TKL_TNNI3K (Serine/threonine-protein kinase TNNI3K)

Total number of chains: 22
Active chains: 1
Uniprot: TNI3K_HUMAN
Kinase Domain Residues: 463 - 721
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 14 63.6% AF-Q59H18-K3A
DFGout BBAminus 8 36.4% 7MGJA

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
TNNI3K AF-Q59H18-K3A Q59H18 455 729 835.0 No_ligand No_ligand Active DFGin 6.6962 13.8804 BLAminus -139.07, 177.24 54.32, 90.68 -94.1, 12.35 288.15, 91.72 -60.08, -34.83 in-in in 8.1877 Saltbr-in 2.7503 HRD-in -78.12, -43.64 70.08, -16.01 in-in-in SNCiii in-in ActLoopNT-in 2.8812 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -78.58, 153.21 APE9-dihe-na 68.3, -167.13 APE8-dihe-in -85.53, 115.08 APE8-rot-na 194.71 APE67-dihe-in -69.96, -26.34 -49.24, -34.71 APE12-dist-in 10.0753 APE11-dist-in 11.1028 APE10-dist-in 5.413 APE9-dist-in 3.8317 None None None AF2 -1.0 1.0 1.0 A 275.0 275.0 0 29 29 0 [[463, 721]] 1.0 AF-Q59H18-K3 TKL_TNNI3K_HUMAN TKL 9.6e-78 267.3 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K AF-Q59H18-K1A Q59H18 455 729 835.0 No_ligand No_ligand Inactive DFGin 6.9673 14.2132 BLAminus -137.24, 177.07 58.03, 78.77 -90.1, 16.58 289.46, 86.3 -61.99, -35.76 in-in in 8.4036 Saltbr-in 2.841 HRD-in -76.03, -43.57 65.98, -16.11 in-in-out SNCiio in-out ActLoopNT-in 2.9244 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -71.99, 139.8 APE9-dihe-na -71.23, -158.5 APE8-dihe-in -64.75, 109.31 APE8-rot-na 193.38 APE67-dihe-in -73.05, -29.32 -52.87, -33.11 APE12-dist-in 12.5994 APE11-dist-out 7.6494 APE10-dist-out 10.2409 APE9-dist-in 4.0266 None None None AF2 -1.0 1.0 1.0 A 275.0 275.0 0 29 29 0 [[463, 721]] 1.0 AF-Q59H18-K1 TKL_TNNI3K_HUMAN TKL 9.6e-78 267.3 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFFC Q59H18 452 725 835.0 4CV:801 Type1 Inactive DFGin 6.9042 14.2898 BLAminus -137.59, 177.85 57.57, 83.21 -93.61, 21.97 283.02, 76.58 -61.87, -21.22 in-in in 8.7546 Saltbr-in 2.6479 HRD-in -73.89, -42.66 73.16, 1.89 in-in-out SNCiio in-out ActLoopNT-in 2.8756 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nooo APE10-dihe-na -68.61, 136.84 APE9-dihe-na -80.53, -15.93 APE8-dihe-out -53.66, -37.06 APE8-rot-na 53.41 APE67-dihe-in -65.33, -27.85 -42.42, -33.67 APE12-dist-none 999.0 APE11-dist-out 28.6607 APE10-dist-out 28.0999 APE9-dist-out 29.2755 None None None XRAY 3.07 0.211 0.251 C 311.0 258.0 16 29 21 8 [[463, 721]] 1.0 4yff TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFFD Q59H18 452 726 835.0 4CV:801 Type1 Inactive DFGin 6.9196 14.2606 BLAminus -138.19, 176.18 59.05, 82.1 -92.69, 22.93 284.26, 76.55 -62.07, -21.96 in-in in 8.6995 Saltbr-in 2.6737 HRD-in -72.99, -42.85 72.57, 4.93 in-in-out SNCiio in-out ActLoopNT-in 2.8824 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -20.75 APE8-dihe-out -51.62, -40.33 APE8-rot-na 51.44 APE67-dihe-in -65.2, -25.35 -42.12, -32.96 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 29.4216 None None None XRAY 3.07 0.211 0.251 D 311.0 257.0 18 29 19 10 [[463, 721]] 1.0 4yff TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 6B5JA Q59H18 445 726 835.0 CV4:801 Type1 Inactive DFGin 6.8129 13.8645 BLAminus -126.38, 171.36 62.48, 91.94 -100.05, 34.64 289.93, 73.51 -70.41, -26.85 in-in in 8.5373 Saltbr-in 3.0165 HRD-in -69.61, -48.01 72.35, -18.59 in-in-out SNCiio in-out ActLoopNT-in 2.9554 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -156.21 APE8-dihe-in -96.29, 132.1 APE8-rot-na 189.83 APE67-dihe-in -67.3, -25.63 -78.42, -19.47 