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| PDB | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 6BG2A | 336 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.811 | 14.714 | BLAminus | -124.15, 169.14 | 66.07, 88.5 | -100.57, 30.98 | 280.35, 66.41 | -65.35, -25.12 | in-in | in | 9.522 | Saltbr-in | 2.883 | HRD-in | -85.83, -52.95 | 73.29, 9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.851 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.93, 165.57 | APE9-dihe-na | 117.74, 172.78 | APE8-dihe-in | -83.6, 129.51 | APE8-rot-in | 307.46 | APE67-dihe-in | -66.9, -19.23 | -49.63, -41.3 | APE12-dist-in | 8.235 | APE11-dist-in | 11.512 | APE10-dist-in | 6.041 | APE9-dist-in | 4.269 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | A | 347 | 336 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 6BG2B | 346 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 6.001 | 13.81 | BLAminus | -122.67, 175.58 | 65.94, 84.43 | -99.77, 30.78 | 285.96, 70.42 | -64.93, -24.07 | in-in | in | 8.944 | Saltbr-in | 2.743 | HRD-in | -86.95, -52.47 | 73.99, 7.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.924 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.61, 163.67 | APE9-dihe-na | 118.96, 172.39 | APE8-dihe-in | -86.94, 131.94 | APE8-rot-in | 306.51 | APE67-dihe-in | -68.79, -20.88 | -48.58, -41.68 | APE12-dist-in | 7.826 | APE11-dist-in | 11.215 | APE10-dist-in | 5.769 | APE9-dist-in | 4.008 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | B | 347 | 326 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 6BG2C | 337 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.746 | 14.057 | BLAminus | -122.99, 175.03 | 65.66, 84.22 | -99.61, 30.7 | 281.62, 66.26 | -64.81, -23.57 | in-in | in | 8.742 | Saltbr-in | 2.723 | HRD-in | -85.99, -53.51 | 74.31, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.951 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.66, 165.85 | APE9-dihe-na | 118.46, 173.18 | APE8-dihe-in | -87.41, 130.75 | APE8-rot-in | 306.63 | APE67-dihe-in | -67.71, -19.03 | -48.39, -42.55 | APE12-dist-in | 7.972 | APE11-dist-in | 11.385 | APE10-dist-in | 5.857 | APE9-dist-in | 3.861 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | C | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 6BG2D | 344 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.71 | 14.012 | BLAminus | -124.49, 174.79 | 65.67, 84.87 | -99.37, 30.45 | 283.38, 66.11 | -64.13, -22.3 | in-in | in | 8.754 | Saltbr-in | 2.644 | HRD-in | -85.68, -52.69 | 74.16, 8.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.92, 166.42 | APE9-dihe-na | 119.53, 169.97 | APE8-dihe-in | -84.81, 130.45 | APE8-rot-in | 305.19 | APE67-dihe-in | -66.29, -19.88 | -48.13, -43.31 | APE12-dist-in | 7.988 | APE11-dist-in | 11.327 | APE10-dist-in | 5.784 | APE9-dist-in | 3.81 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | D | 347 | 328 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7LV3A | 57 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.851 | 14.036 | BLAminus | -116.97, 177.04 | 63.26, 88.72 | -106.87, 28.72 | 283.22, 63.7 | -62.95, -24.33 | in-in | in | 8.624 | Saltbr-in | 2.891 | HRD-in | -87.82, -54.22 | 74.26, 7.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.911 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.98 | APE9-dihe-na | 157.95, -145.59 | APE8-dihe-in | -124.73, 128.61 | APE8-rot-in | 299.79 | APE67-dihe-in | -58.37, -20.06 | -47.89, -51.97 | APE12-dist-in | 7.972 | APE11-dist-in | 11.057 | APE10-dist-in | 5.469 | APE9-dist-in | 3.811 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | A | 617 | 600 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7lv3 | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7LV3B | 58 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.634 | 13.962 | BLAminus | -116.52, 178.28 | 63.3, 90.17 | -108.68, 29.08 | 283.48, 65.02 | -62.88, -23.93 | in-in | in | 8.883 | Saltbr-in | 2.824 | HRD-in | -86.48, -52.9 | 74.97, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.21 | APE9-dihe-na | 157.62, -145.94 | APE8-dihe-in | -123.75, 129.22 | APE8-rot-in | 300.73 | APE67-dihe-in | -59.05, -19.44 | -46.41, -52.49 | APE12-dist-in | 8.134 | APE11-dist-in | 11.198 | APE10-dist-in | 5.604 | APE9-dist-in | 3.787 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | B | 617 | 593 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7lv3 | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4VB | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Active | DFGin | 6.191 | 14.848 | BLAminus | -117.12, 164.99 | 68.84, 100.49 | -114.63, 44.2 | 282.85, 73.02 | -69.55, -49.58 | in-in | in | 9.876 | Saltbr-in | 3.02 | HRD-in | -85.46, -53.89 | 74.22, -39.