Ligand: 824

Total number of chains: 7
Active chains: 0
Total number of genes: 3
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 5 71.4% 2X7FB
DFGin ABAminus 1 14.3% 4C58A
DFGin None 1 14.3% 2X7FE

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
OTHER GAK GAK_HUMAN 4C58A O14976 27 333 1311.0 824:1336 Type1.5_Back Inactive DFGin 5.7769 13.7982 ABAminus -132.89, -19.04 -95.75, 85.27 -100.86, 19.52 307.21, 107.98 -74.39, -16.9 in-in in 8.74 Saltbr-in 2.9557 HRD-in -74.87, -50.0 69.14, -1.84 in-in-none SNCiin in-none ActLoopNT-in 2.8465 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.16 0.182 0.242 A 340.0 267.0 40 40 13 27 [[40, 313]] 1.0 4c58 OTHER_GAK_HUMAN CAMK 5.3e-44 156.7 3.0 252.0 250.0 190 191 192 194 196 69 85 89 170 172 171 173.0 245 230 225 224 223 222 221 220 219 124 Cyclin-G-associated kinase
OTHER WEE1 WEE1_HUMAN 1X8BA P30291 291 569 646.0 824:901 Type1 Inactive DFGin 5.1383 12.0784 BLAminus -126.44, -167.26 52.99, 80.97 -90.02, 18.86 302.17, 14.25 -66.11, -12.47 in-in in 8.7986 Saltbr-in 2.7294 HRD-in -82.83, -50.09 72.75, 8.93 in-in-out SNCiio in-out ActLoopNT-in 2.9206 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -58.07, 132.65 APE9-dihe-na -83.92, -172.43 APE8-dihe-in -49.42, 128.03 APE8-rot-na 195.04 APE67-dihe-in -69.68, -24.37 -54.98, -30.74 APE12-dist-in 8.1542 APE11-dist-out 5.6134 APE10-dist-out 9.1378 APE9-dist-in 3.2091 None None None XRAY 1.81 0.219 0.237 A 289.0 259.0 20 24 24 0 [[299, 569]] 1.0 1x8b OTHER_WEE1_HUMAN OTHER 1.4e-37 135.5 1.0 258.0 258.0 462 463 464 466 468 328 346 350 423 425 424 426.0 499 486 481 480 479 478 477 476 475 377 Wee1-like protein kinase
STE TNIK TNIK_HUMAN 2X7FA Q9UKE5 15 313 1360.0 824:500 Type1 Inactive DFGin 6.7876 14.6427 BLAminus -125.93, 176.2 60.97, 100.67 -114.36, 23.27 288.61, 85.46 -68.11, -48.66 in-none in 9.2041 Saltbr-none 999.0 HRD-in -65.92, -41.18 69.14, -4.02 none-out-out SNCnoo out-out ActLoopNT-out 6.167 ActLoopCT-out nonTYR APEdihe_aaini APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -150.84 APE8-dihe-in -101.28, 96.29 APE8-rot-none 999.0 APE67-dihe-in -52.7, -32.64 -83.9, 2.97 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 10.9208 None None None XRAY 2.8 0.21 0.229 A 326.0 276.0 23 28 15 13 [[25, 289]] 1.0 2x7f STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FB Q9UKE5 13 313 1360.0 824:500 Type1 Inactive DFGin 6.759 14.6163 BLAminus -125.8, 175.96 61.22, 100.42 -113.19, 24.28 288.37, 86.39 -68.54, -48.18 in-none in 9.1073 Saltbr-none 999.0 HRD-in -67.06, -42.58 70.38, -4.99 none-out-out SNCnoo out-out ActLoopNT-out 6.1902 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 154.09 APE8-dihe-in -121.12, 111.62 APE8-rot-out 48.12 APE67-dihe-in -53.26, -31.37 -96.48, 3.58 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.5142 None None None XRAY 2.8 0.21 0.229 B 326.0 288.0 13 28 16 12 [[25, 289]] 1.0 2x7f STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FC Q9UKE5 14 313 1360.0 824:500 Type1 Inactive DFGin 6.7637 14.765 BLAminus -124.84, 175.84 60.69, 100.51 -112.75, 22.89 287.95, 85.81 -67.51, -48.09 in-none in 9.1407 Saltbr-none 999.0 HRD-in -67.07, -40.49 68.23, -3.68 none-out-none SNCnon out-none ActLoopNT-out 6.1705 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 118.77 APE8-rot-none 999.0 APE67-dihe-in -54.15, -31.45 -96.1, 4.16 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.8 0.21 0.229 C 326.0 285.0 15 28 14 14 [[25, 289]] 1.0 2x7f STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FD Q9UKE5 17 306 1360.0 824:500 Type1 None DFGin 6.6469 15.0461 BLAminus -124.52, 178.85 56.71, 102.04 -114.11, 22.87 287.2, 83.98 -65.42, -48.91 in-none in 9.4441 Saltbr-none 999.0 HRD-in -66.67, -40.26 66.21, -2.06 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 119.49 APE8-rot-none 999.0 APE67-dihe-in -52.92, -32.7 -93.58, 2.88 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.8 0.21 0.229 D 326.0 236.0 51 28 13 15 [[25, 289]] 1.0 2x7f STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FE Q9UKE5 14 309 1360.0 824:500 Type1 Inactive DFGin 6.6596 14.7942 None -124.38, 176.52 58.71, 103.53 -115.64, 999.0 286.98, 84.26 999.0, 999.0 in-none in 9.525 Saltbr-none 999.0 HRD-in -65.29, -41.79 67.65, -3.62 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 128.45 APE8-rot-none 999.0 APE67-dihe-in -51.92, -33.29 -95.18, 3.25 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.8 0.21 0.229 E 326.0 251.0 45 28 10 18 [[25, 289]] 1.0 2x7f STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase

