CMGC_CLK1 (Dual specificity protein kinase CLK1)

Total number of chains: 61
Active chains: 39
Uniprot: CLK1_HUMAN
Kinase Domain Residues: 161 - 477
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 59 96.7% AF-P49759-K3A
DFGin ABAminus 1 1.6% 6KHDC
DFGin None 1 1.6% 6KHDA

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CLK1 AF-P49759-K3A P49759 153 484 484.0 No_ligand No_ligand Active DFGin 6.9434 14.1501 BLAminus -132.48, 177.39 60.27, 71.57 -85.18, 10.53 300.3, 105.86 -66.37, -11.95 in-in in 8.4417 Saltbr-in 2.7174 HRD-in -74.62, -35.37 68.27, -12.7 in-in-in SNCiii in-in ActLoopNT-in 2.9068 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -118.72, 174.26 APE9-dihe-na 63.43, 136.97 APE8-dihe-in -54.83, 138.19 APE8-rot-in 291.39 APE67-dihe-in -67.82, -20.27 -52.33, -42.8 APE12-dist-in 13.8915 APE11-dist-in 11.5231 APE10-dist-in 7.7323 APE9-dist-in 3.0057 None None None AF2 -1.0 1.0 1.0 A 332.0 332.0 0 25 25 0 [[161, 477]] 1.0 AF-P49759-K3 CMGC_CLK1_HUMAN CMGC 1.8e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6YTDA P49759 148 484 484.0 EAE:60501 Type1 Active DFGin 7.2177 14.6236 BLAminus -129.04, -179.37 68.43, 75.26 -99.43, 5.66 289.75, 100.38 -57.22, -23.43 in-in in 8.7889 Saltbr-in 2.7429 HRD-in -67.84, -52.77 79.42, -15.7 in-in-in SNCiii in-in ActLoopNT-in 2.9558 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.91, 160.56 APE9-dihe-na 78.51, 152.43 APE8-dihe-in -82.58, 136.21 APE8-rot-in 297.75 APE67-dihe-in -72.13, -8.69 -31.46, -59.55 APE12-dist-in 13.4088 APE11-dist-in 11.1174 APE10-dist-in 7.4109 APE9-dist-in 2.9862 V324A None None XRAY 2.0 0.182 0.228 A 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6ytd CMGC_CLK1_HUMAN CMGC 1.5e-93 319.2 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6QTYA P49759 149 481 484.0 V25:501 Type1 Active DFGin 7.1891 13.8275 BLAminus -129.69, 172.83 71.11, 83.55 -99.13, 16.45 297.38, 96.6 -71.94, -15.11 in-in in 8.3243 Saltbr-in 2.6508 HRD-in -69.24, -51.3 77.68, -14.79 in-in-in SNCiii in-in ActLoopNT-in 2.9043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.16, 166.1 APE9-dihe-na 76.64, 158.21 APE8-dihe-in -87.0, 137.14 APE8-rot-in 293.42 APE67-dihe-in -62.6, -10.5 -44.79, -53.3 APE12-dist-in 12.9806 APE11-dist-in 11.463 APE10-dist-in 7.4777 APE9-dist-in 3.0885 None None None XRAY 1.65 0.139 0.203 A 337.0 333.0 0 25 25 0 [[161, 477]] 1.0 6qty CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6R3DA P49759 152 481 484.0 JQW:901 Type1 Active DFGin 7.2355 14.0134 BLAminus -122.46, 176.35 64.69, 84.91 -101.75, 18.8 296.55, 100.55 -62.91, -23.24 in-in in 8.2719 Saltbr-in 2.9375 HRD-in -66.66, -51.76 77.65, -11.03 in-in-in SNCiii in-in ActLoopNT-in 2.8299 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.87, 173.33 APE9-dihe-na 73.0, 159.5 APE8-dihe-in -89.36, 141.36 APE8-rot-in 302.1 APE67-dihe-in -68.09, -12.73 -48.4, -46.85 APE12-dist-in 13.1776 APE11-dist-in 11.688 APE10-dist-in 7.5691 APE9-dist-in 2.9938 None None None XRAY 1.85 0.223 0.265 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 6r3d CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6R6EA P49759 153 481 484.0 JTQ:901 Type1 Active DFGin 7.2885 14.2962 BLAminus -128.0, 174.1 72.24, 79.12 -104.06, 19.03 290.47, 84.52 -68.66, -15.84 in-in in 8.4091 Saltbr-in 2.7454 HRD-in -60.82, -42.83 67.21, -15.33 in-in-in SNCiii in-in ActLoopNT-in 2.7501 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.15, 166.85 APE9-dihe-na 79.69, 155.93 APE8-dihe-in -74.39, 146.66 APE8-rot-in 301.47 APE67-dihe-in -66.87, -19.64 -52.56, -47.56 APE12-dist-in 13.1772 APE11-dist-in 11.7084 APE10-dist-in 7.6156 APE9-dist-in 3.0911 None None None XRAY 2.25 0.209 0.258 A 337.0 327.0 2 25 25 0 [[161, 477]] 1.0 6r6e CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6R6XA P49759 152 481 484.0 JU8:901 Type1 Active DFGin 7.1913 13.8821 BLAminus -123.65, 175.5 67.74, 78.23 -100.49, 14.01 300.01, 96.17 -58.94, -19.36 in-in in 8.4365 Saltbr-in 2.7463 HRD-in -67.05, -47.28 77.18, -15.83 in-in-in SNCiii in-in ActLoopNT-in 2.8079 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.71, 173.64 APE9-dihe-na 76.22, 157.17 APE8-dihe-in -81.77, 144.6 APE8-rot-in 304.54 APE67-dihe-in -66.2, -13.27 -49.16, -50.71 APE12-dist-in 12.9882 APE11-dist-in 11.6232 APE10-dist-in 7.4897 APE9-dist-in 3.0418 None None None XRAY 2.05 0.201 0.247 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 6r6x CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 7O9YA P49759 152 481 484.0 V5T:501 Type1 Active DFGin 7.2462 13.6868 BLAminus -122.5, 174.1 68.65, 82.2 -100.77, 14.37 301.76, 93.94 -56.91, -24.51 in-in in 8.1529 Saltbr-in 2.7617 HRD-in -69.77, -51.58 81.58, -12.75 in-in-in SNCiii in-in ActLoopNT-in 2.8507 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.84, 169.0 APE9-dihe-na 74.97, 161.24 APE8-dihe-in -86.97, 141.45 APE8-rot-in 302.46 APE67-dihe-in -63.2, -13.37 -47.79, -52.2 APE12-dist-in 12.972 APE11-dist-in 11.507 APE10-dist-in 7.4864 APE9-dist-in 3.0804 None None None XRAY 1.66 0.219 0.246 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 7o9y CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 7OA0AAA P49759 152 481 484.0 JTQ:501 Type1 Active DFGin 7.2082 13.8687 BLAminus -123.62, 171.83 70.68, 87.81 -105.24, 18.66 295.8, 102.89 -75.22, -10.65 in-in in 8.2485 Saltbr-in 2.7502 HRD-in -68.11, -52.1 81.61, -13.16 in-in-in SNCiii in-in ActLoopNT-in 2.8593 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.31, 171.34 APE9-dihe-na 77.29, 158.23 APE8-dihe-in -81.59, 143.88 APE8-rot-in 304.32 APE67-dihe-in -62.82, -8.69 -51.01, -53.79 APE12-dist-in 13.0487 APE11-dist-in 11.5697 APE10-dist-in 7.4745 APE9-dist-in 3.03 None None None XRAY 1.81 0.195 0.242 AAA 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 7oa0 CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 1Z57A P49759 148 482 484.0 DBQ:60001 Type1 Active DFGin 6.9813 14.002 BLAminus -125.78, 172.53 74.79, 89.46 -108.53, 21.5 296.6, 99.61 -72.51, -21.17 in-in in 8.4658 Saltbr-in 2.7879 HRD-in -70.25, -52.83 80.14, -14.55 in-in-in SNCiii in-in ActLoopNT-in 2.9435 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.0, 169.19 APE9-dihe-na 76.16, 157.77 APE8-dihe-in -82.83, 140.18 APE8-rot-in 294.7 APE67-dihe-in -63.99, -15.88 -47.28, -50.61 APE12-dist-in 13.3216 APE11-dist-in 11.2235 APE10-dist-in 7.313 APE9-dist-in 3.0014 None None None XRAY 1.7 0.14 0.186 A 339.0 331.0 4 25 25 0 [[161, 477]] 1.0 1z57 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5J1VA P49759 148 483 484.0 6FD:60501 Type1 Active DFGin 7.1 14.1716 BLAminus -126.87, 172.93 72.75, 87.91 -109.91, 21.95 296.61, 87.13 -77.69, -9.89 in-in in 8.5266 Saltbr-in 2.7359 HRD-in -74.36, -52.4 82.96, -16.81 in-in-in SNCiii in-in ActLoopNT-in 2.8778 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.9, 168.51 APE9-dihe-na 72.23, 149.39 APE8-dihe-in -71.93, 136.52 APE8-rot-in 285.15 APE67-dihe-in -66.67, -20.56 -35.82, -53.71 APE12-dist-in 13.5279 APE11-dist-in 11.4445 APE10-dist-in 7.2811 APE9-dist-in 3.0427 None None None XRAY 2.52 0.201 0.244 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 5j1v CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5J1VB P49759 148 482 484.0 6FD:60501 Type1 Active DFGin 7.1093 14.1198 BLAminus -126.74, 175.0 70.24, 87.64 -108.44, 20.05 295.73, 90.04 -77.7, -8.55 in-in in 8.5763 Saltbr-in 2.7543 HRD-in -73.08, -51.15 80.15, -14.17 in-in-in SNCiii in-in ActLoopNT-in 2.8769 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.41, 168.72 APE9-dihe-na 72.72, 151.05 APE8-dihe-in -70.92, 135.35 APE8-rot-in 286.36 APE67-dihe-in -65.82, -21.41 -37.05, -51.94 APE12-dist-in 13.782 APE11-dist-in 11.5423 APE10-dist-in 7.3562 APE9-dist-in 3.0498 None None None XRAY 2.52 0.201 0.244 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 5j1v CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5J1WA P49759 148 483 484.0 6FB:60506 Type1 Active DFGin 7.1724 14.3259 BLAminus -121.81, 173.7 71.87, 86.58 -105.02, 20.94 296.61, 84.3 -77.49, -14.22 in-in in 8.5488 Saltbr-in 2.5641 HRD-in -71.53, -50.92 81.49, -14.91 in-in-in SNCiii in-in ActLoopNT-in 2.9036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.47, 167.51 APE9-dihe-na 77.02, 140.17 APE8-dihe-in -56.28, 137.97 APE8-rot-in 295.84 APE67-dihe-in -62.06, -22.4 -61.94, -35.28 APE12-dist-in 13.6052 APE11-dist-in 11.4365 APE10-dist-in 7.2516 APE9-dist-in 3.0421 None None None XRAY 2.42 0.191 0.228 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 5j1w CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5J1WB P49759 148 482 484.0 6FB:60503 Type1 Active DFGin 7.2901 14.2646 BLAminus -120.99, 173.46 72.42, 86.12 -105.34, 21.92 296.07, 87.01 -75.02, -15.34 in-in in 8.5851 Saltbr-in 2.5852 HRD-in -69.32, -50.91 80.3, -14.73 in-in-in SNCiii in-in ActLoopNT-in 2.8972 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.41, 167.18 APE9-dihe-na 77.9, 139.82 APE8-dihe-in -54.28, 138.17 APE8-rot-in 296.7 APE67-dihe-in -62.44, -21.37 -62.69, -34.82 APE12-dist-in 13.6477 APE11-dist-in 11.342 APE10-dist-in 7.196 APE9-dist-in 3.035 None None None XRAY 2.42 0.191 0.228 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 5j1w CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6FT8A P49759 148 483 484.0 E6T:60501 Type1 Active DFGin 7.0417 14.1532 BLAminus -123.69, 179.12 66.02, 80.75 -102.66, 23.58 296.94, 92.84 -75.28, -12.2 in-in in 8.4476 Saltbr-in 2.7433 HRD-in -68.91, -53.98 78.36, -16.69 in-in-in SNCiii in-in ActLoopNT-in 2.9408 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.28, 167.17 APE9-dihe-na 78.21, 159.73 APE8-dihe-in -85.1, 140.33 APE8-rot-in 293.05 APE67-dihe-in -66.99, -12.12 -49.73, -45.92 APE12-dist-in 13.2816 APE11-dist-in 11.5166 APE10-dist-in 7.3272 APE9-dist-in 3.0294 None None None XRAY 1.45 0.166 0.195 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6ft8 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6FT9A P49759 148 482 484.0 E6W:60501 Type1 Active DFGin 7.2322 14.2998 BLAminus -125.02, 175.42 67.64, 86.22 -106.42, 22.86 292.22, 81.03 -75.21, -13.41 in-in in 8.4297 Saltbr-in 2.7125 HRD-in -69.31, -51.72 79.55, -13.59 in-in-in SNCiii in-in ActLoopNT-in 2.8663 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.87, 168.01 APE9-dihe-na 73.7, 150.41 APE8-dihe-in -70.08, 140.16 APE8-rot-in 296.52 APE67-dihe-in -66.14, -21.84 -44.66, -47.8 APE12-dist-in 13.556 APE11-dist-in 11.2182 APE10-dist-in 7.2792 APE9-dist-in 2.9326 None None None XRAY 1.87 0.168 0.202 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6ft9 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6FT9B P49759 148 482 484.0 E6W:60501 Type1 Active DFGin 7.2936 14.3139 BLAminus -123.52, 178.1 65.34, 85.29 -106.33, 21.22 292.88, 84.42 -75.16, -8.95 in-in in 8.4862 Saltbr-in 2.7077 HRD-in -71.01, -50.08 80.37, -13.57 in-in-in SNCiii in-in ActLoopNT-in 2.834 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.43, 168.15 APE9-dihe-na 75.76, 149.1 APE8-dihe-in -68.06, 138.01 APE8-rot-in 296.86 APE67-dihe-in -65.44, -22.15 -43.68, -46.72 APE12-dist-in 13.7449 APE11-dist-in 11.2771 APE10-dist-in 7.2841 APE9-dist-in 2.9662 None None None XRAY 1.87 0.168 0.202 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6ft9 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5HA P49759 148 481 484.0 H3N:60507 Type1 Active DFGin 6.9359 13.9902 BLAminus -127.91, 175.49 70.62, 86.84 -104.99, 23.28 297.7, 98.27 -76.67, -15.26 in-in in 8.6705 Saltbr-in 2.7942 HRD-in -71.42, -54.52 81.98, -15.98 in-in-in SNCiii in-in ActLoopNT-in 2.9892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.5, 162.59 APE9-dihe-na 81.01, 150.81 APE8-dihe-in -73.05, 137.12 APE8-rot-in 298.85 APE67-dihe-in -65.31, -13.64 -50.7, -47.04 APE12-dist-in 12.9825 APE11-dist-in 11.3246 APE10-dist-in 7.2343 APE9-dist-in 3.0974 None None None XRAY 1.49 0.179 0.206 A 339.0 323.0 11 25 25 0 [[161, 477]] 1.0 6i5h CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5IA P49759 148 483 484.0 H3E:60501 Type1 Active DFGin 6.9087 13.9494 BLAminus -127.6, 172.7 71.85, 87.8 -102.42, 20.37 300.05, 101.13 -74.42, -16.22 in-in in 8.7126 Saltbr-in 2.693 HRD-in -75.53, -52.34 81.22, -14.82 in-in-in SNCiii in-in ActLoopNT-in 2.9983 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.19, 164.34 APE9-dihe-na 79.5, 152.78 APE8-dihe-in -78.57, 135.82 APE8-rot-in 292.41 APE67-dihe-in -65.9, -11.23 -46.6, -47.35 APE12-dist-in 13.1135 APE11-dist-in 11.2837 APE10-dist-in 7.2519 APE9-dist-in 3.0736 None None None XRAY 1.6 0.166 0.196 A 339.0 333.0 3 25 25 0 [[161, 477]] 1.0 6i5i CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5KB P49759 148 481 484.0 H3H:60504 Type1 Active DFGin 7.006 14.3591 BLAminus -126.82, 178.06 66.53, 84.63 -104.0, 26.37 299.27, 91.89 -80.46, -16.31 in-in in 9.0291 Saltbr-in 2.6927 HRD-in -71.59, -48.77 75.18, -11.75 in-in-in SNCiii in-in ActLoopNT-in 2.9844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.96, 164.13 APE9-dihe-na 74.43, 150.15 APE8-dihe-in -66.68, 137.66 APE8-rot-in 303.78 APE67-dihe-in -77.74, -18.3 -54.0, -31.51 APE12-dist-in 13.8442 APE11-dist-in 11.2244 APE10-dist-in 7.3953 APE9-dist-in 3.093 None None None XRAY 2.3 0.197 0.224 B 