 6VM:500 Type1 Active DFGin 7.1408 14.6384 BLAminus -142.12, 178.63 60.71, 81.6 -96.16, 22.05 281.72, 76.19 -66.25, -7.91 in-in in 8.6086 Saltbr-in 2.5806 HRD-in -65.22, -49.2 64.23, 7.63 in-in-in SNCiii in-in ActLoopNT-in 2.9931 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.34, 163.89 APE9-dihe-na 62.78, 158.8 APE8-dihe-in -77.09, 139.57 APE8-rot-in 302.93 APE67-dihe-in -64.17, -18.23 -41.12, -52.04 APE12-dist-in 13.5592 APE11-dist-in 11.9721 APE10-dist-in 7.4703 APE9-dist-in 3.1928 None PTR216 PTR216 XRAY 2.69 0.178 0.24 B 424.0 346.0 3 27 27 0 [[56, 340]] 1.0 5kpm Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4IQ6A P49841 37 382 420.0 IQ6:501 Type1 Active DFGin 7.0678 14.0082 BLAminus -142.1, 176.37 68.23, 72.95 -88.9, 16.75 291.61, 92.77 -55.61, -37.28 in-in in 8.5737 Saltbr-in 2.8412 HRD-in -66.67, -43.42 72.45, -14.35 in-in-in SNCiii in-in ActLoopNT-in 3.0118 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -77.44, 163.79 APE9-dihe-na 84.06, 140.31 APE8-dihe-in -95.86, 141.6 APE8-rot-in 294.32 APE67-dihe-inflip 102.08, -40.06 -38.49, 130.32 APE12-dist-in 13.2141 APE11-dist-in 11.0068 APE10-dist-in 6.1934 APE9-dist-in 3.1668 None None None XRAY 3.12 0.188 0.227 A 426.0 324.0 22 27 27 0 [[56, 340]] 1.0 4iq6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3SAYA P49841 35 384 420.0 OFT:431 Type1 Active DFGin 6.9238 14.2084 BLAminus -134.06, -176.24 58.1, 80.75 -95.49, 24.69 285.79, 80.8 -58.99, -23.52 in-in in 8.7646 Saltbr-in 2.6835 HRD-in -76.77, -47.73 71.86, 15.98 in-in-in SNCiii in-in ActLoopNT-in 2.8872 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.28, 177.68 APE9-dihe-na 70.36, 150.2 APE8-dihe-in -70.69, 142.5 APE8-rot-in 303.06 APE67-dihe-in -64.8, -21.63 -53.21, -43.25 APE12-dist-in 13.4747 APE11-dist-in 11.7676 APE10-dist-in 6.4744 APE9-dist-in 3.1409 None PTR216 PTR216 XRAY 2.231 0.202 0.23 A 430.0 348.0 2 27 27 0 [[56, 340]] 1.0 3say Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3SAYB P49841 35 382 420.0 OFT:431 Type1 Active DFGin 7.0946 14.2081 BLAminus -125.43, -174.49 59.4, 82.08 -94.07, 22.41 283.95, 82.11 -68.04, -11.91 in-in in 8.7759 Saltbr-in 2.5965 HRD-in -71.92, -46.59 68.83, 6.83 in-in-in SNCiii in-in ActLoopNT-in 2.9773 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.5, 172.68 APE9-dihe-na 72.51, 152.54 APE8-dihe-in -66.45, 133.95 APE8-rot-in 293.34 APE67-dihe-in -62.41, -25.02 -42.21, -48.58 APE12-dist-in 13.5034 APE11-dist-in 11.8296 APE10-dist-in 6.7035 APE9-dist-in 3.0926 None PTR216 PTR216 XRAY 2.231 0.202 0.23 B 430.0 348.0 0 27 27 0 [[56, 340]] 1.0 3say Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.5e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4PTCA P49841 36 381 420.0 2WE:501 Type1 Active DFGin 6.9363 14.3975 BLAminus -147.73, -174.11 62.98, 81.81 -100.26, 25.83 284.28, 79.03 -59.65, -43.28 in-in in 9.1619 Saltbr-in 2.729 HRD-in -73.84, -45.42 69.86, 9.93 in-in-in SNCiii in-in ActLoopNT-in 2.77 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -85.04, 172.51 APE9-dihe-na 77.59, 144.28 APE8-dihe-in -89.54, 156.63 APE8-rot-in 297.82 APE67-dihe-inflip 95.7, -27.15 -58.15, 143.88 APE12-dist-in 13.0497 APE11-dist-in 10.7791 APE10-dist-in 6.0041 APE9-dist-in 3.2718 None None None XRAY 2.711 0.217 0.281 A 441.0 342.0 4 27 27 0 [[56, 340]] 1.0 4ptc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4PTCB P49841 35 385 420.0 2WE:501 Type1 Active DFGin 7.2125 14.6055 BLAminus -123.82, -167.89 50.38, 80.91 -94.33, 28.59 284.85, 71.64 -64.12, -29.45 in-in in 8.9235 Saltbr-in 2.4023 HRD-in -67.43, -42.31 63.02, 14.07 in-in-in SNCiii in-in ActLoopNT-in 2.9358 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.89, 173.71 APE9-dihe-na 81.21, 152.66 APE8-dihe-in -112.25, 156.82 APE8-rot-in 292.56 APE67-dihe-inflip 100.85, -22.79 -44.26, 123.15 APE12-dist-in 13.0829 APE11-dist-in 10.9184 APE10-dist-in 5.8898 APE9-dist-in 3.2799 None None None XRAY 2.711 0.217 0.281 B 441.0 347.0 4 27 27 0 [[56, 340]] 1.0 4ptc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4PTEA P49841 36 382 420.0 2WF:501 Type1 Active DFGin 6.9317 14.0172 BLAminus -141.21, 178.04 57.99, 89.39 -100.23, 24.26 286.38, 75.9 -68.08, -19.02 in-in in 8.7161 Saltbr-in 2.6354 HRD-in -73.56, -44.45 69.11, 4.74 in-in-in SNCiii in-in ActLoopNT-in 2.7924 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.74, 175.98 APE9-dihe-na 75.98, 148.82 APE8-dihe-in -103.79, 152.51 APE8-rot-in 295.33 APE67-dihe-inflip 95.08, -28.26 -38.95, 126.56 APE12-dist-in 12.9786 APE11-dist-in 10.8902 APE10-dist-in 5.8826 APE9-dist-in 3.0881 None None None XRAY 2.033 0.17 0.195 A 441.0 341.0 6 27 27 0 [[56, 340]] 1.0 4pte Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4PTEB P49841 36 385 420.0 2WF:501 Type1 Active DFGin 6.9181 13.9369 BLAminus -137.07, 179.43 58.52, 88.98 -101.38, 27.88 284.28, 76.88 -69.85, -20.65 in-in in 8.4836 Saltbr-in 2.6854 HRD-in -70.9, -46.61 73.05, 2.3 in-in-in SNCiii in-in ActLoopNT-in 2.8872 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.76, 178.59 APE9-dihe-na 72.73, 147.77 APE8-dihe-in -103.48, 150.66 APE8-rot-in 296.89 APE67-dihe-inflip 94.67, -27.57 -36.66, 125.81 APE12-dist-in 12.9354 APE11-dist-in 10.8805 APE10-dist-in 5.8765 APE9-dist-in 3.1539 None None None XRAY 2.033 0.17 0.195 B 441.0 347.0 3 27 27 0 [[56, 340]] 1.0 4pte Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4PTGA P49841 36 382 420.0 2WG:501 Type1 Active DFGin 7.0033 13.9163 BLAminus -132.5, 179.85 66.28, 92.0 -106.7, 26.9 285.24, 77.28 -68.07, -25.88 in-in in 8.5408 Saltbr-in 2.8279 HRD-in -68.57, -44.88 68.54, 10.31 in-in-in SNCiii in-in ActLoopNT-in 2.939 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -81.39, 169.96 APE9-dihe-na 80.02, 147.16 APE8-dihe-in -96.08, 142.52 APE8-rot-in 290.31 APE67-dihe-inflip 90.23, -35.22 -45.66, 142.01 APE12-dist-in 13.0565 APE11-dist-in 11.0186 APE10-dist-in 6.1199 APE9-dist-in 3.284 None None None XRAY 2.361 0.173 0.211 A 441.0 333.0 14 27 27 0 [[56, 340]] 1.0 4ptg Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4PTGB P49841 37 385 420.0 2WG:501 Type1 Active DFGin 6.9512 13.863 BLAminus -136.28, -175.42 57.62, 87.0 -101.31, 27.32 285.42, 76.21 -67.67, -26.13 in-in in 8.437 Saltbr-in 2.705 HRD-in -71.07, -46.44 71.76, 6.12 in-in-in SNCiii in-in ActLoopNT-in 2.8995 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -89.44, 175.88 APE9-dihe-na 76.35, 149.91 APE8-dihe-in -109.95, 151.08 APE8-rot-in 289.69 APE67-dihe-inflip 91.44, -30.76 -44.23, 136.59 APE12-dist-in 12.9878 APE11-dist-in 11.0088 APE10-dist-in 5.9105 APE9-dist-in 3.1601 None None None XRAY 2.361 0.173 0.211 B 441.0 332.0 17 27 27 0 [[56, 340]] 1.0 4ptg Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8DJCA P49841 35 382 420.0 UAU:501 Type1 Active DFGin 7.1066 13.6454 BLAminus -130.93, 175.08 68.46, 84.27 -99.8, 25.87 290.84, 77.95 -66.29, -22.25 in-in in 8.4422 Saltbr-in 2.6994 HRD-in -67.33, -44.59 69.12, 7.74 in-in-in SNCiii in-in ActLoopNT-in 2.984 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 169.18 APE9-dihe-na 83.11, 139.06 APE8-dihe-in -86.29, 148.88 APE8-rot-in 301.44 APE67-dihe-inflip 95.96, -28.78 -50.91, 136.23 APE12-dist-in 12.9117 APE11-dist-in 10.8312 APE10-dist-in 5.8045 APE9-dist-in 3.2569 None None None XRAY 2.463 0.217 0.242 A 441.0 331.0 17 27 27 0 [[56, 340]] 1.0 8djc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8DJCB P49841 35 385 420.0 UAU:501 Type1 Active DFGin 7.1252 13.6329 BLAminus -137.19, 179.71 59.65, 83.27 -96.94, 27.03 290.51, 79.22 -67.53, -21.56 in-in in 8.3277 Saltbr-in 2.738 HRD-in -65.99, -44.91 69.53, 7.25 in-in-in SNCiii in-in ActLoopNT-in 2.9859 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.05, 167.49 APE9-dihe-na 82.24, 138.29 APE8-dihe-in -85.04, 145.47 APE8-rot-in 300.63 APE67-dihe-inflip 98.12, -32.04 -46.91, 135.02 APE12-dist-in 12.9423 APE11-dist-in 10.8879 APE10-dist-in 5.9441 APE9-dist-in 3.2585 None None None XRAY 2.463 0.217 0.242 B 441.0 332.0 19 27 27 0 [[56, 340]] 1.0 8djc Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8DJDA P49841 36 383 420.0 U3E:501 Type1 Active DFGin 7.1826 13.8782 BLAminus -134.36, -179.72 59.88, 85.28 -97.18, 26.66 285.76, 75.79 -65.91, -27.91 in-in in 8.3565 Saltbr-in 2.7038 HRD-in -66.89, -45.93 70.71, 8.73 in-in-in SNCiii in-in