Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_HUMAN | 5N23A | P17612 | 9 | 351 | 351.0 | 35R:60401 | Type1 | Active | DFGin | 5.421 | 13.864 | BLAminus | -109.83, 165.02 | 72.7, 94.27 | -97.78, 24.01 | 286.85, 71.32 | -58.73, -25.18 | in-in | in | 9.5 | Saltbr-in | 2.927 | HRD-in | -90.99, -49.74 | 71.93, 9.7 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.878 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.89, 153.96 | APE9-dihe-na | 137.51, -163.29 | APE8-dihe-in | -116.51, 133.79 | APE8-rot-in | 303.7 | APE67-dihe-in | -56.98, -24.74 | -46.64, -52.33 | APE12-dist-in | 8.056 | APE11-dist-in | 11.585 | APE10-dist-in | 5.945 | APE9-dist-in | 3.654 | K48R,L96Q,M121L,V124A,Q182K,T184A | SEP11,SEP140,TPO198,SEP339 | SEP11,SEP140,TPO198,SEP339 | XRAY | 2.088 | 0.192 | 0.239 | A | 352 | 337 | 0 | 0 | 0 | 0 | [[44, 298]] | 1.0 | 5n23 | AGC_PRKACA_HUMAN | AGC | 5.3e-93 | 316.9 | 1 | 260 | 260 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| CAMK | AURKA | AURKA_HUMAN | 6CPGA | O14965 | 127 | 387 | 403.0 | 35R:501 | Type1 | Inactive | DFGinter | 6.711 | 9.485 | None | -140.02, 96.03 | -108.44, 103.16 | -141.15, -67.9 | 302.74, 112.44 | 175.19, -125.6 | out-out | out | 12.429 | Saltbr-out | 10.941 | HRD-out | 55.39, 71.59 | -104.21, 123.45 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnoo | APE10-dihe-na | 999.0, -80.02 | APE9-dihe-na | 97.77, -146.55 | APE8-dihe-out | -62.97, -12.48 | APE8-rot-none | 999.0 | APE67-dihe-in | -58.41, -29.26 | -54.85, -41.27 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 17.041 | APE9-dist-out | 13.657 | None | None | None | XRAY | 2.8 | 0.285 | 0.335 | A | 285 | 249 | 12 | 0 | 0 | 12 | [[133, 383]] | 1.0 | 6cpg | CAMK_AURKA_HUMAN | CAMK | 7.7e-80 | 273.8 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | AURKA | AURKA_HUMAN | 6CPGD | O14965 | 127 | 388 | 403.0 | 35R:501 | Type1 | Inactive | DFGinter | 6.404 | 9.772 | None | -125.89, 77.36 | -98.94, 84.58 | -127.68, 52.17 | 302.92, 103.94 | 97.64, -149.27 | out-out | out | 11.62 | Saltbr-out | 12.775 | HRD-out | 61.84, 98.64 | -116.43, 122.15 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nooo | APE10-dihe-na | -115.97, 178.85 | APE9-dihe-na | -115.52, -132.49 | APE8-dihe-out | -76.59, 1.28 | APE8-rot-out | 68.27 | APE67-dihe-in | -65.85, -12.72 | -75.15, -27.74 | APE12-dist-none | 999.0 | APE11-dist-out | 19.388 | APE10-dist-out | 16.46 | APE9-dist-out | 14.83 | None | None | None | XRAY | 2.8 | 0.285 | 0.335 | D | 285 | 252 | 10 | 0 | 0 | 10 | [[133, 383]] | 1.0 | 6cpg | CAMK_AURKA_HUMAN | CAMK | 7.7e-80 | 273.8 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| STE | STK24 | STK24_HUMAN | 4QMMA | Q9Y6E0 | 18 | 309 | 443.0 | 35R:60401 | Type1 | Active | DFGin | 6.456 | 14.869 | BLAminus | -136.1, 172.57 | 56.6, 85.7 | -97.18, 29.33 | 287.89, 78.12 | -60.54, -24.23 | in-in | in | 9.035 | Saltbr-in | 2.726 | HRD-in | -73.78, -49.7 | 70.31, 2.