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.2764 None None None XRAY 2.97 0.204 0.258 A 311.0 263.0 19 29 19 10 [[463, 721]] 1.0 6b5j TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 6B5JC Q59H18 451 726 835.0 CV4:801 Type1 Inactive DFGin 6.8466 14.3196 BLAminus -130.93, 173.95 56.3, 85.73 -92.89, 28.95 283.96, 71.94 -60.28, -23.99 in-in in 8.6566 Saltbr-in 2.8227 HRD-in -75.55, -36.97 68.66, 0.24 in-in-out SNCiio in-out ActLoopNT-in 2.9103 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nooo APE10-dihe-na -69.92, 151.63 APE9-dihe-na -59.24, -28.73 APE8-dihe-out -64.35, -20.05 APE8-rot-na 73.57 APE67-dihe-in -70.47, -24.58 -56.79, -26.65 APE12-dist-none 999.0 APE11-dist-out 28.0382 APE10-dist-out 28.6445 APE9-dist-out 29.6749 None None None XRAY 2.97 0.204 0.258 C 311.0 260.0 16 29 22 7 [[463, 721]] 1.0 6b5j TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 6B5JD Q59H18 452 726 835.0 CV4:801 Type1 Inactive DFGin 6.8408 14.2648 BLAminus -132.12, 173.84 58.27, 85.6 -93.97, 30.79 285.02, 72.35 -64.62, -22.56 in-in in 8.6488 Saltbr-in 2.796 HRD-in -73.89, -40.9 71.61, 1.26 in-in-out SNCiio in-out ActLoopNT-in 2.966 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -50.25 APE8-dihe-out -60.76, -16.48 APE8-rot-na 57.99 APE67-dihe-in -64.06, -34.42 -74.64, -18.94 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 30.2472 None None None XRAY 2.97 0.204 0.258 D 311.0 257.0 18 29 19 10 [[463, 721]] 1.0 6b5j TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFIA Q59H18 441 726 835.0 4CW:801 Type1 Inactive DFGin 7.1477 14.0773 BLAminus -134.84, 175.79 58.1, 92.29 -99.47, 27.9 285.94, 73.67 -68.71, -26.95 in-in in 8.2146 Saltbr-in 2.9555 HRD-in -84.08, -48.18 75.05, 0.66 in-in-out SNCiio in-out ActLoopNT-in 3.0202 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -162.01 APE8-dihe-in -79.92, 138.7 APE8-rot-na 192.61 APE67-dihe-in -56.79, -31.79 -77.63, -30.03 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 26.9145 None None None XRAY 2.7 0.217 0.261 A 330.0 268.0 18 29 18 11 [[463, 721]] 1.0 4yfi TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFIB Q59H18 451 729 835.0 4CW:801 Type1 Inactive DFGin 7.0749 14.5653 BLAminus -121.54, 177.03 56.79, 87.27 -99.8, 31.09 284.15, 68.4 -68.89, -25.59 in-in in 8.5901 Saltbr-in 2.8471 HRD-in -63.87, -47.95 70.39, 1.06 in-in-out SNCiio in-out ActLoopNT-in 2.9046 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -68.32 APE8-dihe-out -66.38, -17.23 APE8-rot-na 67.92 APE67-dihe-in -62.92, -25.6 -64.1, -31.48 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 30.8384 None None None XRAY 2.7 0.217 0.261 B 330.0 262.0 17 29 19 10 [[463, 721]] 1.0 4yfi TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFIC Q59H18 441 726 835.0 4CW:801 Type1 Inactive DFGin 7.029 14.0468 BLAminus -119.12, 170.12 62.73, 94.49 -102.41, 18.34 284.63, 68.96 -60.63, -21.51 in-in in 8.3499 Saltbr-in 2.7933 HRD-in -81.8, -51.75 73.29, 8.93 in-in-out SNCiio in-out ActLoopNT-in 2.9284 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -166.83 APE8-dihe-in -85.58, 133.55 APE8-rot-na 183.6 APE67-dihe-in -63.19, -28.24 -74.71, -24.38 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.3503 None None None XRAY 2.7 0.217 0.261 C 330.0 269.0 17 29 19 10 [[463, 721]] 1.0 4yfi TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFID Q59H18 451 729 835.0 4CW:801 Type1 Inactive DFGin 6.9827 14.4988 BLAminus -132.3, -176.25 57.34, 76.41 -86.69, 32.24 287.65, 73.81 -68.32, -29.28 in-in in 8.4514 Saltbr-in 3.0842 HRD-in -70.86, -49.92 74.99, 