Ligand: 824

Total number of chains: 7
Active chains: 0
Total number of genes: 3
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 5 71.4% 2X7FB
DFGin ABAminus 1 14.3% 4C58A
DFGin None 1 14.3% 2X7FE

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
OTHER GAK GAK_HUMAN 4C58A O14976 27 333 1311.0 824:1336 Type1.5_Back Inactive DFGin 5.7769 13.7982 ABAminus -132.89, -19.04 -95.75, 85.27 -100.86, 19.52 307.21, 107.98 -74.39, -16.9 in-in in 8.74 Saltbr-in 2.9557 HRD-in -74.87, -50.0 69.14, -1.84 in-in-none SNCiin in-none ActLoopNT-in 2.8465 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.16 0.182 0.242 A 340.0 267.0 40 40 13 27 [[40, 313]] 1.0 4c58 Homo sapiens OTHER_GAK_HUMAN CAMK 5.3e-44 156.7 3.0 252.0 250.0 190 191 192 194 196 69 85 89 170 172 171 173.0 245 230 225 224 223 222 221 220 219 124 Cyclin-G-associated kinase
OTHER WEE1 WEE1_HUMAN 1X8BA P30291 291 569 646.0 824:901 Type1 Inactive DFGin 5.1383 12.0784 BLAminus -126.44, -167.26 52.99, 80.97 -90.02, 18.86 302.17, 14.25 -66.11, -12.47 in-in in 8.7986 Saltbr-in 2.7294 HRD-in -82.83, -50.09 72.75, 8.93 in-in-out SNCiio in-out ActLoopNT-in 2.9206 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -58.07, 132.65 APE9-dihe-na -83.92, -172.43 APE8-dihe-in -49.42, 128.03 APE8-rot-na 195.04 APE67-dihe-in -69.68, -24.37 -54.98, -30.74 APE12-dist-in 8.1542 APE11-dist-out 5.6134 APE10-dist-out 9.1378 APE9-dist-in 3.2091 None None None XRAY 1.81 0.219 0.237 A 289.0 259.0 20 24 24 0 [[299, 569]] 1.0 1x8b Homo sapiens OTHER_WEE1_HUMAN OTHER 1.4e-37 135.5 1.0 258.0 258.0 462 463 464 466 468 328 346 350 423 425 424 426.0 499 486 481 480 479 478 477 476 475 377 Wee1-like protein kinase
STE TNIK TNIK_HUMAN 2X7FA Q9UKE5 15 313 1360.0 824:500 Type1 Inactive DFGin 6.7876 14.6427 BLAminus -125.93, 176.2 60.97, 100.67 -114.36, 23.27 288.61, 85.46 -68.11, -48.66 in-none in 9.2041 Saltbr-none 999.0 HRD-in -65.92, -41.18 69.14, -4.02 none-out-out SNCnoo out-out ActLoopNT-out 6.167 ActLoopCT-out nonTYR APEdihe_aaini APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -150.84 APE8-dihe-in -101.28, 96.29 APE8-rot-none 999.0 APE67-dihe-in -52.7, -32.64 -83.9, 2.97 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 10.9208 None None None XRAY 2.8 0.21 0.229 A 326.0 276.0 23 28 15 13 [[25, 289]] 1.0 2x7f Homo sapiens STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FB Q9UKE5 13 313 1360.0 824:500 Type1 Inactive DFGin 