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 6i5k CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5KC P49759 148 483 484.0 H3H:60504 Type1 Active DFGin 6.9865 14.3514 BLAminus -125.41, 178.1 66.91, 85.45 -105.62, 25.72 298.18, 84.65 -79.89, -19.48 in-in in 8.919 Saltbr-in 2.6659 HRD-in -72.35, -49.89 76.53, -11.56 in-in-in SNCiii in-in ActLoopNT-in 3.0005 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.9, 163.92 APE9-dihe-na 72.8, 149.97 APE8-dihe-in -66.75, 139.4 APE8-rot-in 303.5 APE67-dihe-in -77.85, -17.5 -52.64, -34.11 APE12-dist-in 13.6161 APE11-dist-in 11.124 APE10-dist-in 7.3407 APE9-dist-in 3.1121 None None None XRAY 2.3 0.197 0.224 C 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6i5k CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5LB P49759 148 481 484.0 H3Q:60502 Type1 Active DFGin 6.9284 14.418 BLAminus -123.55, 178.93 67.48, 93.05 -113.53, 21.71 295.78, 85.8 -74.38, -22.09 in-in in 8.9824 Saltbr-in 2.7395 HRD-in -69.85, -49.79 74.87, -13.88 in-in-in SNCiii in-in ActLoopNT-in 2.9995 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.82, 165.73 APE9-dihe-na 81.08, 146.54 APE8-dihe-in -62.76, 135.54 APE8-rot-in 302.63 APE67-dihe-in -68.98, -24.89 -54.53, -33.68 APE12-dist-in 13.8519 APE11-dist-in 11.4167 APE10-dist-in 7.226 APE9-dist-in 3.1016 None None None XRAY 2.55 0.195 0.221 B 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 6i5l CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5LC P49759 148 483 484.0 H3Q:60502 Type1 Active DFGin 6.9131 14.3839 BLAminus -123.57, 177.17 68.91, 92.22 -114.6, 21.5 296.12, 85.91 -74.75, -23.49 in-in in 8.8781 Saltbr-in 2.7107 HRD-in -71.08, -49.61 75.52, -13.95 in-in-in SNCiii in-in ActLoopNT-in 3.0208 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.58, 165.38 APE9-dihe-na 80.23, 146.0 APE8-dihe-in -62.57, 137.3 APE8-rot-in 302.62 APE67-dihe-in -70.1, -23.69 -53.95, -35.33 APE12-dist-in 13.6577 APE11-dist-in 11.3372 APE10-dist-in 7.1791 APE9-dist-in 3.1361 None None None XRAY 2.55 0.195 0.221 C 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6i5l CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Q8KA P49759 148 484 484.0 FG9:60502 Type1 Active DFGin 7.0383 14.0726 BLAminus -126.96, 173.92 68.96, 94.14 -110.91, 19.67 299.22, 86.31 -70.74, -15.36 in-in in 8.7893 Saltbr-in 2.6969 HRD-in -64.71, -54.26 80.91, -18.18 in-in-in SNCiii in-in ActLoopNT-in 2.9149 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.28, 157.45 APE9-dihe-na 83.98, 154.49 APE8-dihe-in -77.73, 126.84 APE8-rot-in 298.77 APE67-dihe-in -63.27, -22.97 -33.76, -49.02 APE12-dist-in 13.3669 APE11-dist-in 11.2855 APE10-dist-in 7.4682 APE9-dist-in 3.1111 None None None XRAY 2.29 0.191 0.259 A 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6q8k CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6YTAA P49759 148 483 484.0 IYZ:60702 Type1 Active DFGin 6.9349 13.7248 BLAminus -125.39, 175.02 66.16, 92.34 -102.15, 17.18 301.41, 98.15 -60.08, -20.3 in-in in 8.3168 Saltbr-in 2.6989 HRD-in -68.08, -57.05 83.09, -18.57 in-in-in SNCiii in-in ActLoopNT-in 2.8997 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.65, 155.94 APE9-dihe-na 83.67, 157.83 APE8-dihe-in -84.55, 129.06 APE8-rot-in 292.9 APE67-dihe-in -62.02, -24.22 -28.74, -53.35 APE12-dist-in 13.2113 APE11-dist-in 11.6634 APE10-dist-in 7.3747 APE9-dist-in 3.1591 None None None XRAY 2.3 0.194 0.275 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6yta CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6YTEC P49759 148 484 484.0 EAE:60501 Type1 Active DFGin 7.1447 14.1109 BLAminus -123.36, 172.5 72.26, 86.11 -107.09, 11.71 295.65, 98.47 -58.29, -17.8 in-in in 8.5445 Saltbr-in 2.2253 HRD-in -60.42, -59.86 88.88, -8.99 in-in-in SNCiii in-in ActLoopNT-in 3.0048 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.24, 160.76 APE9-dihe-na 81.35, 157.72 APE8-dihe-in -87.96, 130.83 APE8-rot-in 293.05 APE67-dihe-in -54.77, -23.25 -31.22, -65.53 APE12-dist-in 13.3746 APE11-dist-in 11.4404 APE10-dist-in 7.3205 APE9-dist-in 3.082 None None None XRAY 2.3 0.184 0.258 C 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6yte CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6YTIA P49759 150 482 484.0 7A7:605 Type1 Active DFGin 7.2921 14.242 BLAminus -134.7, 172.33 69.03, 94.12 -110.31, 22.0 290.95, 98.93 -72.82, -22.05 in-in in 8.6449 Saltbr-in 2.6167 HRD-in -68.46, -54.35 84.41, -17.31 in-in-in SNCiii in-in ActLoopNT-in 2.8883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.78, 154.97 APE9-dihe-na 84.02, 157.2 APE8-dihe-in -78.01, 116.07 APE8-rot-in 301.91 APE67-dihe-in -65.16, -18.0 -14.75, -58.2 APE12-dist-in 13.4174 APE11-dist-in 11.0368 APE10-dist-in 7.4563 APE9-dist-in 3.0199 None None None XRAY 2.4 0.198 0.256 A 339.0 329.0 4 25 25 0 [[161, 477]] 1.0 6yti CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Z4ZA P49759 148 482 484.0 PQ5:60505 Type1 Active DFGin 7.046 14.2363 BLAminus -126.68, 179.24 66.69, 82.0 -103.33, 19.73 297.68, 94.61 -71.59, -13.97 in-in in 8.4611 Saltbr-in 2.7642 HRD-in -69.38, -51.98 76.89, -13.79 in-in-in SNCiii in-in ActLoopNT-in 2.9245 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.91, 169.84 APE9-dihe-na 70.81, 154.45 APE8-dihe-in -79.18, 136.44 APE8-rot-in 295.15 APE67-dihe-in -64.16, -17.67 -45.6, -49.57 APE12-dist-in 13.5127 APE11-dist-in 11.3594 APE10-dist-in 7.327 APE9-dist-in 3.0405 None None None XRAY 2.07 0.177 0.213 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6z4z CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Z4ZB P49759 148 484 484.0 PQ5:60501 Type1 Active DFGin 7.0483 14.168 BLAminus -127.78, 179.44 66.36, 84.49 -106.02, 23.22 298.83, 96.06 -73.86, -11.97 in-in in 8.4214 Saltbr-in 2.7252 HRD-in -70.61, -51.12 77.5, -15.65 in-in-in SNCiii in-in ActLoopNT-in 2.9096 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, 168.57 APE9-dihe-na 73.19, 152.9 APE8-dihe-in -77.75, 136.06 APE8-rot-in 294.47 APE67-dihe-in -61.42, -18.21 -47.63, -47.77 APE12-dist-in 13.4848 APE11-dist-in 11.247 APE10-dist-in 7.2192 APE9-dist-in 3.0518 None None None XRAY 2.07 0.177 0.213 B 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6z4z CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Z4ZC P49759 148 482 484.0 PQ5:60502 Type1 Active DFGin 7.1081 14.2491 BLAminus -126.87, 178.82 67.48, 81.17 -101.74, 18.48 298.94, 95.28 -65.75, -17.47 in-in in 8.5666 Saltbr-in 2.7627 HRD-in -67.93, -52.14 78.08, -12.45 in-in-in SNCiii in-in ActLoopNT-in 2.8763 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.01, 169.28 APE9-dihe-na 73.05, 151.25 APE8-dihe-in -74.69, 135.04 APE8-rot-in 294.69 APE67-dihe-in -63.57, -18.13 -46.66, -45.93 APE12-dist-in 13.7076 APE11-dist-in 11.4576 APE10-dist-in 7.407 APE9-dist-in 3.0276 None None None XRAY 2.07 0.177 0.213 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6z4z CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6ZLNA P49759 148 484 484.0 PKB:60503 Type1 Active DFGin 7.0057 14.1924 BLAminus -125.63, 176.89 76.78, 75.35 -103.44, 16.76 293.35, 98.15 -70.81, -12.33 in-in in 8.6634 Saltbr-in 2.7072 HRD-in -67.73, -49.47 78.97, -14.05 in-in-in SNCiii in-in ActLoopNT-in 2.9351 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.54, 162.21 APE9-dihe-na 79.84, 163.79 APE8-dihe-in -96.39, 123.92 APE8-rot-in 291.96 APE67-dihe-in -72.31, -12.72 -20.91, -56.58 APE12-dist-in 13.2334 APE11-dist-in 10.9238 APE10-dist-in 7.2166 APE9-dist-in 3.0919 None None None XRAY 1.7 0.171 0.199 A 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6zln CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 7AK3A P49759 148 483 484.0 RH8:60501 Type1 Active DFGin 7.3197 14.2837 BLAminus -128.56, 172.37 67.01, 84.33 -103.74, 27.34 296.18, 85.72 -72.52, -23.23 in-in in 8.6033 Saltbr-in 2.8652 HRD-in -61.61, -53.86 89.68, -14.81 in-in-in SNCiii in-in ActLoopNT-in 2.9582 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.68, 162.47 APE9-dihe-na 75.05, 158.38 APE8-dihe-in -88.77, 128.79 APE8-rot-in 301.95 APE67-dihe-in -60.58, -28.09 -3.93, -77.31 APE12-dist-in 13.3868 APE11-dist-in 11.1501 APE10-dist-in 7.274 APE9-dist-in 2.9982 None None None XRAY 2.5 0.213 0.26 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 7ak3 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 7OPGA P49759 148 482 484.0 06N:60501 Type1 Active DFGin 7.0787 14.3372 BLAminus -125.23, 174.99 68.34, 89.35 -108.55, 22.34 294.5, 84.43 -74.9, -16.57 in-in in 8.8275 Saltbr-in 2.697 HRD-in -68.7, -53.19 79.41, -13.79 in-in-in SNCiii in-in ActLoopNT-in 2.8637 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.87, 169.9 APE9-dihe-na 72.2, 152.58 APE8-dihe-in -74.2, 140.4 APE8-rot-in 296.34 APE67-dihe-in -64.01, -18.08 -47.78, -49.23 APE12-dist-in 13.4538 APE11-dist-in 11.205 APE10-dist-in 7.2886 APE9-dist-in 3.0135 None None None XRAY 1.93 0.176 0.208 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 7opg CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 7OPGB P49759 148 483 484.0 06N:60501 Type1 Active DFGin 7.0918 14.2954 BLAminus -128.58, 171.98 71.57, 88.89 -110.25, 21.49 294.73, 85.57 -73.38, -14.32 in-in in 8.7933 Saltbr-in 2.6848 HRD-in -66.06, -53.32 81.87, -15.7 in-in-in SNCiii in-in ActLoopNT-in 2.843 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.09, 167.09 APE9-dihe-na 74.85, 150.04 APE8-dihe-in -76.84, 138.69 APE8-rot-in 295.58 APE67-dihe-in -61.09, -19.4 -51.05, -46.51 APE12-dist-in 13.2757 APE11-dist-in 11.1509 APE10-dist-in 7.227 APE9-dist-in 3.0505 None None None XRAY 1.93 0.176 0.208 B 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 7opg CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 7OPGC P49759 148 482 484.0 06N:60501 Type1 Active DFGin 7.1396 14.3181 BLAminus -126.92, 172.88 71.54, 91.0 -109.11, 17.42 294.29, 87.52 -72.35, -14.96 in-in in 8.8983 Saltbr-in 2.7034 HRD-in -68.36, -53.23 82.74, -14.25 in-in-in SNCiii in-in ActLoopNT-in 2.8367 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.58, 169.34 APE9-dihe-na 74.62, 150.8 APE8-dihe-in -72.07, 139.48 APE8-rot-in 296.41 APE67-dihe-in -63.14, -17.95 -50.02, -46.94 APE12-dist-in 13.4592 APE11-dist-in 11.323 APE10-dist-in 7.3831 APE9-dist-in 3.0248 None None None XRAY 1.93 0.176 0.208 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 7opg CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6FYOA P49759 148 481 484.0 EAQ:501 Type1 Active DFGin 7.1303 14.6092 BLAminus -126.41, -177.97 57.7, 79.82 -101.45, 23.66 290.45, 86.2 -71.99, -23.62 in-in in 8.2538 Saltbr-in 2.8261 HRD-in -67.73, -44.39 69.27, -21.51 in-in-in SNCiii in-in ActLoopNT-in 2.7761 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.41, 162.2 APE9-dihe-na 76.62, 158.52 APE8-dihe-in -81.15, 137.38 APE8-rot-in 320.28 APE67-dihe-in -54.52, -12.47 -37.95, -53.62 APE12-dist-in 13.1043 APE11-dist-in 11.2911 APE10-dist-in 7.0165 APE9-dist-in 3.2103 None None None XRAY 2.32 0.204 0.234 A 339.0 331.0 3 25 25 0 [[161, 477]] 1.0 6fyo CMGC_CLK1_HUMAN CMGC 2e-93 318.8 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5X8IA P49759 154 481 484.0 SQZ:501 Type1 Active DFGin 7.3534 13.9989 BLAminus -122.66, 172.48 71.45, 69.85 -89.46, 19.16 303.2, 86.95 -71.61, -17.76 in-in in 8.3789 Saltbr-in 2.5421 HRD-in -68.32, -52.49 79.94, -11.57 in-in-in SNCiii in-in ActLoopNT-in 2.8658 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.32, 168.72 APE9-dihe-na 74.05, 158.08 APE8-dihe-in -81.53, 144.19 APE8-rot-in 300.53 APE67-dihe-in -65.15, -11.28 -51.71, -50.28 APE12-dist-in 13.0833 APE11-dist-in 11.6511 APE10-dist-in 7.533 APE9-dist-in 3.016 R432A None None XRAY 1.902 0.168 0.206 A 346.0 328.0 0 25 25 0 [[161, 477]] 1.0 5x8i CMGC_CLK1_HUMAN CMGC 2.7e-93 318.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5X8IB P49759 155 481 484.0 SQZ:501 Type1 Active DFGin 7.3842 13.9802 BLAminus -126.45, 170.69 71.83, 69.37 -88.36, 11.76 302.43, 89.48 -69.31, -18.97 in-in in 8.3824 Saltbr-in 2.41 HRD-in -67.27, -52.41 79.09, -12.7 in-in-in SNCiii in-in ActLoopNT-in 2.8887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.02, 169.54 APE9-dihe-na 72.76, 157.49 APE8-dihe-in -80.25, 143.44 APE8-rot-in 301.33 APE67-dihe-in -65.52, -10.3 -49.82, -50.77 APE12-dist-in 13.1161 APE11-dist-in 11.6767 APE10-dist-in 7.4994 APE9-dist-in 3.0166 R432A None None XRAY 1.902 0.168 0.206 B 346.0 327.0 0 25 25 0 [[161, 477]] 1.0 5x8i CMGC_CLK1_HUMAN CMGC 2.7e-93 318.