| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| PRKG1 | 6BG2A | Q13976 | 336 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.8108 | 14.7141 | BLAminus | -124.15, 169.14 | 66.07, 88.5 | -100.57, 30.98 | 280.35, 66.41 | -65.35, -25.12 | in-in | in | 9.5223 | Saltbr-in | 2.8826 | HRD-in | -85.83, -52.95 | 73.29, 9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8514 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.93, 165.57 | APE9-dihe-na | 117.74, 172.78 | APE8-dihe-in | -83.6, 129.51 | APE8-rot-in | 307.46 | APE67-dihe-in | -66.9, -19.23 | -49.63, -41.3 | APE12-dist-in | 8.2348 | APE11-dist-in | 11.5121 | APE10-dist-in | 6.0409 | APE9-dist-in | 4.269 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | A | 347.0 | 336.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 6BG2B | Q13976 | 346 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 6.0006 | 13.8103 | BLAminus | -122.67, 175.58 | 65.94, 84.43 | -99.77, 30.78 | 285.96, 70.42 | -64.93, -24.07 | in-in | in | 8.944 | Saltbr-in | 2.7425 | HRD-in | -86.95, -52.47 | 73.99, 7.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9238 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.61, 163.67 | APE9-dihe-na | 118.96, 172.39 | APE8-dihe-in | -86.94, 131.94 | APE8-rot-in | 306.51 | APE67-dihe-in | -68.79, -20.88 | -48.58, -41.68 | APE12-dist-in | 7.8257 | APE11-dist-in | 11.2147 | APE10-dist-in | 5.7688 | APE9-dist-in | 4.0083 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | B | 347.0 | 326.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 6BG2C | Q13976 | 337 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.7459 | 14.0572 | BLAminus | -122.99, 175.03 | 65.66, 84.22 | -99.61, 30.7 | 281.62, 66.26 | -64.81, -23.57 | in-in | in | 8.7415 | Saltbr-in | 2.7233 | HRD-in | -85.99, -53.51 | 74.31, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9506 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.66, 165.85 | APE9-dihe-na | 118.46, 173.18 | APE8-dihe-in | -87.41, 130.75 | APE8-rot-in | 306.63 | APE67-dihe-in | -67.71, -19.03 | -48.39, -42.55 | APE12-dist-in | 7.9723 | APE11-dist-in | 11.3847 | APE10-dist-in | 5.8567 | APE9-dist-in | 3.8612 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | C | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 6BG2D | Q13976 | 344 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.7098 | 14.0124 | BLAminus | -124.49, 174.79 | 65.67, 84.87 | -99.37, 30.45 | 283.38, 66.11 | -64.13, -22.3 | in-in | in | 8.754 | Saltbr-in | 2.6441 | HRD-in | -85.68, -52.69 | 74.16, 8.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9303 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.92, 166.42 | APE9-dihe-na | 119.53, 169.97 | APE8-dihe-in | -84.81, 130.45 | APE8-rot-in | 305.19 | APE67-dihe-in | -66.29, -19.88 | -48.13, -43.31 | APE12-dist-in | 7.9878 | APE11-dist-in | 11.3267 | APE10-dist-in | 5.7839 | APE9-dist-in | 3.8102 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | D | 347.0 | 328.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7LV3A | Q13976 | 57 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.8509 | 14.0363 | BLAminus | -116.97, 177.04 | 63.26, 88.72 | -106.87, 28.72 | 283.22, 63.7 | -62.95, -24.33 | in-in | in | 8.6241 | Saltbr-in | 2.891 | HRD-in | -87.82, -54.22 | 74.26, 7.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.911 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.98 | APE9-dihe-na | 157.95, -145.59 | APE8-dihe-in | -124.73, 128.61 | APE8-rot-in | 299.79 | APE67-dihe-in | -58.37, -20.06 | -47.89, -51.97 | APE12-dist-in | 7.9724 | APE11-dist-in | 11.0568 | APE10-dist-in | 5.4693 | APE9-dist-in | 3.8106 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | A | 617.0 | 600.