ActLoopNT-in 2.9738 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -97.03, 169.31 APE9-dihe-na 77.5, 142.18 APE8-dihe-in -93.09, 155.03 APE8-rot-in 301.61 APE67-dihe-inflip 94.8, -31.52 -52.67, 137.81 APE12-dist-in 13.0595 APE11-dist-in 11.0394 APE10-dist-in 6.1287 APE9-dist-in 3.198 None None None XRAY 2.205 0.209 0.222 A 441.0 338.0 10 27 27 0 [[56, 340]] 1.0 8djd Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8DJDB P49841 36 384 420.0 U3E:501 Type1 Active DFGin 7.129 13.9195 BLAminus -133.17, 179.77 59.91, 85.17 -97.09, 26.57 285.62, 75.36 -66.56, -27.45 in-in in 8.3472 Saltbr-in 2.6969 HRD-in -66.65, -46.07 70.85, 8.52 in-in-in SNCiii in-in ActLoopNT-in 2.9199 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.46, 170.54 APE9-dihe-na 79.57, 140.07 APE8-dihe-in -94.46, 154.56 APE8-rot-in 301.16 APE67-dihe-inflip 94.52, -31.07 -52.58, 138.22 APE12-dist-in 13.0861 APE11-dist-in 11.08 APE10-dist-in 6.0775 APE9-dist-in 3.2169 None None None XRAY 2.205 0.209 0.222 B 441.0 341.0 8 27 27 0 [[56, 340]] 1.0 8djd Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8DJEA P49841 36 384 420.0 U6S:501 Type1 Active DFGin 7.2598 13.3694 BLAminus -139.51, 175.88 67.17, 88.55 -102.31, 22.49 287.71, 78.25 -63.99, -27.99 in-in in 8.3126 Saltbr-in 2.7163 HRD-in -68.38, -45.52 70.24, 12.16 in-in-in SNCiii in-in ActLoopNT-in 2.8928 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -84.85, 166.32 APE9-dihe-na 87.14, 140.36 APE8-dihe-in -88.6, 149.46 APE8-rot-in 293.07 APE67-dihe-inflip 99.13, -30.7 -44.53, 124.89 APE12-dist-in 12.957 APE11-dist-in 10.8666 APE10-dist-in 6.0436 APE9-dist-in 3.3533 None None None XRAY 2.374 0.201 0.227 A 441.0 347.0 2 27 27 0 [[56, 340]] 1.0 8dje Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8DJEB P49841 36 385 420.0 U6S:501 Type1 Active DFGin 7.2394 13.4205 BLAminus -137.87, 177.52 63.92, 86.56 -101.17, 24.78 290.39, 74.84 -68.33, -25.47 in-in in 8.2646 Saltbr-in 2.7355 HRD-in -65.34, -46.08 68.76, 12.58 in-in-in SNCiii in-in ActLoopNT-in 2.8895 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.12, 167.71 APE9-dihe-na 84.3, 145.94 APE8-dihe-in -98.8, 148.34 APE8-rot-in 293.36 APE67-dihe-inflip 97.13, -37.27 -40.76, 129.94 APE12-dist-in 12.9575 APE11-dist-in 10.9317 APE10-dist-in 5.908 APE9-dist-in 3.263 None None None XRAY 2.374 0.201 0.227 B 441.0 343.0 7 27 27 0 [[56, 340]] 1.0 8dje Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8FF8A P49841 36 382 420.0 XV0:501 Type1 Active DFGin 7.2002 13.7357 BLAminus -135.89, 175.65 65.86, 84.5 -97.83, 25.7 284.17, 77.94 -66.05, -27.44 in-in in 8.341 Saltbr-in 2.7523 HRD-in -68.43, -43.4 70.29, 3.62 in-in-in SNCiii in-in ActLoopNT-in 2.8419 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.65, 167.87 APE9-dihe-na 84.02, 136.04 APE8-dihe-in -86.03, 151.96 APE8-rot-in 298.92 APE67-dihe-inflip 95.48, -31.71 -43.39, 129.41 APE12-dist-in 12.7414 APE11-dist-in 10.7529 APE10-dist-in 5.7907 APE9-dist-in 3.2113 None None None XRAY 2.33 0.198 0.217 A 441.0 347.0 0 27 27 0 [[56, 340]] 1.0 8ff8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8FF8B P49841 36 385 420.0 XV0:501 Type1 Active DFGin 7.2005 13.8111 BLAminus -130.19, -175.53 57.72, 85.5 -98.92, 25.25 283.55, 78.69 -65.7, -29.77 in-in in 8.3387 Saltbr-in 2.7464 HRD-in -67.11, -43.98 70.41, 3.15 in-in-in SNCiii in-in ActLoopNT-in 2.825 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -83.86, 169.83 APE9-dihe-na 81.04, 142.01 APE8-dihe-in -96.19, 150.13 APE8-rot-in 300.46 APE67-dihe-inflip 95.56, -32.32 -40.34, 130.68 APE12-dist-in 12.779 APE11-dist-in 10.7843 APE10-dist-in 5.8246 APE9-dist-in 3.2182 None None None XRAY 2.33 0.198 0.217 B 441.0 346.0 4 27 27 0 [[56, 340]] 1.0 8ff8 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.7e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3F88A P49841 35 383 420.0 3HT:999 Type1 Active DFGin 7.2474 13.7299 BLAminus -137.96, -171.11 53.2, 96.02 -109.46, 31.55 277.23, 77.74 -85.58, 3.2 in-in in 8.6202 Saltbr-in 2.5161 HRD-in -66.41, -48.84 71.78, 26.38 in-in-in SNCiii in-in ActLoopNT-in 3.1406 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.98, 165.73 APE9-dihe-na 69.33, 171.05 APE8-dihe-in -86.85, 130.82 APE8-rot-in 314.66 APE67-dihe-in -71.94, -20.16 -24.55, -52.13 APE12-dist-in 13.5473 APE11-dist-in 12.041 APE10-dist-in 7.3411 APE9-dist-in 3.5985 None PTR216 PTR216 XRAY 2.6 0.204 0.281 A 349.0 341.0 8 27 27 0 [[56, 340]] 1.0 3f88 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3F88B P49841 35 383 420.0 3HT:999 Type1 Active DFGin 6.9996 13.6509 BLAminus -143.93, 176.87 66.18, 95.41 -113.06, 21.86 281.61, 81.82 -72.47, -7.16 in-in in 8.7652 Saltbr-in 2.6705 HRD-in -64.13, -56.14 79.67, 28.55 in-in-in SNCiii in-in ActLoopNT-in 3.1764 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.92, 167.15 APE9-dihe-na 65.97, 165.61 APE8-dihe-in -80.57, 145.62 APE8-rot-in 308.56 APE67-dihe-in -71.31, -21.5 -44.75, -45.4 APE12-dist-in 13.509 APE11-dist-in 11.9668 APE10-dist-in 7.2567 APE9-dist-in 3.4061 None PTR216 PTR216 XRAY 2.6 0.204 0.281 B 349.0 341.0 8 27 27 0 [[56, 340]] 1.0 3f88 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.9e-70 243.0 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACCA P49841 35 385 420.0 7YG:1387 Type1 Active DFGin 7.1831 13.5808 BLAminus -136.28, 179.66 61.59, 88.25 -100.04, 20.56 281.3, 79.98 -65.9, -21.03 in-in in 8.3469 Saltbr-in 2.7616 HRD-in -66.74, -44.81 68.93, 1.06 in-in-in SNCiii in-in ActLoopNT-in 2.8975 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.14, 170.6 APE9-dihe-na 77.6, 138.09 APE8-dihe-in -85.62, 145.43 APE8-rot-in 296.7 APE67-dihe-inflip 94.96, -30.16 -47.88, 136.19 APE12-dist-in 13.0341 APE11-dist-in 10.957 APE10-dist-in 5.8889 APE9-dist-in 3.171 None None None XRAY 2.21 0.191 0.219 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acc Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACCB P49841 35 385 420.0 7YG:1386 Type1 Active DFGin 7.2279 13.5244 BLAminus -136.66, 179.59 61.79, 88.29 -99.73, 21.22 281.91, 80.18 -66.08, -22.29 in-in in 8.2447 Saltbr-in 2.8714 HRD-in -66.61, -45.06 69.24, 1.05 in-in-in SNCiii in-in ActLoopNT-in 2.8922 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -79.27, 172.02 APE9-dihe-na 75.79, 137.96 APE8-dihe-in -86.62, 146.41 APE8-rot-in 295.61 APE67-dihe-inflip 93.46, -30.62 -49.23, 136.97 APE12-dist-in 13.056 APE11-dist-in 11.009 APE10-dist-in 5.9124 APE9-dist-in 3.1824 None None None XRAY 2.21 0.191 0.219 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acc Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACDA P49841 35 385 420.0 GR9:1385 Type1 Active DFGin 7.1862 13.3568 BLAminus -142.44, 176.49 66.05, 88.14 -100.25, 16.93 286.04, 81.9 -64.04, -24.03 in-in in 8.3063 Saltbr-in 2.9365 HRD-in -63.25, -48.42 73.67, 5.76 in-in-in SNCiii in-in ActLoopNT-in 2.8831 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -87.94, 167.01 APE9-dihe-na 78.77, 128.64 APE8-dihe-in -74.85, 143.25 APE8-rot-in 302.95 APE67-dihe-inflip 99.55, -31.6 -49.31, 132.99 APE12-dist-in 12.8767 APE11-dist-in 10.8678 APE10-dist-in 5.9097 APE9-dist-in 3.2101 None None None XRAY 2.6 0.18 0.226 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acd Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACDB P49841 35 385 420.0 GR9:1385 Type1 Active DFGin 7.1414 13.3767 BLAminus -142.06, 177.81 64.05, 89.32 -100.31, 16.47 285.95, 82.89 -62.46, -26.08 in-in in 8.2225 Saltbr-in 2.9412 HRD-in -62.52, -48.15 72.88, 6.33 in-in-in SNCiii in-in ActLoopNT-in 2.8916 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -86.53, 167.96 APE9-dihe-na 77.33, 127.92 APE8-dihe-in -74.4, 143.25 APE8-rot-in 302.61 APE67-dihe-inflip 99.75, -32.16 -47.58, 132.33 APE12-dist-in 12.9284 APE11-dist-in 10.9465 APE10-dist-in 5.956 APE9-dist-in 3.211 None None None XRAY 2.6 0.18 0.226 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acd Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACGA P49841 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.0033 13.7172 BLAminus -136.29, 179.17 66.16, 92.5 -104.82, 26.85 285.89, 83.54 -71.26, -31.7 in-in in 8.2753 Saltbr-in 2.8663 HRD-in -62.3, -47.68 71.35, 0.06 in-in-in SNCiii in-in ActLoopNT-in 2.9897 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.26, 169.3 APE9-dihe-na 82.24, 136.71 