12.01 in-in-out SNCiio in-out ActLoopNT-in 2.8072 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -77.73 APE8-dihe-out -78.4, -7.06 APE8-rot-na 86.27 APE67-dihe-in -68.67, -26.29 -70.22, -28.38 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 31.2769 None None None XRAY 2.7 0.217 0.261 D 330.0 261.0 18 29 19 10 [[463, 721]] 1.0 4yfi TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGKA Q59H18 444 726 835.0 ZGD:801 Type2 Inactive DFGout 15.0236 10.3486 BBAminus -136.11, -167.43 -161.58, 104.18 -68.96, -17.69 283.06, 90.36 80.74, 69.7 in-in in 7.8889 Saltbr-in 3.1395 HRD-in -62.84, -47.58 72.31, -16.61 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -171.11 APE8-dihe-in -86.32, 127.94 APE8-rot-na 191.21 APE67-dihe-in -60.28, -29.5 -75.53, -21.14 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.1525 None None None XRAY 3.1 0.198 0.239 A 311.0 262.0 21 29 13 16 [[463, 721]] 1.0 7mgk TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGKB Q59H18 444 727 835.0 ZGD:801 Type2 Inactive DFGout 14.6369 9.2616 BBAminus -136.1, -166.0 -163.89, 103.37 -69.12, -14.28 283.44, 87.76 84.95, 110.73 in-in in 8.2266 Saltbr-in 3.0963 HRD-in -63.33, -46.59 72.46, -18.58 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -171.17 APE8-dihe-in -84.68, 125.14 APE8-rot-na 191.2 APE67-dihe-in -61.15, -29.7 -78.96, -24.17 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 26.9334 None None None XRAY 3.1 0.198 0.239 B 311.0 261.0 23 29 13 16 [[463, 721]] 1.0 7mgk TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGKC Q59H18 445 726 835.0 ZGD:801 Type2 Inactive DFGout 15.2687 10.0615 BBAminus -135.81, -167.53 -162.54, 105.05 -66.31, -16.16 281.98, 90.65 80.81, 29.43 in-in in 8.0128 Saltbr-in 3.0708 HRD-in -63.3, -46.14 71.73, -18.15 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 128.83 APE8-rot-na 191.34 APE67-dihe-in -60.85, -29.89 -76.21, -23.31 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 3.1 0.198 0.239 C 311.0 260.0 22 29 13 16 [[463, 721]] 1.0 7mgk TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGKD Q59H18 444 727 835.0 ZGD:801 Type2 Inactive DFGout 14.8417 9.6948 BBAminus -121.51, -163.82 -171.47, 92.6 -57.07, -16.06 289.23, 82.11 84.14, 81.99 in-in in 8.1085 Saltbr-in 2.8017 HRD-in -61.83, -47.27 63.18, 0.84 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoo APE10-dihe-na 999.0, -105.6 APE9-dihe-na 75.02, 174.66 APE8-dihe-in -97.98, 119.78 APE8-rot-na 187.47 APE67-dihe-in -53.23, -38.91 -67.14, -31.62 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 30.6699 APE9-dist-out 26.8313 None None None XRAY 3.1 0.198 0.239 D 311.0 263.0 21 29 15 14 [[463, 721]] 1.0 7mgk TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGJA Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.8582 9.5819 BBAminus -134.42, -179.18 -141.04, 112.0 -72.43, -1.46 272.54, 97.9 75.05, 22.83 in-in in 7.7537 Saltbr-in 2.6724 HRD-in -64.15, -45.05 73.18, -17.04 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -171.97 APE8-dihe-in -104.46, 123.1 APE8-rot-na 189.02 APE67-dihe-in -59.47, -32.71 -67.71, -22.35 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.3356 None None None XRAY 2.95 0.197 0.228 A 330.0 262.0 20 29 13 16 [[463, 721]] 1.0 7mgj TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGJB Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.5602 9.2473 BBAminus -135.63, -179.46 -142.92, 111.63 -76.44, -17.08 273.4, 86.62 76.35, 79.73 in-in in 7.8588 Saltbr-in 2.9045 HRD-in -64.65, -46.97 73.32, -12.56 