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.74, 158.6 | APE9-dihe-na | 131.64, -167.88 | APE8-dihe-in | -113.08, 118.53 | APE8-rot-in | 307.24 | APE67-dihe-in | -61.4, -26.15 | -38.81, -50.43 | APE12-dist-in | 8.458 | APE11-dist-in | 10.893 | APE10-dist-in | 5.077 | APE9-dist-in | 3.296 | None | TPO190 | TPO190 | XRAY | 1.852 | 0.141 | 0.198 | A | 310 | 289 | 0 | 0 | 0 | 0 | [[36, 286]] | 1.0 | 4qmm | STE_STK24_HUMAN | STE | 3.9e-100 | 340.4 | 1 | 257 | 257 | 173 | 174 | 175 | 177 | 179 | 65 | 82 | 86 | 153 | 155 | 154 | 156 | 213 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 112 | Serine/threonine-protein kinase 24 |
| TYR | JAK2-1 | JAK2_HUMAN | 6D2IA | O60674 | 536 | 808 | 1132.0 | 35R:901 | Type1 | Pseudo | DFGin | 6.552 | 13.651 | None | -85.6, -168.64 | -71.02, 159.25 | -67.8, -19.61 | 341.93, 32.5 | 72.61, -145.53 | in-na | in | 9.639 | Saltbr-na | 999.0 | HRD-in | -88.15, -70.56 | 100.36, -8.76 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.7 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -69.19, -30.63 | APE9-dihe-out | -73.76, -13.56 | APE8-dihe-out | -89.52, 2.58 | APE8-rot-na | 300.29 | APE67-dihe-out | -99.98, 28.53 | -66.76, 135.82 | APE12-dist-na | 10.52 | APE11-dist-na | 11.514 | APE10-dist-na | 16.315 | APE9-dist-out | 13.019 | W659A,W777A,F794H | None | None | XRAY | 3.192 | 0.272 | 0.29 | A | 273 | 273 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 6d2i | TYR_JAK2-1_HUMAN | TYR | 2.9e-64 | 222.8 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 6D2IB | O60674 | 537 | 808 | 1132.0 | 35R:901 | Type1 | Pseudo | DFGin | 6.745 | 13.508 | None | -83.97, -172.62 | -69.78, 158.02 | -65.46, -20.62 | 341.26, 32.34 | 71.79, -145.54 | in-na | in | 9.436 | Saltbr-na | 999.0 | HRD-in | -84.58, -69.97 | 97.0, -6.55 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.449 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -68.97, -30.79 | APE9-dihe-out | -72.59, -17.09 | APE8-dihe-out | -89.77, 2.61 | APE8-rot-na | 301.92 | APE67-dihe-out | -99.31, 27.86 | -67.19, 135.78 | APE12-dist-na | 10.586 | APE11-dist-na | 11.89 | APE10-dist-na | 16.65 | APE9-dist-out | 12.896 | W659A,W777A,F794H | None | None | XRAY | 3.192 | 0.272 | 0.29 | B | 273 | 272 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 6d2i | TYR_JAK2-1_HUMAN | TYR | 2.9e-64 | 222.8 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 5WIMA | O60674 | 536 | 809 | 1132.0 | 35R:901 | Type1 | Pseudo | DFGin | 7.752 | 13.585 | None | -93.28, 176.5 | -38.24, 151.14 | -78.63, -21.68 | 29.2, 149.11 | 81.15, -169.97 | out-na | out | 10.568 | Saltbr-na | 999.0 | HRD-in | -83.09, -66.39 | 96.8, 0.86 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.85 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -105.18, -10.47 | APE9-dihe-out | -83.98, -20.52 | APE8-dihe-out | -80.31, 9.26 | APE8-rot-na | 299.8 | APE67-dihe-out | -97.29, 28.98 | -67.31, 132.23 | APE12-dist-na | 9.833 | APE11-dist-na | 11.542 | APE10-dist-na | 15.898 | APE9-dist-out | 12.889 | W659A,W777A,F794H | None | None | XRAY | 2.55 | 0.211 | 0.258 | A | 277 | 274 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 5wim | TYR_JAK2-1_HUMAN | TYR | 1.6e-64 | 223.6 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 5UT0A | O60674 | 537 | 808 | 1132.0 | 35R:903 | Type1 | Pseudo | DFGin | 7.594 | 13.572 | None | -93.9, 174.39 | -69.93, 155.11 | -74.3, -13.06 | 28.06, 143.5 | 77.21, -173.63 | in-na | in | 9.939 | Saltbr-na | 999.0 | HRD-in | -83.57, -61.23 | 99.02, -12.98 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.966 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -63.47, -40.74 | APE9-dihe-out | -59.34, -26.03 | APE8-dihe-out | -86.35, 4.34 | APE8-rot-na | 287.5 | APE67-dihe-out | -101.06, 28.12 | -64.23, 136.97 | APE12-dist-na | 10.005 | APE11-dist-na | 11.478 | APE10-dist-na | 16.135 | APE9-dist-out | 12.932 | W659A,W777A,F794H | None | None | XRAY | 2.102 | 0.171 | 0.226 | A | 289 | 272 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 5ut0 | TYR_JAK2-1_HUMAN | TYR | 1.9e-64 | 223.4 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_HUMAN | 5N23A | P17612 | 9 | 351 | 351.0 | 35R:60401 | Type1 | Active | DFGin | 5.421 | 13.864 | BLAminus | -109.83, 165.02 | 72.7, 94.27 | -97.78, 24.01 | 286.85, 71.32 | -58.73, -25.18 | in-in | in | 9.5 | Saltbr-in | 2.927 | HRD-in | -90.99, -49.74 | 71.93, 9.7 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.878 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.89, 153.96 | APE9-dihe-na | 137.51, -163.29 | APE8-dihe-in | -116.51, 133.79 | APE8-rot-in | 303.7 | APE67-dihe-in | -56.98, -24.74 | -46.64, -52.33 | APE12-dist-in | 8.056 | APE11-dist-in | 11.585 | APE10-dist-in | 5.945 | APE9-dist-in | 3.654 | K48R,L96Q,M121L,V124A,Q182K,T184A | SEP11,SEP140,TPO198,SEP339 | SEP11,SEP140,TPO198,SEP339 | XRAY | 2.088 | 0.192 | 0.239 | A | 352 | 337 | 0 | 0 | 0 | 0 | [[44, 298]] | 1.0 | 5n23 | Homo sapiens | AGC_PRKACA_HUMAN | AGC | 5.3e-93 | 316.9 | 1 | 260 | 260 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| CAMK | AURKA | AURKA_HUMAN | 6CPGA | O14965 | 127 | 387 | 403.0 | 35R:501 | Type1 | Inactive | DFGinter | 6.711 | 9.485 | None | -140.02, 96.03 | -108.44, 103.16 | -141.15, -67.9 | 302.74, 112.44 | 175.19, -125.6 | out-out | out | 12.429 | Saltbr-out | 10.941 | HRD-out | 55.39, 71.59 | -104.21, 123.45 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaoni | APEdist_nnoo | APE10-dihe-na | 999.0, -80.02 | APE9-dihe-na | 97.77, -146.55 | APE8-dihe-out | -62.97, -12.48 | APE8-rot-none | 999.0 | APE67-dihe-in | -58.41, -29.26 | -54.85, -41.27 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-out | 17.041 | APE9-dist-out | 13.657 | None | None | None | XRAY | 2.8 | 0.285 | 0.335 | A | 285 | 249 | 12 | 0 | 0 | 12 | [[133, 383]] | 1.0 | 6cpg | Homo sapiens | CAMK_AURKA_HUMAN | CAMK | 7.7e-80 | 273.8 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| CAMK | AURKA | AURKA_HUMAN | 6CPGD | O14965 | 127 | 388 | 403.0 | 35R:501 | Type1 | Inactive | DFGinter | 6.404 | 9.772 | None | -125.89, 77.36 | -98.94, 84.58 | -127.68, 52.17 | 302.92, 103.94 | 97.64, -149.27 | out-out | out | 11.62 | Saltbr-out | 12.775 | HRD-out | 61.84, 98.64 | -116.43, 122.15 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aaooi | APEdist_nooo | APE10-dihe-na | -115.97, 178.85 | APE9-dihe-na | -115.52, -132.49 | APE8-dihe-out | -76.59, 1.28 | APE8-rot-out | 68.27 | APE67-dihe-in | -65.85, -12.72 | -75.15, -27.74 | APE12-dist-none | 999.0 | APE11-dist-out | 19.388 | APE10-dist-out | 16.46 | APE9-dist-out | 14.83 | None | None | None | XRAY | 2.8 | 0.285 | 0.335 | D | 285 | 252 | 10 | 0 | 0 | 10 | [[133, 383]] | 1.0 | 6cpg | Homo sapiens | CAMK_AURKA_HUMAN | CAMK | 7.7e-80 | 273.8 | 1 | 256 | 256 | 273 | 274 | 275 | 277 | 279 | 162 | 181 | 185 | 253 | 255 | 254 | 256 | 311 | 299 | 294 | 293 | 292 | 291 | 290 | 289 | 288 | 211 | Aurora kinase A |
| STE | STK24 | STK24_HUMAN | 4QMMA | Q9Y6E0 | 18 | 309 | 443.0 | 35R:60401 | Type1 | Active | DFGin | 6.456 | 14.869 | BLAminus | -136.1, 172.57 | 56.6, 85.7 | -97.18, 29.33 | 287.89, 78.12 | -60.54, -24.23 | in-in | in | 9.035 | Saltbr-in | 2.726 | HRD-in | -73.78, -49.7 | 70.31, 2.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.74, 158.6 | APE9-dihe-na | 131.64, -167.88 | APE8-dihe-in | -113.08, 118.53 | APE8-rot-in | 307.24 | APE67-dihe-in | -61.4, -26.15 | -38.81, -50.43 | APE12-dist-in | 8.458 | APE11-dist-in | 10.893 | APE10-dist-in | 5.077 | APE9-dist-in | 3.296 | None | TPO190 | TPO190 | XRAY | 1.852 | 0.141 | 0.198 | A | 310 | 289 | 0 | 0 | 0 | 0 | [[36, 286]] | 1.0 | 4qmm | Homo sapiens | STE_STK24_HUMAN | STE | 3.9e-100 | 340.4 | 1 | 257 | 257 | 173 | 174 | 175 | 177 | 179 | 65 | 82 | 86 | 153 | 155 | 154 | 156 | 213 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 112 | Serine/threonine-protein kinase 24 |
| TYR | JAK2-1 | JAK2_HUMAN | 6D2IA | O60674 | 536 | 808 | 1132.0 | 35R:901 | Type1 | Pseudo | DFGin | 6.552 | 13.651 | None | -85.6, -168.64 | -71.02, 159.25 | -67.8, -19.61 | 341.93, 32.5 | 72.61, -145.53 | in-na | in | 9.639 | Saltbr-na | 999.0 | HRD-in | -88.15, -70.56 | 100.36, -8.76 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.7 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -69.19, -30.63 | APE9-dihe-out | -73.76, -13.56 | APE8-dihe-out | -89.52, 2.58 | APE8-rot-na | 300.29 | APE67-dihe-out | -99.98, 28.53 | -66.76, 135.82 | APE12-dist-na | 10.52 | APE11-dist-na | 11.514 | APE10-dist-na | 16.315 | APE9-dist-out | 13.019 | W659A,W777A,F794H | None | None | XRAY | 3.192 | 0.272 | 0.29 | A | 273 | 273 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 6d2i | Homo sapiens | TYR_JAK2-1_HUMAN | TYR | 2.9e-64 | 222.8 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 6D2IB | O60674 | 537 | 808 | 1132.0 | 35R:901 | Type1 | Pseudo | DFGin | 6.745 | 13.508 | None | -83.97, -172.62 | -69.78, 158.02 | -65.46, -20.62 | 341.26, 32.34 | 71.79, -145.54 | in-na | in | 9.436 | Saltbr-na | 999.0 | HRD-in | -84.58, -69.97 | 97.0, -6.55 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.449 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -68.97, -30.79 | APE9-dihe-out | -72.59, -17.09 | APE8-dihe-out | -89.77, 2.61 | APE8-rot-na | 301.92 | APE67-dihe-out | -99.31, 27.86 | -67.19, 135.78 | APE12-dist-na | 10.586 | APE11-dist-na | 11.89 | APE10-dist-na | 16.65 | APE9-dist-out | 12.896 | W659A,W777A,F794H | None | None | XRAY | 3.192 | 0.272 | 0.29 | B | 273 | 272 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 6d2i | Homo sapiens | TYR_JAK2-1_HUMAN | TYR | 2.9e-64 | 222.8 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 5WIMA | O60674 | 536 | 809 | 1132.0 | 35R:901 | Type1 | Pseudo | DFGin | 7.752 | 13.585 | None | -93.28, 176.5 | -38.24, 151.14 | -78.63, -21.68 | 29.2, 149.11 | 81.15, -169.97 | out-na | out | 10.568 | Saltbr-na | 999.0 | HRD-in | -83.09, -66.39 | 96.8, 0.86 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.85 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -105.18, -10.47 | APE9-dihe-out | -83.98, -20.52 | APE8-dihe-out | -80.31, 9.26 | APE8-rot-na | 299.8 | APE67-dihe-out | -97.29, 28.98 | -67.31, 132.23 | APE12-dist-na | 9.833 | APE11-dist-na | 11.542 | APE10-dist-na | 15.898 | APE9-dist-out | 12.889 | W659A,W777A,F794H | None | None | XRAY | 2.55 | 0.211 | 0.258 | A | 277 | 274 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 5wim | Homo sapiens | TYR_JAK2-1_HUMAN | TYR | 1.6e-64 | 223.6 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| TYR | JAK2-1 | JAK2_HUMAN | 5UT0A | O60674 | 537 | 808 | 1132.0 | 35R:903 | Type1 | Pseudo | DFGin | 7.594 | 13.572 | None | -93.9, 174.39 | -69.93, 155.11 | -74.3, -13.06 | 28.06, 143.5 | 77.21, -173.63 | in-na | in | 9.939 | Saltbr-na | 999.0 | HRD-in | -83.57, -61.23 | 99.02, -12.98 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.966 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -63.47, -40.74 | APE9-dihe-out | -59.34, -26.03 | APE8-dihe-out | -86.35, 4.34 | APE8-rot-na | 287.5 | APE67-dihe-out | -101.06, 28.12 | -64.23, 136.97 | APE12-dist-na | 10.005 | APE11-dist-na | 11.478 | APE10-dist-na | 16.135 | APE9-dist-out | 12.932 | W659A,W777A,F794H | None | None | XRAY | 2.102 | 0.171 | 0.226 | A | 289 | 272 | 0 | 0 | 0 | 0 | [[545, 807], [849, 1125]] | 2.0 | 5ut0 | Homo sapiens | TYR_JAK2-1_HUMAN | TYR | 1.9e-64 | 223.4 | 2 | 260 | 259 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
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Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
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