APE8-dihe-in -91.92, 145.05 APE8-rot-in 294.1 APE67-dihe-inflip 97.4, -31.68 -47.8, 134.4 APE12-dist-in 12.9461 APE11-dist-in 10.9812 APE10-dist-in 5.9282 APE9-dist-in 3.2924 None None None XRAY 2.6 0.177 0.225 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acg Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACGB P49841 35 385 420.0 6LQ:1385 Type1 Active DFGin 7.0603 13.6101 BLAminus -135.89, 178.4 67.23, 92.34 -105.78, 27.09 285.23, 82.98 -71.05, -30.43 in-in in 8.3794 Saltbr-in 2.9801 HRD-in -63.74, -47.68 70.98, 1.15 in-in-in SNCiii in-in ActLoopNT-in 2.9729 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -92.69, 168.91 APE9-dihe-na 83.12, 137.88 APE8-dihe-in -91.66, 145.04 APE8-rot-in 292.39 APE67-dihe-inflip 98.28, -31.78 -48.39, 133.48 APE12-dist-in 12.9182 APE11-dist-in 10.9335 APE10-dist-in 5.917 APE9-dist-in 3.2904 None None None XRAY 2.6 0.177 0.225 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4acg Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACHA P49841 35 385 420.0 KDI:1386 Type1 Active DFGin 7.1308 13.8433 BLAminus -136.87, 179.55 65.58, 91.16 -104.2, 25.64 286.28, 84.07 -69.39, -35.2 in-in in 8.2337 Saltbr-in 2.9352 HRD-in -61.5, -48.36 72.42, -0.28 in-in-in SNCiii in-in ActLoopNT-in 2.9817 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -90.62, 166.44 APE9-dihe-na 83.56, 135.36 APE8-dihe-in -86.16, 143.31 APE8-rot-in 295.11 APE67-dihe-inflip 98.78, -32.06 -48.27, 133.26 APE12-dist-in 12.998 APE11-dist-in 11.0588 APE10-dist-in 5.9833 APE9-dist-in 3.3216 None None None XRAY 2.6 0.231 0.252 A 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4ach Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4ACHB P49841 35 385 420.0 KDI:1386 Type1 Active DFGin 7.0809 13.7158 BLAminus -136.91, 178.72 65.4, 91.31 -104.6, 25.63 285.26, 83.9 -68.47, -34.59 in-in in 8.3598 Saltbr-in 2.9378 HRD-in -60.93, -48.9 72.19, 0.38 in-in-in SNCiii in-in ActLoopNT-in 2.9768 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -91.1, 166.35 APE9-dihe-na 83.22, 136.77 APE8-dihe-in -87.16, 144.14 APE8-rot-in 294.96 APE67-dihe-inflip 98.6, -31.77 -49.65, 133.73 APE12-dist-in 12.9349 APE11-dist-in 10.9849 APE10-dist-in 5.9381 APE9-dist-in 3.2896 None None None XRAY 2.6 0.231 0.252 B 465.0 351.0 0 27 27 0 [[56, 340]] 1.0 4ach Homo sapiens CMGC_GSK3B_HUMAN CMGC 4.4e-70 242.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5OY4A P49841 36 385 420.0 B4K:504 Type1.5_Back Active DFGin 6.9988 13.8215 BLAminus -130.87, 178.64 57.91, 86.19 -95.47, 21.04 282.05, 81.42 -63.36, -27.5 in-in in 8.0884 Saltbr-in 2.722 HRD-in -68.24, -44.36 63.28, 15.03 in-in-in SNCiii in-in ActLoopNT-in 2.8882 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.23, 157.34 APE9-dihe-na 87.05, 159.63 APE8-dihe-in -83.83, 115.67 APE8-rot-in 295.36 APE67-dihe-in -60.03, -25.52 -23.01, -56.29 APE12-dist-in 13.5581 APE11-dist-in 11.6893 APE10-dist-in 7.0579 APE9-dist-in 3.4463 None PTR216 PTR216 XRAY 3.2 0.196 0.229 A 420.0 350.0 0 27 27 0 [[56, 340]] 1.0 5oy4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4IQ6B P49841 37 382 420.0 IQ6:501 Type1.5_Back Active DFGin 7.0646 14.0574 BLAminus -142.54, 175.49 69.06, 72.09 -88.69, 16.42 291.37, 92.47 -54.24, -38.91 in-in in 8.6089 Saltbr-in 2.85 HRD-in -66.96, -42.68 72.42, -15.31 in-in-in SNCiii in-in ActLoopNT-in 3.0094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.08, 167.69 APE9-dihe-na 81.68, 134.42 APE8-dihe-in -80.06, 146.43 APE8-rot-in 285.37 APE67-dihe-inflip 104.71, -27.8 -48.51, 126.71 APE12-dist-in 13.1481 APE11-dist-in 10.9082 APE10-dist-in 6.2442 APE9-dist-in 3.1149 None None None XRAY 3.12 0.188 0.227 B 426.0 332.0 14 27 27 0 [[56, 340]] 1.0 4iq6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.4e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6Y9SA P49841 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.7588 13.6151 ABAminus -144.68, -36.37 -95.25, 102.78 -104.54, 22.52 286.7, 80.89 -71.31, -22.3 in-in in 8.4688 Saltbr-in 2.731 HRD-in -69.96, -46.79 66.16, 22.69 in-in-out SNCiio in-out ActLoopNT-in 2.8691 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.41, 160.13 APE9-dihe-na 78.21, 163.56 APE8-dihe-in -74.57, 133.14 APE8-rot-out 174.03 APE67-dihe-in -60.25, -21.67 -45.31, -52.5 APE12-dist-in 13.3908 APE11-dist-in 11.6341 APE10-dist-in 6.8152 APE9-dist-in 3.2172 None PTR216 PTR216 XRAY 2.03 0.204 0.249 A 350.0 344.0 5 27 27 0 [[56, 340]] 1.0 6y9s Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6Y9SB P49841 35 383 420.0 OHK:401 Type1 Inactive DFGin 6.4656 13.6443 ABAminus -142.08, -29.11 -101.71, 107.32 -109.34, 26.02 290.64, 79.47 -70.13, -24.37 in-in in 8.6267 Saltbr-in 2.6258 HRD-in -62.98, -47.75 66.63, 19.7 in-in-out SNCiio in-out ActLoopNT-in 2.8706 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -149.54, 160.17 APE9-dihe-na 74.78, 156.26 APE8-dihe-in -72.21, 136.72 APE8-rot-out 179.96 APE67-dihe-in -63.91, -18.81 -47.88, -49.22 APE12-dist-in 13.498 APE11-dist-in 11.6964 APE10-dist-in 6.9402 APE9-dist-in 3.1721 None PTR216 PTR216 XRAY 2.03 0.204 0.249 B 350.0 340.0 9 27 27 0 [[56, 340]] 1.0 6y9s Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4NM0A P49841 26 383 420.0 ADP:60408 ATPlike Inactive DFGin 6.641 14.2129 BLAminus -133.4, -174.33 56.9, 85.51 -105.72, 27.83 287.31, 80.39 -76.48, -2.57 in-in in 8.774 Saltbr-in 3.0941 HRD-in -69.87, -45.12 67.03, 14.87 in-in-out SNCiio in-out ActLoopNT-in 2.9268 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -71.29, 168.54 APE9-dihe-na 70.19, 144.11 APE8-dihe-in -96.47, 160.21 APE8-rot-out 64.82 APE67-dihe-inflip 78.46, -27.02 -43.67, 149.07 APE12-dist-in 13.0905 APE11-dist-in 10.885 APE10-dist-in 6.5705 APE9-dist-in 3.1347 None None None XRAY 2.5 0.193 0.239 A 389.0 355.0 0 27 27 0 [[56, 340]] 1.0 4nm0 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.5e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8XN6B P49841 26 386 420.0 ANP:501 ATPlike Inactive DFGin 6.5384 13.6503 BLAminus -128.79, 173.26 73.68, 79.74 -95.9, 22.51 291.63, 80.46 -68.54, -21.83 in-in in 8.3292 Saltbr-in 2.8234 HRD-in -66.59, -53.03 79.09, 5.6 in-in-out SNCiio in-out ActLoopNT-in 2.9512 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -88.32, 165.9 APE9-dihe-na 83.63, 132.42 APE8-dihe-in -59.67, 147.17 APE8-rot-out 189.94 APE67-dihe-in -64.51, -21.68 -60.38, -49.59 APE12-dist-in 13.0235 APE11-dist-in 10.9696 APE10-dist-in 5.846 APE9-dist-in 3.0807 None None None XRAY 2.4 0.194 0.242 B 421.0 359.0 2 27 27 0 [[56, 340]] 1.0 8xn6 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1I09B P49841 37 382 420.0 No_ligand No_ligand Inactive DFGin 6.8606 14.0248 BLAminus -135.93, 178.35 61.75, 84.0 -100.67, 24.72 288.55, 74.93 -64.65, -15.56 in-in in 8.4828 Saltbr-in 2.7113 HRD-in -62.69, -41.62 66.11, 9.61 in-in-out SNCiio in-out ActLoopNT-in 2.9529 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.33, -45.22 APE9-dihe-na -71.78, 167.71 APE8-dihe-in -94.58, 171.33 APE8-rot-out 74.32 APE67-dihe-in -65.52, -17.17 -44.16, -80.97 APE12-dist-in 12.7638 APE11-dist-in 11.113 APE10-dist-in 6.2214 APE9-dist-in 3.37 None None None XRAY 2.7 0.242 0.274 B 420.0 341.0 5 27 27 0 [[56, 340]] 1.0 1i09 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6HK7A P49841 36 382 420.0 G8N:403 Type1 Inactive DFGin 7.1812 13.9264 BLAminus -137.45, -171.56 51.7, 92.53 -104.06, 22.16 271.05, 85.97 -65.5, -26.28 in-in in 8.435 Saltbr-in 2.7671 HRD-in -53.21, -66.83 89.97, 19.54 in-in-out SNCiio in-out ActLoopNT-in 2.957 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -85.73, 172.92 APE9-dihe-na 79.4, 146.18 APE8-dihe-in -92.07, 85.52 APE8-rot-in 243.21 APE67-dihe-out 35.1, -40.06 22.07, -158.21 APE12-dist-in 13.2898 APE11-dist-in 11.4463 APE10-dist-in 6.7807 APE9-dist-in 3.3203 None PTR216 PTR216 XRAY 3.2 0.204 0.286 A 347.0 347.0 0 27 27 0 [[56, 340]] 1.0 6hk7 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7SXHA P49841 37 383 420.0 D1E:501 Type1 Inactive DFGin 6.6502 13.9439 BLAminus -139.68, -175.41 60.2, 74.18 -88.43, 22.79 288.62, 86.11 -74.83, -15.81 in-in in 8.1673 Saltbr-in 2.8585 HRD-in -67.33, -47.27 70.7, 6.58 in-in-out SNCiio in-out ActLoopNT-in 2.863 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -126.8, 168.99 APE9-dihe-na 70.82, 157.42 APE8-dihe-in -70.74, 147.57 