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoo APE10-dihe-na 999.0, -80.9 APE9-dihe-na 83.07, -177.24 APE8-dihe-in -105.62, 120.49 APE8-rot-na 192.96 APE67-dihe-in -61.56, -34.4 -69.66, -24.07 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 30.6715 APE9-dist-out 26.8043 None None None XRAY 2.95 0.197 0.228 B 330.0 260.0 22 29 14 15 [[463, 721]] 1.0 7mgj TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGJC Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.6969 9.6665 BBAminus -137.79, -177.03 -141.64, 110.69 -73.01, -3.0 273.24, 93.94 74.23, 29.77 in-in in 7.8989 Saltbr-in 2.91 HRD-in -66.15, -44.57 73.37, -16.84 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 119.35 APE8-rot-na 190.99 APE67-dihe-in -61.3, -34.66 -68.53, -21.6 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.95 0.197 0.228 C 330.0 261.0 21 29 13 16 [[463, 721]] 1.0 7mgj TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 7MGJD Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.5321 9.688 BBAminus -144.03, 179.53 -144.45, 109.82 -73.53, -9.7 276.8, 74.13 75.18, 64.15 in-in in 7.7498 Saltbr-in 2.6424 HRD-in -65.07, -45.42 74.54, -12.51 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoo APE10-dihe-na 999.0, -81.24 APE9-dihe-na 82.5, -174.24 APE8-dihe-in -103.92, 121.0 APE8-rot-na 193.26 APE67-dihe-in -60.88, -34.79 -69.71, -24.61 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 31.3479 APE9-dist-out 27.2314 None None None XRAY 2.95 0.197 0.228 D 330.0 261.0 21 29 15 14 [[463, 721]] 1.0 7mgj TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFFA Q59H18 445 726 835.0 4CV:801 Type1 None DFGin 6.8965 13.8872 BLAminus -127.46, 175.49 57.0, 94.25 -101.84, 21.43 285.11, 76.86 -67.58, -12.19 in-in in 8.3049 Saltbr-in 2.5732 HRD-in -72.29, -48.61 68.2, 11.99 in-in-none SNCiin in-none ActLoopNT-in 2.7517 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 133.81 APE8-rot-na 181.89 APE67-dihe-in -64.26, -21.67 -83.98, -17.01 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 3.07 0.211 0.251 A 311.0 264.0 18 29 18 11 [[463, 721]] 1.0 4yff TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 4YFFB Q59H18 445 726 835.0 4CV:801 Type1 None DFGin 6.8476 13.8816 BLAminus -128.82, 174.1 57.67, 94.34 -100.02, 21.13 285.48, 77.01 -67.5, -10.8 in-in in 8.3585 Saltbr-in 2.6026 HRD-in -72.09, -48.38 68.6, 12.37 in-in-none SNCiin in-none ActLoopNT-in 2.7622 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 137.74 APE8-rot-none 999.0 APE67-dihe-in -59.76, -26.5 -86.26, -18.43 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 3.07 0.211 0.251 B 311.0 264.0 18 29 17 12 [[463, 721]] 1.0 4yff TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K 6B5JB Q59H18 445 726 835.0 CV4:801 Type1 None DFGin 6.7764 13.8842 BLAminus -127.39, 170.23 63.58, 89.42 -96.67, 32.19 290.95, 72.96 -66.8, -26.81 in-in in 8.6163 Saltbr-in 3.0489 HRD-in -67.53, -48.98 70.48, -12.85 in-in-none SNCiin in-none ActLoopNT-in 2.9262 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 129.15 APE8-rot-na 200.19 APE67-dihe-in -61.72, -25.21 -84.18, -18.08 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.97 0.204 0.258 B 311.0 264.0 18 29 17 12 [[463, 721]] 1.0 6b5j TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K

TKL_TNNI3K (Serine/threonine-protein kinase TNNI3K)

Total number of chains: 22
Active chains: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 14 63.6% AF-Q59H18-K3A
DFGout BBAminus 8 36.4% 7MGJA

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
