| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TKL | BRAF | BRAF_HUMAN | 6P7GA | 2.65 | Inactive | DFGout‑BBAminus | in-in | none-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | E7M | Type2 | 449 - 720 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 6P7GC | 2.65 | Inactive | DFGout‑BBAminus | in-in | none-out | nonTYR | APEdihe_aaoii | APEdist_nnno | E7M | Type2 | 449 - 721 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 6P7GD | 2.65 | Inactive | DFGout‑BBAminus | in-in | none-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | E7M | Type2 | 449 - 721 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf |
| TKL | BRAF | BRAF_HUMAN | 6P7GB | 2.65 | Inactive | DFGout‑BBAminus | in-in | out-out | nonTYR | APEdihe_aaoii | APEdist_iooo | E7M, NHE | Type2, Allosteric | 449 - 721 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf |
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TKL | BRAF | BRAF_HUMAN | 6P7GA | 2.65 | Inactive | DFGout‑BBAminus | in-in | none-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | E7M | Type2 | 449 - 720 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf | Homo sapiens |
| TKL | BRAF | BRAF_HUMAN | 6P7GC | 2.65 | Inactive | DFGout‑BBAminus | in-in | none-out | nonTYR | APEdihe_aaoii | APEdist_nnno | E7M | Type2 | 449 - 721 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf | Homo sapiens |
| TKL | BRAF | BRAF_HUMAN | 6P7GD | 2.65 | Inactive | DFGout‑BBAminus | in-in | none-out | nonTYR | APEdihe_aaoii | APEdist_nnoo | E7M | Type2 | 449 - 721 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf | Homo sapiens |
| TKL | BRAF | BRAF_HUMAN | 6P7GB | 2.65 | Inactive | DFGout‑BBAminus | in-in | out-out | nonTYR | APEdihe_aaoii | APEdist_iooo | E7M, NHE | Type2, Allosteric | 449 - 721 | 0 | None | I543A,I544S,I551K,Q562R,L588N,V600E,K630S,F667E,Y673S,A688R,L706S,Q709R,S713E,L716E,S720E,P722S,K723G | Serine/threonine-protein kinase B-raf | Homo sapiens |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Family | Gene | UniprotID | PDB | Resolution | Activity | Spatial-Dihedral | Chelix-SaltBridge | ActLoopNT-ActLoopCT | APEtype | APEdihe | APEdist | Ligand | Ligand Type | Residues in structure | Unresolved residues in A-loop | Phosphorylation | Mutation | Protein | Organism |
|---|