APE8-rot-out 190.63 APE67-dihe-in -58.92, -21.73 -57.82, -47.78 APE12-dist-in 13.7709 APE11-dist-in 11.9746 APE10-dist-in 7.3712 APE9-dist-in 3.4319 None PTR216 PTR216 XRAY 2.09 0.216 0.255 A 347.0 341.0 6 27 27 0 [[56, 340]] 1.0 7sxh Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.7e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3F7ZA P49841 35 383 420.0 34O:63000 Type1 Inactive DFGin 7.116 13.8181 BLAminus -134.47, 172.11 69.02, 81.68 -97.3, 19.46 284.39, 70.02 -68.92, -10.86 in-in in 8.4854 Saltbr-in 2.5753 HRD-in -62.81, -48.18 67.57, 12.21 in-in-out SNCiio in-out ActLoopNT-in 2.9498 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -139.18, 179.1 APE9-dihe-na 69.89, 157.17 APE8-dihe-in -75.28, 142.37 APE8-rot-out 185.5 APE67-dihe-in -55.86, -28.19 -45.56, -57.07 APE12-dist-in 13.5001 APE11-dist-in 12.029 APE10-dist-in 6.8149 APE9-dist-in 3.3141 None PTR216 PTR216 XRAY 2.4 0.206 0.253 A 350.0 339.0 10 27 27 0 [[56, 340]] 1.0 3f7z Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3SD0A P49841 35 384 420.0 TSK:400 Type1 Inactive DFGin 6.8934 13.6777 BLAminus -139.29, -172.59 62.67, 82.92 -94.93, 18.52 283.9, 73.87 -68.11, -17.74 in-in in 8.4187 Saltbr-in 2.8235 HRD-in -68.02, -47.17 76.6, 11.56 in-in-out SNCiio in-out ActLoopNT-in 2.7996 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -82.28, 176.65 APE9-dihe-na 71.42, 130.7 APE8-dihe-in -100.53, 166.25 APE8-rot-out 29.1 APE67-dihe-inflip 91.12, -25.82 -31.67, 128.67 APE12-dist-in 12.9104 APE11-dist-in 10.8103 APE10-dist-in 5.7793 APE9-dist-in 3.0415 None None None XRAY 2.7 0.179 0.254 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 3sd0 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3ZDIA P49841 36 384 420.0 UGJ:61386 Type1 Inactive DFGin 7.0898 14.0106 BLAminus -139.08, 169.73 59.85, 93.36 -102.57, 31.03 284.51, 75.61 -74.44, -6.01 in-in in 8.7186 Saltbr-in 2.7736 HRD-in -66.47, -49.36 70.61, -12.05 in-in-out SNCiio in-out ActLoopNT-in 2.8737 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.6, -176.4 APE9-dihe-na 57.27, -141.25 APE8-dihe-in -136.89, 135.85 APE8-rot-out 188.96 APE67-dihe-in -60.18, -28.67 -48.24, -43.31 APE12-dist-in 13.7771 APE11-dist-in 12.1156 APE10-dist-in 7.549 APE9-dist-in 3.0939 None PTR216 PTR216 XRAY 2.645 0.204 0.242 A 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 3zdi Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4B7TA P49841 35 384 420.0 CWT:1385 Type1 Inactive DFGin 6.733 14.135 BLAminus -139.29, -173.55 55.51, 80.28 -97.98, 26.2 284.11, 78.64 -70.02, -22.23 in-in in 8.8256 Saltbr-in 2.732 HRD-in -65.66, -45.08 68.98, -4.07 in-in-out SNCiio in-out ActLoopNT-in 3.0218 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -80.96, 174.72 APE9-dihe-na 79.02, 153.66 APE8-dihe-in -90.72, 141.08 APE8-rot-out 219.61 APE67-dihe-inflip 82.28, -25.01 -65.77, 158.92 APE12-dist-in 13.1502 APE11-dist-in 11.3146 APE10-dist-in 6.5521 APE9-dist-in 3.1216 None None None XRAY 2.772 0.197 0.235 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 4b7t Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6HK3A P49841 35 384 420.0 G8B:401 Type1 Inactive DFGin 6.9186 13.7488 BLAminus -140.26, -177.42 53.43, 89.98 -101.44, 26.95 281.28, 77.81 -71.94, -4.92 in-in in 8.2647 Saltbr-in 2.5202 HRD-in -65.54, -43.12 59.71, 15.8 in-in-out SNCiio in-out ActLoopNT-in 2.9314 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -120.05, -174.23 APE9-dihe-na 65.54, 142.28 APE8-dihe-in -62.37, 137.73 APE8-rot-out 183.0 APE67-dihe-in -57.53, -32.37 -39.19, -57.21 APE12-dist-in 13.3885 APE11-dist-in 11.7623 APE10-dist-in 6.4209 APE9-dist-in 3.2183 None PTR216 PTR216 XRAY 2.35 0.206 0.234 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6hk3 Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6Y9RA P49841 35 384 420.0 OH8:401 Type1 Inactive DFGin 7.2128 13.9564 BLAminus -128.7, 177.14 64.74, 83.75 -99.31, 22.7 285.39, 75.74 -67.18, -22.12 in-in in 8.3866 Saltbr-in 2.7599 HRD-in -68.2, -47.94 70.12, 17.05 in-in-out SNCiio in-out ActLoopNT-in 2.9695 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -147.41, 164.13 APE9-dihe-na 71.55, 162.91 APE8-dihe-in -81.0, 136.61 APE8-rot-out 173.09 APE67-dihe-in -62.95, -25.51 -45.24, -50.14 APE12-dist-in 13.6836 APE11-dist-in 12.0385 APE10-dist-in 7.353 APE9-dist-in 3.2948 None PTR216 PTR216 XRAY 2.08 0.191 0.226 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 6y9r Homo sapiens CMGC_GSK3B_HUMAN CMGC 1.8e-70 243.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1O9UA P49841 35 384 420.0 ADZ:1386 Type1 Inactive DFGin 6.69 14.4088 BLAminus -135.58, -170.77 57.68, 80.28 -97.17, 18.56 286.56, 73.24 -63.89, -4.57 in-in in 8.9184 Saltbr-in 3.2524 HRD-in -60.54, -48.22 66.04, 11.65 in-in-out SNCiio in-out ActLoopNT-in 2.9648 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.51, 167.48 APE9-dihe-na 74.14, -178.83 APE8-dihe-in -103.59, 140.85 APE8-rot-out 179.41 APE67-dihe-in -52.99, -22.64 -16.1, -87.79 APE12-dist-in 13.762 APE11-dist-in 11.7056 APE10-dist-in 7.3617 APE9-dist-in 2.8623 None PTR216 PTR216 XRAY 2.4 0.233 0.26 A 350.0 350.0 0 27 27 0 [[56, 340]] 1.0 1o9u Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-69 240.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9PE9A P49841 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.0716 14.2287 BLAminus -128.7, -179.96 59.31, 84.1 -97.11, 26.91 283.64, 74.63 -73.69, -18.15 in-in in 8.351 Saltbr-in 2.7255 HRD-in -68.62, -45.57 65.7, 16.55 in-in-out SNCiio in-out ActLoopNT-in 2.9248 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -143.94, 165.33 APE9-dihe-na 76.34, 152.28 APE8-dihe-in -69.82, 130.62 APE8-rot-out 176.66 APE67-dihe-in -58.68, -26.71 -39.69, -56.4 APE12-dist-in 13.2799 APE11-dist-in 11.7578 APE10-dist-in 7.0929 APE9-dist-in 3.1547 None PTR216 PTR216 XRAY 2.11 0.221 0.247 A 359.0 332.0 13 27 27 0 [[56, 340]] 1.0 9pe9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9PE9B P49841 36 382 420.0 A1CIF:900 Type1 Inactive DFGin 7.0575 14.2183 BLAminus -128.76, -179.81 59.6, 84.42 -97.78, 27.09 283.79, 74.38 -73.25, -17.71 in-in in 8.3532 Saltbr-in 2.7132 HRD-in -68.49, -44.82 64.55, 18.32 in-in-out SNCiio in-out ActLoopNT-in 2.9402 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -144.27, 163.74 APE9-dihe-na 77.64, 152.05 APE8-dihe-in -69.14, 130.82 APE8-rot-out 177.12 APE67-dihe-in -58.92, -26.81 -39.96, -55.88 APE12-dist-in 13.3604 APE11-dist-in 11.8241 APE10-dist-in 7.1609 APE9-dist-in 3.1723 None PTR216 PTR216 XRAY 2.11 0.221 0.247 B 359.0 332.0 13 27 27 0 [[56, 340]] 1.0 9pe9 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7Z1FA P49841 28 383 420.0 3NG:60401 Type1 Inactive DFGin 7.1722 14.3874 BLAminus -140.61, -172.17 56.83, 67.31 -90.44, 24.59 283.96, 78.9 -70.58, -34.2 in-in in 8.5891 Saltbr-in 2.7064 HRD-in -70.71, -48.08 68.23, 20.67 in-in-out SNCiio in-out ActLoopNT-in 2.8765 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -121.77, -56.1 APE9-dihe-na -73.95, 173.6 APE8-dihe-in -71.54, 133.95 APE8-rot-out 205.24 APE67-dihe-in -54.78, -22.55 -52.86, -47.6 APE12-dist-in 13.7113 APE11-dist-in 11.9213 APE10-dist-in 7.2574 APE9-dist-in 3.4781 None PTR216 PTR216 XRAY 3.0 0.224 0.249 A 364.0 354.0 2 27 27 0 [[56, 340]] 1.0 7z1f Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 7Z1FB P49841 38 382 420.0 3NG:60401 Type1 Inactive DFGin 6.8696 14.4685 BLAminus -141.12, -171.82 52.8, 73.11 -90.49, 20.89 285.47, 81.84 -62.59, -35.1 in-in in 9.0255 Saltbr-in 2.7633 HRD-in -68.41, -52.97 70.54, 14.05 in-in-out SNCiio in-out ActLoopNT-in 3.0394 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.34, -53.99 APE9-dihe-na -75.88, 165.71 APE8-dihe-in -64.92, 136.76 APE8-rot-out 179.7 APE67-dihe-in -58.44, -19.64 -54.95, -47.33 APE12-dist-in 13.527 APE11-dist-in 11.8588 APE10-dist-in 7.1538 APE9-dist-in 3.5583 None PTR216 PTR216 XRAY 3.0 0.224 0.249 B 364.0 321.0 24 27 27 0 [[56, 340]] 1.0 7z1f Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8AV1A P49841 27 381 420.0 O9L:406 Type1 Inactive DFGin 7.0048 13.8018 BLAminus -134.83, 176.12 61.29, 85.31 -97.92, 27.58 284.57, 74.39 -70.18, -20.31 in-in in 8.4199 Saltbr-in 2.6588 HRD-in -72.82, -53.06 75.09, 11.93 in-in-out SNCiio in-out ActLoopNT-in 2.8108 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -162.3, 