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.744 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.05, 169.08 | APE9-dihe-na | 104.88, 162.74 | APE8-dihe-in | -71.34, 125.86 | APE8-rot-in | 297.46 | APE67-dihe-in | -57.61, -28.56 | -42.75, -43.02 | APE12-dist-in | 8.264 | APE11-dist-in | 11.663 | APE10-dist-in | 6.268 | APE9-dist-in | 5.216 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | B | 469 | 464 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4v | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| AF-Q13976-K1A | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 6.271 | 14.18 | BLAminus | -115.7, -171.89 | 41.6, 86.13 | -92.63, 18.96 | 285.01, 78.59 | -59.54, -30.9 | in-in | in | 9.607 | Saltbr-in | 2.712 | HRD-in | -90.69, -50.22 | 66.05, 7.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.881 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.15, 172.71 | APE9-dihe-na | 108.43, 171.02 | APE8-dihe-in | -80.49, 129.57 | APE8-rot-in | 300.74 | APE67-dihe-in | -68.04, -21.28 | -48.8, -41.85 | APE12-dist-in | 8.214 | APE11-dist-in | 11.197 | APE10-dist-in | 5.629 | APE9-dist-in | 3.53 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276 | 276 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K1 | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| AF-Q13976-K3A | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 5.906 | 13.923 | BLAminus | -115.45, -173.31 | 41.39, 87.3 | -90.8, 19.58 | 282.99, 76.21 | -58.78, -31.1 | in-in | in | 9.248 | Saltbr-in | 2.714 | HRD-in | -91.17, -53.27 | 69.22, 14.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.87 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.96, 169.62 | APE9-dihe-na | 104.72, 167.78 | APE8-dihe-in | -75.94, 135.6 | APE8-rot-in | 283.37 | APE67-dihe-in | -66.68, -21.92 | -49.58, -45.16 | APE12-dist-in | 7.888 | APE11-dist-in | 11.013 | APE10-dist-in | 5.444 | APE9-dist-in | 3.338 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276 | 276 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K3 | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4UA | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.893 | 14.511 | ABAminus | -110.98, -36.23 | -113.94, 119.68 | -109.65, 38.15 | 284.57, 73.72 | -68.19, -46.47 | in-in | in | 9.753 | Saltbr-in | 2.944 | HRD-in | -80.27, -49.41 | 62.96, -11.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.82, 170.87 | APE9-dihe-na | 95.36, 163.3 | APE8-dihe-in | -65.83, 127.77 | APE8-rot-in | 297.19 | APE67-dihe-in | -61.65, -25.18 | -50.5, -36.94 | APE12-dist-in | 8.302 | APE11-dist-in | 11.55 | APE10-dist-in | 5.886 | APE9-dist-in | 5.043 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | A | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4u | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4UB | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.882 | 14.671 | ABAminus | -116.42, -27.15 | -112.65, 115.98 | -107.16, 33.12 | 284.12, 70.33 | -62.23, -46.18 | in-in | in | 9.761 | Saltbr-in | 2.921 | HRD-in | -79.97, -49.4 | 62.99, -11.