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7lv3 | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7LV3B | Q13976 | 58 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.6336 | 13.9624 | BLAminus | -116.52, 178.28 | 63.3, 90.17 | -108.68, 29.08 | 283.48, 65.02 | -62.88, -23.93 | in-in | in | 8.8833 | Saltbr-in | 2.8237 | HRD-in | -86.48, -52.9 | 74.97, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9589 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.21 | APE9-dihe-na | 157.62, -145.94 | APE8-dihe-in | -123.75, 129.22 | APE8-rot-in | 300.73 | APE67-dihe-in | -59.05, -19.44 | -46.41, -52.49 | APE12-dist-in | 8.1341 | APE11-dist-in | 11.1978 | APE10-dist-in | 5.6042 | APE9-dist-in | 3.7871 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | B | 617.0 | 593.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7lv3 | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4VB | Q13976 | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Active | DFGin | 6.191 | 14.8482 | BLAminus | -117.12, 164.99 | 68.84, 100.49 | -114.63, 44.2 | 282.85, 73.02 | -69.55, -49.58 | in-in | in | 9.8759 | Saltbr-in | 3.02 | HRD-in | -85.46, -53.89 | 74.22, -39.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.744 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.05, 169.08 | APE9-dihe-na | 104.88, 162.74 | APE8-dihe-in | -71.34, 125.86 | APE8-rot-in | 297.46 | APE67-dihe-in | -57.61, -28.56 | -42.75, -43.02 | APE12-dist-in | 8.2638 | APE11-dist-in | 11.6633 | APE10-dist-in | 6.268 | APE9-dist-in | 5.2162 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | B | 469.0 | 464.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4v | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | AF-Q13976-K1A | Q13976 | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 6.2706 | 14.18 | BLAminus | -115.7, -171.89 | 41.6, 86.13 | -92.63, 18.96 | 285.01, 78.59 | -59.54, -30.9 | in-in | in | 9.6067 | Saltbr-in | 2.7119 | HRD-in | -90.69, -50.22 | 66.05, 7.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8812 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.15, 172.71 | APE9-dihe-na | 108.43, 171.02 | APE8-dihe-in | -80.49, 129.57 | APE8-rot-in | 300.74 | APE67-dihe-in | -68.04, -21.28 | -48.8, -41.85 | APE12-dist-in | 8.2142 | APE11-dist-in | 11.1969 | APE10-dist-in | 5.629 | APE9-dist-in | 3.5295 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K1 | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | AF-Q13976-K3A | Q13976 | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 5.9061 | 13.9228 | BLAminus | -115.45, -173.31 | 41.39, 87.3 | -90.8, 19.58 | 282.99, 76.21 | -58.78, -31.1 | in-in | in | 9.2484 | Saltbr-in | 2.7136 | HRD-in | -91.17, -53.27 | 69.22, 14.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8698 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.96, 169.62 | APE9-dihe-na | 104.72, 167.78 | APE8-dihe-in | -75.94, 135.6 | APE8-rot-in | 283.37 | APE67-dihe-in | -66.68, -21.92 | -49.58, -45.16 | APE12-dist-in | 7.8884 | APE11-dist-in | 11.013 | APE10-dist-in | 5.4435 | APE9-dist-in | 3.3379 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K3 | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4UA | Q13976 | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.8928 | 14.5109 | ABAminus | -110.98, -36.23 | -113.94, 119.68 | -109.65, 38.15 | 284.57, 73.72 | -68.19, -46.47 | in-in | in | 9.7533 | Saltbr-in | 2.9444 | HRD-in | -80.27, -49.41 | 62.96, -11.