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6YTGA P49759 148 483 484.0 KHC:60501,KHC:60502 Type1,Allosteric Active DFGin 7.1086 14.3781 BLAminus -123.68, -179.19 66.81, 76.1 -102.89, 15.19 291.91, 90.06 -75.03, -12.8 in-in in 8.5496 Saltbr-in 2.696 HRD-in -64.66, -54.29 85.54, -10.78 in-in-in SNCiii in-in ActLoopNT-in 2.8316 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -106.45, 156.23 APE9-dihe-na 81.17, 153.49 APE8-dihe-in -77.75, 128.48 APE8-rot-in 300.43 APE67-dihe-in -69.97, -17.37 -12.96, -64.06 APE12-dist-in 13.337 APE11-dist-in 11.4029 APE10-dist-in 7.7563 APE9-dist-in 2.9823 None None None XRAY 1.95 0.207 0.261 A 339.0 329.0 7 25 25 0 [[161, 477]] 1.0 6ytg CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6R8JA P49759 152 481 484.0 JUW:501,JUW:502 Type1,Type1 Active DFGin 7.1717 13.6765 BLAminus -124.23, 172.49 72.75, 83.0 -102.73, 17.52 298.34, 101.12 -64.7, -21.81 in-in in 8.1336 Saltbr-in 2.8945 HRD-in -66.22, -54.05 83.24, -16.78 in-in-in SNCiii in-in ActLoopNT-in 2.8729 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.97, 169.66 APE9-dihe-na 75.96, 160.32 APE8-dihe-in -86.77, 141.55 APE8-rot-in 304.05 APE67-dihe-in -66.39, -13.17 -48.7, -48.98 APE12-dist-in 13.0103 APE11-dist-in 11.5266 APE10-dist-in 7.5479 APE9-dist-in 2.9805 None None None XRAY 1.75 0.218 0.263 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 6r8j CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6KHDC P49759 150 479 484.0 3NG:1000 Type1 Inactive DFGin 7.0261 14.4118 ABAminus -125.6, -45.1 -89.27, 107.55 -111.64, 19.23 292.41, 98.32 -77.1, 0.74 in-in in 8.7674 Saltbr-in 2.9039 HRD-in -53.74, -54.41 89.98, -20.88 in-in-out SNCiio in-out ActLoopNT-in 2.895 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iioo APE10-dihe-na -118.02, -81.8 APE9-dihe-na -80.38, 126.35 APE8-dihe-in -130.72, 139.1 APE8-rot-out 73.02 APE67-dihe-in -49.48, -32.44 -62.98, -36.18 APE12-dist-in 13.3713 APE11-dist-in 9.0973 APE10-dist-out 11.3298 APE9-dist-out 7.8489 None None None XRAY 2.7 0.204 0.274 C 484.0 325.0 5 25 25 0 [[161, 477]] 1.0 6khd CMGC_CLK1_HUMAN CMGC 8.2e-93 317.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 AF-P49759-K1A P49759 153 484 484.0 No_ligand No_ligand Inactive DFGin 7.0737 14.19 BLAminus -127.24, 176.41 62.19, 72.99 -88.32, 9.55 297.11, 102.62 -68.31, -9.87 in-in in 8.4508 Saltbr-in 2.696 HRD-in -72.36, -39.16 64.91, -10.55 in-in-out SNCiio in-out ActLoopNT-in 2.9091 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oiii APE10-dihe-na -123.01, 174.5 APE9-dihe-na 65.72, 145.79 APE8-dihe-in -57.06, 135.18 APE8-rot-in 292.86 APE67-dihe-in -70.16, -18.82 -51.52, -41.74 APE12-dist-out 14.1099 APE11-dist-in 11.8348 APE10-dist-in 7.5822 APE9-dist-in 2.9068 None None None AF2 -1.0 1.0 1.0 A 332.0 332.0 0 25 25 0 [[161, 477]] 1.0 AF-P49759-K1 CMGC_CLK1_HUMAN CMGC 1.8e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 2VAGA P49759 148 481 484.0 V25:61482 Type1 Inactive DFGin 7.1077 14.0258 BLAminus -129.43, 175.64 66.18, 85.97 -104.96, 23.22 293.24, 95.17 -73.67, -15.41 in-in in 8.37 Saltbr-in 2.6268 HRD-in -71.48, -53.18 82.14, -13.71 in-in-out SNCiio in-out ActLoopNT-in 2.8437 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oioo APE10-dihe-na -88.11, 138.68 APE9-dihe-na -83.4, -165.24 APE8-dihe-in -49.62, 134.22 APE8-rot-none 999.0 APE67-dihe-out -47.82, -50.26 -151.88, 142.32 APE12-dist-out 14.0645 APE11-dist-in 12.8642 APE10-dist-out 9.7767 APE9-dist-out 8.6182 None SEP341,TPO342 SEP341,TPO342 XRAY 1.8 0.182 0.225 A 339.0 331.0 3 25 25 0 [[161, 477]] 1.0 2vag CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5J1VC P49759 148 483 484.0 6FD:60501 Type1 Inactive DFGin 7.0653 14.1863 BLAminus -127.76, 172.5 71.94, 87.97 -108.84, 22.87 296.53, 88.54 -79.84, -9.02 in-in in 8.5354 Saltbr-in 2.7469 HRD-in -76.64, -52.07 83.95, -17.44 in-in-out SNCiio in-out ActLoopNT-in 2.8928 ActLoopCT-out nonTYR APEdihe_aannn APEdist_oion APE10-dihe-na -156.89, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, -20.42 999.0, 999.0 APE12-dist-out 14.2512 APE11-dist-in 11.6023 APE10-dist-out 9.6806 APE9-dist-none 999.0 None None None XRAY 2.52 0.201 0.244 C 339.0 312.0 24 25 22 3 [[161, 477]] 1.0 5j1v CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6FT9C P49759 148 482 484.0 E6W:60501 Type1 Inactive DFGin 7.2141 14.2533 BLAminus -122.85, 177.29 65.92, 85.07 -105.77, 22.23 295.06, 82.45 -71.81, -8.98 in-in in 8.3694 Saltbr-in 2.6709 HRD-in -69.43, -51.23 80.08, -14.43 in-in-out SNCiio in-out ActLoopNT-in 2.8644 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -129.97, 131.35 APE9-dihe-na -47.51, 149.39 APE8-dihe-in -75.79, 135.36 APE8-rot-in 303.89 APE67-dihe-out -54.68, -26.4 -154.15, 148.3 APE12-dist-out 14.7393 APE11-dist-in 12.4265 APE10-dist-out 9.6939 APE9-dist-out 8.7023 None None None XRAY 1.87 0.168 0.202 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6ft9 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6G33A P49759 148 482 484.0 5ID:60501 Type1 Inactive DFGin 7.0386 14.0293 BLAminus -127.31, 176.31 68.38, 85.72 -104.03, 25.47 298.82, 93.66 -74.89, -17.97 in-in in 8.3822 Saltbr-in 2.7246 HRD-in -70.1, -50.84 78.28, -13.18 in-in-out SNCiio in-out ActLoopNT-in 2.8482 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oioo APE10-dihe-na -128.78, 136.1 APE9-dihe-na -77.1, 148.33 APE8-dihe-in -66.51, 123.5 APE8-rot-none 999.0 APE67-dihe-out -66.2, -20.29 -135.8, 167.22 APE12-dist-out 14.7008 APE11-dist-in 12.3537 APE10-dist-out 9.4988 APE9-dist-out 8.7999 None SEP341,TPO342 SEP341,TPO342 XRAY 2.05 0.19 0.218 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6g33 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6G33B P49759 148 482 484.0 5ID:60501 Type1 Inactive DFGin 7.0769 13.9786 BLAminus -125.16, 175.81 68.83, 87.13 -106.27, 24.24 297.31, 93.02 -76.58, -16.07 in-in in 8.3864 Saltbr-in 2.6996 HRD-in -69.85, -51.6 75.98, -11.49 in-in-out SNCiio in-out ActLoopNT-in 2.8786 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iioo APE10-dihe-na -123.97, 135.36 APE9-dihe-na -72.42, 114.42 APE8-dihe-in -42.53, 141.22 APE8-rot-in 302.44 APE67-dihe-out -66.45, -16.55 -136.36, 149.49 APE12-dist-in 13.8836 APE11-dist-in 11.9062 APE10-dist-out 10.3491 APE9-dist-out 9.743 None None None XRAY 2.05 0.19 0.218 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6g33 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6G33C P49759 148 482 484.0 5ID:60501 Type1 Inactive DFGin 7.1529 14.0498 BLAminus -127.31, 175.45 68.57, 84.45 -104.42, 25.23 297.23, 96.23 -74.84, -18.72 in-in in 8.4304 Saltbr-in 2.707 HRD-in -68.44, -51.98 75.83, -9.76 in-in-out SNCiio in-out ActLoopNT-in 2.8328 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oioi APE10-dihe-na -158.67, 144.43 APE9-dihe-na 80.91, 147.02 APE8-dihe-in -56.89, 133.87 APE8-rot-none 999.0 APE67-dihe-in -70.75, -20.64 -58.82, -30.99 APE12-dist-out 14.1296 APE11-dist-in 11.4642 APE10-dist-out 8.2148 APE9-dist-in 3.07 None None None XRAY 2.05 0.19 0.218 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6g33 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5KA P49759 148 482 484.0 H3H:60503 Type1 Inactive DFGin 7.0191 14.2807 BLAminus -127.95, 177.21 67.34, 85.43 -106.5, 25.82 299.72, 92.63 -80.22, -14.39 in-in in 8.8988 Saltbr-in 2.6726 HRD-in -72.89, -48.86 76.37, -11.75 in-in-out SNCiio in-out ActLoopNT-in 3.0079 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -139.66, 157.93 APE9-dihe-na -83.57, -145.55 APE8-dihe-in -77.05, 120.2 APE8-rot-in 311.82 APE67-dihe-out -112.74, 31.9 -178.22, 144.22 APE12-dist-out 14.3954 APE11-dist-in 12.6175 APE10-dist-out 8.7668 APE9-dist-out 8.7264 None None None XRAY 2.3 0.197 0.224 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6i5k CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6I5LA P49759 148 483 484.0 H3Q:60503 Type1 Inactive DFGin 6.9146 14.3203 BLAminus -124.28, 177.5 67.34, 93.35 -114.57, 21.88 295.56, 86.41 -76.53, -21.33 in-in in 8.8454 Saltbr-in 2.712 HRD-in -70.91, -49.07 76.68, -14.69 in-in-out SNCiio in-out ActLoopNT-in 3.01 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -133.89, 159.24 APE9-dihe-na -106.72, -141.34 APE8-dihe-in -74.35, 99.26 APE8-rot-in 314.71 APE67-dihe-out -134.72, 40.5 -167.53, 148.17 APE12-dist-out 14.5511 APE11-dist-in 12.2796 APE10-dist-out 9.5559 APE9-dist-out 8.8533 None None None XRAY 2.55 0.195 0.221 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6i5l CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Q8PB P49759 148 483 484.0 HQB:60501 Type1 Inactive DFGin 6.6661 14.0806 BLAminus -123.82, 175.86 66.42, 98.63 -122.53, 30.35 298.66, 86.39 -77.45, -10.39 in-in in 8.7879 Saltbr-in 2.9933 HRD-in -68.29, -44.12 72.95, -22.76 in-in-out SNCiio in-out ActLoopNT-in 3.0122 ActLoopCT-out nonTYR APEdihe_aannn APEdist_oion APE10-dihe-na -125.35, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -60.69, -36.51 999.0, -33.63 APE12-dist-out 14.4348 APE11-dist-in 12.4103 APE10-dist-out 9.3984 APE9-dist-none 999.0 None None None XRAY 3.0 0.201 0.244 B 339.0 331.0 5 25 23 2 [[161, 477]] 1.0 6q8p CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6RAAA P49759 148 481 484.0 JWN:60501 Type1 Inactive DFGin 6.8873 13.7549 BLAminus -129.66, 171.4 69.19, 92.86 -107.95, 20.85 301.15, 106.22 -67.28, -18.14 in-in in 8.302 Saltbr-in 2.9175 HRD-in -72.74, -49.16 79.77, -9.47 in-in-out SNCiio in-out ActLoopNT-in 2.9284 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.73, 160.54 APE9-dihe-na 78.15, 152.31 APE8-dihe-in -85.85, 139.96 APE8-rot-out 71.85 APE67-dihe-in -63.36, -27.28 -38.74, -49.54 APE12-dist-in 13.2788 APE11-dist-in 11.3142 APE10-dist-in 7.2917 APE9-dist-in 3.081 None None None XRAY 2.1 0.19 0.233 A 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 6raa CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6TW2E P49759 148 484 484.0 V25:62301 Type1 Inactive DFGin 7.1046 14.057 BLAminus -132.08, 175.35 68.1, 86.44 -104.28, 22.11 293.58, 88.16 -72.28, -16.22 in-in in 8.3715 Saltbr-in 2.6068 HRD-in -73.71, -50.29 77.69, -11.9 in-in-out SNCiio in-out ActLoopNT-in 2.8741 ActLoopCT-out nonTYR APEdihe_aanao APEdist_oioo APE10-dihe-na -119.46, 133.12 APE9-dihe-na 999.0, -6.85 APE8-dihe-none 999.0, 103.3 APE8-rot-na 296.95 APE67-dihe-out -59.07, -41.0 14.44, 142.85 APE12-dist-out 14.8499 APE11-dist-in 13.5831 APE10-dist-out 9.9466 APE9-dist-out 8.7917 None SEP341,TPO342 SEP341,TPO342 XRAY 1.8 0.183 0.223 E 339.0 333.0 4 25 25 0 [[161, 477]] 1.0 6tw2 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Z50A P49759 149 481 484.0 Q7K:501 Type1 Inactive DFGin 7.4479 14.9506 BLAminus -124.17, 179.68 61.85, 81.91 -99.95, 20.34 287.34, 80.47 -70.86, -16.42 in-out in 8.7095 Saltbr-out 4.4776 HRD-in -69.04, -50.58 79.9, -14.59 out-in-in SNCoii in-in ActLoopNT-in 2.9642 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.92, 168.17 APE9-dihe-na 76.04, 153.68 APE8-dihe-in -72.55, 139.47 APE8-rot-in 294.1 APE67-dihe-in -67.47, -19.59 -46.45, -46.57 APE12-dist-in 13.5434 APE11-dist-in 11.5441 APE10-dist-in 7.5172 APE9-dist-in 2.9892 None None None XRAY 1.6 0.152 0.179 A 339.0 333.0 0 25 25 0 [[161, 477]] 1.0 6z50 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 8P04A P49759 148 481 484.0 WAK:60501 Type1 Inactive DFGin 6.7708 13.6576 BLAminus -133.01, 172.38 67.05, 96.19 -115.13, 17.91 300.74, 102.47 -73.76, -12.51 in-in in 8.4668 Saltbr-in 2.8428 HRD-in -68.49, -47.59 68.4, -9.92 in-in-out SNCiio in-out ActLoopNT-in 2.9261 ActLoopCT-out nonTYR APEdihe_aaono APEdist_nnni APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 12.77 APE8-dihe-out 175.17, 160.57 APE8-rot-none 999.0 APE67-dihe-out -106.6, 0.77 -150.85, -100.34 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-in 3.6373 None None None XRAY 2.6 0.212 0.259 A 339.0 320.0 14 25 19 6 [[161, 477]] 1.0 8p04 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 8P08A P49759 148 481 484.0 WAZ:60501 Type1 Inactive DFGin 6.9169 13.8251 BLAminus -129.66, 178.06 64.59, 93.43 -115.04, 31.69 303.49, 95.34 -73.89, -25.33 in-in in 8.6245 Saltbr-in 2.6771 HRD-in -76.48, -42.72 69.48, -15.82 in-in-out SNCiio in-out ActLoopNT-in 2.8847 ActLoopCT-out nonTYR APEdihe_aaoio APEdist_iioo APE10-dihe-na -73.7, -173.61 APE9-dihe-na -62.64, 77.27 APE8-dihe-out -66.74, -40.98 APE8-rot-in 246.46 APE67-dihe-out -59.36, 9.02 163.87, 172.03 APE12-dist-in 12.905 APE11-dist-in 9.2029 APE10-dist-out 8.8464 APE9-dist-out 9.0208 None None None XRAY 2.4 0.211 0.26 A 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 8p08 CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 8UWNA P49759 148 482 484.0 XQX:1002 Type1 Inactive DFGin 6.9694 14.2923 BLAminus -127.28, 178.92 66.55, 91.52 -112.74, 24.76 300.27, 94.07 -77.25, -18.47 in-in in 8.7247 Saltbr-in 2.6923 HRD-in -67.24, -52.59 80.23, -15.08 in-in-out SNCiio in-out ActLoopNT-in 2.9502 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oioo APE10-dihe-na -75.07, 130.75 APE9-dihe-na -78.49, -168.23 APE8-dihe-in -60.11, 132.08 APE8-rot-none 999.0 APE67-dihe-out -60.44, -48.1 -144.72, 138.81 APE12-dist-out 14.5997 APE11-dist-in 13.7486 APE10-dist-out 10.0881 APE9-dist-out 8.8511 None SEP341,TPO342 SEP341,TPO342 XRAY 1.8 0.18 0.24 A 360.0 335.0 0 25 25 0 [[161, 477]] 1.0 8uwn CMGC_CLK1_HUMAN CMGC 3.1e-93 318.2 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6KHDB P49759 149 482 484.0 3NG:1000 Type1 Inactive DFGin 6.9078 14.0758 BLAminus -116.48, -175.0 67.35, 80.01 -102.96, 15.9 292.23, 100.48 -53.02, -40.84 in-in in 8.5827 Saltbr-in 2.6359 HRD-in -57.21, -57.72 79.07, -3.09 in-in-out SNCiio in-out ActLoopNT-in 2.9181 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -136.88, 104.05 APE9-dihe-na 173.26, -145.7 APE8-dihe-in -145.78, 56.63 APE8-rot-in 325.36 APE67-dihe-out -165.57, -36.7 24.99, 58.5 APE12-dist-in 13.5825 APE11-dist-in 11.8902 APE10-dist-in 6.8247 APE9-dist-in 3.7474 None None None XRAY 2.7 0.204 0.274 B 484.0 332.0 2 25 25 0 [[161, 477]] 1.0 6khd CMGC_CLK1_HUMAN CMGC 8.2e-93 317.