Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 1 | 8BURB |
DFGin | ABAminus | 1 | 8BURE |
DFGin | None | 1 | 8BURH |
Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|
CMGC | CDK12 | CDK12_HUMAN | Cyclin-dependent kinase 12 | 8BURE | 3.64 | Inactive | DFGin | ABAminus | in-in | in-in | RQU | Type1 |
CMGC | CDK12 | CDK12_HUMAN | Cyclin-dependent kinase 12 | 8BURB | 3.64 | Active | DFGin | BLAminus | in-in | in-in | RQU | Type1 |
CMGC | CDK12 | CDK12_HUMAN | Cyclin-dependent kinase 12 | 8BURH | 3.64 | Inactive | DFGin | None | in-in | in-in | RQU | Type1 |
Spatial | Dihedral | Chains | Representative |
---|---|---|---|
DFGin | BLAminus | 1 | 8BURB |
DFGin | ABAminus | 1 | 8BURE |
DFGin | None | 1 | 8BURH |
Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Homo sapiens | CMGC | CDK12 | CDK12_HUMAN | Cyclin-dependent kinase 12 | 8BURE | 3.64 | Inactive | DFGin | ABAminus | in-in | in-in | RQU | Type1 |
Homo sapiens | CMGC | CDK12 | CDK12_HUMAN | Cyclin-dependent kinase 12 | 8BURB | 3.64 | Active | DFGin | BLAminus | in-in | in-in | RQU | Type1 |
Homo sapiens | CMGC | CDK12 | CDK12_HUMAN | Cyclin-dependent kinase 12 | 8BURH | 3.64 | Inactive | DFGin | None | in-in | in-in | RQU | Type1 |
Spatial | Dihedral | Chains | Representative |
---|
Organism | Group | Gene | UniprotID | Protein | PDB | Resolu | Activity Label | Spatial Label | Dihedral Label | Chelix-SaltBridge | ActLoopNT-ActLoopCT | Ligand | Type |
---|