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9436 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.82, 170.87 | APE9-dihe-na | 95.36, 163.3 | APE8-dihe-in | -65.83, 127.77 | APE8-rot-in | 297.19 | APE67-dihe-in | -61.65, -25.18 | -50.5, -36.94 | APE12-dist-in | 8.3016 | APE11-dist-in | 11.5495 | APE10-dist-in | 5.8864 | APE9-dist-in | 5.0426 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | A | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4u | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4UB | Q13976 | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.8817 | 14.6709 | ABAminus | -116.42, -27.15 | -112.65, 115.98 | -107.16, 33.12 | 284.12, 70.33 | -62.23, -46.18 | in-in | in | 9.7607 | Saltbr-in | 2.9206 | HRD-in | -79.97, -49.4 | 62.99, -11.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9244 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.62, 162.77 | APE9-dihe-na | 104.48, 162.22 | APE8-dihe-in | -65.39, 128.54 | APE8-rot-in | 296.86 | APE67-dihe-in | -62.65, -24.95 | -50.24, -36.77 | APE12-dist-in | 8.2598 | APE11-dist-in | 11.5735 | APE10-dist-in | 5.9624 | APE9-dist-in | 5.0144 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | B | 469.0 | 461.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4u | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4WA | Q13976 | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.2029 | 14.6561 | ABAminus | -120.51, -49.82 | -94.54, 125.75 | -115.2, 38.22 | 287.71, 71.79 | -69.94, -44.46 | in-in | in | 9.8677 | Saltbr-in | 3.4624 | HRD-in | -82.07, -59.56 | 68.33, -9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0314 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.57, 172.99 | APE9-dihe-na | 100.31, 156.35 | APE8-dihe-in | -58.55, 123.29 | APE8-rot-in | 292.59 | APE67-dihe-in | -70.67, -20.63 | -47.72, -29.8 | APE12-dist-in | 8.0748 | APE11-dist-in | 11.4987 | APE10-dist-in | 6.2222 | APE9-dist-in | 4.9178 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | A | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4w | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4WB | Q13976 | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.1666 | 14.645 | ABAminus | -115.45, -45.68 | -98.44, 117.3 | -111.38, 33.0 | 288.61, 72.93 | -65.23, -44.36 | in-in | in | 9.884 | Saltbr-in | 3.465 | HRD-in | -84.88, -51.35 | 65.14, -16.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.45, 173.1 | APE9-dihe-na | 100.13, 155.73 | APE8-dihe-in | -59.24, 124.2 | APE8-rot-in | 292.57 | APE67-dihe-in | -70.75, -20.56 | -47.95, -29.59 | APE12-dist-in | 8.0863 | APE11-dist-in | 11.5137 | APE10-dist-in | 6.2502 | APE9-dist-in | 4.8978 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | B | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4w | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4TA | Q13976 | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.8055 | 14.9328 | ABAminus | -123.17, -29.2 | -107.96, 118.17 | -112.33, 30.1 | 285.53, 74.3 | -67.24, -29.77 | in-in | in | 9.5568 | Saltbr-in | 3.3803 | HRD-in | -86.67, -51.63 | 61.2, 10.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8595 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -166.89, 164.61 | APE9-dihe-na | 124.7, -170.63 | APE8-dihe-in | -100.54, 134.31 | APE8-rot-in | 302.38 | APE67-dihe-in | -67.0, -27.98 | -44.1, -43.89 | APE12-dist-in | 7.9413 | APE11-dist-in | 10.7126 | APE10-dist-in | 5.3076 | APE9-dist-in | 3.712 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | A | 469.0 | 453.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4t | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4TB | Q13976 | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.8004 | 14.8112 | ABAminus | -121.38, -38.76 | -100.76, 117.73 | -112.4, 30.34 | 285.48, 73.71 | -68.75, -29.12 | in-in | in | 9.4009 | Saltbr-in | 3.3105 | HRD-in | -86.82, -51.68 | 61.52, 10.