153.55 APE9-dihe-na 79.71, 140.85 APE8-dihe-in -55.94, 133.71 APE8-rot-out 187.25 APE67-dihe-in -61.14, -25.49 -46.06, -52.45 APE12-dist-in 13.2676 APE11-dist-in 11.4128 APE10-dist-in 6.8843 APE9-dist-in 3.0607 None PTR216 PTR216 XRAY 2.15 0.18 0.21 A 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8av1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8AV1B P49841 27 381 420.0 O9L:405 Type1 Inactive DFGin 7.0411 13.8178 BLAminus -134.53, 176.17 61.15, 83.84 -96.42, 28.03 285.62, 75.68 -72.4, -19.61 in-in in 8.3507 Saltbr-in 2.6481 HRD-in -70.84, -52.05 73.58, 16.86 in-in-out SNCiio in-out ActLoopNT-in 2.809 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -159.36, 152.7 APE9-dihe-na 82.35, 142.4 APE8-dihe-in -57.42, 133.83 APE8-rot-out 184.71 APE67-dihe-in -59.68, -24.96 -48.86, -51.78 APE12-dist-in 13.2597 APE11-dist-in 11.441 APE10-dist-in 6.8498 APE9-dist-in 3.0597 None PTR216 PTR216 XRAY 2.15 0.18 0.21 B 365.0 351.0 4 27 27 0 [[56, 340]] 1.0 8av1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6GN1A P49841 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.9399 14.3347 BLAminus -135.29, 179.1 59.47, 89.49 -98.73, 29.98 286.18, 72.49 -75.74, -10.8 in-in in 8.608 Saltbr-in 3.0396 HRD-in -74.24, -44.22 64.59, 22.98 in-in-out SNCiio in-out ActLoopNT-in 2.9401 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -143.03, -18.16 APE9-dihe-na -103.04, 175.18 APE8-dihe-in -67.81, 136.03 APE8-rot-out 187.31 APE67-dihe-in -61.67, -27.65 -44.51, -52.79 APE12-dist-out 14.0101 APE11-dist-in 12.3553 APE10-dist-in 7.3869 APE9-dist-in 3.5875 None PTR216 PTR216 XRAY 2.6 0.224 0.259 A 368.0 340.0 8 27 27 0 [[56, 340]] 1.0 6gn1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6GN1B P49841 36 383 420.0 F4N:502 Type1 Inactive DFGin 6.9439 14.317 BLAminus -135.3, 179.27 59.56, 89.49 -98.78, 30.1 286.37, 73.15 -75.82, -10.91 in-in in 8.6216 Saltbr-in 3.0339 HRD-in -74.17, -44.23 64.47, 22.86 in-in-out SNCiio in-out ActLoopNT-in 2.9462 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oiii APE10-dihe-na -129.39, -14.9 APE9-dihe-na -108.68, -179.33 APE8-dihe-in -68.02, 134.54 APE8-rot-out 210.75 APE67-dihe-in -62.25, -27.68 -44.3, -51.95 APE12-dist-out 14.0238 APE11-dist-in 12.1834 APE10-dist-in 7.4033 APE9-dist-in 3.6999 None PTR216 PTR216 XRAY 2.6 0.224 0.259 B 368.0 340.0 8 27 27 0 [[56, 340]] 1.0 6gn1 Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.1e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 2O5KA P49841 35 384 420.0 HBM:0 Type1 Inactive DFGin 6.7209 13.939 BLAminus -127.34, -179.9 54.97, 85.31 -97.88, 27.22 279.56, 72.26 -63.78, -54.26 in-in in 8.3524 Saltbr-in 3.3761 HRD-in -66.17, -47.55 59.21, 39.45 in-in-out SNCiio in-out ActLoopNT-in 2.9464 ActLoopCT-out nonTYR APEdihe_aaoii APEdist_iiii APE10-dihe-na 170.93, -156.16 APE9-dihe-na 30.47, -152.36 APE8-dihe-out -134.5, -176.14 APE8-rot-in 306.82 APE67-dihe-in -73.05, -7.32 -59.58, -80.34 APE12-dist-in 12.6788 APE11-dist-in 9.1805 APE10-dist-in 5.885 APE9-dist-in 3.0373 None None None XRAY 3.2 0.251 0.309 A 372.0 350.0 0 27 27 0 [[56, 340]] 1.0 2o5k Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.2e-70 243.4 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 1UV5A P49841 35 383 420.0 BRW:1383 Type1 Inactive DFGin 6.9015 14.0788 BLAminus -144.35, -177.14 59.35, 81.04 -94.26, 27.94 286.0, 72.94 -59.18, -36.48 in-in in 8.299 Saltbr-in 2.5611 HRD-in -65.61, -42.55 70.5, 0.98 in-in-out SNCiio in-out ActLoopNT-in 2.8842 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -98.47, 172.31 APE9-dihe-na 85.56, 133.89 APE8-dihe-in -66.16, 126.55 APE8-rot-out 191.14 APE67-dihe-in -61.71, -20.34 -21.78, -65.88 APE12-dist-in 12.7631 APE11-dist-in 10.9893 APE10-dist-in 5.7154 APE9-dist-in 3.2357 None None None XRAY 2.8 0.193 0.226 A 350.0 349.0 0 27 27 0 [[56, 340]] 1.0 1uv5 Homo sapiens CMGC_GSK3B_HUMAN CMGC 7.4e-70 241.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6GJOA P49841 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.1764 14.254 BLAminus -136.61, 169.82 63.4, 86.22 -103.46, 25.41 276.6, 83.48 -69.91, -39.25 in-in in 8.6359 Saltbr-in 2.8102 HRD-in -57.84, -41.83 58.98, 16.97 in-in-out SNCiio in-out ActLoopNT-in 3.0119 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.92, 162.15 APE9-dihe-na 71.93, 161.47 APE8-dihe-in -78.01, 132.19 APE8-rot-out 37.25 APE67-dihe-in -62.57, -18.8 -29.28, -56.31 APE12-dist-in 13.62 APE11-dist-in 11.8617 APE10-dist-in 6.9452 APE9-dist-in 3.4449 None None None XRAY 2.91 0.218 0.237 A 414.0 349.0 0 27 27 0 [[56, 340]] 1.0 6gjo Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 6GJOB P49841 35 383 420.0 F1B:501 Type1 Inactive DFGin 7.4783 14.2513 BLAminus -136.82, 170.18 63.9, 83.46 -101.86, 22.92 278.62, 83.32 -68.81, -38.47 in-in in 8.4049 Saltbr-in 3.0839 HRD-in -57.78, -41.9 58.99, 17.22 in-in-out SNCiio in-out ActLoopNT-in 3.0124 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.67, 163.61 APE9-dihe-na 73.76, 161.78 APE8-dihe-in -77.57, 137.96 APE8-rot-out 184.23 APE67-dihe-in -62.17, -20.4 -36.29, -55.68 APE12-dist-in 13.4495 APE11-dist-in 11.7843 APE10-dist-in 6.8542 APE9-dist-in 3.4366 None None None XRAY 2.91 0.218 0.237 B 414.0 343.0 6 27 27 0 [[56, 340]] 1.0 6gjo Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.1e-70 242.9 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 3M1SA P49841 35 385 420.0 DW1:421 Type1 Inactive DFGin 7.021 13.7099 BLAminus -149.21, -179.05 55.83, 87.87 -101.26, 23.04 292.92, 65.81 -62.39, -0.11 in-in in 8.7264 Saltbr-in 2.9756 HRD-in -71.98, -44.05 63.65, 18.92 in-in-out SNCiio in-out ActLoopNT-in 3.0324 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -100.39, 171.9 APE9-dihe-na 82.48, 144.37 APE8-dihe-in -94.3, 96.58 APE8-rot-in 285.71 APE67-dihe-out 116.42, -45.78 9.38, 103.41 APE12-dist-in 13.6493 APE11-dist-in 11.7091 APE10-dist-in 6.707 APE9-dist-in 3.4451 None None None XRAY 3.134 0.171 0.228 A 420.0 348.0 3 27 27 0 [[56, 340]] 1.0 3m1s Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 9HUKA P49841 25 385 420.0 A1IXL:501 Type1 Inactive DFGin 7.0533 14.0777 BLAminus -135.25, -177.02 57.0, 94.14 -110.6, 20.82 285.12, 72.82 -66.1, -13.46 in-out in 8.1101 Saltbr-out 3.6586 HRD-in -70.91, -39.46 63.28, 18.66 out-in-in SNCoii in-in ActLoopNT-in 3.1574 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -82.9, 179.26 APE9-dihe-na 68.03, 135.17 APE8-dihe-in -69.47, 168.34 APE8-rot-in 295.64 APE67-dihe-inflip 67.51, -44.25 -66.67, 175.58 APE12-dist-in 13.1194 APE11-dist-in 10.9456 APE10-dist-in 5.924 APE9-dist-in 3.2016 None None None XRAY 3.5 0.219 0.25 A 442.0 361.0 0 27 27 0 [[56, 340]] 1.0 9huk Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.8e-70 242.6 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4J71A P49841 36 383 420.0 1JX:501 Type1 Inactive DFGin 6.9292 14.0341 BLAminus -134.37, 178.91 60.63, 80.22 -96.96, 24.92 284.72, 75.18 -68.29, -15.66 in-in in 8.4479 Saltbr-in 3.0956 HRD-in -74.9, -47.0 72.06, 4.98 in-in-out SNCiio in-out ActLoopNT-in 2.7141 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.32, 163.35 APE9-dihe-na 76.45, 151.25 APE8-dihe-in -65.19, 140.55 APE8-rot-out 188.84 APE67-dihe-in -55.99, -28.06 -50.85, -54.43 APE12-dist-in 13.3964 APE11-dist-in 11.8958 APE10-dist-in 7.1633 APE9-dist-in 2.9983 None PTR216 PTR216 XRAY 2.31 0.191 0.234 A 424.0 348.0 0 27 27 0 [[56, 340]] 1.0 4j71 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4J71B P49841 36 383 420.0 1JX:501 Type1 Inactive DFGin 7.043 13.8316 BLAminus -140.62, 179.7 59.87, 90.62 -104.73, 25.33 288.76, 76.25 -66.71, -17.33 in-in in 8.3305 Saltbr-in 2.8961 HRD-in -77.92, -46.29 72.36, 3.7 in-in-out SNCiio in-out ActLoopNT-in 2.834 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -141.74, 169.96 APE9-dihe-na 69.52, 149.79 APE8-dihe-in -68.04, 134.18 APE8-rot-out 173.06 APE67-dihe-in -53.62, -29.43 -43.81, -55.09 APE12-dist-in 13.2129 APE11-dist-in 11.9572 APE10-dist-in 7.1265 APE9-dist-in 2.9738 None PTR216 PTR216 XRAY 2.31 0.191 0.234 B 424.0 348.0 0 27 27 0 [[56, 340]] 1.0 4j71 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5HLNB P49841 37 383 420.0 65C:501 Type1 Inactive DFGin 6.8475 13.3316 BLAminus -143.06, -174.61 53.09, 90.34 -103.45, 33.01 288.97, 83.64 -74.69, -34.84 in-in in 8.9958 