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 5J1WC P49759 148 483 484.0 6FB:60505,6FB:60506 Type1,Allosteric Inactive DFGin 7.1425 14.2862 BLAminus -122.18, 173.27 71.94, 86.76 -106.83, 22.04 296.04, 87.14 -77.19, -12.48 in-in in 8.5036 Saltbr-in 2.5683 HRD-in -74.28, -51.47 84.87, -18.08 in-in-out SNCiio in-out ActLoopNT-in 2.8804 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -128.25, 150.31 APE9-dihe-na -78.45, -169.37 APE8-dihe-in -56.02, 117.75 APE8-rot-in 301.81 APE67-dihe-out -74.26, -11.87 -128.54, 128.96 APE12-dist-out 14.7541 APE11-dist-in 12.3342 APE10-dist-out 9.2098 APE9-dist-out 8.676 None None None XRAY 2.42 0.191 0.228 C 339.0 314.0 22 25 25 0 [[161, 477]] 1.0 5j1w CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6KHDA P49759 149 481 484.0 3NG:1000 Type1 Inactive DFGin 6.8618 14.4848 None -115.36, -74.37 -61.99, 112.36 -110.01, 19.25 292.55, 104.1 -59.59, -27.31 in-in in 8.7531 Saltbr-in 2.4552 HRD-in -79.61, -40.92 65.39, -11.49 in-in-out SNCiio in-out ActLoopNT-in 2.9802 ActLoopCT-out nonTYR APEdihe_aannn APEdist_ioon APE10-dihe-na -162.31, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -85.78, 10.46 999.0, -15.39 APE12-dist-in 11.8684 APE11-dist-out 7.0432 APE10-dist-out 11.6347 APE9-dist-none 999.0 None None None XRAY 2.7 0.204 0.274 A 484.0 322.0 11 25 23 2 [[161, 477]] 1.0 6khd CMGC_CLK1_HUMAN CMGC 8.2e-93 317.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Q8PA P49759 148 482 484.0 HQB:60501 Type1 None DFGin 7.1106 14.5328 BLAminus -124.47, -177.12 56.99, 94.11 -115.67, 29.05 294.23, 87.9 -80.98, -10.13 in-in in 9.0127 Saltbr-in 3.4176 HRD-in -77.51, -42.79 69.43, -19.47 in-in-none SNCiin in-none ActLoopNT-in 3.1315 ActLoopCT-none nonTYR APEdihe_aanii APEdist_iiin APE10-dihe-na -135.51, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 147.79 APE8-rot-in 323.11 APE67-dihe-in -68.72, -18.82 -64.59, -40.03 APE12-dist-in 13.2041 APE11-dist-in 11.2012 APE10-dist-in 7.2881 APE9-dist-none 999.0 None None None XRAY 3.0 0.201 0.244 A 339.0 334.0 1 25 24 1 [[161, 477]] 1.0 6q8p CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 6Q8PC P49759 148 483 484.0 HQB:60501 Type1 None DFGin 7.2607 13.9451 BLAminus -128.5, 178.53 59.41, 97.23 -121.71, 37.79 304.27, 105.41 -86.72, -22.18 in-in in 8.6759 Saltbr-in 3.006 HRD-in -68.24, -39.01 69.57, -23.21 in-in-none SNCiin in-none ActLoopNT-in 2.9528 ActLoopCT-none nonTYR APEdihe_aanii APEdist_iiin APE10-dihe-na -136.11, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 147.77 APE8-rot-in 314.52 APE67-dihe-in -61.24, -29.44 -57.39, -46.95 APE12-dist-in 13.763 APE11-dist-in 11.1263 APE10-dist-in 7.2951 APE9-dist-none 999.0 None None None XRAY 3.0 0.201 0.244 C 339.0 333.0 3 25 24 1 [[161, 477]] 1.0 6q8p CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1

CMGC_CLK1 (Dual specificity protein kinase CLK1)

Total number of chains: 77
Active chains: 45
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 75 97.4% AF-P49759-K3A
DFGin ABAminus 1 1.3% 6KHDC
DFGin None 1 1.3% 6KHDA

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CLK1 CLK1_HUMAN AF-P49759-K3A P49759 153 484 484.0 No_ligand No_ligand Active DFGin 6.9434 14.1501 BLAminus -132.48, 177.39 60.27, 71.57 -85.18, 10.53 300.3, 105.86 -66.37, -11.95 in-in in 8.4417 Saltbr-in 2.7174 HRD-in -74.62, -35.37 68.27, -12.7 in-in-in SNCiii in-in ActLoopNT-in 2.9068 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -118.72, 174.26 APE9-dihe-na 63.43, 136.97 APE8-dihe-in -54.83, 138.19 APE8-rot-in 291.39 APE67-dihe-in -67.82, -20.27 -52.33, -42.8 APE12-dist-in 13.8915 APE11-dist-in 11.5231 APE10-dist-in 7.7323 APE9-dist-in 3.0057 None None None AF2 -1.0 1.0 1.0 A 332.0 332.0 0 25 25 0 [[161, 477]] 1.0 AF-P49759-K3 Homo sapiens CMGC_CLK1_HUMAN CMGC 1.8e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6YTDA P49759 148 484 484.0 EAE:60501 Type1 Active DFGin 7.2177 14.6236 BLAminus -129.04, -179.37 68.43, 75.26 -99.43, 5.66 289.75, 100.38 -57.22, -23.43 in-in in 8.7889 Saltbr-in 2.7429 HRD-in -67.84, -52.77 79.42, -15.7 in-in-in SNCiii in-in ActLoopNT-in 2.9558 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -135.91, 160.56 APE9-dihe-na 78.51, 152.43 APE8-dihe-in -82.58, 136.21 APE8-rot-in 297.75 APE67-dihe-in -72.13, -8.69 -31.46, -59.55 APE12-dist-in 13.4088 APE11-dist-in 11.1174 APE10-dist-in 7.4109 APE9-dist-in 2.9862 V324A None None XRAY 2.0 0.182 0.228 A 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6ytd Homo sapiens CMGC_CLK1_HUMAN CMGC 1.5e-93 319.2 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6QTYA P49759 149 481 484.0 V25:501 Type1 Active DFGin 7.1891 13.8275 BLAminus -129.69, 172.83 71.11, 83.55 -99.13, 16.45 297.38, 96.6 -71.94, -15.11 in-in in 8.3243 Saltbr-in 2.6508 HRD-in -69.24, -51.3 77.68, -14.79 in-in-in SNCiii in-in ActLoopNT-in 2.9043 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.16, 166.1 APE9-dihe-na 76.64, 158.21 APE8-dihe-in -87.0, 137.14 APE8-rot-in 293.42 APE67-dihe-in -62.6, -10.5 -44.79, -53.3 APE12-dist-in 12.9806 APE11-dist-in 11.463 APE10-dist-in 7.4777 APE9-dist-in 3.0885 None None None XRAY 1.65 0.139 0.203 A 337.0 333.0 0 25 25 0 [[161, 477]] 1.0 6qty Homo sapiens CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6R3DA P49759 152 481 484.0 JQW:901 Type1 Active DFGin 7.2355 14.0134 BLAminus -122.46, 176.35 64.69, 84.91 -101.75, 18.8 296.55, 100.55 -62.91, -23.24 in-in in 8.2719 Saltbr-in 2.9375 HRD-in -66.66, -51.76 77.65, -11.03 in-in-in SNCiii in-in ActLoopNT-in 2.8299 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.87, 173.33 APE9-dihe-na 73.0, 159.5 APE8-dihe-in -89.36, 141.36 APE8-rot-in 302.1 APE67-dihe-in -68.09, -12.73 -48.4, -46.85 APE12-dist-in 13.1776 APE11-dist-in 11.688 APE10-dist-in 7.5691 APE9-dist-in 2.9938 None None None XRAY 1.85 0.223 0.265 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 6r3d Homo sapiens CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6R6EA P49759 153 481 484.0 JTQ:901 Type1 Active DFGin 7.2885 14.2962 BLAminus -128.0, 174.1 72.24, 79.12 -104.06, 19.03 290.47, 84.52 -68.66, -15.84 in-in in 8.4091 Saltbr-in 2.7454 HRD-in -60.82, -42.83 67.21, -15.33 in-in-in SNCiii in-in ActLoopNT-in 2.7501 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.15, 166.85 APE9-dihe-na 79.69, 155.93 APE8-dihe-in -74.39, 146.66 APE8-rot-in 301.47 APE67-dihe-in -66.87, -19.64 -52.56, -47.56 APE12-dist-in 13.1772 APE11-dist-in 11.7084 APE10-dist-in 7.6156 APE9-dist-in 3.0911 None None None XRAY 2.25 0.209 0.258 A 337.0 327.0 2 25 25 0 [[161, 477]] 1.0 6r6e Homo sapiens CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6R6XA P49759 152 481 484.0 JU8:901 Type1 Active DFGin 7.1913 13.8821 BLAminus -123.65, 175.5 67.74, 78.23 -100.49, 14.01 300.01, 96.17 -58.94, -19.36 in-in in 8.4365 Saltbr-in 2.7463 HRD-in -67.05, -47.28 77.18, -15.83 in-in-in SNCiii in-in ActLoopNT-in 2.8079 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.71, 173.64 APE9-dihe-na 76.22, 157.17 APE8-dihe-in -81.77, 144.6 APE8-rot-in 304.54 APE67-dihe-in -66.2, -13.27 -49.16, -50.71 APE12-dist-in 12.9882 APE11-dist-in 11.6232 APE10-dist-in 7.4897 APE9-dist-in 3.0418 None None None XRAY 2.05 0.201 0.247 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 6r6x Homo sapiens CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 7O9YA P49759 152 481 484.0 V5T:501 Type1 Active DFGin 7.2462 13.6868 BLAminus -122.5, 174.1 68.65, 82.2 -100.77, 14.37 301.76, 93.94 -56.91, -24.51 in-in in 8.1529 Saltbr-in 2.7617 HRD-in -69.77, -51.58 81.58, -12.75 in-in-in SNCiii in-in ActLoopNT-in 2.8507 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.84, 169.0 APE9-dihe-na 74.97, 161.24 APE8-dihe-in -86.97, 141.45 APE8-rot-in 302.46 APE67-dihe-in -63.2, -13.37 -47.79, -52.2 APE12-dist-in 12.972 APE11-dist-in 11.507 APE10-dist-in 7.4864 APE9-dist-in 3.0804 None None None XRAY 1.66 0.219 0.246 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 7o9y Homo sapiens CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 7OA0AAA P49759 152 481 484.0 JTQ:501 Type1 Active DFGin 7.2082 13.8687 BLAminus -123.62, 171.83 70.68, 87.81 -105.24, 18.66 295.8, 102.89 -75.22, -10.65 in-in in 8.2485 Saltbr-in 2.7502 HRD-in -68.11, -52.1 81.61, -13.16 in-in-in SNCiii in-in ActLoopNT-in 2.8593 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.31, 171.34 APE9-dihe-na 77.29, 158.23 APE8-dihe-in -81.59, 143.88 APE8-rot-in 304.32 APE67-dihe-in -62.82, -8.69 -51.01, -53.79 APE12-dist-in 13.0487 APE11-dist-in 11.5697 APE10-dist-in 7.4745 APE9-dist-in 3.03 None None None XRAY 1.81 0.195 0.242 AAA 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 7oa0 Homo sapiens CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 1Z57A P49759 148 482 484.0 DBQ:60001 Type1 Active DFGin 6.9813 14.002 BLAminus -125.78, 172.53 74.79, 89.46 -108.53, 21.5 296.6, 99.61 -72.51, -21.17 in-in in 8.4658 Saltbr-in 2.7879 HRD-in -70.25, -52.83 80.14, -14.55 in-in-in SNCiii in-in ActLoopNT-in 2.9435 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.0, 169.19 APE9-dihe-na 76.16, 157.77 APE8-dihe-in -82.83, 140.18 APE8-rot-in 294.7 APE67-dihe-in -63.99, -15.88 -47.28, -50.61 APE12-dist-in 13.3216 APE11-dist-in 11.2235 APE10-dist-in 7.313 APE9-dist-in 3.0014 None None None XRAY 1.7 0.14 0.186 A 339.0 331.0 4 25 25 0 [[161, 477]] 1.0 1z57 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5J1VA P49759 148 483 484.0 6FD:60501 Type1 Active DFGin 7.1 14.1716 BLAminus -126.87, 172.93 72.75, 87.91 -109.91, 21.95 296.61, 87.13 -77.69, -9.89 in-in in 8.5266 Saltbr-in 2.7359 HRD-in -74.36, -52.4 82.96, -16.81 in-in-in SNCiii in-in ActLoopNT-in 2.8778 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.9, 168.51 APE9-dihe-na 72.23, 149.39 APE8-dihe-in -71.93, 136.52 APE8-rot-in 285.15 APE67-dihe-in -66.67, -20.56 -35.82, -53.71 APE12-dist-in 13.5279 APE11-dist-in 11.4445 APE10-dist-in 7.2811 APE9-dist-in 3.0427 None None None XRAY 2.52 0.201 0.244 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 5j1v Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5J1VB P49759 148 482 484.0 6FD:60501 Type1 Active DFGin 7.1093 14.1198 BLAminus -126.74, 175.0 70.24, 87.64 -108.44, 20.05 295.73, 90.04 -77.7, -8.55 in-in in 8.5763 Saltbr-in 2.7543 HRD-in -73.08, -51.15 80.15, -14.17 in-in-in SNCiii in-in ActLoopNT-in 2.8769 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.41, 168.72 APE9-dihe-na 72.72, 151.05 APE8-dihe-in -70.92, 135.35 APE8-rot-in 286.36 APE67-dihe-in -65.82, -21.41 -37.05, -51.94 APE12-dist-in 13.782 APE11-dist-in 11.5423 APE10-dist-in 7.3562 APE9-dist-in 3.0498 None None None XRAY 2.52 0.201 0.244 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 5j1v Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5J1WA P49759 148 483 484.0 6FB:60506 Type1 Active DFGin 7.1724 14.3259 BLAminus -121.81, 173.7 71.87, 86.58 -105.02, 20.94 296.61, 84.3 -77.49, -14.22 in-in in 8.5488 Saltbr-in 2.5641 HRD-in -71.53, -50.92 81.49, -14.91 in-in-in SNCiii in-in ActLoopNT-in 2.9036 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.47, 167.51 APE9-dihe-na 77.02, 140.17 APE8-dihe-in -56.28, 137.97 APE8-rot-in 295.84 APE67-dihe-in -62.06, -22.4 -61.94, -35.28 APE12-dist-in 13.6052 APE11-dist-in 11.4365 APE10-dist-in 7.2516 APE9-dist-in 3.0421 None None None XRAY 2.42 0.191 0.228 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 5j1w Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5J1WB P49759 148 482 484.0 6FB:60503 Type1 Active DFGin 7.2901 14.2646 BLAminus -120.99, 173.46 72.42, 86.12 -105.34, 21.92 296.07, 87.01 -75.02, -15.34 in-in in 8.5851 Saltbr-in 2.5852 HRD-in -69.32, -50.91 80.3, -14.73 in-in-in SNCiii in-in ActLoopNT-in 2.8972 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.41, 167.18 APE9-dihe-na 77.9, 139.82 APE8-dihe-in -54.28, 138.17 APE8-rot-in 296.7 APE67-dihe-in -62.44, -21.37 -62.69, -34.82 APE12-dist-in 13.6477 APE11-dist-in 11.342 APE10-dist-in 7.196 APE9-dist-in 3.035 None None None XRAY 2.42 0.191 0.228 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 5j1w Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6FT8A P49759 148 483 484.0 E6T:60501 Type1 Active DFGin 7.0417 14.1532 BLAminus -123.69, 179.12 66.02, 80.75 -102.66, 23.58 296.94, 92.84 -75.28, -12.2 in-in in 8.4476 Saltbr-in 2.7433 HRD-in -68.91, -53.98 78.36, -16.69 in-in-in SNCiii in-in ActLoopNT-in 2.9408 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.28, 167.17 APE9-dihe-na 78.21, 159.73 APE8-dihe-in -85.1, 140.33 APE8-rot-in 293.05 APE67-dihe-in -66.99, -12.12 -49.73, -45.92 APE12-dist-in 13.2816 APE11-dist-in 11.5166 APE10-dist-in 7.3272 APE9-dist-in 3.0294 None None None XRAY 1.45 0.166 0.195 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6ft8 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6FT9A P49759 148 482 484.0 E6W:60501 Type1 Active DFGin 7.2322 14.2998 BLAminus -125.02, 175.42 67.64, 86.22 -106.42, 22.86 292.22, 81.03 -75.21, -13.41 in-in in 8.4297 Saltbr-in 2.7125 HRD-in -69.31, -51.72 79.55, -13.59 in-in-in SNCiii in-in ActLoopNT-in 2.8663 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.87, 168.01 APE9-dihe-na 73.7, 150.41 APE8-dihe-in -70.08, 140.16 