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8534 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -165.5, 164.27 | APE9-dihe-na | 124.32, -169.95 | APE8-dihe-in | -101.18, 134.26 | APE8-rot-in | 302.8 | APE67-dihe-in | -67.54, -26.94 | -44.3, -44.01 | APE12-dist-in | 7.9575 | APE11-dist-in | 10.7572 | APE10-dist-in | 5.3357 | APE9-dist-in | 3.7168 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | B | 469.0 | 453.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4t | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 7T4VA | Q13976 | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Inactive | DFGin | 6.1797 | 14.758 | BLAminus | -117.38, 165.11 | 68.06, 101.28 | -115.37, 45.06 | 282.61, 73.13 | -70.13, -49.07 | in-in | in | 9.8385 | Saltbr-in | 2.9792 | HRD-in | -86.09, -51.09 | 71.54, -55.93 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7416 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -158.12, 169.74 | APE9-dihe-na | 104.56, 162.71 | APE8-dihe-in | -70.69, 125.48 | APE8-rot-in | 298.14 | APE67-dihe-in | -57.19, -28.82 | -42.61, -42.82 | APE12-dist-in | 8.5561 | APE11-dist-in | 11.7139 | APE10-dist-in | 6.3175 | APE9-dist-out | 6.0312 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | A | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4v | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 6BDLA | Q13976 | 337 | 671 | 671.0 | No_ligand | No_ligand | Inactive | DFGin | 5.7129 | 14.5128 | BLAminus | -122.27, 166.18 | 66.21, 96.03 | -109.78, 28.36 | 280.09, 66.52 | -59.53, -32.57 | in-in | in | 9.5651 | Saltbr-in | 2.7123 | HRD-in | -93.15, -47.43 | 77.49, -41.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.821 | ActLoopCT-out | nonTYR | APEdihe_aaini | APEdist_iiio | APE10-dihe-na | -113.85, 160.0 | APE9-dihe-na | 86.62, 160.7 | APE8-dihe-in | -68.44, 153.87 | APE8-rot-none | 999.0 | APE67-dihe-in | -67.03, -17.86 | -55.61, -25.3 | APE12-dist-in | 7.7646 | APE11-dist-in | 11.2183 | APE10-dist-in | 5.6044 | APE9-dist-out | 6.2314 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | A | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bdl | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 6C0TA | Q13976 | 337 | 671 | 671.0 | EE4:701 | Type1.5_Front | Inactive | DFGin | 5.9004 | 14.2567 | BLAminus | -131.41, 173.3 | 67.52, 81.76 | -101.27, 23.85 | 278.07, 65.63 | -65.26, -23.23 | in-in | in | 8.9348 | Saltbr-in | 2.7968 | HRD-in | -100.02, -51.71 | 77.78, -11.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7896 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -144.5, 158.55 | APE9-dihe-na | 107.94, 162.3 | APE8-dihe-in | -69.48, 141.18 | APE8-rot-out | 79.81 | APE67-dihe-in | -72.66, -16.0 | -52.58, -33.36 | APE12-dist-in | 7.7396 | APE11-dist-in | 11.364 | APE10-dist-in | 5.9865 | APE9-dist-in | 4.8195 | None | TPO517 | TPO517 | XRAY | 1.98 | 0.21 | 0.244 | A | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6c0t | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | 6BDLB | Q13976 | 337 | 671 | 671.0 | No_ligand | No_ligand | None | DFGin | 5.7574 | 14.6582 | BLAminus | -124.78, 164.72 | 65.46, 95.48 | -109.07, 28.23 | 278.78, 64.61 | -59.31, -33.14 | in-in | in | 9.3371 | Saltbr-in | 2.902 | HRD-in | -92.19, -47.19 | 78.26, -40.54 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8769 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_iiii | APE10-dihe-na | -122.13, 167.41 | APE9-dihe-na | 91.21, 161.43 | APE8-dihe-in | -67.63, 145.68 | APE8-rot-none | 999.0 | APE67-dihe-in | -70.27, -17.78 | -60.28, -30.02 | APE12-dist-in | 7.5984 | APE11-dist-in | 11.396 | APE10-dist-in | 5.7947 | APE9-dist-in | 5.4685 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | B | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bdl | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| PRKG1 | KGP1_HUMAN | 6BG2A | Q13976 | 336 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.8108 | 14.7141 | BLAminus | -124.15, 169.14 | 66.07, 88.5 | -100.57, 30.98 | 280.35, 66.41 | -65.35, -25.12 | in-in | in | 9.5223 | Saltbr-in | 2.8826 | HRD-in | -85.83, -52.95 | 73.29, 9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8514 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.93, 165.57 | APE9-dihe-na | 117.74, 172.78 | APE8-dihe-in | -83.6, 129.51 | APE8-rot-in | 307.46 | APE67-dihe-in | -66.9, -19.23 | -49.63, -41.3 | APE12-dist-in | 8.2348 | APE11-dist-in | 11.5121 | APE10-dist-in | 6.0409 | APE9-dist-in | 4.269 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | A | 347.0 | 336.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 6BG2B | Q13976 | 346 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 6.0006 | 13.8103 | BLAminus | -122.67, 175.58 | 65.94, 84.43 | -99.77, 30.78 | 285.96, 70.42 | -64.93, -24.07 | in-in | in | 8.944 | Saltbr-in | 2.7425 | HRD-in | -86.95, -52.47 | 73.99, 7.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9238 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.61, 163.67 | APE9-dihe-na | 118.96, 172.39 | APE8-dihe-in | -86.94, 131.94 | APE8-rot-in | 306.51 | APE67-dihe-in | -68.79, -20.88 | -48.58, -41.68 | APE12-dist-in | 7.8257 | APE11-dist-in | 11.2147 | APE10-dist-in | 5.7688 | APE9-dist-in | 4.0083 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | B | 347.0 | 326.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 6BG2C | Q13976 | 337 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.7459 | 14.0572 | BLAminus | -122.99, 175.03 | 65.66, 84.22 | -99.61, 30.7 | 281.62, 66.26 | -64.81, -23.57 | in-in | in | 8.7415 | Saltbr-in | 2.7233 | HRD-in | -85.99, -53.51 | 74.31, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9506 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.66, 165.85 | APE9-dihe-na | 118.46, 173.18 | APE8-dihe-in | -87.41, 130.75 | APE8-rot-in | 306.63 | APE67-dihe-in | -67.71, -19.03 | -48.39, -42.55 | APE12-dist-in | 7.9723 | APE11-dist-in | 11.3847 | APE10-dist-in | 5.8567 | APE9-dist-in | 3.8612 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | C | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 6BG2D | Q13976 | 344 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.7098 | 14.0124 | BLAminus | -124.49, 174.79 | 65.67, 84.87 | -99.37, 30.45 | 283.38, 66.11 | -64.13, -22.3 | in-in | in | 8.754 | Saltbr-in | 2.6441 | HRD-in | -85.68, -52.69 | 74.16, 8.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9303 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.92, 166.42 | APE9-dihe-na | 119.53, 169.97 | APE8-dihe-in | -84.81, 130.45 | APE8-rot-in | 305.19 | APE67-dihe-in | -66.29, -19.88 | -48.13, -43.31 | APE12-dist-in | 7.9878 | APE11-dist-in | 11.3267 | APE10-dist-in | 5.7839 | APE9-dist-in | 3.8102 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | D | 347.0 | 328.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7LV3A | Q13976 | 57 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.8509 | 14.0363 | BLAminus | -116.97, 177.04 | 63.26, 88.72 | -106.87, 28.72 | 283.22, 63.7 | -62.95, -24.33 | in-in | in | 8.6241 | Saltbr-in | 2.891 | HRD-in | -87.82, -54.22 | 74.26, 7.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.911 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.98 | APE9-dihe-na | 157.95, -145.59 | APE8-dihe-in | -124.73, 128.61 | APE8-rot-in | 299.79 | APE67-dihe-in | -58.37, -20.06 | -47.89, -51.97 | APE12-dist-in | 7.9724 | APE11-dist-in | 11.0568 | APE10-dist-in | 5.4693 | APE9-dist-in | 3.8106 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | A | 617.0 | 600.