| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4V04B | P11362 | 458 | 765 | 822.0 | 0LI:1771 | Type2 | Inactive | DFGout | 13.974 | 9.8725 | BBAminus | -127.4, -173.98 | -164.99, 120.92 | -104.35, 44.71 | 306.97, 107.67 | 29.41, -12.23 | in-in | in | 7.692 | Saltbr-in | 3.0147 | HRD-in | -72.1, -51.88 | 81.11, -15.75 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.55, 155.16 | APE9-dihe-in | -98.03, 109.95 | APE8-dihe-out | -52.12, -21.56 | APE8-rot-na | 329.22 | APE67-dihe-in | -70.06, -7.36 | -58.08, -24.0 | APE12-dist-na | 19.5141 | APE11-dist-na | 20.9701 | APE10-dist-na | 19.2978 | APE9-dist-out | 11.5913 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | B | 309.0 | 289.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V04A | P11362 | 463 | 765 | 822.0 | 0LI:1772 | Type2 | Inactive | DFGout | 14.0506 | 10.3941 | None | -127.25, -179.24 | -145.47, 116.11 | -167.94, 35.9 | 26.55, 54.39 | 23.93, -5.2 | in-in | in | 7.8637 | Saltbr-in | 3.2056 | HRD-in | -65.2, -58.04 | 83.28, -16.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.41, 155.12 | APE9-dihe-in | -98.09, 110.26 | APE8-dihe-out | -52.77, -21.99 | APE8-rot-na | 329.65 | APE67-dihe-in | -70.41, -8.08 | -56.89, -24.83 | APE12-dist-na | 19.6385 | APE11-dist-na | 21.0205 | APE10-dist-na | 19.3218 | APE9-dist-out | 11.7003 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | A | 309.0 | 293.0 | 10 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4V04B | P11362 | 458 | 765 | 822.0 | 0LI:1771 | Type2 | Inactive | DFGout | 13.974 | 9.8725 | BBAminus | -127.4, -173.98 | -164.99, 120.92 | -104.35, 44.71 | 306.97, 107.67 | 29.41, -12.23 | in-in | in | 7.692 | Saltbr-in | 3.0147 | HRD-in | -72.1, -51.88 | 81.11, -15.75 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.55, 155.16 | APE9-dihe-in | -98.03, 109.95 | APE8-dihe-out | -52.12, -21.56 | APE8-rot-na | 329.22 | APE67-dihe-in | -70.06, -7.36 | -58.08, -24.0 | APE12-dist-na | 19.5141 | APE11-dist-na | 20.9701 | APE10-dist-na | 19.2978 | APE9-dist-out | 11.5913 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | B | 309.0 | 289.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V04A | P11362 | 463 | 765 | 822.0 | 0LI:1772 | Type2 | Inactive | DFGout | 14.0506 | 10.3941 | None | -127.25, -179.24 | -145.47, 116.11 | -167.94, 35.9 | 26.55, 54.39 | 23.93, -5.2 | in-in | in | 7.8637 | Saltbr-in | 3.2056 | HRD-in | -65.2, -58.04 | 83.28, -16.96 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -102.41, 155.12 | APE9-dihe-in | -98.09, 110.26 | APE8-dihe-out | -52.77, -21.99 | APE8-rot-na | 329.65 | APE67-dihe-in | -70.41, -8.08 | -56.89, -24.83 | APE12-dist-na | 19.6385 | APE11-dist-na | 21.0205 | APE10-dist-na | 19.3218 | APE9-dist-out | 11.7003 | C488A,C584S | None | None | XRAY | 2.12 | 0.188 | 0.228 | A | 309.0 | 293.0 | 10 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4v04 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|