6.759 14.6163 BLAminus -125.8, 175.96 61.22, 100.42 -113.19, 24.28 288.37, 86.39 -68.54, -48.18 in-none in 9.1073 Saltbr-none 999.0 HRD-in -67.06, -42.58 70.38, -4.99 none-out-out SNCnoo out-out ActLoopNT-out 6.1902 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 154.09 APE8-dihe-in -121.12, 111.62 APE8-rot-out 48.12 APE67-dihe-in -53.26, -31.37 -96.48, 3.58 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 11.5142 None None None XRAY 2.8 0.21 0.229 B 326.0 288.0 13 28 16 12 [[25, 289]] 1.0 2x7f Homo sapiens STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FC Q9UKE5 14 313 1360.0 824:500 Type1 Inactive DFGin 6.7637 14.765 BLAminus -124.84, 175.84 60.69, 100.51 -112.75, 22.89 287.95, 85.81 -67.51, -48.09 in-none in 9.1407 Saltbr-none 999.0 HRD-in -67.07, -40.49 68.23, -3.68 none-out-none SNCnon out-none ActLoopNT-out 6.1705 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 118.77 APE8-rot-none 999.0 APE67-dihe-in -54.15, -31.45 -96.1, 4.16 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.8 0.21 0.229 C 326.0 285.0 15 28 14 14 [[25, 289]] 1.0 2x7f Homo sapiens STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FD Q9UKE5 17 306 1360.0 824:500 Type1 None DFGin 6.6469 15.0461 BLAminus -124.52, 178.85 56.71, 102.04 -114.11, 22.87 287.2, 83.98 -65.42, -48.91 in-none in 9.4441 Saltbr-none 999.0 HRD-in -66.67, -40.26 66.21, -2.06 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 119.49 APE8-rot-none 999.0 APE67-dihe-in -52.92, -32.7 -93.58, 2.88 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.8 0.21 0.229 D 326.0 236.0 51 28 13 15 [[25, 289]] 1.0 2x7f Homo sapiens STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase
STE TNIK TNIK_HUMAN 2X7FE Q9UKE5 14 309 1360.0 824:500 Type1 Inactive DFGin 6.6596 14.7942 None -124.38, 176.52 58.71, 103.53 -115.64, 999.0 286.98, 84.26 999.0, 999.0 in-none in 9.525 Saltbr-none 999.0 HRD-in -65.29, -41.79 67.65, -3.62 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 128.45 APE8-rot-none 999.0 APE67-dihe-in -51.92, -33.29 -95.18, 3.25 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.8 0.21 0.229 E 326.0 251.0 45 28 10 18 [[25, 289]] 1.0 2x7f Homo sapiens STE_TNIK_HUMAN STE 3.7e-105 356.8 1.0 257.0 257.0 170 171 172 174 176 54 69 73 150 152 151 153.0 215 198 193 192 191 190 189 188 187 106 TRAF2 and NCK-interacting protein kinase

Ligand: 824

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name