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7lv3 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7LV3B | Q13976 | 58 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.6336 | 13.9624 | BLAminus | -116.52, 178.28 | 63.3, 90.17 | -108.68, 29.08 | 283.48, 65.02 | -62.88, -23.93 | in-in | in | 8.8833 | Saltbr-in | 2.8237 | HRD-in | -86.48, -52.9 | 74.97, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9589 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.21 | APE9-dihe-na | 157.62, -145.94 | APE8-dihe-in | -123.75, 129.22 | APE8-rot-in | 300.73 | APE67-dihe-in | -59.05, -19.44 | -46.41, -52.49 | APE12-dist-in | 8.1341 | APE11-dist-in | 11.1978 | APE10-dist-in | 5.6042 | APE9-dist-in | 3.7871 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | B | 617.0 | 593.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7lv3 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4VB | Q13976 | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Active | DFGin | 6.191 | 14.8482 | BLAminus | -117.12, 164.99 | 68.84, 100.49 | -114.63, 44.2 | 282.85, 73.02 | -69.55, -49.58 | in-in | in | 9.8759 | Saltbr-in | 3.02 | HRD-in | -85.46, -53.89 | 74.22, -39.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.744 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.05, 169.08 | APE9-dihe-na | 104.88, 162.74 | APE8-dihe-in | -71.34, 125.86 | APE8-rot-in | 297.46 | APE67-dihe-in | -57.61, -28.56 | -42.75, -43.02 | APE12-dist-in | 8.2638 | APE11-dist-in | 11.6633 | APE10-dist-in | 6.268 | APE9-dist-in | 5.2162 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | B | 469.0 | 464.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4v | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | AF-Q13976-K1A | Q13976 | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 6.2706 | 14.18 | BLAminus | -115.7, -171.89 | 41.6, 86.13 | -92.63, 18.96 | 285.01, 78.59 | -59.54, -30.9 | in-in | in | 9.6067 | Saltbr-in | 2.7119 | HRD-in | -90.69, -50.22 | 66.05, 7.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8812 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.15, 172.71 | APE9-dihe-na | 108.43, 171.02 | APE8-dihe-in | -80.49, 129.57 | APE8-rot-in | 300.74 | APE67-dihe-in | -68.04, -21.28 | -48.8, -41.85 | APE12-dist-in | 8.2142 | APE11-dist-in | 11.1969 | APE10-dist-in | 5.629 | APE9-dist-in | 3.5295 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K1 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | AF-Q13976-K3A | Q13976 | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 5.9061 | 13.9228 | BLAminus | -115.45, -173.31 | 41.39, 87.3 | -90.8, 19.58 | 282.99, 76.21 | -58.78, -31.1 | in-in | in | 9.2484 | Saltbr-in | 2.7136 | HRD-in | -91.17, -53.27 | 69.22, 14.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8698 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.96, 169.62 | APE9-dihe-na | 104.72, 167.78 | APE8-dihe-in | -75.94, 135.6 | APE8-rot-in | 283.37 | APE67-dihe-in | -66.68, -21.92 | -49.58, -45.16 | APE12-dist-in | 7.8884 | APE11-dist-in | 11.013 | APE10-dist-in | 5.4435 | APE9-dist-in | 3.3379 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276.0 | 276.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K3 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4UA | Q13976 | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.8928 | 14.5109 | ABAminus | -110.98, -36.23 | -113.94, 119.68 | -109.65, 38.15 | 284.57, 73.72 | -68.19, -46.47 | in-in | in | 9.7533 | Saltbr-in | 2.9444 | HRD-in | -80.27, -49.41 | 62.96, -11.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9436 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.82, 170.87 | APE9-dihe-na | 95.36, 163.3 | APE8-dihe-in | -65.83, 127.77 | APE8-rot-in | 297.19 | APE67-dihe-in | -61.65, -25.18 | -50.5, -36.94 | APE12-dist-in | 8.3016 | APE11-dist-in | 11.5495 | APE10-dist-in | 5.8864 | APE9-dist-in | 5.0426 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | A | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4u | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4UB | Q13976 | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.8817 | 14.6709 | ABAminus | -116.42, -27.15 | -112.65, 115.98 | -107.16, 33.12 | 284.12, 70.33 | -62.23, -46.18 | in-in | in | 9.7607 | Saltbr-in | 2.9206 | HRD-in | -79.97, -49.4 | 62.99, -11.