APE8-rot-in 296.52 APE67-dihe-in -66.14, -21.84 -44.66, -47.8 APE12-dist-in 13.556 APE11-dist-in 11.2182 APE10-dist-in 7.2792 APE9-dist-in 2.9326 None None None XRAY 1.87 0.168 0.202 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6ft9 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6FT9B P49759 148 482 484.0 E6W:60501 Type1 Active DFGin 7.2936 14.3139 BLAminus -123.52, 178.1 65.34, 85.29 -106.33, 21.22 292.88, 84.42 -75.16, -8.95 in-in in 8.4862 Saltbr-in 2.7077 HRD-in -71.01, -50.08 80.37, -13.57 in-in-in SNCiii in-in ActLoopNT-in 2.834 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.43, 168.15 APE9-dihe-na 75.76, 149.1 APE8-dihe-in -68.06, 138.01 APE8-rot-in 296.86 APE67-dihe-in -65.44, -22.15 -43.68, -46.72 APE12-dist-in 13.7449 APE11-dist-in 11.2771 APE10-dist-in 7.2841 APE9-dist-in 2.9662 None None None XRAY 1.87 0.168 0.202 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6ft9 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5HA P49759 148 481 484.0 H3N:60507 Type1 Active DFGin 6.9359 13.9902 BLAminus -127.91, 175.49 70.62, 86.84 -104.99, 23.28 297.7, 98.27 -76.67, -15.26 in-in in 8.6705 Saltbr-in 2.7942 HRD-in -71.42, -54.52 81.98, -15.98 in-in-in SNCiii in-in ActLoopNT-in 2.9892 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.5, 162.59 APE9-dihe-na 81.01, 150.81 APE8-dihe-in -73.05, 137.12 APE8-rot-in 298.85 APE67-dihe-in -65.31, -13.64 -50.7, -47.04 APE12-dist-in 12.9825 APE11-dist-in 11.3246 APE10-dist-in 7.2343 APE9-dist-in 3.0974 None None None XRAY 1.49 0.179 0.206 A 339.0 323.0 11 25 25 0 [[161, 477]] 1.0 6i5h Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5IA P49759 148 483 484.0 H3E:60501 Type1 Active DFGin 6.9087 13.9494 BLAminus -127.6, 172.7 71.85, 87.8 -102.42, 20.37 300.05, 101.13 -74.42, -16.22 in-in in 8.7126 Saltbr-in 2.693 HRD-in -75.53, -52.34 81.22, -14.82 in-in-in SNCiii in-in ActLoopNT-in 2.9983 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.19, 164.34 APE9-dihe-na 79.5, 152.78 APE8-dihe-in -78.57, 135.82 APE8-rot-in 292.41 APE67-dihe-in -65.9, -11.23 -46.6, -47.35 APE12-dist-in 13.1135 APE11-dist-in 11.2837 APE10-dist-in 7.2519 APE9-dist-in 3.0736 None None None XRAY 1.6 0.166 0.196 A 339.0 333.0 3 25 25 0 [[161, 477]] 1.0 6i5i Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5KB P49759 148 481 484.0 H3H:60504 Type1 Active DFGin 7.006 14.3591 BLAminus -126.82, 178.06 66.53, 84.63 -104.0, 26.37 299.27, 91.89 -80.46, -16.31 in-in in 9.0291 Saltbr-in 2.6927 HRD-in -71.59, -48.77 75.18, -11.75 in-in-in SNCiii in-in ActLoopNT-in 2.9844 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.96, 164.13 APE9-dihe-na 74.43, 150.15 APE8-dihe-in -66.68, 137.66 APE8-rot-in 303.78 APE67-dihe-in -77.74, -18.3 -54.0, -31.51 APE12-dist-in 13.8442 APE11-dist-in 11.2244 APE10-dist-in 7.3953 APE9-dist-in 3.093 None None None XRAY 2.3 0.197 0.224 B 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 6i5k Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5KC P49759 148 483 484.0 H3H:60504 Type1 Active DFGin 6.9865 14.3514 BLAminus -125.41, 178.1 66.91, 85.45 -105.62, 25.72 298.18, 84.65 -79.89, -19.48 in-in in 8.919 Saltbr-in 2.6659 HRD-in -72.35, -49.89 76.53, -11.56 in-in-in SNCiii in-in ActLoopNT-in 3.0005 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.9, 163.92 APE9-dihe-na 72.8, 149.97 APE8-dihe-in -66.75, 139.4 APE8-rot-in 303.5 APE67-dihe-in -77.85, -17.5 -52.64, -34.11 APE12-dist-in 13.6161 APE11-dist-in 11.124 APE10-dist-in 7.3407 APE9-dist-in 3.1121 None None None XRAY 2.3 0.197 0.224 C 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6i5k Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5LB P49759 148 481 484.0 H3Q:60502 Type1 Active DFGin 6.9284 14.418 BLAminus -123.55, 178.93 67.48, 93.05 -113.53, 21.71 295.78, 85.8 -74.38, -22.09 in-in in 8.9824 Saltbr-in 2.7395 HRD-in -69.85, -49.79 74.87, -13.88 in-in-in SNCiii in-in ActLoopNT-in 2.9995 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.82, 165.73 APE9-dihe-na 81.08, 146.54 APE8-dihe-in -62.76, 135.54 APE8-rot-in 302.63 APE67-dihe-in -68.98, -24.89 -54.53, -33.68 APE12-dist-in 13.8519 APE11-dist-in 11.4167 APE10-dist-in 7.226 APE9-dist-in 3.1016 None None None XRAY 2.55 0.195 0.221 B 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 6i5l Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5LC P49759 148 483 484.0 H3Q:60502 Type1 Active DFGin 6.9131 14.3839 BLAminus -123.57, 177.17 68.91, 92.22 -114.6, 21.5 296.12, 85.91 -74.75, -23.49 in-in in 8.8781 Saltbr-in 2.7107 HRD-in -71.08, -49.61 75.52, -13.95 in-in-in SNCiii in-in ActLoopNT-in 3.0208 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.58, 165.38 APE9-dihe-na 80.23, 146.0 APE8-dihe-in -62.57, 137.3 APE8-rot-in 302.62 APE67-dihe-in -70.1, -23.69 -53.95, -35.33 APE12-dist-in 13.6577 APE11-dist-in 11.3372 APE10-dist-in 7.1791 APE9-dist-in 3.1361 None None None XRAY 2.55 0.195 0.221 C 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6i5l Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Q8KA P49759 148 484 484.0 FG9:60502 Type1 Active DFGin 7.0383 14.0726 BLAminus -126.96, 173.92 68.96, 94.14 -110.91, 19.67 299.22, 86.31 -70.74, -15.36 in-in in 8.7893 Saltbr-in 2.6969 HRD-in -64.71, -54.26 80.91, -18.18 in-in-in SNCiii in-in ActLoopNT-in 2.9149 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.28, 157.45 APE9-dihe-na 83.98, 154.49 APE8-dihe-in -77.73, 126.84 APE8-rot-in 298.77 APE67-dihe-in -63.27, -22.97 -33.76, -49.02 APE12-dist-in 13.3669 APE11-dist-in 11.2855 APE10-dist-in 7.4682 APE9-dist-in 3.1111 None None None XRAY 2.29 0.191 0.259 A 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6q8k Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6YTAA P49759 148 483 484.0 IYZ:60702 Type1 Active DFGin 6.9349 13.7248 BLAminus -125.39, 175.02 66.16, 92.34 -102.15, 17.18 301.41, 98.15 -60.08, -20.3 in-in in 8.3168 Saltbr-in 2.6989 HRD-in -68.08, -57.05 83.09, -18.57 in-in-in SNCiii in-in ActLoopNT-in 2.8997 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.65, 155.94 APE9-dihe-na 83.67, 157.83 APE8-dihe-in -84.55, 129.06 APE8-rot-in 292.9 APE67-dihe-in -62.02, -24.22 -28.74, -53.35 APE12-dist-in 13.2113 APE11-dist-in 11.6634 APE10-dist-in 7.3747 APE9-dist-in 3.1591 None None None XRAY 2.3 0.194 0.275 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6yta Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6YTEC P49759 148 484 484.0 EAE:60501 Type1 Active DFGin 7.1447 14.1109 BLAminus -123.36, 172.5 72.26, 86.11 -107.09, 11.71 295.65, 98.47 -58.29, -17.8 in-in in 8.5445 Saltbr-in 2.2253 HRD-in -60.42, -59.86 88.88, -8.99 in-in-in SNCiii in-in ActLoopNT-in 3.0048 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.24, 160.76 APE9-dihe-na 81.35, 157.72 APE8-dihe-in -87.96, 130.83 APE8-rot-in 293.05 APE67-dihe-in -54.77, -23.25 -31.22, -65.53 APE12-dist-in 13.3746 APE11-dist-in 11.4404 APE10-dist-in 7.3205 APE9-dist-in 3.082 None None None XRAY 2.3 0.184 0.258 C 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6yte Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6YTIA P49759 150 482 484.0 7A7:605 Type1 Active DFGin 7.2921 14.242 BLAminus -134.7, 172.33 69.03, 94.12 -110.31, 22.0 290.95, 98.93 -72.82, -22.05 in-in in 8.6449 Saltbr-in 2.6167 HRD-in -68.46, -54.35 84.41, -17.31 in-in-in SNCiii in-in ActLoopNT-in 2.8883 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.78, 154.97 APE9-dihe-na 84.02, 157.2 APE8-dihe-in -78.01, 116.07 APE8-rot-in 301.91 APE67-dihe-in -65.16, -18.0 -14.75, -58.2 APE12-dist-in 13.4174 APE11-dist-in 11.0368 APE10-dist-in 7.4563 APE9-dist-in 3.0199 None None None XRAY 2.4 0.198 0.256 A 339.0 329.0 4 25 25 0 [[161, 477]] 1.0 6yti Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Z4ZA P49759 148 482 484.0 PQ5:60505 Type1 Active DFGin 7.046 14.2363 BLAminus -126.68, 179.24 66.69, 82.0 -103.33, 19.73 297.68, 94.61 -71.59, -13.97 in-in in 8.4611 Saltbr-in 2.7642 HRD-in -69.38, -51.98 76.89, -13.79 in-in-in SNCiii in-in ActLoopNT-in 2.9245 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.91, 169.84 APE9-dihe-na 70.81, 154.45 APE8-dihe-in -79.18, 136.44 APE8-rot-in 295.15 APE67-dihe-in -64.16, -17.67 -45.6, -49.57 APE12-dist-in 13.5127 APE11-dist-in 11.3594 APE10-dist-in 7.327 APE9-dist-in 3.0405 None None None XRAY 2.07 0.177 0.213 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6z4z Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Z4ZB P49759 148 484 484.0 PQ5:60501 Type1 Active DFGin 7.0483 14.168 BLAminus -127.78, 179.44 66.36, 84.49 -106.02, 23.22 298.83, 96.06 -73.86, -11.97 in-in in 8.4214 Saltbr-in 2.7252 HRD-in -70.61, -51.12 77.5, -15.65 in-in-in SNCiii in-in ActLoopNT-in 2.9096 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.17, 168.57 APE9-dihe-na 73.19, 152.9 APE8-dihe-in -77.75, 136.06 APE8-rot-in 294.47 APE67-dihe-in -61.42, -18.21 -47.63, -47.77 APE12-dist-in 13.4848 APE11-dist-in 11.247 APE10-dist-in 7.2192 APE9-dist-in 3.0518 None None None XRAY 2.07 0.177 0.213 B 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6z4z Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Z4ZC P49759 148 482 484.0 PQ5:60502 Type1 Active DFGin 7.1081 14.2491 BLAminus -126.87, 178.82 67.48, 81.17 -101.74, 18.48 298.94, 95.28 -65.75, -17.47 in-in in 8.5666 Saltbr-in 2.7627 HRD-in -67.93, -52.14 78.08, -12.45 in-in-in SNCiii in-in ActLoopNT-in 2.8763 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.01, 169.28 APE9-dihe-na 73.05, 151.25 APE8-dihe-in -74.69, 135.04 APE8-rot-in 294.69 APE67-dihe-in -63.57, -18.13 -46.66, -45.93 APE12-dist-in 13.7076 APE11-dist-in 11.4576 APE10-dist-in 7.407 APE9-dist-in 3.0276 None None None XRAY 2.07 0.177 0.213 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6z4z Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6ZLNA P49759 148 484 484.0 PKB:60503 Type1 Active DFGin 7.0057 14.1924 BLAminus -125.63, 176.89 76.78, 75.35 -103.44, 16.76 293.35, 98.15 -70.81, -12.33 in-in in 8.6634 Saltbr-in 2.7072 HRD-in -67.73, -49.47 78.97, -14.05 in-in-in SNCiii in-in ActLoopNT-in 2.9351 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.54, 162.21 APE9-dihe-na 79.84, 163.79 APE8-dihe-in -96.39, 123.92 APE8-rot-in 291.96 APE67-dihe-in -72.31, -12.72 -20.91, -56.58 APE12-dist-in 13.2334 APE11-dist-in 10.9238 APE10-dist-in 7.2166 APE9-dist-in 3.0919 None None None XRAY 1.7 0.171 0.199 A 339.0 337.0 0 25 25 0 [[161, 477]] 1.0 6zln Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 7AK3A P49759 148 483 484.0 RH8:60501 Type1 Active DFGin 7.3197 14.2837 BLAminus -128.56, 172.37 67.01, 84.33 -103.74, 27.34 296.18, 85.72 -72.52, -23.23 in-in in 8.6033 Saltbr-in 2.8652 HRD-in -61.61, -53.86 89.68, -14.81 in-in-in SNCiii in-in ActLoopNT-in 2.9582 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.68, 162.47 APE9-dihe-na 75.05, 158.38 APE8-dihe-in -88.77, 128.79 APE8-rot-in 301.95 APE67-dihe-in -60.58, -28.09 -3.93, -77.31 APE12-dist-in 13.3868 APE11-dist-in 11.1501 APE10-dist-in 7.274 APE9-dist-in 2.9982 None None None XRAY 2.5 0.213 0.26 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 7ak3 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 7OPGA P49759 148 482 484.0 06N:60501 Type1 Active DFGin 7.0787 14.3372 BLAminus -125.23, 174.99 68.34, 89.35 -108.55, 22.34 294.5, 84.43 -74.9, -16.57 in-in in 8.8275 Saltbr-in 2.697 HRD-in -68.7, -53.19 79.41, -13.79 in-in-in SNCiii in-in ActLoopNT-in 2.8637 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.87, 169.9 APE9-dihe-na 72.2, 152.58 APE8-dihe-in -74.2, 140.4 APE8-rot-in 296.34 APE67-dihe-in -64.01, -18.08 -47.78, -49.23 APE12-dist-in 13.4538 APE11-dist-in 11.205 APE10-dist-in 7.2886 APE9-dist-in 3.0135 None None None XRAY 1.93 0.176 0.208 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 7opg Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 7OPGB P49759 148 483 484.0 06N:60501 Type1 Active DFGin 7.0918 14.2954 BLAminus -128.58, 171.98 71.57, 88.89 -110.25, 21.49 294.73, 85.57 -73.38, -14.32 in-in in 8.7933 Saltbr-in 2.6848 HRD-in -66.06, -53.32 81.87, -15.7 in-in-in SNCiii in-in ActLoopNT-in 2.843 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.09, 167.09 APE9-dihe-na 74.85, 150.04 APE8-dihe-in -76.84, 138.69 APE8-rot-in 295.58 APE67-dihe-in -61.09, -19.4 -51.05, -46.51 APE12-dist-in 13.2757 APE11-dist-in 11.1509 APE10-dist-in 7.227 APE9-dist-in 3.0505 None None None XRAY 1.93 0.176 0.208 B 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 7opg Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 7OPGC P49759 148 482 484.0 06N:60501 Type1 Active DFGin 7.1396 14.3181 BLAminus -126.92, 172.88 71.54, 91.0 -109.11, 17.42 294.29, 87.52 -72.35, -14.96 in-in in 8.8983 Saltbr-in 2.7034 HRD-in -68.36, -53.23 82.74, -14.25 in-in-in SNCiii in-in ActLoopNT-in 2.8367 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.58, 169.34 APE9-dihe-na 74.62, 150.8 APE8-dihe-in -72.07, 139.48 APE8-rot-in 296.41 APE67-dihe-in -63.14, -17.95 -50.02, -46.94 APE12-dist-in 13.4592 APE11-dist-in 11.323 APE10-dist-in 7.3831 APE9-dist-in 3.0248 None None None XRAY 1.93 0.176 0.208 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 7opg Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6FYOA P49759 148 481 484.0 EAQ:501 Type1 Active DFGin 7.1303 14.6092 BLAminus -126.41, -177.97 57.7, 79.82 -101.45, 23.66 290.45, 86.2 -71.99, -23.62 in-in in 8.2538 Saltbr-in 2.8261 HRD-in -67.73, -44.39 69.27, -21.51 in-in-in SNCiii in-in ActLoopNT-in 2.7761 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.41, 162.2 APE9-dihe-na 76.62, 158.52 APE8-dihe-in -81.15, 137.38 APE8-rot-in 320.28 APE67-dihe-in -54.52, -12.47 -37.95, -53.62 APE12-dist-in 13.1043 APE11-dist-in 11.2911 APE10-dist-in 7.0165 APE9-dist-in 3.2103 None None None XRAY 2.32 0.204 0.234 A 339.0 331.0 3 25 25 0 [[161, 477]] 1.0 6fyo Homo sapiens CMGC_CLK1_HUMAN CMGC 2e-93 318.8 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5X8IA P49759 154 481 484.0 SQZ:501 Type1 Active DFGin 7.3534 13.9989 BLAminus -122.66, 172.48 71.45, 69.85 -89.46, 19.16 303.2, 86.95 -71.61, -17.76 in-in in 8.3789 Saltbr-in 2.5421 HRD-in -68.32, -52.49 79.94, -11.57 in-in-in SNCiii in-in ActLoopNT-in 2.8658 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.32, 168.72 APE9-dihe-na 74.05, 158.08 APE8-dihe-in -81.53, 144.19 APE8-rot-in 300.53 APE67-dihe-in -65.15, -11.28 -51.71, -50.28 APE12-dist-in 13.0833 APE11-dist-in 11.6511 APE10-dist-in 7.533 APE9-dist-in 3.016 R432A None None XRAY 1.902 0.168 0.206 A 346.0 328.0 0 25 25 0 [[161, 477]] 1.0 5x8i Homo sapiens CMGC_CLK1_HUMAN CMGC 2.7e-93 318.