Saltbr-in 2.6044 HRD-in -68.15, -40.04 65.1, 19.28 in-in-out SNCiio in-out ActLoopNT-in 2.9629 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -137.65, -62.86 APE9-dihe-na -78.36, 171.11 APE8-dihe-in -56.52, 151.93 APE8-rot-out 161.85 APE67-dihe-in -56.43, -28.42 -72.24, -45.62 APE12-dist-in 13.5983 APE11-dist-in 11.8341 APE10-dist-in 7.3737 APE9-dist-in 3.4156 None PTR216 PTR216 XRAY 3.1 0.173 0.236 B 424.0 347.0 0 27 27 0 [[56, 340]] 1.0 5hln Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.3e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 5OY4B P49841 30 384 420.0 B4K:502 Type1.5_Back Inactive DFGin 7.0077 13.7409 BLAminus -131.51, 177.88 58.43, 85.84 -94.85, 21.53 281.4, 81.96 -63.5, -26.63 in-in in 7.965 Saltbr-in 2.7509 HRD-in -68.43, -44.24 63.59, 14.9 in-in-out SNCiio in-out ActLoopNT-in 2.8689 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -145.82, 158.71 APE9-dihe-na 86.22, 156.23 APE8-dihe-in -75.92, 122.37 APE8-rot-out 226.12 APE67-dihe-in -60.14, -24.48 -28.85, -54.97 APE12-dist-in 13.5037 APE11-dist-in 11.6211 APE10-dist-in 7.0093 APE9-dist-in 3.404 None PTR216 PTR216 XRAY 3.2 0.196 0.229 B 420.0 354.0 1 27 27 0 [[56, 340]] 1.0 5oy4 Homo sapiens CMGC_GSK3B_HUMAN CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 8QJIA P49841 36 381 420.0 VNG:401 Type1 Inactive DFGin 6.9495 14.1959 None -92.57, -90.5 -72.82, 155.73 -144.36, 17.02 276.05, 102.26 -73.85, -19.5 in-in in 8.3845 Saltbr-in 2.6943 HRD-in -65.27, -43.08 63.67, 22.78 in-in-out SNCiio in-out ActLoopNT-in 3.34 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -115.54, 179.17 APE9-dihe-na 65.4, 161.24 APE8-dihe-in -68.89, 150.02 APE8-rot-out 175.4 APE67-dihe-in -64.21, -18.12 -58.7, -47.99 APE12-dist-in 13.3857 APE11-dist-in 12.0024 APE10-dist-in 7.07 APE9-dist-in 3.4473 None PTR216 PTR216 XRAY 3.02 0.253 0.289 A 364.0 340.0 6 27 27 0 [[56, 340]] 1.0 8qji Homo sapiens CMGC_GSK3B_HUMAN CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_HUMAN 4DITA P49841 35 387 420.0 0KD:501 Type1 None DFGin 6.8051 13.9479 BLAminus -145.37, 179.76 65.92, 81.37 -105.97, 22.54 288.96, 82.14 -68.29, -17.95 in-in in 8.8255 Saltbr-in 2.717 HRD-in -69.87, -50.6 73.87, 5.2 in-in-none SNCiin in-none ActLoopNT-in 2.9388 ActLoopCT-none nonTYR APEdihe_aannn APEdist_iinn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 14.5 999.0, 999.0 APE12-dist-in 13.4889 APE11-dist-in 10.3847 APE10-dist-none 999.0 APE9-dist-none 999.0 None PTR216 PTR216 XRAY 2.6 0.243 0.304 A 382.0 329.0 24 27 23 4 [[56, 340]] 1.0 4dit Homo sapiens CMGC_GSK3B_HUMAN CMGC 2.4e-70 243.3 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 8VMFA Q9WV60 27 383 420.0 ADP:60504 ATPlike Active DFGin 6.6121 14.0996 BLAminus -148.4, -167.57 58.53, 66.72 -90.57, 24.21 287.49, 78.37 -75.04, -7.89 in-in in 8.6601 Saltbr-in 2.678 HRD-in -67.34, -47.3 70.6, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.8401 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.01, -20.74 APE9-dihe-na -93.16, -168.14 APE8-dihe-in -112.8, 164.36 APE8-rot-in 304.6 APE67-dihe-inflip 78.98, -8.38 -56.8, 140.56 APE12-dist-in 13.183 APE11-dist-in 10.9487 APE10-dist-in 6.514 APE9-dist-in 3.3085 None None None XRAY 2.5 0.21 0.251 A 364.0 354.0 0 27 27 0 [[56, 340]] 1.0 8vmf Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 8VMGA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 7.0002 13.9987 BLAminus -139.67, -176.86 60.44, 73.06 -89.27, 27.07 283.1, 81.19 -73.23, -12.63 in-in in 8.478 Saltbr-in 2.6881 HRD-in -67.64, -48.38 72.75, 3.36 in-in-in SNCiii in-in ActLoopNT-in 2.8435 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.26, 164.63 APE9-dihe-na 72.45, 142.8 APE8-dihe-in -66.41, 146.08 APE8-rot-in 307.07 APE67-dihe-in -64.3, -22.81 -57.43, -46.54 APE12-dist-in 13.2782 APE11-dist-in 11.627 APE10-dist-in 6.9412 APE9-dist-in 2.9838 None None None XRAY 2.45 0.195 0.23 A 364.0 358.0 0 27 27 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 8VMEA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 6.469 13.8439 BLAminus -131.0, -171.33 63.41, 73.0 -92.56, 22.88 289.27, 83.61 -79.03, -1.02 in-in in 8.7532 Saltbr-in 2.7802 HRD-in -67.9, -47.67 70.4, 7.52 in-in-in SNCiii in-in ActLoopNT-in 2.7313 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.18, 168.01 APE9-dihe-na 68.83, 161.19 APE8-dihe-in -90.7, 152.54 APE8-rot-in 290.93 APE67-dihe-inflip 82.32, -22.26 -51.38, 150.9 APE12-dist-in 13.2878 APE11-dist-in 12.0712 APE10-dist-in 6.9342 APE9-dist-in 3.2916 None None None XRAY 2.3 0.183 0.23 A 365.0 355.0 0 27 27 0 [[56, 340]] 1.0 8vme Mus musculus CMGC_GSK3B_MOUSE CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 4NU1A Q9WV60 6 383 420.0 ADP:405 ATPlike Active DFGin 6.1094 13.6771 BLAminus -140.27, -172.8 60.29, 88.19 -108.14, 24.39 289.57, 88.21 -68.01, -14.99 in-in in 8.691 Saltbr-in 2.7928 HRD-in -66.76, -45.51 62.96, 19.85 in-in-in SNCiii in-in ActLoopNT-in 2.6824 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.38, 172.68 APE9-dihe-na 66.76, 153.81 APE8-dihe-in -82.08, 156.46 APE8-rot-in 299.93 APE67-dihe-inflip 76.53, -25.22 -54.39, 158.45 APE12-dist-in 13.5101 APE11-dist-in 11.6207 APE10-dist-in 7.1263 APE9-dist-in 3.1496 None SEP9 SEP9 XRAY 2.5 0.194 0.245 A 389.0 357.0 2 27 27 0 [[56, 340]] 1.0 4nu1 Mus musculus CMGC_GSK3B_MOUSE CMGC 2.5e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3D Q9WV60 36 382 420.0 No_ligand No_ligand Active DFGin 6.8462 14.3954 BLAminus -141.83, -176.77 60.2, 77.49 -89.39, 22.71 281.69, 81.03 -67.16, -17.62 in-in in 8.5972 Saltbr-in 2.9198 HRD-in -66.38, -49.02 71.39, 7.08 in-in-in SNCiii in-in ActLoopNT-in 3.0257 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.65, -50.64 APE9-dihe-na -86.99, 177.5 APE8-dihe-in -52.77, 135.95 APE8-rot-in 241.34 APE67-dihe-in -60.13, -26.01 -56.25, -47.64 APE12-dist-in 13.5374 APE11-dist-in 11.7665 APE10-dist-in 7.2779 APE9-dist-in 3.256 None PTR216 PTR216 XRAY 2.14 0.192 0.226 D 420.0 333.0 13 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 5AIRB Q9WV60 22 384 420.0 No_ligand No_ligand Active DFGin 7.2132 14.6827 BLAminus -135.77, 173.37 62.69, 75.87 -94.37, 22.65 282.98, 71.43 -62.58, -24.12 in-in in 8.743 Saltbr-in 3.1941 HRD-in -72.7, -48.08 74.63, 8.38 in-in-in SNCiii in-in ActLoopNT-in 3.0783 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.78, -34.05 APE9-dihe-na -91.23, 159.66 APE8-dihe-in -80.14, 164.39 APE8-rot-in 286.43 APE67-dihe-in -76.71, -12.41 -69.97, -37.36 APE12-dist-in 12.7248 APE11-dist-in 10.7707 APE10-dist-in 5.7984 APE9-dist-in 3.2801 None None None XRAY 2.53 0.215 0.26 B 430.0 361.0 2 27 27 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 5AIRA Q9WV60 26 383 420.0 No_ligand No_ligand Inactive DFGin 6.9865 14.3368 ABAminus -142.69, -19.87 -113.16, 97.17 -94.15, 12.11 276.77, 85.56 -67.43, -12.28 in-in in 8.7803 Saltbr-in 2.843 HRD-in -76.77, -43.42 72.44, 6.11 in-in-in SNCiii in-in ActLoopNT-in 2.9198 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.55, -31.48 APE9-dihe-na -99.45, 158.56 APE8-dihe-in -79.74, 161.48 APE8-rot-in 283.68 APE67-dihe-in -67.71, -13.15 -61.56, -52.85 APE12-dist-in 12.7446 APE11-dist-in 10.5629 APE10-dist-in 5.8016 APE9-dist-in 3.2157 None None None XRAY 2.53 0.215 0.26 A 430.0 353.0 2 27 27 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 8VMGB Q9WV60 35 383 420.0 No_ligand No_ligand Inactive DFGin 7.0355 14.1047 BLAminus -148.77, -175.26 61.58, 69.86 -88.49, 24.73 286.58, 81.46 -68.41, -21.39 in-in in 8.5062 Saltbr-in 2.8221 HRD-in -64.17, -52.24 74.94, 4.57 in-in-out SNCiio in-out ActLoopNT-in 2.7514 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -148.65, 168.87 APE9-dihe-na 71.82, 140.54 APE8-dihe-in -63.28, 148.93 APE8-rot-out 168.42 APE67-dihe-in -62.52, -22.04 -64.28, -46.93 APE12-dist-in 13.4966 APE11-dist-in 11.8072 APE10-dist-in 7.0074 APE9-dist-in 3.0097 None None None XRAY 2.45 0.195 0.23 B 364.0 349.0 0 27 27 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3C Q9WV60 37 383 420.0 No_ligand No_ligand Inactive DFGin 7.0852 14.2465 BLAminus -138.84, 177.7 70.47, 68.34 -81.63, 23.64 278.71, 79.84 -68.29, -26.67 in-in in 8.5431 Saltbr-in 3.0998 HRD-in -63.75, -49.26 68.09, 4.78 in-in-out SNCiio in-out ActLoopNT-in 2.9308 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.25, -51.04 