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9244 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.62, 162.77 | APE9-dihe-na | 104.48, 162.22 | APE8-dihe-in | -65.39, 128.54 | APE8-rot-in | 296.86 | APE67-dihe-in | -62.65, -24.95 | -50.24, -36.77 | APE12-dist-in | 8.2598 | APE11-dist-in | 11.5735 | APE10-dist-in | 5.9624 | APE9-dist-in | 5.0144 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | B | 469.0 | 461.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4u | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4WA | Q13976 | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.2029 | 14.6561 | ABAminus | -120.51, -49.82 | -94.54, 125.75 | -115.2, 38.22 | 287.71, 71.79 | -69.94, -44.46 | in-in | in | 9.8677 | Saltbr-in | 3.4624 | HRD-in | -82.07, -59.56 | 68.33, -9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0314 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.57, 172.99 | APE9-dihe-na | 100.31, 156.35 | APE8-dihe-in | -58.55, 123.29 | APE8-rot-in | 292.59 | APE67-dihe-in | -70.67, -20.63 | -47.72, -29.8 | APE12-dist-in | 8.0748 | APE11-dist-in | 11.4987 | APE10-dist-in | 6.2222 | APE9-dist-in | 4.9178 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | A | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4w | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4WB | Q13976 | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.1666 | 14.645 | ABAminus | -115.45, -45.68 | -98.44, 117.3 | -111.38, 33.0 | 288.61, 72.93 | -65.23, -44.36 | in-in | in | 9.884 | Saltbr-in | 3.465 | HRD-in | -84.88, -51.35 | 65.14, -16.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.45, 173.1 | APE9-dihe-na | 100.13, 155.73 | APE8-dihe-in | -59.24, 124.2 | APE8-rot-in | 292.57 | APE67-dihe-in | -70.75, -20.56 | -47.95, -29.59 | APE12-dist-in | 8.0863 | APE11-dist-in | 11.5137 | APE10-dist-in | 6.2502 | APE9-dist-in | 4.8978 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | B | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4w | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4TA | Q13976 | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.8055 | 14.9328 | ABAminus | -123.17, -29.2 | -107.96, 118.17 | -112.33, 30.1 | 285.53, 74.3 | -67.24, -29.77 | in-in | in | 9.5568 | Saltbr-in | 3.3803 | HRD-in | -86.67, -51.63 | 61.2, 10.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8595 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -166.89, 164.61 | APE9-dihe-na | 124.7, -170.63 | APE8-dihe-in | -100.54, 134.31 | APE8-rot-in | 302.38 | APE67-dihe-in | -67.0, -27.98 | -44.1, -43.89 | APE12-dist-in | 7.9413 | APE11-dist-in | 10.7126 | APE10-dist-in | 5.3076 | APE9-dist-in | 3.712 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | A | 469.0 | 453.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4t | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4TB | Q13976 | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.8004 | 14.8112 | ABAminus | -121.38, -38.76 | -100.76, 117.73 | -112.4, 30.34 | 285.48, 73.71 | -68.75, -29.12 | in-in | in | 9.4009 | Saltbr-in | 3.3105 | HRD-in | -86.82, -51.68 | 61.52, 10.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8534 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -165.5, 164.27 | APE9-dihe-na | 124.32, -169.95 | APE8-dihe-in | -101.18, 134.26 | APE8-rot-in | 302.8 | APE67-dihe-in | -67.54, -26.94 | -44.3, -44.01 | APE12-dist-in | 7.9575 | APE11-dist-in | 10.7572 | APE10-dist-in | 5.3357 | APE9-dist-in | 3.7168 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | B | 469.0 | 453.