TNNI3K TNI3K_HUMAN AF-Q59H18-K3A Q59H18 455 729 835.0 No_ligand No_ligand Active DFGin 6.6962 13.8804 BLAminus -139.07, 177.24 54.32, 90.68 -94.1, 12.35 288.15, 91.72 -60.08, -34.83 in-in in 8.1877 Saltbr-in 2.7503 HRD-in -78.12, -43.64 70.08, -16.01 in-in-in SNCiii in-in ActLoopNT-in 2.8812 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -78.58, 153.21 APE9-dihe-na 68.3, -167.13 APE8-dihe-in -85.53, 115.08 APE8-rot-na 194.71 APE67-dihe-in -69.96, -26.34 -49.24, -34.71 APE12-dist-in 10.0753 APE11-dist-in 11.1028 APE10-dist-in 5.413 APE9-dist-in 3.8317 None None None AF2 -1.0 1.0 1.0 A 275.0 275.0 0 29 29 0 [[463, 721]] 1.0 AF-Q59H18-K3 Homo sapiens TKL_TNNI3K_HUMAN TKL 9.6e-78 267.3 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN AF-Q59H18-K1A Q59H18 455 729 835.0 No_ligand No_ligand Inactive DFGin 6.9673 14.2132 BLAminus -137.24, 177.07 58.03, 78.77 -90.1, 16.58 289.46, 86.3 -61.99, -35.76 in-in in 8.4036 Saltbr-in 2.841 HRD-in -76.03, -43.57 65.98, -16.11 in-in-out SNCiio in-out ActLoopNT-in 2.9244 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -71.99, 139.8 APE9-dihe-na -71.23, -158.5 APE8-dihe-in -64.75, 109.31 APE8-rot-na 193.38 APE67-dihe-in -73.05, -29.32 -52.87, -33.11 APE12-dist-in 12.5994 APE11-dist-out 7.6494 APE10-dist-out 10.2409 APE9-dist-in 4.0266 None None None AF2 -1.0 1.0 1.0 A 275.0 275.0 0 29 29 0 [[463, 721]] 1.0 AF-Q59H18-K1 Homo sapiens TKL_TNNI3K_HUMAN TKL 9.6e-78 267.3 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFFC Q59H18 452 725 835.0 4CV:801 Type1 Inactive DFGin 6.9042 14.2898 BLAminus -137.59, 177.85 57.57, 83.21 -93.61, 21.97 283.02, 76.58 -61.87, -21.22 in-in in 8.7546 Saltbr-in 2.6479 HRD-in -73.89, -42.66 73.16, 1.89 in-in-out SNCiio in-out ActLoopNT-in 2.8756 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nooo APE10-dihe-na -68.61, 136.84 APE9-dihe-na -80.53, -15.93 APE8-dihe-out -53.66, -37.06 APE8-rot-na 53.41 APE67-dihe-in -65.33, -27.85 -42.42, -33.67 APE12-dist-none 999.0 APE11-dist-out 28.6607 APE10-dist-out 28.0999 APE9-dist-out 29.2755 None None None XRAY 3.07 0.211 0.251 C 311.0 258.0 16 29 21 8 [[463, 721]] 1.0 4yff Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFFD Q59H18 452 726 835.0 4CV:801 Type1 Inactive DFGin 6.9196 14.2606 BLAminus -138.19, 176.18 59.05, 82.1 -92.69, 22.93 284.26, 76.55 -62.07, -21.96 in-in in 8.6995 Saltbr-in 2.6737 HRD-in -72.99, -42.85 72.57, 4.93 in-in-out SNCiio in-out ActLoopNT-in 2.8824 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -20.75 APE8-dihe-out -51.62, -40.33 APE8-rot-na 51.44 APE67-dihe-in -65.2, -25.35 -42.12, -32.96 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 29.4216 None None None XRAY 3.07 0.211 0.251 D 311.0 257.0 18 29 19 10 [[463, 721]] 1.0 4yff Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 6B5JA Q59H18 445 726 835.0 CV4:801 Type1 Inactive DFGin 6.8129 13.8645 BLAminus -126.38, 171.36 62.48, 91.94 -100.05, 34.64 289.93, 73.51 -70.41, -26.85 in-in in 8.5373 Saltbr-in 3.0165 HRD-in -69.61, -48.01 72.35, -18.59 in-in-out SNCiio in-out ActLoopNT-in 2.9554 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -156.21 APE8-dihe-in -96.29, 132.1 APE8-rot-na 189.83 APE67-dihe-in -67.3, -25.63 -78.42, -19.47 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.2764 None None None XRAY 2.97 0.204 0.258 A 311.0 263.0 19 29 19 10 [[463, 721]] 1.0 6b5j Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 6B5JC Q59H18 451 726 835.0 CV4:801 Type1 Inactive DFGin 6.8466 14.3196 BLAminus -130.93, 173.95 56.3, 85.73 -92.89, 28.95 283.96, 71.94 -60.28, -23.99 in-in in 8.6566 Saltbr-in 2.8227 HRD-in -75.55, -36.97 68.66, 0.24 in-in-out SNCiio in-out ActLoopNT-in 2.9103 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nooo APE10-dihe-na -69.92, 151.63 APE9-dihe-na -59.24, -28.73 APE8-dihe-out -64.35, -20.05 APE8-rot-na 73.57 APE67-dihe-in -70.47, -24.58 -56.79, -26.65 APE12-dist-none 999.0 APE11-dist-out 28.0382 APE10-dist-out 28.6445 APE9-dist-out 29.6749 None None None XRAY 2.97 0.204 0.258 C 311.0 260.0 16 29 22 7 [[463, 721]] 1.0 6b5j Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 6B5JD Q59H18 452 726 835.0 CV4:801 Type1 Inactive DFGin 6.8408 14.2648 BLAminus -132.12, 173.84 58.27, 85.6 -93.97, 30.79 285.02, 72.35 -64.62, -22.56 in-in in 8.6488 Saltbr-in 2.796 HRD-in -73.89, -40.9 71.61, 1.26 in-in-out SNCiio in-out ActLoopNT-in 2.966 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -50.25 APE8-dihe-out -60.76, -16.48 APE8-rot-na 57.99 APE67-dihe-in -64.06, -34.42 -74.64, -18.94 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 30.2472 None None None XRAY 2.97 0.204 0.258 D 311.0 257.0 18 29 19 10 [[463, 721]] 1.0 6b5j Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFIA Q59H18 441 726 835.0 4CW:801 Type1 Inactive DFGin 7.1477 14.0773 BLAminus -134.84, 175.79 58.1, 92.29 -99.47, 27.9 285.94, 73.67 -68.71, -26.95 in-in in 8.2146 Saltbr-in 2.9555 HRD-in -84.08, -48.18 75.05, 0.66 in-in-out SNCiio in-out ActLoopNT-in 3.0202 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -162.01 APE8-dihe-in -79.92, 138.7 APE8-rot-na 192.61 APE67-dihe-in -56.79, -31.79 -77.63, -30.03 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 26.9145 None None None XRAY 2.7 0.217 0.261 A 330.0 268.0 18 29 18 11 [[463, 721]] 1.0 4yfi Homo sapiens TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFIB Q59H18 451 729 835.0 4CW:801 Type1 Inactive DFGin 7.0749 14.5653 BLAminus -121.54, 177.03 56.79, 87.27 -99.8, 31.09 284.15, 68.4 -68.89, -25.59 in-in in 8.5901 Saltbr-in 2.8471 HRD-in -63.87, -47.95 70.39, 1.06 in-in-out SNCiio in-out ActLoopNT-in 2.9046 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -68.32 APE8-dihe-out -66.38, -17.23 APE8-rot-na 67.92 APE67-dihe-in -62.92, -25.6 -64.1, -31.48 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 30.8384 None None None XRAY 2.7 0.217 0.261 B 330.0 262.0 17 29 19 10 [[463, 721]] 1.0 4yfi Homo sapiens TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFIC Q59H18 441 726 835.0 4CW:801 Type1 Inactive DFGin 7.029 14.0468 BLAminus -119.12, 170.12 62.73, 94.49 -102.41, 18.34 284.63, 68.96 -60.63, -21.51 in-in in 8.3499 Saltbr-in 2.7933 HRD-in -81.8, -51.75 73.29, 8.93 in-in-out SNCiio in-out ActLoopNT-in 2.9284 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -166.83 APE8-dihe-in -85.58, 133.55 APE8-rot-na 183.6 APE67-dihe-in -63.19, -28.24 -74.71, -24.38 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.3503 None None None XRAY 2.7 0.217 0.261 C 330.0 269.0 17 29 19 10 [[463, 721]] 1.0 4yfi Homo sapiens TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFID Q59H18 451 729 835.0 4CW:801 Type1 Inactive DFGin 6.9827 14.4988 BLAminus -132.3, -176.25 57.34, 76.41 -86.69, 32.24 287.65, 73.81 -68.32, -29.28 in-in in 8.4514 Saltbr-in 3.0842 HRD-in -70.86, -49.92 74.99, 12.01 in-in-out SNCiio in-out ActLoopNT-in 2.8072 ActLoopCT-out nonTYR APEdihe_aaoai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -77.73 APE8-dihe-out -78.4, -7.06 APE8-rot-na 86.27 APE67-dihe-in -68.67, -26.29 -70.22, -28.38 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 