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.924 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.62, 162.77 | APE9-dihe-na | 104.48, 162.22 | APE8-dihe-in | -65.39, 128.54 | APE8-rot-in | 296.86 | APE67-dihe-in | -62.65, -24.95 | -50.24, -36.77 | APE12-dist-in | 8.26 | APE11-dist-in | 11.573 | APE10-dist-in | 5.962 | APE9-dist-in | 5.014 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | B | 469 | 461 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4u | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4WA | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.203 | 14.656 | ABAminus | -120.51, -49.82 | -94.54, 125.75 | -115.2, 38.22 | 287.71, 71.79 | -69.94, -44.46 | in-in | in | 9.868 | Saltbr-in | 3.462 | HRD-in | -82.07, -59.56 | 68.33, -9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.031 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.57, 172.99 | APE9-dihe-na | 100.31, 156.35 | APE8-dihe-in | -58.55, 123.29 | APE8-rot-in | 292.59 | APE67-dihe-in | -70.67, -20.63 | -47.72, -29.8 | APE12-dist-in | 8.075 | APE11-dist-in | 11.499 | APE10-dist-in | 6.222 | APE9-dist-in | 4.918 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | A | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4w | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4WB | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.167 | 14.645 | ABAminus | -115.45, -45.68 | -98.44, 117.3 | -111.38, 33.0 | 288.61, 72.93 | -65.23, -44.36 | in-in | in | 9.884 | Saltbr-in | 3.465 | HRD-in | -84.88, -51.35 | 65.14, -16.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.986 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.45, 173.1 | APE9-dihe-na | 100.13, 155.73 | APE8-dihe-in | -59.24, 124.2 | APE8-rot-in | 292.57 | APE67-dihe-in | -70.75, -20.56 | -47.95, -29.59 | APE12-dist-in | 8.086 | APE11-dist-in | 11.514 | APE10-dist-in | 6.25 | APE9-dist-in | 4.898 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | B | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4w | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4TA | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.806 | 14.933 | ABAminus | -123.17, -29.2 | -107.96, 118.17 | -112.33, 30.1 | 285.53, 74.3 | -67.24, -29.77 | in-in | in | 9.557 | Saltbr-in | 3.38 | HRD-in | -86.67, -51.63 | 61.2, 10.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.86 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -166.89, 164.61 | APE9-dihe-na | 124.7, -170.63 | APE8-dihe-in | -100.54, 134.31 | APE8-rot-in | 302.38 | APE67-dihe-in | -67.0, -27.98 | -44.1, -43.89 | APE12-dist-in | 7.941 | APE11-dist-in | 10.713 | APE10-dist-in | 5.308 | APE9-dist-in | 3.712 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | A | 469 | 453 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4t | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4TB | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.8 | 14.811 | ABAminus | -121.38, -38.76 | -100.76, 117.73 | -112.4, 30.34 | 285.48, 73.71 | -68.75, -29.12 | in-in | in | 9.401 | Saltbr-in | 3.311 | HRD-in | -86.82, -51.68 | 61.52, 10.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.853 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -165.5, 164.27 | APE9-dihe-na | 124.32, -169.95 | APE8-dihe-in | -101.18, 134.26 | APE8-rot-in | 302.8 | APE67-dihe-in | -67.54, -26.94 | -44.3, -44.01 | APE12-dist-in | 7.957 | APE11-dist-in | 10.757 | APE10-dist-in | 5.336 | APE9-dist-in | 3.717 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | B | 469 | 453 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4t | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 7T4VA | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Inactive | DFGin | 6.18 | 14.758 | BLAminus | -117.38, 165.11 | 68.06, 101.28 | -115.37, 45.06 | 282.61, 73.13 | -70.13, -49.07 | in-in | in | 9.838 | Saltbr-in | 2.979 | HRD-in | -86.09, -51.09 | 71.54, -55.93 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.742 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -158.12, 169.74 | APE9-dihe-na | 104.56, 162.71 | APE8-dihe-in | -70.69, 125.48 | APE8-rot-in | 298.14 | APE67-dihe-in | -57.19, -28.82 | -42.61, -42.82 | APE12-dist-in | 8.556 | APE11-dist-in | 11.714 | APE10-dist-in | 6.317 | APE9-dist-out | 6.031 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | A | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4v | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 6BDLA | 337 | 671 | 671.0 | No_ligand | No_ligand | Inactive | DFGin | 5.713 | 14.513 | BLAminus | -122.27, 166.18 | 66.21, 96.03 | -109.78, 28.36 | 280.09, 66.52 | -59.53, -32.57 | in-in | in | 9.565 | Saltbr-in | 2.712 | HRD-in | -93.15, -47.43 | 77.49, -41.