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4t | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 7T4VA | Q13976 | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Inactive | DFGin | 6.1797 | 14.758 | BLAminus | -117.38, 165.11 | 68.06, 101.28 | -115.37, 45.06 | 282.61, 73.13 | -70.13, -49.07 | in-in | in | 9.8385 | Saltbr-in | 2.9792 | HRD-in | -86.09, -51.09 | 71.54, -55.93 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7416 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -158.12, 169.74 | APE9-dihe-na | 104.56, 162.71 | APE8-dihe-in | -70.69, 125.48 | APE8-rot-in | 298.14 | APE67-dihe-in | -57.19, -28.82 | -42.61, -42.82 | APE12-dist-in | 8.5561 | APE11-dist-in | 11.7139 | APE10-dist-in | 6.3175 | APE9-dist-out | 6.0312 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | A | 469.0 | 467.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 7t4v | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 6BDLA | Q13976 | 337 | 671 | 671.0 | No_ligand | No_ligand | Inactive | DFGin | 5.7129 | 14.5128 | BLAminus | -122.27, 166.18 | 66.21, 96.03 | -109.78, 28.36 | 280.09, 66.52 | -59.53, -32.57 | in-in | in | 9.5651 | Saltbr-in | 2.7123 | HRD-in | -93.15, -47.43 | 77.49, -41.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.821 | ActLoopCT-out | nonTYR | APEdihe_aaini | APEdist_iiio | APE10-dihe-na | -113.85, 160.0 | APE9-dihe-na | 86.62, 160.7 | APE8-dihe-in | -68.44, 153.87 | APE8-rot-none | 999.0 | APE67-dihe-in | -67.03, -17.86 | -55.61, -25.3 | APE12-dist-in | 7.7646 | APE11-dist-in | 11.2183 | APE10-dist-in | 5.6044 | APE9-dist-out | 6.2314 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | A | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bdl | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 6C0TA | Q13976 | 337 | 671 | 671.0 | EE4:701 | Type1.5_Front | Inactive | DFGin | 5.9004 | 14.2567 | BLAminus | -131.41, 173.3 | 67.52, 81.76 | -101.27, 23.85 | 278.07, 65.63 | -65.26, -23.23 | in-in | in | 8.9348 | Saltbr-in | 2.7968 | HRD-in | -100.02, -51.71 | 77.78, -11.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7896 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -144.5, 158.55 | APE9-dihe-na | 107.94, 162.3 | APE8-dihe-in | -69.48, 141.18 | APE8-rot-out | 79.81 | APE67-dihe-in | -72.66, -16.0 | -52.58, -33.36 | APE12-dist-in | 7.7396 | APE11-dist-in | 11.364 | APE10-dist-in | 5.9865 | APE9-dist-in | 4.8195 | None | TPO517 | TPO517 | XRAY | 1.98 | 0.21 | 0.244 | A | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6c0t | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| PRKG1 | KGP1_HUMAN | 6BDLB | Q13976 | 337 | 671 | 671.0 | No_ligand | No_ligand | None | DFGin | 5.7574 | 14.6582 | BLAminus | -124.78, 164.72 | 65.46, 95.48 | -109.07, 28.23 | 278.78, 64.61 | -59.31, -33.14 | in-in | in | 9.3371 | Saltbr-in | 2.902 | HRD-in | -92.19, -47.19 | 78.26, -40.54 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8769 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_iiii | APE10-dihe-na | -122.13, 167.41 | APE9-dihe-na | 91.21, 161.43 | APE8-dihe-in | -67.63, 145.68 | APE8-rot-none | 999.0 | APE67-dihe-in | -70.27, -17.78 | -60.28, -30.02 | APE12-dist-in | 7.5984 | APE11-dist-in | 11.396 | APE10-dist-in | 5.7947 | APE9-dist-in | 5.4685 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | B | 347.0 | 335.0 | 0 | 27 | 27 | 0 | [[360, 619]] | 1.0 | 6bdl | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1.0 | 260.0 | 260.0 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484.0 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|