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5X8IB P49759 155 481 484.0 SQZ:501 Type1 Active DFGin 7.3842 13.9802 BLAminus -126.45, 170.69 71.83, 69.37 -88.36, 11.76 302.43, 89.48 -69.31, -18.97 in-in in 8.3824 Saltbr-in 2.41 HRD-in -67.27, -52.41 79.09, -12.7 in-in-in SNCiii in-in ActLoopNT-in 2.8887 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.02, 169.54 APE9-dihe-na 72.76, 157.49 APE8-dihe-in -80.25, 143.44 APE8-rot-in 301.33 APE67-dihe-in -65.52, -10.3 -49.82, -50.77 APE12-dist-in 13.1161 APE11-dist-in 11.6767 APE10-dist-in 7.4994 APE9-dist-in 3.0166 R432A None None XRAY 1.902 0.168 0.206 B 346.0 327.0 0 25 25 0 [[161, 477]] 1.0 5x8i Homo sapiens CMGC_CLK1_HUMAN CMGC 2.7e-93 318.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6YTGA P49759 148 483 484.0 KHC:60501,KHC:60502 Type1,Allosteric Active DFGin 7.1086 14.3781 BLAminus -123.68, -179.19 66.81, 76.1 -102.89, 15.19 291.91, 90.06 -75.03, -12.8 in-in in 8.5496 Saltbr-in 2.696 HRD-in -64.66, -54.29 85.54, -10.78 in-in-in SNCiii in-in ActLoopNT-in 2.8316 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -106.45, 156.23 APE9-dihe-na 81.17, 153.49 APE8-dihe-in -77.75, 128.48 APE8-rot-in 300.43 APE67-dihe-in -69.97, -17.37 -12.96, -64.06 APE12-dist-in 13.337 APE11-dist-in 11.4029 APE10-dist-in 7.7563 APE9-dist-in 2.9823 None None None XRAY 1.95 0.207 0.261 A 339.0 329.0 7 25 25 0 [[161, 477]] 1.0 6ytg Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6R8JA P49759 152 481 484.0 JUW:501,JUW:502 Type1,Type1 Active DFGin 7.1717 13.6765 BLAminus -124.23, 172.49 72.75, 83.0 -102.73, 17.52 298.34, 101.12 -64.7, -21.81 in-in in 8.1336 Saltbr-in 2.8945 HRD-in -66.22, -54.05 83.24, -16.78 in-in-in SNCiii in-in ActLoopNT-in 2.8729 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.97, 169.66 APE9-dihe-na 75.96, 160.32 APE8-dihe-in -86.77, 141.55 APE8-rot-in 304.05 APE67-dihe-in -66.39, -13.17 -48.7, -48.98 APE12-dist-in 13.0103 APE11-dist-in 11.5266 APE10-dist-in 7.5479 APE9-dist-in 2.9805 None None None XRAY 1.75 0.218 0.263 A 337.0 330.0 0 25 25 0 [[161, 477]] 1.0 6r8j Homo sapiens CMGC_CLK1_HUMAN CMGC 1.9e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6KHDC P49759 150 479 484.0 3NG:1000 Type1 Inactive DFGin 7.0261 14.4118 ABAminus -125.6, -45.1 -89.27, 107.55 -111.64, 19.23 292.41, 98.32 -77.1, 0.74 in-in in 8.7674 Saltbr-in 2.9039 HRD-in -53.74, -54.41 89.98, -20.88 in-in-out SNCiio in-out ActLoopNT-in 2.895 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iioo APE10-dihe-na -118.02, -81.8 APE9-dihe-na -80.38, 126.35 APE8-dihe-in -130.72, 139.1 APE8-rot-out 73.02 APE67-dihe-in -49.48, -32.44 -62.98, -36.18 APE12-dist-in 13.3713 APE11-dist-in 9.0973 APE10-dist-out 11.3298 APE9-dist-out 7.8489 None None None XRAY 2.7 0.204 0.274 C 484.0 325.0 5 25 25 0 [[161, 477]] 1.0 6khd Homo sapiens CMGC_CLK1_HUMAN CMGC 8.2e-93 317.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN AF-P49759-K1A P49759 153 484 484.0 No_ligand No_ligand Inactive DFGin 7.0737 14.19 BLAminus -127.24, 176.41 62.19, 72.99 -88.32, 9.55 297.11, 102.62 -68.31, -9.87 in-in in 8.4508 Saltbr-in 2.696 HRD-in -72.36, -39.16 64.91, -10.55 in-in-out SNCiio in-out ActLoopNT-in 2.9091 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oiii APE10-dihe-na -123.01, 174.5 APE9-dihe-na 65.72, 145.79 APE8-dihe-in -57.06, 135.18 APE8-rot-in 292.86 APE67-dihe-in -70.16, -18.82 -51.52, -41.74 APE12-dist-out 14.1099 APE11-dist-in 11.8348 APE10-dist-in 7.5822 APE9-dist-in 2.9068 None None None AF2 -1.0 1.0 1.0 A 332.0 332.0 0 25 25 0 [[161, 477]] 1.0 AF-P49759-K1 Homo sapiens CMGC_CLK1_HUMAN CMGC 1.8e-93 318.9 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 2VAGA P49759 148 481 484.0 V25:61482 Type1 Inactive DFGin 7.1077 14.0258 BLAminus -129.43, 175.64 66.18, 85.97 -104.96, 23.22 293.24, 95.17 -73.67, -15.41 in-in in 8.37 Saltbr-in 2.6268 HRD-in -71.48, -53.18 82.14, -13.71 in-in-out SNCiio in-out ActLoopNT-in 2.8437 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oioo APE10-dihe-na -88.11, 138.68 APE9-dihe-na -83.4, -165.24 APE8-dihe-in -49.62, 134.22 APE8-rot-none 999.0 APE67-dihe-out -47.82, -50.26 -151.88, 142.32 APE12-dist-out 14.0645 APE11-dist-in 12.8642 APE10-dist-out 9.7767 APE9-dist-out 8.6182 None SEP341,TPO342 SEP341,TPO342 XRAY 1.8 0.182 0.225 A 339.0 331.0 3 25 25 0 [[161, 477]] 1.0 2vag Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5J1VC P49759 148 483 484.0 6FD:60501 Type1 Inactive DFGin 7.0653 14.1863 BLAminus -127.76, 172.5 71.94, 87.97 -108.84, 22.87 296.53, 88.54 -79.84, -9.02 in-in in 8.5354 Saltbr-in 2.7469 HRD-in -76.64, -52.07 83.95, -17.44 in-in-out SNCiio in-out ActLoopNT-in 2.8928 ActLoopCT-out nonTYR APEdihe_aannn APEdist_oion APE10-dihe-na -156.89, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, -20.42 999.0, 999.0 APE12-dist-out 14.2512 APE11-dist-in 11.6023 APE10-dist-out 9.6806 APE9-dist-none 999.0 None None None XRAY 2.52 0.201 0.244 C 339.0 312.0 24 25 22 3 [[161, 477]] 1.0 5j1v Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6FT9C P49759 148 482 484.0 E6W:60501 Type1 Inactive DFGin 7.2141 14.2533 BLAminus -122.85, 177.29 65.92, 85.07 -105.77, 22.23 295.06, 82.45 -71.81, -8.98 in-in in 8.3694 Saltbr-in 2.6709 HRD-in -69.43, -51.23 80.08, -14.43 in-in-out SNCiio in-out ActLoopNT-in 2.8644 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -129.97, 131.35 APE9-dihe-na -47.51, 149.39 APE8-dihe-in -75.79, 135.36 APE8-rot-in 303.89 APE67-dihe-out -54.68, -26.4 -154.15, 148.3 APE12-dist-out 14.7393 APE11-dist-in 12.4265 APE10-dist-out 9.6939 APE9-dist-out 8.7023 None None None XRAY 1.87 0.168 0.202 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6ft9 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6G33A P49759 148 482 484.0 5ID:60501 Type1 Inactive DFGin 7.0386 14.0293 BLAminus -127.31, 176.31 68.38, 85.72 -104.03, 25.47 298.82, 93.66 -74.89, -17.97 in-in in 8.3822 Saltbr-in 2.7246 HRD-in -70.1, -50.84 78.28, -13.18 in-in-out SNCiio in-out ActLoopNT-in 2.8482 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oioo APE10-dihe-na -128.78, 136.1 APE9-dihe-na -77.1, 148.33 APE8-dihe-in -66.51, 123.5 APE8-rot-none 999.0 APE67-dihe-out -66.2, -20.29 -135.8, 167.22 APE12-dist-out 14.7008 APE11-dist-in 12.3537 APE10-dist-out 9.4988 APE9-dist-out 8.7999 None SEP341,TPO342 SEP341,TPO342 XRAY 2.05 0.19 0.218 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6g33 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6G33B P49759 148 482 484.0 5ID:60501 Type1 Inactive DFGin 7.0769 13.9786 BLAminus -125.16, 175.81 68.83, 87.13 -106.27, 24.24 297.31, 93.02 -76.58, -16.07 in-in in 8.3864 Saltbr-in 2.6996 HRD-in -69.85, -51.6 75.98, -11.49 in-in-out SNCiio in-out ActLoopNT-in 2.8786 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iioo APE10-dihe-na -123.97, 135.36 APE9-dihe-na -72.42, 114.42 APE8-dihe-in -42.53, 141.22 APE8-rot-in 302.44 APE67-dihe-out -66.45, -16.55 -136.36, 149.49 APE12-dist-in 13.8836 APE11-dist-in 11.9062 APE10-dist-out 10.3491 APE9-dist-out 9.743 None None None XRAY 2.05 0.19 0.218 B 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6g33 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6G33C P49759 148 482 484.0 5ID:60501 Type1 Inactive DFGin 7.1529 14.0498 BLAminus -127.31, 175.45 68.57, 84.45 -104.42, 25.23 297.23, 96.23 -74.84, -18.72 in-in in 8.4304 Saltbr-in 2.707 HRD-in -68.44, -51.98 75.83, -9.76 in-in-out SNCiio in-out ActLoopNT-in 2.8328 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oioi APE10-dihe-na -158.67, 144.43 APE9-dihe-na 80.91, 147.02 APE8-dihe-in -56.89, 133.87 APE8-rot-none 999.0 APE67-dihe-in -70.75, -20.64 -58.82, -30.99 APE12-dist-out 14.1296 APE11-dist-in 11.4642 APE10-dist-out 8.2148 APE9-dist-in 3.07 None None None XRAY 2.05 0.19 0.218 C 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6g33 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5KA P49759 148 482 484.0 H3H:60503 Type1 Inactive DFGin 7.0191 14.2807 BLAminus -127.95, 177.21 67.34, 85.43 -106.5, 25.82 299.72, 92.63 -80.22, -14.39 in-in in 8.8988 Saltbr-in 2.6726 HRD-in -72.89, -48.86 76.37, -11.75 in-in-out SNCiio in-out ActLoopNT-in 3.0079 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -139.66, 157.93 APE9-dihe-na -83.57, -145.55 APE8-dihe-in -77.05, 120.2 APE8-rot-in 311.82 APE67-dihe-out -112.74, 31.9 -178.22, 144.22 APE12-dist-out 14.3954 APE11-dist-in 12.6175 APE10-dist-out 8.7668 APE9-dist-out 8.7264 None None None XRAY 2.3 0.197 0.224 A 339.0 335.0 0 25 25 0 [[161, 477]] 1.0 6i5k Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6I5LA P49759 148 483 484.0 H3Q:60503 Type1 Inactive DFGin 6.9146 14.3203 BLAminus -124.28, 177.5 67.34, 93.35 -114.57, 21.88 295.56, 86.41 -76.53, -21.33 in-in in 8.8454 Saltbr-in 2.712 HRD-in -70.91, -49.07 76.68, -14.69 in-in-out SNCiio in-out ActLoopNT-in 3.01 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -133.89, 159.24 APE9-dihe-na -106.72, -141.34 APE8-dihe-in -74.35, 99.26 APE8-rot-in 314.71 APE67-dihe-out -134.72, 40.5 -167.53, 148.17 APE12-dist-out 14.5511 APE11-dist-in 12.2796 APE10-dist-out 9.5559 APE9-dist-out 8.8533 None None None XRAY 2.55 0.195 0.221 A 339.0 336.0 0 25 25 0 [[161, 477]] 1.0 6i5l Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Q8PB P49759 148 483 484.0 HQB:60501 Type1 Inactive DFGin 6.6661 14.0806 BLAminus -123.82, 175.86 66.42, 98.63 -122.53, 30.35 298.66, 86.39 -77.45, -10.39 in-in in 8.7879 Saltbr-in 2.9933 HRD-in -68.29, -44.12 72.95, -22.76 in-in-out SNCiio in-out ActLoopNT-in 3.0122 ActLoopCT-out nonTYR APEdihe_aannn APEdist_oion APE10-dihe-na -125.35, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -60.69, -36.51 999.0, -33.63 APE12-dist-out 14.4348 APE11-dist-in 12.4103 APE10-dist-out 9.3984 APE9-dist-none 999.0 None None None XRAY 3.0 0.201 0.244 B 339.0 331.0 5 25 23 2 [[161, 477]] 1.0 6q8p Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6RAAA P49759 148 481 484.0 JWN:60501 Type1 Inactive DFGin 6.8873 13.7549 BLAminus -129.66, 171.4 69.19, 92.86 -107.95, 20.85 301.15, 106.22 -67.28, -18.14 in-in in 8.302 Saltbr-in 2.9175 HRD-in -72.74, -49.16 79.77, -9.47 in-in-out SNCiio in-out ActLoopNT-in 2.9284 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -136.73, 160.54 APE9-dihe-na 78.15, 152.31 APE8-dihe-in -85.85, 139.96 APE8-rot-out 71.85 APE67-dihe-in -63.36, -27.28 -38.74, -49.54 APE12-dist-in 13.2788 APE11-dist-in 11.3142 APE10-dist-in 7.2917 APE9-dist-in 3.081 None None None XRAY 2.1 0.19 0.233 A 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 6raa Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6TW2E P49759 148 484 484.0 V25:62301 Type1 Inactive DFGin 7.1046 14.057 BLAminus -132.08, 175.35 68.1, 86.44 -104.28, 22.11 293.58, 88.16 -72.28, -16.22 in-in in 8.3715 Saltbr-in 2.6068 HRD-in -73.71, -50.29 77.69, -11.9 in-in-out SNCiio in-out ActLoopNT-in 2.8741 ActLoopCT-out nonTYR APEdihe_aanao APEdist_oioo APE10-dihe-na -119.46, 133.12 APE9-dihe-na 999.0, -6.85 APE8-dihe-none 999.0, 103.3 APE8-rot-na 296.95 APE67-dihe-out -59.07, -41.0 14.44, 142.85 APE12-dist-out 14.8499 APE11-dist-in 13.5831 APE10-dist-out 9.9466 APE9-dist-out 8.7917 None SEP341,TPO342 SEP341,TPO342 XRAY 1.8 0.183 0.223 E 339.0 333.0 4 25 25 0 [[161, 477]] 1.0 6tw2 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Z50A P49759 149 481 484.0 Q7K:501 Type1 Inactive DFGin 7.4479 14.9506 BLAminus -124.17, 179.68 61.85, 81.91 -99.95, 20.34 287.34, 80.47 -70.86, -16.42 in-out in 8.7095 Saltbr-out 4.4776 HRD-in -69.04, -50.58 79.9, -14.59 out-in-in SNCoii in-in ActLoopNT-in 2.9642 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.92, 168.17 APE9-dihe-na 76.04, 153.68 APE8-dihe-in -72.55, 139.47 APE8-rot-in 294.1 APE67-dihe-in -67.47, -19.59 -46.45, -46.57 APE12-dist-in 13.5434 APE11-dist-in 11.5441 APE10-dist-in 7.5172 APE9-dist-in 