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.821 | ActLoopCT-out | nonTYR | APEdihe_aaini | APEdist_iiio | APE10-dihe-na | -113.85, 160.0 | APE9-dihe-na | 86.62, 160.7 | APE8-dihe-in | -68.44, 153.87 | APE8-rot-none | 999.0 | APE67-dihe-in | -67.03, -17.86 | -55.61, -25.3 | APE12-dist-in | 7.765 | APE11-dist-in | 11.218 | APE10-dist-in | 5.604 | APE9-dist-out | 6.231 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | A | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bdl | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 6C0TA | 337 | 671 | 671.0 | EE4:701 | Type1.5_Front | Inactive | DFGin | 5.9 | 14.257 | BLAminus | -131.41, 173.3 | 67.52, 81.76 | -101.27, 23.85 | 278.07, 65.63 | -65.26, -23.23 | in-in | in | 8.935 | Saltbr-in | 2.797 | HRD-in | -100.02, -51.71 | 77.78, -11.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.79 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -144.5, 158.55 | APE9-dihe-na | 107.94, 162.3 | APE8-dihe-in | -69.48, 141.18 | APE8-rot-out | 79.81 | APE67-dihe-in | -72.66, -16.0 | -52.58, -33.36 | APE12-dist-in | 7.74 | APE11-dist-in | 11.364 | APE10-dist-in | 5.987 | APE9-dist-in | 4.819 | None | TPO517 | TPO517 | XRAY | 1.98 | 0.21 | 0.244 | A | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6c0t | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| 6BDLB | 337 | 671 | 671.0 | No_ligand | No_ligand | None | DFGin | 5.757 | 14.658 | BLAminus | -124.78, 164.72 | 65.46, 95.48 | -109.07, 28.23 | 278.78, 64.61 | -59.31, -33.14 | in-in | in | 9.337 | Saltbr-in | 2.902 | HRD-in | -92.19, -47.19 | 78.26, -40.54 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.877 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_iiii | APE10-dihe-na | -122.13, 167.41 | APE9-dihe-na | 91.21, 161.43 | APE8-dihe-in | -67.63, 145.68 | APE8-rot-none | 999.0 | APE67-dihe-in | -70.27, -17.78 | -60.28, -30.02 | APE12-dist-in | 7.598 | APE11-dist-in | 11.396 | APE10-dist-in | 5.795 | APE9-dist-in | 5.468 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | B | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bdl | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| KGP1_HUMAN | 6BG2A | Q13976 | 336 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.811 | 14.714 | BLAminus | -124.15, 169.14 | 66.07, 88.5 | -100.57, 30.98 | 280.35, 66.41 | -65.35, -25.12 | in-in | in | 9.522 | Saltbr-in | 2.883 | HRD-in | -85.83, -52.95 | 73.29, 9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.851 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.93, 165.57 | APE9-dihe-na | 117.74, 172.78 | APE8-dihe-in | -83.6, 129.51 | APE8-rot-in | 307.46 | APE67-dihe-in | -66.9, -19.23 | -49.63, -41.3 | APE12-dist-in | 8.235 | APE11-dist-in | 11.512 | APE10-dist-in | 6.041 | APE9-dist-in | 4.269 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | A | 347 | 336 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 6BG2B | Q13976 | 346 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 6.001 | 13.81 | BLAminus | -122.67, 175.58 | 65.94, 84.43 | -99.77, 30.78 | 285.96, 70.42 | -64.93, -24.07 | in-in | in | 8.944 | Saltbr-in | 2.743 | HRD-in | -86.95, -52.47 | 73.99, 7.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.924 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.61, 163.67 | APE9-dihe-na | 118.96, 172.39 | APE8-dihe-in | -86.94, 131.94 | APE8-rot-in | 306.51 | APE67-dihe-in | -68.79, -20.88 | -48.58, -41.68 | APE12-dist-in | 7.826 | APE11-dist-in | 11.215 | APE10-dist-in | 5.769 | APE9-dist-in | 4.008 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | B | 347 | 326 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 6BG2C | Q13976 | 337 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.746 | 14.057 | BLAminus | -122.99, 175.03 | 65.66, 84.22 | -99.61, 30.7 | 281.62, 66.26 | -64.81, -23.57 | in-in | in | 8.742 | Saltbr-in | 2.723 | HRD-in | -85.99, -53.51 | 74.31, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.951 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.66, 165.85 | APE9-dihe-na | 118.46, 173.18 | APE8-dihe-in | -87.41, 130.75 | APE8-rot-in | 306.63 | APE67-dihe-in | -67.71, -19.03 | -48.39, -42.55 | APE12-dist-in | 7.972 | APE11-dist-in | 11.385 | APE10-dist-in | 5.857 | APE9-dist-in | 3.861 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | C | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 6BG2D | Q13976 | 344 | 671 | 671.0 | ANP:700 | ATPlike | Active | DFGin | 5.71 | 14.012 | BLAminus | -124.49, 174.79 | 65.67, 84.87 | -99.37, 30.45 | 283.38, 66.11 | -64.13, -22.3 | in-in | in | 8.754 | Saltbr-in | 2.644 | HRD-in | -85.68, -52.69 | 74.16, 8.