APE9-dihe-na -75.73, 169.64 APE8-dihe-in -64.7, 134.47 APE8-rot-out 205.91 APE67-dihe-in -59.9, -28.79 -47.43, -50.42 APE12-dist-in 13.3567 APE11-dist-in 11.8202 APE10-dist-in 6.6175 APE9-dist-in 3.4159 None PTR216 PTR216 XRAY 2.14 0.192 0.226 C 420.0 332.0 14 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3A Q9WV60 36 387 420.0 MRI:501 Type1 Inactive DFGin 6.8942 14.102 BLAminus -136.0, 177.47 66.33, 76.64 -88.44, 20.33 285.85, 84.43 -66.44, -23.98 in-in in 8.8767 Saltbr-in 2.9541 HRD-in -71.52, -49.56 71.35, 12.25 in-in-out SNCiio in-out ActLoopNT-in 3.032 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.99, -47.87 APE9-dihe-na -84.23, -172.24 APE8-dihe-in -75.59, 135.74 APE8-rot-out 167.98 APE67-dihe-in -65.02, -21.79 -52.52, -47.78 APE12-dist-in 13.6917 APE11-dist-in 12.0236 APE10-dist-in 7.3136 APE9-dist-in 3.3344 None PTR216 PTR216 XRAY 2.14 0.192 0.226 A 420.0 348.0 4 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3B Q9WV60 36 384 420.0 MRI:501 Type1 Inactive DFGin 6.7389 14.0903 BLAminus -133.31, 179.77 64.96, 75.18 -85.96, 22.4 281.26, 80.21 -65.67, -27.09 in-in in 8.9797 Saltbr-in 3.0191 HRD-in -70.11, -50.99 71.74, 15.55 in-in-out SNCiio in-out ActLoopNT-in 2.9225 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.24, -38.47 APE9-dihe-na -87.03, 178.23 APE8-dihe-in -68.15, 134.76 APE8-rot-out 177.54 APE67-dihe-in -64.59, -23.54 -47.57, -47.97 APE12-dist-in 13.6259 APE11-dist-in 11.9079 APE10-dist-in 6.6939 APE9-dist-in 3.4142 None PTR216 PTR216 XRAY 2.14 0.192 0.226 B 420.0 344.0 5 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B A0A125YY75_TOXGG 9HVXA A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.8122 13.7389 BLAminus -151.79, -170.99 58.28, 71.83 -90.67, 23.31 282.96, 81.43 -68.24, -23.58 in-in in 7.973 Saltbr-in 2.6702 HRD-in -79.27, -44.62 69.75, 6.05 in-in-out SNCiio in-out ActLoopNT-in 2.9155 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -133.04, -39.68 APE9-dihe-na -85.38, 168.26 APE8-dihe-in -65.75, 139.05 APE8-rot-out 179.82 APE67-dihe-in -62.31, -27.06 -57.82, -44.69 APE12-dist-in 13.5047 APE11-dist-in 11.8681 APE10-dist-in 7.3712 APE9-dist-in 3.4994 None PTR211 PTR211 XRAY 2.1 0.203 0.25 A 350.0 323.0 16 27 27 0 [[47, 344]] 1.0 9hvx Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 6.4e-71 244.9 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6A A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.5538 13.5143 BLAminus -159.29, -172.81 63.26, 75.9 -98.23, 18.12 289.64, 83.03 -60.9, -17.5 in-in in 8.2475 Saltbr-in 2.9128 HRD-in -74.22, -42.3 70.91, -2.75 in-in-out SNCiio in-out ActLoopNT-in 2.7786 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -107.29, 145.01 APE9-dihe-na -102.07, 19.34 APE8-dihe-in -80.82, 138.15 APE8-rot-out 53.99 APE67-dihe-in -80.29, -18.75 -104.8, -54.34 APE12-dist-none 999.0 APE11-dist-in 10.1113 APE10-dist-in 7.183 APE9-dist-out 8.8047 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 A 373.0 332.0 7 27 24 3 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6B A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.9687 13.759 BLAminus -158.71, -175.52 61.04, 75.48 -97.8, 20.68 289.3, 83.48 -61.51, -18.44 in-in in 8.3397 Saltbr-in 2.533 HRD-in -73.25, -38.58 70.21, -4.6 in-in-out SNCiio in-out ActLoopNT-in 2.9566 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnio APE10-dihe-na 999.0, 137.93 APE9-dihe-na -128.88, -94.97 APE8-dihe-out 8.76, 102.73 APE8-rot-out 52.93 APE67-dihe-in -72.89, -15.66 -99.47, -15.26 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 6.6732 APE9-dist-out 7.8742 None PTR211 PTR211 XRAY 2.9 0.207 0.26 B 373.0 332.0 7 27 21 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6D A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.7524 13.5451 BLAminus -157.98, -176.25 63.15, 72.4 -94.88, 18.71 288.21, 86.06 -60.77, -17.66 in-in in 8.448 Saltbr-in 3.0006 HRD-in -74.85, -41.94 71.3, -1.92 in-in-out SNCiio in-out ActLoopNT-in 2.8531 ActLoopCT-out nonTYR APEdihe_aaooo APEdist_nnio APE10-dihe-na 999.0, -28.71 APE9-dihe-na 70.23, 60.42 APE8-dihe-out -136.17, -56.82 APE8-rot-out 132.32 APE67-dihe-out -77.45, -28.23 69.46, -39.41 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 7.0768 APE9-dist-out 8.5822 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 D 373.0 327.0 12 27 18 9 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6F A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.9801 13.8202 BLAminus -156.62, -174.56 59.51, 71.39 -97.24, 16.48 288.27, 84.06 -60.16, -18.79 in-in in 8.206 Saltbr-in 2.7353 HRD-in -76.38, -41.74 71.66, -4.7 in-in-out SNCiio in-out ActLoopNT-in 2.744 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -146.52, 154.45 APE9-dihe-na -92.11, 49.24 APE8-dihe-in -83.14, 134.37 APE8-rot-out 54.49 APE67-dihe-in -77.45, -15.85 -109.34, -69.31 APE12-dist-none 999.0 APE11-dist-in 9.9364 APE10-dist-in 6.6737 APE9-dist-out 9.0418 None PTR211 PTR211 XRAY 2.9 0.207 0.26 F 373.0 325.0 14 27 21 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK

CMGC_GSK3B (Glycogen synthase kinase-3 beta)

Total number of chains: 16
Active chains: 6
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 15 93.8% 8VMEA
DFGin ABAminus 1 6.2% 5AIRA

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GSK3B GSK3B_MOUSE 8VMFA Q9WV60 27 383 420.0 ADP:60504 ATPlike Active DFGin 6.6121 14.0996 BLAminus -148.4, -167.57 58.53, 66.72 -90.57, 24.21 287.49, 78.37 -75.04, -7.89 in-in in 8.6601 Saltbr-in 2.678 HRD-in -67.34, -47.3 70.6, 6.45 in-in-in SNCiii in-in ActLoopNT-in 2.8401 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -98.01, -20.74 APE9-dihe-na -93.16, -168.14 APE8-dihe-in -112.8, 164.36 APE8-rot-in 304.6 APE67-dihe-inflip 78.98, -8.38 -56.8, 140.56 APE12-dist-in 13.183 APE11-dist-in 10.9487 APE10-dist-in 6.514 APE9-dist-in 3.3085 None None None XRAY 2.5 0.21 0.251 A 364.0 354.0 0 27 27 0 [[56, 340]] 1.0 8vmf Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 8VMGA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 7.0002 13.9987 BLAminus -139.67, -176.86 60.44, 73.06 -89.27, 27.07 283.1, 81.19 -73.23, -12.63 in-in in 8.478 Saltbr-in 2.6881 HRD-in -67.64, -48.38 72.75, 3.36 in-in-in SNCiii in-in ActLoopNT-in 2.8435 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.26, 164.63 APE9-dihe-na 72.45, 142.8 APE8-dihe-in -66.41, 146.08 APE8-rot-in 307.07 APE67-dihe-in -64.3, -22.81 -57.43, -46.54 APE12-dist-in 13.2782 APE11-dist-in 11.627 APE10-dist-in 6.9412 APE9-dist-in 2.9838 None None None XRAY 2.45 0.195 0.23 A 364.0 358.0 0 27 27 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 8VMEA Q9WV60 26 383 420.0 ADP:60401 ATPlike Active DFGin 6.469 13.8439 BLAminus -131.0, -171.33 63.41, 73.0 -92.56, 22.88 289.27, 83.61 -79.03, -1.02 in-in in 8.7532 Saltbr-in 2.7802 HRD-in -67.9, -47.67 70.4, 7.52 in-in-in SNCiii in-in ActLoopNT-in 2.7313 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.18, 168.01 APE9-dihe-na 68.83, 161.19 APE8-dihe-in -90.7, 152.54 APE8-rot-in 290.93 APE67-dihe-inflip 82.32, -22.26 -51.38, 150.9 APE12-dist-in 13.2878 APE11-dist-in 12.0712 APE10-dist-in 6.9342 APE9-dist-in 3.2916 None None None XRAY 2.3 0.183 0.23 A 365.0 355.0 0 27 27 0 [[56, 340]] 1.0 8vme Mus musculus CMGC_GSK3B_MOUSE CMGC 2.1e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 4NU1A Q9WV60 6 383 420.0 ADP:405 ATPlike Active DFGin 6.1094 13.6771 BLAminus -140.27, -172.8 60.29, 88.19 -108.14, 24.39 289.57, 88.21 -68.01, -14.99 in-in in 8.691 Saltbr-in 2.7928 HRD-in -66.76, -45.51 62.96, 19.85 in-in-in SNCiii in-in ActLoopNT-in 2.6824 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.38, 172.68 APE9-dihe-na 66.76, 153.81 APE8-dihe-in -82.08, 156.46 APE8-rot-in 299.93 APE67-dihe-inflip 76.53, -25.22 -54.39, 158.45 APE12-dist-in 13.5101 APE11-dist-in 11.6207 APE10-dist-in 7.1263 APE9-dist-in 3.1496 None SEP9 SEP9 XRAY 2.5 0.194 0.245 A 389.0 357.0 2 27 27 0 [[56, 340]] 1.0 4nu1 Mus musculus CMGC_GSK3B_MOUSE CMGC 2.5e-70 243.2 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3D Q9WV60 36 382 420.0 No_ligand No_ligand Active DFGin 6.8462 14.3954 BLAminus -141.83, -176.77 60.2, 77.49 -89.39, 22.71 281.69, 81.03 -67.16, -17.62 in-in in 8.5972 Saltbr-in 2.9198 HRD-in -66.38, -49.02 71.39, 7.08 in-in-in SNCiii in-in ActLoopNT-in 