2.9892 None None None XRAY 1.6 0.152 0.179 A 339.0 333.0 0 25 25 0 [[161, 477]] 1.0 6z50 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 8P04A P49759 148 481 484.0 WAK:60501 Type1 Inactive DFGin 6.7708 13.6576 BLAminus -133.01, 172.38 67.05, 96.19 -115.13, 17.91 300.74, 102.47 -73.76, -12.51 in-in in 8.4668 Saltbr-in 2.8428 HRD-in -68.49, -47.59 68.4, -9.92 in-in-out SNCiio in-out ActLoopNT-in 2.9261 ActLoopCT-out nonTYR APEdihe_aaono APEdist_nnni APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 12.77 APE8-dihe-out 175.17, 160.57 APE8-rot-none 999.0 APE67-dihe-out -106.6, 0.77 -150.85, -100.34 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-in 3.6373 None None None XRAY 2.6 0.212 0.259 A 339.0 320.0 14 25 19 6 [[161, 477]] 1.0 8p04 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 8P08A P49759 148 481 484.0 WAZ:60501 Type1 Inactive DFGin 6.9169 13.8251 BLAminus -129.66, 178.06 64.59, 93.43 -115.04, 31.69 303.49, 95.34 -73.89, -25.33 in-in in 8.6245 Saltbr-in 2.6771 HRD-in -76.48, -42.72 69.48, -15.82 in-in-out SNCiio in-out ActLoopNT-in 2.8847 ActLoopCT-out nonTYR APEdihe_aaoio APEdist_iioo APE10-dihe-na -73.7, -173.61 APE9-dihe-na -62.64, 77.27 APE8-dihe-out -66.74, -40.98 APE8-rot-in 246.46 APE67-dihe-out -59.36, 9.02 163.87, 172.03 APE12-dist-in 12.905 APE11-dist-in 9.2029 APE10-dist-out 8.8464 APE9-dist-out 9.0208 None None None XRAY 2.4 0.211 0.26 A 339.0 334.0 0 25 25 0 [[161, 477]] 1.0 8p08 Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 8UWNA P49759 148 482 484.0 XQX:1002 Type1 Inactive DFGin 6.9694 14.2923 BLAminus -127.28, 178.92 66.55, 91.52 -112.74, 24.76 300.27, 94.07 -77.25, -18.47 in-in in 8.7247 Saltbr-in 2.6923 HRD-in -67.24, -52.59 80.23, -15.08 in-in-out SNCiio in-out ActLoopNT-in 2.9502 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oioo APE10-dihe-na -75.07, 130.75 APE9-dihe-na -78.49, -168.23 APE8-dihe-in -60.11, 132.08 APE8-rot-none 999.0 APE67-dihe-out -60.44, -48.1 -144.72, 138.81 APE12-dist-out 14.5997 APE11-dist-in 13.7486 APE10-dist-out 10.0881 APE9-dist-out 8.8511 None SEP341,TPO342 SEP341,TPO342 XRAY 1.8 0.18 0.24 A 360.0 335.0 0 25 25 0 [[161, 477]] 1.0 8uwn Homo sapiens CMGC_CLK1_HUMAN CMGC 3.1e-93 318.2 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6KHDB P49759 149 482 484.0 3NG:1000 Type1 Inactive DFGin 6.9078 14.0758 BLAminus -116.48, -175.0 67.35, 80.01 -102.96, 15.9 292.23, 100.48 -53.02, -40.84 in-in in 8.5827 Saltbr-in 2.6359 HRD-in -57.21, -57.72 79.07, -3.09 in-in-out SNCiio in-out ActLoopNT-in 2.9181 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_iiii APE10-dihe-na -136.88, 104.05 APE9-dihe-na 173.26, -145.7 APE8-dihe-in -145.78, 56.63 APE8-rot-in 325.36 APE67-dihe-out -165.57, -36.7 24.99, 58.5 APE12-dist-in 13.5825 APE11-dist-in 11.8902 APE10-dist-in 6.8247 APE9-dist-in 3.7474 None None None XRAY 2.7 0.204 0.274 B 484.0 332.0 2 25 25 0 [[161, 477]] 1.0 6khd Homo sapiens CMGC_CLK1_HUMAN CMGC 8.2e-93 317.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 5J1WC P49759 148 483 484.0 6FB:60505,6FB:60506 Type1,Allosteric Inactive DFGin 7.1425 14.2862 BLAminus -122.18, 173.27 71.94, 86.76 -106.83, 22.04 296.04, 87.14 -77.19, -12.48 in-in in 8.5036 Saltbr-in 2.5683 HRD-in -74.28, -51.47 84.87, -18.08 in-in-out SNCiio in-out ActLoopNT-in 2.8804 ActLoopCT-out nonTYR APEdihe_aaiio APEdist_oioo APE10-dihe-na -128.25, 150.31 APE9-dihe-na -78.45, -169.37 APE8-dihe-in -56.02, 117.75 APE8-rot-in 301.81 APE67-dihe-out -74.26, -11.87 -128.54, 128.96 APE12-dist-out 14.7541 APE11-dist-in 12.3342 APE10-dist-out 9.2098 APE9-dist-out 8.676 None None None XRAY 2.42 0.191 0.228 C 339.0 314.0 22 25 25 0 [[161, 477]] 1.0 5j1w Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6KHDA P49759 149 481 484.0 3NG:1000 Type1 Inactive DFGin 6.8618 14.4848 None -115.36, -74.37 -61.99, 112.36 -110.01, 19.25 292.55, 104.1 -59.59, -27.31 in-in in 8.7531 Saltbr-in 2.4552 HRD-in -79.61, -40.92 65.39, -11.49 in-in-out SNCiio in-out ActLoopNT-in 2.9802 ActLoopCT-out nonTYR APEdihe_aannn APEdist_ioon APE10-dihe-na -162.31, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -85.78, 10.46 999.0, -15.39 APE12-dist-in 11.8684 APE11-dist-out 7.0432 APE10-dist-out 11.6347 APE9-dist-none 999.0 None None None XRAY 2.7 0.204 0.274 A 484.0 322.0 11 25 23 2 [[161, 477]] 1.0 6khd Homo sapiens CMGC_CLK1_HUMAN CMGC 8.2e-93 317.4 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Q8PA P49759 148 482 484.0 HQB:60501 Type1 None DFGin 7.1106 14.5328 BLAminus -124.47, -177.12 56.99, 94.11 -115.67, 29.05 294.23, 87.9 -80.98, -10.13 in-in in 9.0127 Saltbr-in 3.4176 HRD-in -77.51, -42.79 69.43, -19.47 in-in-none SNCiin in-none ActLoopNT-in 3.1315 ActLoopCT-none nonTYR APEdihe_aanii APEdist_iiin APE10-dihe-na -135.51, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 147.79 APE8-rot-in 323.11 APE67-dihe-in -68.72, -18.82 -64.59, -40.03 APE12-dist-in 13.2041 APE11-dist-in 11.2012 APE10-dist-in 7.2881 APE9-dist-none 999.0 None None None XRAY 3.0 0.201 0.244 A 339.0 334.0 1 25 24 1 [[161, 477]] 1.0 6q8p Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 CLK1_HUMAN 6Q8PC P49759 148 483 484.0 HQB:60501 Type1 None DFGin 7.2607 13.9451 BLAminus -128.5, 178.53 59.41, 97.23 -121.71, 37.79 304.27, 105.41 -86.72, -22.18 in-in in 8.6759 Saltbr-in 3.006 HRD-in -68.24, -39.01 69.57, -23.21 in-in-none SNCiin in-none ActLoopNT-in 2.9528 ActLoopCT-none nonTYR APEdihe_aanii APEdist_iiin APE10-dihe-na -136.11, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 147.77 APE8-rot-in 314.52 APE67-dihe-in -61.24, -29.44 -57.39, -46.95 APE12-dist-in 13.763 APE11-dist-in 11.1263 APE10-dist-in 7.2951 APE9-dist-none 999.0 None None None XRAY 3.0 0.201 0.244 C 339.0 333.0 3 25 24 1 [[161, 477]] 1.0 6q8p Homo sapiens CMGC_CLK1_HUMAN CMGC 2.5e-93 318.5 1.0 301.0 301.0 324 325 326 328 330 191 206 210 285 287 286 288.0 361 349 344 343 342 341 340 339 338 242 Dual specificity protein kinase CLK1
CLK1 Q382U0_TRYB2 6Q2AD Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.4763 13.7883 BLAminus -119.9, -168.35 59.48, 71.83 -95.76, 15.53 257.41, 49.17 -69.28, -32.09 in-in in 8.7697 Saltbr-in 2.5559 HRD-in -77.83, -52.64 69.75, -5.64 in-in-in SNCiii in-in ActLoopNT-in 2.7715 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.39, 176.32 APE9-dihe-na 74.78, 146.92 APE8-dihe-in -63.78, 143.48 APE8-rot-in 298.53 APE67-dihe-in -58.91, -29.46 -58.64, -38.04 APE12-dist-in 10.3181 APE11-dist-in 11.6994 APE10-dist-in 7.6506 APE9-dist-in 3.0228 None None None XRAY 2.6 0.268 0.313 D 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AE Q382U0 127 465 465.0 5XH:504 Type1 Active DFGin 5.0906 13.0633 BLAminus -121.78, -169.06 62.52, 72.68 -96.4, 15.33 297.74, 13.76 -68.04, -32.18 in-in in 8.6394 Saltbr-in 2.8288 HRD-in -76.83, -49.95 71.59, -7.8 in-in-in SNCiii in-in ActLoopNT-in 3.0535 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.17, 173.06 APE9-dihe-na 75.56, 145.89 APE8-dihe-in -62.51, 142.36 APE8-rot-in 293.21 APE67-dihe-in -55.52, -31.54 -58.16, -36.13 APE12-dist-in 10.6347 APE11-dist-in 11.984 APE10-dist-in 7.4646 APE9-dist-in 3.0395 None None None XRAY 2.6 0.268 0.313 E 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AG Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.5763 13.1058 BLAminus -121.56, -172.32 65.3, 68.19 -94.07, 20.09 303.8, 13.18 -67.3, -31.23 in-in in 8.869 Saltbr-in 2.8754 HRD-in -76.86, -53.07 69.99, -8.5 in-in-in SNCiii in-in ActLoopNT-in 2.9764 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.65, 172.86 APE9-dihe-na 73.21, 147.32 APE8-dihe-in -64.07, 143.32 APE8-rot-in 299.51 APE67-dihe-in -56.19, -31.74 -58.99, -37.58 APE12-dist-in 10.3939 APE11-dist-in 11.506 APE10-dist-in 7.4224 APE9-dist-in 3.0612 None None None XRAY 2.6 0.268 0.313 G 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AM Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.5827 13.2601 BLAminus -122.03, -174.12 52.78, 74.93 -90.64, 21.24 302.72, 9.96 -64.44, -28.74 in-in in 8.9092 Saltbr-in 2.9604 HRD-in -77.14, -50.33 71.06, -8.08 in-in-in SNCiii in-in ActLoopNT-in 3.0683 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.19, 174.15 APE9-dihe-na 75.38, 147.9 APE8-dihe-in -64.58, 143.28 APE8-rot-in 295.72 APE67-dihe-in -56.44, -31.75 -57.92, -36.92 APE12-dist-in 10.2372 APE11-dist-in 11.4943 APE10-dist-in 7.1847 APE9-dist-in 3.026 None None None XRAY 2.6 0.268 0.313 M 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AN Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.4065 12.9916 BLAminus -124.15, -169.82 64.49, 69.46 -95.27, 17.53 299.57, 9.78 -67.21, -30.5 in-in in 8.6413 Saltbr-in 2.7936 HRD-in -76.8, -51.18 70.82, -7.75 in-in-in SNCiii in-in ActLoopNT-in 2.6848 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.16, 174.59 APE9-dihe-na 75.11, 146.41 APE8-dihe-in -63.66, 142.73 APE8-rot-in 302.91 APE67-dihe-in -57.03, -31.59 -59.0, -34.83 APE12-dist-in 10.5202 APE11-dist-in 11.754 APE10-dist-in 7.3865 APE9-dist-in 3.0662 None None None XRAY 2.6 0.268 0.313 N 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AP Q382U0 127 465 465.0 5XH:503 Type1 Active DFGin 4.9726 12.9981 BLAminus -119.74, -171.17 57.48, 79.35 -91.82, 17.72 294.71, 29.77 -67.55, -32.34 in-in in 8.9159 Saltbr-in 2.6957 HRD-in -77.24, -50.23 71.33, -8.82 in-in-in SNCiii in-in ActLoopNT-in 3.24 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.12, 173.39 APE9-dihe-na 74.96, 147.22 APE8-dihe-in -63.55, 142.75 APE8-rot-in 299.72 APE67-dihe-in -56.0, -31.74 -59.18, -37.4 APE12-dist-in 10.3587 APE11-dist-in 11.6146 APE10-dist-in 7.2541 APE9-dist-in 3.0283 None None None XRAY 2.6 0.268 0.313 P 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AA Q382U0 127 465 465.0 5XH:501 Type1 Inactive DFGin 5.5862 13.0975 BLAminus -119.0, -171.54 54.11, 74.62 -93.72, 19.87 300.89, 14.65 -66.08, -30.37 in-in in 8.8544 Saltbr-in 2.7914 HRD-in -77.03, -50.56 71.17, -8.06 in-in-out SNCiio in-out ActLoopNT-in 2.8817 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.64, 174.75 APE9-dihe-na 75.26, 147.37 APE8-dihe-in -65.92, 143.03 APE8-rot-out 74.14 APE67-dihe-in -55.49, -31.28 -58.8, -36.72 APE12-dist-in 10.3907 APE11-dist-in 11.4408 APE10-dist-in 7.2675 APE9-dist-in 3.0249 None None None XRAY 2.6 0.268 0.313 A 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AB Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.2005 13.2155 BLAminus -122.26, -169.1 61.88, 72.0 -96.55, 15.55 296.86, 11.1 -68.18, -31.87 in-in in 8.7753 Saltbr-in 3.0883 HRD-in -76.88, -50.01 71.06, -8.09 in-in-out SNCiio in-out ActLoopNT-in 3.0441 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -125.33, 173.18 APE9-dihe-na 75.34, 143.51 APE8-dihe-in -64.84, 144.66 APE8-rot-out 80.25 APE67-dihe-in -55.28, -33.02 -56.45, -35.89 APE12-dist-in 10.5022 APE11-dist-in 12.0176 APE10-dist-in 7.3118 APE9-dist-in 3.0697 None None None XRAY 2.6 0.268 0.313 B 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AC Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.2007 13.1583 BLAminus -125.39, -171.07 59.62, 74.29 -95.85, 16.24 304.87, 9.48 -67.73, -32.34 in-in in 8.7785 Saltbr-in 2.8403 HRD-in -76.59, -49.44 71.53, -6.33 in-in-out SNCiio in-out ActLoopNT-in 2.9471 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -124.5, 171.75 APE9-dihe-na 75.06, 143.62 APE8-dihe-in -62.63, 144.12 APE8-rot-out 37.89 APE67-dihe-in -55.38, -31.81 -57.03, -35.43 APE12-dist-in 10.4637 APE11-dist-in 11.9397 APE10-dist-in 7.2261 APE9-dist-in 2.991 None None None XRAY 2.6 0.268 0.313 C 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AF Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.0559 13.1599 BLAminus -122.68, -169.75 60.12, 71.93 -96.6, 14.84 301.3, 12.28 -68.75, -31.62 in-in in 8.7506 Saltbr-in 2.8964 HRD-in -77.43, -49.63 71.68, -7.89 in-in-out SNCiio in-out ActLoopNT-in 3.0767 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.12, 172.1 APE9-dihe-na 74.75, 142.67 APE8-dihe-in -63.4, 143.66 APE8-rot-out 37.46 APE67-dihe-in -55.26, -30.17 -56.65, -36.03 APE12-dist-in 10.4776 APE11-dist-in 11.9763 APE10-dist-in 7.4697 APE9-dist-in 3.0023 None None None XRAY 2.6 0.268 0.313 F 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AH Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.3012 12.9689 BLAminus -119.28, -168.95 55.7, 73.66 -95.39, 17.15 309.43, 7.35 -67.18, -32.11 in-in in 8.8165 Saltbr-in 2.7338 HRD-in -76.83, -51.18 71.75, -9.17 in-in-out SNCiio in-out ActLoopNT-in 2.8608 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -121.68, 176.4 APE9-dihe-na 76.23, 143.03 APE8-dihe-in -66.5, 142.66 APE8-rot-out 82.58 APE67-dihe-in -55.95, -26.39 -62.57, -37.5 APE12-dist-in 10.3309 APE11-dist-in 11.676 APE10-dist-in 6.9772 APE9-dist-in 3.0963 None None None XRAY 2.6 0.268 0.313 H 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AI Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.3383 13.1671 BLAminus -123.95, -169.7 61.06, 71.5 -97.59, 15.68 299.06, 12.02 -68.31, -31.48 in-in in 8.6034 Saltbr-in 3.0316 HRD-in -77.59, -50.58 70.98, -7.46 in-in-out SNCiio in-out ActLoopNT-in 3.0044 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.44, 171.47 APE9-dihe-na 75.28, 146.19 APE8-dihe-in -60.08, 142.44 APE8-rot-out 41.76 APE67-dihe-in -54.09, -31.47 -60.2, -34.75 APE12-dist-in 10.5488 APE11-dist-in 11.9841 APE10-dist-in 7.5429 APE9-dist-in 3.0032 None None None XRAY 2.6 0.268 0.313 I 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AJ Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.0967 13.0579 BLAminus -122.46, -166.99 62.87, 71.32 -96.61, 15.13 300.0, 9.52 -68.69, -31.3 in-in in 8.5935 Saltbr-in 2.779 HRD-in -74.22, -48.82 70.81, -6.67 in-in-out SNCiio in-out ActLoopNT-in 3.1899 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.88, 173.79 APE9-dihe-na 75.14, 144.51 APE8-dihe-in -64.43, 143.72 APE8-rot-out 36.49 APE67-dihe-in -55.07, -31.92 -56.83, -35.99 APE12-dist-in 10.5267 APE11-dist-in 11.9433 APE10-dist-in 7.3166 APE9-dist-in 3.0415 None None None XRAY 2.6 0.268 0.313 J 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AK Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.1026 13.0927 BLAminus -122.02, -166.89 62.21, 72.06 -96.74, 15.47 298.33, 8.85 -68.2, -31.83 in-in in 8.556 Saltbr-in 2.7606 HRD-in -77.41, -49.89 71.16, -8.73 in-in-out SNCiio in-out ActLoopNT-in 2.9784 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.79, 172.74 APE9-dihe-na 74.63, 143.9 APE8-dihe-in -64.46, 143.69 APE8-rot-out 167.18 APE67-dihe-in -54.47, -31.83 -57.73, -35.29 APE12-dist-in 10.5545 APE11-dist-in 11.9372 APE10-dist-in 7.3678 APE9-dist-in 3.0193 None None None XRAY 2.6 0.268 0.313 K 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AL Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.2474 13.3685 BLAminus -122.21, -170.28 61.23, 72.83 -97.02, 14.92 300.22, 10.25 -68.16, -32.26 in-in in 9.0028 Saltbr-in 2.9498 HRD-in -76.72, -49.17 71.44, -6.95 in-in-out SNCiio in-out ActLoopNT-in 3.0926 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.35, 171.77 APE9-dihe-na 74.63, 144.65 APE8-dihe-in -64.14, 144.88 APE8-rot-out 47.46 APE67-dihe-in -55.18, -32.42 -57.04, -35.3 APE12-dist-in 10.4807 APE11-dist-in 11.9377 APE10-dist-in 7.4477 APE9-dist-in 3.0317 None None None XRAY 2.6 0.268 0.313 L 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AO Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.5654 13.2155 BLAminus -121.28, -170.74 58.31, 73.08 -95.04, 18.11 298.82, 11.51 -65.91, -30.33 in-out in 8.7808 Saltbr-out 4.331 HRD-in -77.63, -51.71 71.45, -7.94 out-in-in SNCoii in-in ActLoopNT-in 3.0314 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.26, 174.14 APE9-dihe-na 75.9, 145.18 APE8-dihe-in -63.27, 142.33 APE8-rot-in 286.67 APE67-dihe-in -54.38, -29.28 -58.19, -37.84 APE12-dist-in 10.3531 APE11-dist-in 11.7284 APE10-dist-in 7.3364 APE9-dist-in 3.0458 None None None XRAY 2.6 0.268 0.313 O 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative

CMGC_CLK1 (Dual specificity protein kinase CLK1)

Total number of chains: 16
Active chains: 6
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 16 100.0% 6Q2AD

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CLK1 Q382U0_TRYB2 6Q2AD Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.4763 13.7883 BLAminus -119.9, -168.35 59.48, 71.83 -95.76, 15.53 257.41, 49.17 -69.28, -32.09 in-in in 8.7697 Saltbr-in 2.5559 HRD-in -77.83, -52.64 69.75, -5.64 in-in-in SNCiii in-in ActLoopNT-in 2.7715 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -117.39, 176.32 APE9-dihe-na 74.78, 146.92 APE8-dihe-in -63.78, 143.48 APE8-rot-in 298.53 APE67-dihe-in -58.91, -29.46 -58.64, -38.04 APE12-dist-in 10.3181 APE11-dist-in 11.6994 APE10-dist-in 7.6506 APE9-dist-in 3.0228 None None None XRAY 2.6 0.268 0.313 D 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AE Q382U0 127 465 465.0 5XH:504 Type1 Active DFGin 5.0906 13.0633 BLAminus -121.78, -169.06 62.52, 72.68 -96.4, 15.33 297.74, 13.76 -68.04, -32.18 in-in in 8.6394 Saltbr-in 2.8288 HRD-in -76.83, -49.95 71.59, -7.8 in-in-in SNCiii in-in ActLoopNT-in 3.0535 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.17, 173.06 APE9-dihe-na 75.56, 145.89 APE8-dihe-in -62.51, 142.36 APE8-rot-in 293.21 APE67-dihe-in -55.52, -31.54 -58.16, -36.13 APE12-dist-in 10.6347 APE11-dist-in 11.984 APE10-dist-in 7.4646 APE9-dist-in 3.0395 None None None XRAY 2.6 0.268 0.313 E 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AG Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.5763 13.1058 BLAminus -121.56, -172.32 65.3, 68.19 -94.07, 20.09 303.8, 13.18 -67.3, -31.23 in-in in 8.869 Saltbr-in 2.8754 HRD-in -76.86, -53.07 69.99, -8.5 in-in-in SNCiii in-in ActLoopNT-in 2.9764 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.65, 172.86 APE9-dihe-na 73.21, 147.32 APE8-dihe-in -64.07, 143.32 APE8-rot-in 299.51 APE67-dihe-in -56.19, -31.74 -58.99, -37.58 APE12-dist-in 10.3939 APE11-dist-in 11.506 APE10-dist-in 7.4224 APE9-dist-in 3.0612 None None None XRAY 2.6 0.268 0.313 G 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AM Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.5827 13.2601 BLAminus -122.03, -174.12 52.78, 74.93 -90.64, 21.24 302.72, 9.96 -64.44, -28.74 in-in in 8.9092 Saltbr-in 2.9604 HRD-in -77.14, -50.33 71.06, -8.08 in-in-in SNCiii in-in ActLoopNT-in 3.0683 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.19, 174.15 APE9-dihe-na 75.38, 147.9 APE8-dihe-in -64.58, 143.28 APE8-rot-in 295.72 APE67-dihe-in -56.44, -31.75 -57.92, -36.92 APE12-dist-in 10.2372 APE11-dist-in 11.4943 APE10-dist-in 7.1847 APE9-dist-in 3.026 None None None XRAY 2.6 0.268 0.313 M 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AN Q382U0 127 465 465.0 5XH:501 Type1 Active DFGin 5.4065 12.9916 BLAminus -124.15, -169.82 64.49, 69.46 -95.27, 17.53 299.57, 9.78 -67.21, -30.5 in-in in 8.6413 Saltbr-in 2.7936 HRD-in -76.8, -51.18 70.82, -7.75 in-in-in SNCiii in-in ActLoopNT-in 2.6848 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.16, 174.59 APE9-dihe-na 75.11, 146.41 APE8-dihe-in -63.66, 142.73 APE8-rot-in 302.91 APE67-dihe-in -57.03, -31.59 -59.0, -34.83 APE12-dist-in 10.5202 APE11-dist-in 11.754 APE10-dist-in 7.3865 APE9-dist-in 3.0662 None None None XRAY 2.6 0.268 0.313 N 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AP Q382U0 127 465 465.0 5XH:503 Type1 Active DFGin 4.9726 12.9981 BLAminus -119.74, -171.17 57.48, 79.35 -91.82, 17.72 294.71, 29.77 -67.55, -32.34 in-in in 8.9159 Saltbr-in 2.6957 HRD-in -77.24, -50.23 71.33, -8.82 in-in-in SNCiii in-in ActLoopNT-in 3.24 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.12, 173.39 APE9-dihe-na 74.96, 147.22 APE8-dihe-in -63.55, 142.75 APE8-rot-in 299.72 APE67-dihe-in -56.0, -31.74 -59.18, -37.4 APE12-dist-in 10.3587 APE11-dist-in 11.6146 APE10-dist-in 7.2541 APE9-dist-in 3.0283 None None None XRAY 2.6 0.268 0.313 P 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AA Q382U0 127 465 465.0 5XH:501 Type1 Inactive DFGin 5.5862 13.0975 BLAminus -119.0, -171.54 54.11, 74.62 -93.72, 19.87 300.89, 14.65 -66.08, -30.37 in-in in 8.8544 Saltbr-in 2.7914 HRD-in -77.03, -50.56 71.17, -8.06 in-in-out SNCiio in-out ActLoopNT-in 2.8817 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.64, 174.75 APE9-dihe-na 75.26, 147.37 APE8-dihe-in -65.92, 143.03 APE8-rot-out 74.14 APE67-dihe-in -55.49, -31.28 -58.8, -36.72 APE12-dist-in 10.3907 APE11-dist-in 11.4408 APE10-dist-in 7.2675 APE9-dist-in 3.0249 None None None XRAY 2.6 0.268 0.313 A 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AB Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.2005 13.2155 BLAminus -122.26, -169.1 61.88, 72.0 -96.55, 15.55 296.86, 11.1 -68.18, -31.87 in-in in 8.7753 Saltbr-in 3.0883 HRD-in -76.88, -50.01 71.06, -8.09 in-in-out SNCiio in-out ActLoopNT-in 3.0441 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -125.33, 173.18 APE9-dihe-na 75.34, 143.51 APE8-dihe-in -64.84, 144.66 APE8-rot-out 80.25 APE67-dihe-in -55.28, -33.02 -56.45, -35.89 APE12-dist-in 10.5022 APE11-dist-in 12.0176 APE10-dist-in 7.3118 APE9-dist-in 3.0697 None None None XRAY 2.6 0.268 0.313 B 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AC Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.2007 13.1583 BLAminus -125.39, -171.07 59.62, 74.29 -95.85, 16.24 304.87, 9.48 -67.73, -32.34 in-in in 8.7785 Saltbr-in 2.8403 HRD-in -76.59, -49.44 71.53, -6.33 in-in-out SNCiio in-out ActLoopNT-in 2.9471 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -124.5, 171.75 APE9-dihe-na 75.06, 143.62 APE8-dihe-in -62.63, 144.12 APE8-rot-out 37.89 APE67-dihe-in -55.38, -31.81 -57.03, -35.43 APE12-dist-in 10.4637 APE11-dist-in 11.9397 APE10-dist-in 7.2261 APE9-dist-in 2.991 None None None XRAY 2.6 0.268 0.313 C 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AF Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.0559 13.1599 BLAminus -122.68, -169.75 60.12, 71.93 -96.6, 14.84 301.3, 12.28 -68.75, -31.62 in-in in 8.7506 Saltbr-in 2.8964 HRD-in -77.43, -49.63 71.68, -7.89 in-in-out SNCiio in-out ActLoopNT-in 3.0767 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.12, 172.1 APE9-dihe-na 74.75, 142.67 APE8-dihe-in -63.4, 143.66 APE8-rot-out 37.46 APE67-dihe-in -55.26, -30.17 -56.65, -36.03 APE12-dist-in 10.4776 APE11-dist-in 11.9763 APE10-dist-in 7.4697 APE9-dist-in 3.0023 None None None XRAY 2.6 0.268 0.313 F 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AH Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.3012 12.9689 BLAminus -119.28, -168.95 55.7, 73.66 -95.39, 17.15 309.43, 7.35 -67.18, -32.11 in-in in 8.8165 Saltbr-in 2.7338 HRD-in -76.83, -51.18 71.75, -9.17 in-in-out SNCiio in-out ActLoopNT-in 2.8608 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -121.68, 176.4 APE9-dihe-na 76.23, 143.03 APE8-dihe-in -66.5, 142.66 APE8-rot-out 82.58 APE67-dihe-in -55.95, -26.39 -62.57, -37.5 APE12-dist-in 10.3309 APE11-dist-in 11.676 APE10-dist-in 6.9772 APE9-dist-in 3.0963 None None None XRAY 2.6 0.268 0.313 H 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AI Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.3383 13.1671 BLAminus -123.95, -169.7 61.06, 71.5 -97.59, 15.68 299.06, 12.02 -68.31, -31.48 in-in in 8.6034 Saltbr-in 3.0316 HRD-in -77.59, -50.58 70.98, -7.46 in-in-out SNCiio in-out ActLoopNT-in 3.0044 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.44, 171.47 APE9-dihe-na 75.28, 146.19 APE8-dihe-in -60.08, 142.44 APE8-rot-out 41.76 APE67-dihe-in -54.09, -31.47 -60.2, -34.75 APE12-dist-in 10.5488 APE11-dist-in 11.9841 APE10-dist-in 7.5429 APE9-dist-in 3.0032 None None None XRAY 2.6 0.268 0.313 I 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AJ Q382U0 127 465 465.0 5XH:504 Type1 Inactive DFGin 5.0967 13.0579 BLAminus -122.46, -166.99 62.87, 71.32 -96.61, 15.13 300.0, 9.52 -68.69, -31.3 in-in in 8.5935 Saltbr-in 2.779 HRD-in -74.22, -48.82 70.81, -6.67 in-in-out SNCiio in-out ActLoopNT-in 3.1899 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.88, 173.79 APE9-dihe-na 75.14, 144.51 APE8-dihe-in -64.43, 143.72 APE8-rot-out 36.49 APE67-dihe-in -55.07, -31.92 -56.83, -35.99 APE12-dist-in 10.5267 APE11-dist-in 11.9433 APE10-dist-in 7.3166 APE9-dist-in 3.0415 None None None XRAY 2.6 0.268 0.313 J 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AK Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.1026 13.0927 BLAminus -122.02, -166.89 62.21, 72.06 -96.74, 15.47 298.33, 8.85 -68.2, -31.83 in-in in 8.556 Saltbr-in 2.7606 HRD-in -77.41, -49.89 71.16, -8.73 in-in-out SNCiio in-out ActLoopNT-in 2.9784 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -123.79, 172.74 APE9-dihe-na 74.63, 143.9 APE8-dihe-in -64.46, 143.69 APE8-rot-out 167.18 APE67-dihe-in -54.47, -31.83 -57.73, -35.29 APE12-dist-in 10.5545 APE11-dist-in 11.9372 APE10-dist-in 7.3678 APE9-dist-in 3.0193 None None None XRAY 2.6 0.268 0.313 K 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AL Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.2474 13.3685 BLAminus -122.21, -170.28 61.23, 72.83 -97.02, 14.92 300.22, 10.25 -68.16, -32.26 in-in in 9.0028 Saltbr-in 2.9498 HRD-in -76.72, -49.17 71.44, -6.95 in-in-out SNCiio in-out ActLoopNT-in 3.0926 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -122.35, 171.77 APE9-dihe-na 74.63, 144.65 APE8-dihe-in -64.14, 144.88 APE8-rot-out 47.46 APE67-dihe-in -55.18, -32.42 -57.04, -35.3 APE12-dist-in 10.4807 APE11-dist-in 11.9377 APE10-dist-in 7.4477 APE9-dist-in 3.0317 None None None XRAY 2.6 0.268 0.313 L 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative
CLK1 Q382U0_TRYB2 6Q2AO Q382U0 127 465 465.0 5XH:503 Type1 Inactive DFGin 5.5654 13.2155 BLAminus -121.28, -170.74 58.31, 73.08 -95.04, 18.11 298.82, 11.51 -65.91, -30.33 in-out in 8.7808 Saltbr-out 4.331 HRD-in -77.63, -51.71 71.45, -7.94 out-in-in SNCoii in-in ActLoopNT-in 3.0314 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -120.26, 174.14 APE9-dihe-na 75.9, 145.18 APE8-dihe-in -63.27, 142.33 APE8-rot-in 286.67 APE67-dihe-in -54.38, -29.28 -58.19, -37.84 APE12-dist-in 10.3531 APE11-dist-in 11.7284 APE10-dist-in 7.3364 APE9-dist-in 3.0458 None None None XRAY 2.6 0.268 0.313 O 354.0 339.0 0 25 25 0 [[129, 439]] 1.0 6q2a Trypanosoma brucei brucei CMGC_CLK1_TRYB2 CMGC 2e-64 223.6 1.0 301.0 301.0 288 289 290 292 294 158 173 177 252 254 253 255.0 325 313 308 307 306 305 304 303 302 210 Protein kinase, putative