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.92, 166.42 | APE9-dihe-na | 119.53, 169.97 | APE8-dihe-in | -84.81, 130.45 | APE8-rot-in | 305.19 | APE67-dihe-in | -66.29, -19.88 | -48.13, -43.31 | APE12-dist-in | 7.988 | APE11-dist-in | 11.327 | APE10-dist-in | 5.784 | APE9-dist-in | 3.81 | None | TPO517 | TPO517 | XRAY | 1.83 | 0.188 | 0.215 | D | 347 | 328 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bg2 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7LV3A | Q13976 | 57 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.851 | 14.036 | BLAminus | -116.97, 177.04 | 63.26, 88.72 | -106.87, 28.72 | 283.22, 63.7 | -62.95, -24.33 | in-in | in | 8.624 | Saltbr-in | 2.891 | HRD-in | -87.82, -54.22 | 74.26, 7.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.911 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.98 | APE9-dihe-na | 157.95, -145.59 | APE8-dihe-in | -124.73, 128.61 | APE8-rot-in | 299.79 | APE67-dihe-in | -58.37, -20.06 | -47.89, -51.97 | APE12-dist-in | 7.972 | APE11-dist-in | 11.057 | APE10-dist-in | 5.469 | APE9-dist-in | 3.811 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | A | 617 | 600 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7lv3 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7LV3B | Q13976 | 58 | 671 | 671.0 | ANP:60803 | ATPlike | Active | DFGin | 5.634 | 13.962 | BLAminus | -116.52, 178.28 | 63.3, 90.17 | -108.68, 29.08 | 283.48, 65.02 | -62.88, -23.93 | in-in | in | 8.883 | Saltbr-in | 2.824 | HRD-in | -86.48, -52.9 | 74.97, 7.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -152.28, 149.21 | APE9-dihe-na | 157.62, -145.94 | APE8-dihe-in | -123.75, 129.22 | APE8-rot-in | 300.73 | APE67-dihe-in | -59.05, -19.44 | -46.41, -52.49 | APE12-dist-in | 8.134 | APE11-dist-in | 11.198 | APE10-dist-in | 5.604 | APE9-dist-in | 3.787 | None | TPO517 | TPO517 | XRAY | 2.41 | 0.201 | 0.238 | B | 617 | 593 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7lv3 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.3e-83 | 286.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4VB | Q13976 | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Active | DFGin | 6.191 | 14.848 | BLAminus | -117.12, 164.99 | 68.84, 100.49 | -114.63, 44.2 | 282.85, 73.02 | -69.55, -49.58 | in-in | in | 9.876 | Saltbr-in | 3.02 | HRD-in | -85.46, -53.89 | 74.22, -39.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.744 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.05, 169.08 | APE9-dihe-na | 104.88, 162.74 | APE8-dihe-in | -71.34, 125.86 | APE8-rot-in | 297.46 | APE67-dihe-in | -57.61, -28.56 | -42.75, -43.02 | APE12-dist-in | 8.264 | APE11-dist-in | 11.663 | APE10-dist-in | 6.268 | APE9-dist-in | 5.216 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | B | 469 | 464 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4v | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | AF-Q13976-K1A | Q13976 | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 6.271 | 14.18 | BLAminus | -115.7, -171.89 | 41.6, 86.13 | -92.63, 18.96 | 285.01, 78.59 | -59.54, -30.9 | in-in | in | 9.607 | Saltbr-in | 2.712 | HRD-in | -90.69, -50.22 | 66.05, 7.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.881 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -159.15, 172.71 | APE9-dihe-na | 108.43, 171.02 | APE8-dihe-in | -80.49, 129.57 | APE8-rot-in | 300.74 | APE67-dihe-in | -68.04, -21.28 | -48.8, -41.85 | APE12-dist-in | 8.214 | APE11-dist-in | 11.197 | APE10-dist-in | 5.629 | APE9-dist-in | 3.53 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276 | 276 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K1 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | AF-Q13976-K3A | Q13976 | 352 | 627 | 671.0 | No_ligand | No_ligand | Active | DFGin | 5.906 | 13.923 | BLAminus | -115.45, -173.31 | 41.39, 87.3 | -90.8, 19.58 | 282.99, 76.21 | -58.78, -31.1 | in-in | in | 9.248 | Saltbr-in | 2.714 | HRD-in | -91.17, -53.27 | 69.22, 14.