31.2769 None None None XRAY 2.7 0.217 0.261 D 330.0 261.0 18 29 19 10 [[463, 721]] 1.0 4yfi Homo sapiens TKL_TNNI3K_HUMAN TKL 2.1e-77 266.2 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGKA Q59H18 444 726 835.0 ZGD:801 Type2 Inactive DFGout 15.0236 10.3486 BBAminus -136.11, -167.43 -161.58, 104.18 -68.96, -17.69 283.06, 90.36 80.74, 69.7 in-in in 7.8889 Saltbr-in 3.1395 HRD-in -62.84, -47.58 72.31, -16.61 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -171.11 APE8-dihe-in -86.32, 127.94 APE8-rot-na 191.21 APE67-dihe-in -60.28, -29.5 -75.53, -21.14 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.1525 None None None XRAY 3.1 0.198 0.239 A 311.0 262.0 21 29 13 16 [[463, 721]] 1.0 7mgk Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGKB Q59H18 444 727 835.0 ZGD:801 Type2 Inactive DFGout 14.6369 9.2616 BBAminus -136.1, -166.0 -163.89, 103.37 -69.12, -14.28 283.44, 87.76 84.95, 110.73 in-in in 8.2266 Saltbr-in 3.0963 HRD-in -63.33, -46.59 72.46, -18.58 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -171.17 APE8-dihe-in -84.68, 125.14 APE8-rot-na 191.2 APE67-dihe-in -61.15, -29.7 -78.96, -24.17 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 26.9334 None None None XRAY 3.1 0.198 0.239 B 311.0 261.0 23 29 13 16 [[463, 721]] 1.0 7mgk Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGKC Q59H18 445 726 835.0 ZGD:801 Type2 Inactive DFGout 15.2687 10.0615 BBAminus -135.81, -167.53 -162.54, 105.05 -66.31, -16.16 281.98, 90.65 80.81, 29.43 in-in in 8.0128 Saltbr-in 3.0708 HRD-in -63.3, -46.14 71.73, -18.15 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 128.83 APE8-rot-na 191.34 APE67-dihe-in -60.85, -29.89 -76.21, -23.31 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 3.1 0.198 0.239 C 311.0 260.0 22 29 13 16 [[463, 721]] 1.0 7mgk Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGKD Q59H18 444 727 835.0 ZGD:801 Type2 Inactive DFGout 14.8417 9.6948 BBAminus -121.51, -163.82 -171.47, 92.6 -57.07, -16.06 289.23, 82.11 84.14, 81.99 in-in in 8.1085 Saltbr-in 2.8017 HRD-in -61.83, -47.27 63.18, 0.84 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoo APE10-dihe-na 999.0, -105.6 APE9-dihe-na 75.02, 174.66 APE8-dihe-in -97.98, 119.78 APE8-rot-na 187.47 APE67-dihe-in -53.23, -38.91 -67.14, -31.62 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 30.6699 APE9-dist-out 26.8313 None None None XRAY 3.1 0.198 0.239 D 311.0 263.0 21 29 15 14 [[463, 721]] 1.0 7mgk Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGJA Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.8582 9.5819 BBAminus -134.42, -179.18 -141.04, 112.0 -72.43, -1.46 272.54, 97.9 75.05, 22.83 in-in in 7.7537 Saltbr-in 2.6724 HRD-in -64.15, -45.05 73.18, -17.04 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -171.97 APE8-dihe-in -104.46, 123.1 APE8-rot-na 189.02 APE67-dihe-in -59.47, -32.71 -67.71, -22.35 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 27.3356 None None None XRAY 2.95 0.197 0.228 A 330.0 262.0 20 29 13 16 [[463, 721]] 1.0 7mgj Homo sapiens TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGJB Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.5602 9.2473 BBAminus -135.63, -179.46 -142.92, 111.63 -76.44, -17.08 273.4, 86.62 76.35, 79.73 in-in in 7.8588 Saltbr-in 2.9045 HRD-in -64.65, -46.97 73.32, -12.56 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoo APE10-dihe-na 999.0, -80.9 APE9-dihe-na 83.07, -177.24 APE8-dihe-in -105.62, 120.49 APE8-rot-na 192.96 APE67-dihe-in -61.56, -34.4 -69.66, -24.07 