3.0257 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.65, -50.64 APE9-dihe-na -86.99, 177.5 APE8-dihe-in -52.77, 135.95 APE8-rot-in 241.34 APE67-dihe-in -60.13, -26.01 -56.25, -47.64 APE12-dist-in 13.5374 APE11-dist-in 11.7665 APE10-dist-in 7.2779 APE9-dist-in 3.256 None PTR216 PTR216 XRAY 2.14 0.192 0.226 D 420.0 333.0 13 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 5AIRB Q9WV60 22 384 420.0 No_ligand No_ligand Active DFGin 7.2132 14.6827 BLAminus -135.77, 173.37 62.69, 75.87 -94.37, 22.65 282.98, 71.43 -62.58, -24.12 in-in in 8.743 Saltbr-in 3.1941 HRD-in -72.7, -48.08 74.63, 8.38 in-in-in SNCiii in-in ActLoopNT-in 3.0783 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -78.78, -34.05 APE9-dihe-na -91.23, 159.66 APE8-dihe-in -80.14, 164.39 APE8-rot-in 286.43 APE67-dihe-in -76.71, -12.41 -69.97, -37.36 APE12-dist-in 12.7248 APE11-dist-in 10.7707 APE10-dist-in 5.7984 APE9-dist-in 3.2801 None None None XRAY 2.53 0.215 0.26 B 430.0 361.0 2 27 27 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 5AIRA Q9WV60 26 383 420.0 No_ligand No_ligand Inactive DFGin 6.9865 14.3368 ABAminus -142.69, -19.87 -113.16, 97.17 -94.15, 12.11 276.77, 85.56 -67.43, -12.28 in-in in 8.7803 Saltbr-in 2.843 HRD-in -76.77, -43.42 72.44, 6.11 in-in-in SNCiii in-in ActLoopNT-in 2.9198 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -94.55, -31.48 APE9-dihe-na -99.45, 158.56 APE8-dihe-in -79.74, 161.48 APE8-rot-in 283.68 APE67-dihe-in -67.71, -13.15 -61.56, -52.85 APE12-dist-in 12.7446 APE11-dist-in 10.5629 APE10-dist-in 5.8016 APE9-dist-in 3.2157 None None None XRAY 2.53 0.215 0.26 A 430.0 353.0 2 27 27 0 [[56, 340]] 1.0 5air Mus musculus CMGC_GSK3B_MOUSE CMGC 3.5e-70 242.7 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 8VMGB Q9WV60 35 383 420.0 No_ligand No_ligand Inactive DFGin 7.0355 14.1047 BLAminus -148.77, -175.26 61.58, 69.86 -88.49, 24.73 286.58, 81.46 -68.41, -21.39 in-in in 8.5062 Saltbr-in 2.8221 HRD-in -64.17, -52.24 74.94, 4.57 in-in-out SNCiio in-out ActLoopNT-in 2.7514 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -148.65, 168.87 APE9-dihe-na 71.82, 140.54 APE8-dihe-in -63.28, 148.93 APE8-rot-out 168.42 APE67-dihe-in -62.52, -22.04 -64.28, -46.93 APE12-dist-in 13.4966 APE11-dist-in 11.8072 APE10-dist-in 7.0074 APE9-dist-in 3.0097 None None None XRAY 2.45 0.195 0.23 B 364.0 349.0 0 27 27 0 [[56, 340]] 1.0 8vmg Mus musculus CMGC_GSK3B_MOUSE CMGC 2e-70 243.5 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3C Q9WV60 37 383 420.0 No_ligand No_ligand Inactive DFGin 7.0852 14.2465 BLAminus -138.84, 177.7 70.47, 68.34 -81.63, 23.64 278.71, 79.84 -68.29, -26.67 in-in in 8.5431 Saltbr-in 3.0998 HRD-in -63.75, -49.26 68.09, 4.78 in-in-out SNCiio in-out ActLoopNT-in 2.9308 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -131.25, -51.04 APE9-dihe-na -75.73, 169.64 APE8-dihe-in -64.7, 134.47 APE8-rot-out 205.91 APE67-dihe-in -59.9, -28.79 -47.43, -50.42 APE12-dist-in 13.3567 APE11-dist-in 11.8202 APE10-dist-in 6.6175 APE9-dist-in 3.4159 None PTR216 PTR216 XRAY 2.14 0.192 0.226 C 420.0 332.0 14 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3A Q9WV60 36 387 420.0 MRI:501 Type1 Inactive DFGin 6.8942 14.102 BLAminus -136.0, 177.47 66.33, 76.64 -88.44, 20.33 285.85, 84.43 -66.44, -23.98 in-in in 8.8767 Saltbr-in 2.9541 HRD-in -71.52, -49.56 71.35, 12.25 in-in-out SNCiio in-out ActLoopNT-in 3.032 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.99, -47.87 APE9-dihe-na -84.23, -172.24 APE8-dihe-in -75.59, 135.74 APE8-rot-out 167.98 APE67-dihe-in -65.02, -21.79 -52.52, -47.78 APE12-dist-in 13.6917 APE11-dist-in 12.0236 APE10-dist-in 7.3136 APE9-dist-in 3.3344 None PTR216 PTR216 XRAY 2.14 0.192 0.226 A 420.0 348.0 4 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B GSK3B_MOUSE 6AE3B Q9WV60 36 384 420.0 MRI:501 Type1 Inactive DFGin 6.7389 14.0903 BLAminus -133.31, 179.77 64.96, 75.18 -85.96, 22.4 281.26, 80.21 -65.67, -27.09 in-in in 8.9797 Saltbr-in 3.0191 HRD-in -70.11, -50.99 71.74, 15.55 in-in-out SNCiio in-out ActLoopNT-in 2.9225 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -132.24, -38.47 APE9-dihe-na -87.03, 178.23 APE8-dihe-in -68.15, 134.76 APE8-rot-out 177.54 APE67-dihe-in -64.59, -23.54 -47.57, -47.97 APE12-dist-in 13.6259 APE11-dist-in 11.9079 APE10-dist-in 6.6939 APE9-dist-in 3.4142 None PTR216 PTR216 XRAY 2.14 0.192 0.226 B 420.0 344.0 5 27 27 0 [[56, 340]] 1.0 6ae3 Mus musculus CMGC_GSK3B_MOUSE CMGC 3.2e-70 242.8 1.0 301.0 301.0 199 200 201 203 205 85 97 101 178 180 179 181.0 239 226 221 220 219 218 217 216 215 133 Glycogen synthase kinase-3 beta
GSK3B A0A125YY75_TOXGG 9HVXA A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.8122 13.7389 BLAminus -151.79, -170.99 58.28, 71.83 -90.67, 23.31 282.96, 81.43 -68.24, -23.58 in-in in 7.973 Saltbr-in 2.6702 HRD-in -79.27, -44.62 69.75, 6.05 in-in-out SNCiio in-out ActLoopNT-in 2.9155 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -133.04, -39.68 APE9-dihe-na -85.38, 168.26 APE8-dihe-in -65.75, 139.05 APE8-rot-out 179.82 APE67-dihe-in -62.31, -27.06 -57.82, -44.69 APE12-dist-in 13.5047 APE11-dist-in 11.8681 APE10-dist-in 7.3712 APE9-dist-in 3.4994 None PTR211 PTR211 XRAY 2.1 0.203 0.25 A 350.0 323.0 16 27 27 0 [[47, 344]] 1.0 9hvx Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 6.4e-71 244.9 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6A A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.5538 13.5143 BLAminus -159.29, -172.81 63.26, 75.9 -98.23, 18.12 289.64, 83.03 -60.9, -17.5 in-in in 8.2475 Saltbr-in 2.9128 HRD-in -74.22, -42.3 70.91, -2.75 in-in-out SNCiio in-out ActLoopNT-in 2.7786 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -107.29, 145.01 APE9-dihe-na -102.07, 19.34 APE8-dihe-in -80.82, 138.15 APE8-rot-out 53.99 APE67-dihe-in -80.29, -18.75 -104.8, -54.34 APE12-dist-none 999.0 APE11-dist-in 10.1113 APE10-dist-in 7.183 APE9-dist-out 8.8047 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 A 373.0 332.0 7 27 24 3 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6B A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.9687 13.759 BLAminus -158.71, -175.52 61.04, 75.48 -97.8, 20.68 289.3, 83.48 -61.51, -18.44 in-in in 8.3397 Saltbr-in 2.533 HRD-in -73.25, -38.58 70.21, -4.6 in-in-out SNCiio in-out ActLoopNT-in 2.9566 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_nnio APE10-dihe-na 999.0, 137.93 APE9-dihe-na -128.88, -94.97 APE8-dihe-out 8.76, 102.73 APE8-rot-out 52.93 APE67-dihe-in -72.89, -15.66 -99.47, -15.26 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 6.6732 APE9-dist-out 7.8742 None PTR211 PTR211 XRAY 2.9 0.207 0.26 B 373.0 332.0 7 27 21 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6D A0A125YY75 46 384 394.0 A1IYF:60402 Type1 Inactive DFGin 6.7524 13.5451 BLAminus -157.98, -176.25 63.15, 72.4 -94.88, 18.71 288.21, 86.06 -60.77, -17.66 in-in in 8.448 Saltbr-in 3.0006 HRD-in -74.85, -41.94 71.3, -1.92 in-in-out SNCiio in-out ActLoopNT-in 2.8531 ActLoopCT-out nonTYR APEdihe_aaooo APEdist_nnio APE10-dihe-na 999.0, -28.71 APE9-dihe-na 70.23, 60.42 APE8-dihe-out -136.17, -56.82 APE8-rot-out 132.32 APE67-dihe-out -77.45, -28.23 69.46, -39.41 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-in 7.0768 APE9-dist-out 8.5822 None PTR211,SEP257 PTR211,SEP257 XRAY 2.9 0.207 0.26 D 373.0 327.0 12 27 18 9 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK
GSK3B A0A125YY75_TOXGG 9HW6F A0A125YY75 46 384 394.0 A1IYF:60401 Type1 Inactive DFGin 6.9801 13.8202 BLAminus -156.62, -174.56 59.51, 71.39 -97.24, 16.48 288.27, 84.06 -60.16, -18.79 in-in in 8.206 Saltbr-in 2.7353 HRD-in -76.38, -41.74 71.66, -4.7 in-in-out SNCiio in-out ActLoopNT-in 2.744 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_niio APE10-dihe-na -146.52, 154.45 APE9-dihe-na -92.11, 49.24 APE8-dihe-in -83.14, 134.37 APE8-rot-out 54.49 APE67-dihe-in -77.45, -15.85 -109.34, -69.31 APE12-dist-none 999.0 APE11-dist-in 9.9364 APE10-dist-in 6.6737 APE9-dist-out 9.0418 None PTR211 PTR211 XRAY 2.9 0.207 0.26 F 373.0 325.0 14 27 21 6 [[47, 344]] 1.0 9hw6 Toxoplasma gondii CMGC_GSK3B_TOXGG CMGC 8e-71 244.6 1.0 301.0 301.0 194 195 196 198 200 76 88 92 173 175 174 176.0 234 221 216 215 214 213 212 211 210 128 Putative cell-cycle-associated protein kinase GSK