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 30.6715 APE9-dist-out 26.8043 None None None XRAY 2.95 0.197 0.228 B 330.0 260.0 22 29 14 15 [[463, 721]] 1.0 7mgj Homo sapiens TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGJC Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.6969 9.6665 BBAminus -137.79, -177.03 -141.64, 110.69 -73.01, -3.0 273.24, 93.94 74.23, 29.77 in-in in 7.8989 Saltbr-in 2.91 HRD-in -66.15, -44.57 73.37, -16.84 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 119.35 APE8-rot-na 190.99 APE67-dihe-in -61.3, -34.66 -68.53, -21.6 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.95 0.197 0.228 C 330.0 261.0 21 29 13 16 [[463, 721]] 1.0 7mgj Homo sapiens TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 7MGJD Q59H18 445 726 835.0 ZFS:801 Type2 Inactive DFGout 14.5321 9.688 BBAminus -144.03, 179.53 -144.45, 109.82 -73.53, -9.7 276.8, 74.13 75.18, 64.15 in-in in 7.7498 Saltbr-in 2.6424 HRD-in -65.07, -45.42 74.54, -12.51 in-none-out SNCino none-out ActLoopNT-none 999.0 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoo APE10-dihe-na 999.0, -81.24 APE9-dihe-na 82.5, -174.24 APE8-dihe-in -103.92, 121.0 APE8-rot-na 193.26 APE67-dihe-in -60.88, -34.79 -69.71, -24.61 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 31.3479 APE9-dist-out 27.2314 None None None XRAY 2.95 0.197 0.228 D 330.0 261.0 21 29 15 14 [[463, 721]] 1.0 7mgj Homo sapiens TKL_TNNI3K_HUMAN TKL 1.9e-77 266.4 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFFA Q59H18 445 726 835.0 4CV:801 Type1 None DFGin 6.8965 13.8872 BLAminus -127.46, 175.49 57.0, 94.25 -101.84, 21.43 285.11, 76.86 -67.58, -12.19 in-in in 8.3049 Saltbr-in 2.5732 HRD-in -72.29, -48.61 68.2, 11.99 in-in-none SNCiin in-none ActLoopNT-in 2.7517 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 133.81 APE8-rot-na 181.89 APE67-dihe-in -64.26, -21.67 -83.98, -17.01 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 3.07 0.211 0.251 A 311.0 264.0 18 29 18 11 [[463, 721]] 1.0 4yff Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 4YFFB Q59H18 445 726 835.0 4CV:801 Type1 None DFGin 6.8476 13.8816 BLAminus -128.82, 174.1 57.67, 94.34 -100.02, 21.13 285.48, 77.01 -67.5, -10.8 in-in in 8.3585 Saltbr-in 2.6026 HRD-in -72.09, -48.38 68.6, 12.37 in-in-none SNCiin in-none ActLoopNT-in 2.7622 ActLoopCT-none nonTYR APEdihe_aanni APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 137.74 APE8-rot-none 999.0 APE67-dihe-in -59.76, -26.5 -86.26, -18.43 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 3.07 0.211 0.251 B 311.0 264.0 18 29 17 12 [[463, 721]] 1.0 4yff Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K
TNNI3K TNI3K_HUMAN 6B5JB Q59H18 445 726 835.0 CV4:801 Type1 None DFGin 6.7764 13.8842 BLAminus -127.39, 170.23 63.58, 89.42 -96.67, 32.19 290.95, 72.96 -66.8, -26.81 in-in in 8.6163 Saltbr-in 3.0489 HRD-in -67.53, -48.98 70.48, -12.85 in-in-none SNCiin in-none ActLoopNT-in 2.9262 ActLoopCT-none nonTYR APEdihe_aanai APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 129.15 APE8-rot-na 200.19 APE67-dihe-in -61.72, -25.21 -84.18, -18.08 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.97 0.204 0.258 B 311.0 264.0 18 29 17 12 [[463, 721]] 1.0 6b5j Homo sapiens TKL_TNNI3K_HUMAN TKL 1.5e-77 266.7 1.0 267.0 267.0 605 606 607 609 611 490 509 513 585 587 586 588.0 647 634 629 628 627 626 625 624 623 540 Serine/threonine-protein kinase TNNI3K

TKL_TNNI3K (Serine/threonine-protein kinase TNNI3K)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name