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.87 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.96, 169.62 | APE9-dihe-na | 104.72, 167.78 | APE8-dihe-in | -75.94, 135.6 | APE8-rot-in | 283.37 | APE67-dihe-in | -66.68, -21.92 | -49.58, -45.16 | APE12-dist-in | 7.888 | APE11-dist-in | 11.013 | APE10-dist-in | 5.444 | APE9-dist-in | 3.338 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 276 | 276 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | AF-Q13976-K3 | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 1.2e-84 | 289.4 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4UA | Q13976 | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.893 | 14.511 | ABAminus | -110.98, -36.23 | -113.94, 119.68 | -109.65, 38.15 | 284.57, 73.72 | -68.19, -46.47 | in-in | in | 9.753 | Saltbr-in | 2.944 | HRD-in | -80.27, -49.41 | 62.96, -11.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.82, 170.87 | APE9-dihe-na | 95.36, 163.3 | APE8-dihe-in | -65.83, 127.77 | APE8-rot-in | 297.19 | APE67-dihe-in | -61.65, -25.18 | -50.5, -36.94 | APE12-dist-in | 8.302 | APE11-dist-in | 11.55 | APE10-dist-in | 5.886 | APE9-dist-in | 5.043 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | A | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4u | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4UB | Q13976 | 205 | 671 | 671.0 | EX6:69901 | Allosteric | Inactive | DFGin | 5.882 | 14.671 | ABAminus | -116.42, -27.15 | -112.65, 115.98 | -107.16, 33.12 | 284.12, 70.33 | -62.23, -46.18 | in-in | in | 9.761 | Saltbr-in | 2.921 | HRD-in | -79.97, -49.4 | 62.99, -11.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.924 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.62, 162.77 | APE9-dihe-na | 104.48, 162.22 | APE8-dihe-in | -65.39, 128.54 | APE8-rot-in | 296.86 | APE67-dihe-in | -62.65, -24.95 | -50.24, -36.77 | APE12-dist-in | 8.26 | APE11-dist-in | 11.573 | APE10-dist-in | 5.962 | APE9-dist-in | 5.014 | None | TPO517 | TPO517 | XRAY | 1.99 | 0.216 | 0.26 | B | 469 | 461 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4u | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4WA | Q13976 | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.203 | 14.656 | ABAminus | -120.51, -49.82 | -94.54, 125.75 | -115.2, 38.22 | 287.71, 71.79 | -69.94, -44.46 | in-in | in | 9.868 | Saltbr-in | 3.462 | HRD-in | -82.07, -59.56 | 68.33, -9.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.031 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.57, 172.99 | APE9-dihe-na | 100.31, 156.35 | APE8-dihe-in | -58.55, 123.29 | APE8-rot-in | 292.59 | APE67-dihe-in | -70.67, -20.63 | -47.72, -29.8 | APE12-dist-in | 8.075 | APE11-dist-in | 11.499 | APE10-dist-in | 6.222 | APE9-dist-in | 4.918 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | A | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4w | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4WB | Q13976 | 205 | 671 | 671.0 | EZJ:69901 | Allosteric | Inactive | DFGin | 6.167 | 14.645 | ABAminus | -115.45, -45.68 | -98.44, 117.3 | -111.38, 33.0 | 288.61, 72.93 | -65.23, -44.36 | in-in | in | 9.884 | Saltbr-in | 3.465 | HRD-in | -84.88, -51.35 | 65.14, -16.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.986 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.45, 173.1 | APE9-dihe-na | 100.13, 155.73 | APE8-dihe-in | -59.24, 124.2 | APE8-rot-in | 292.57 | APE67-dihe-in | -70.75, -20.56 | -47.95, -29.59 | APE12-dist-in | 8.086 | APE11-dist-in | 11.514 | APE10-dist-in | 6.25 | APE9-dist-in | 4.898 | None | TPO517 | TPO517 | XRAY | 2.23 | 0.207 | 0.267 | B | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4w | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4TA | Q13976 | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.806 | 14.933 | ABAminus | -123.17, -29.2 | -107.96, 118.17 | -112.33, 30.1 | 285.53, 74.3 | -67.24, -29.77 | in-in | in | 9.557 | Saltbr-in | 3.38 | HRD-in | -86.67, -51.63 | 61.2, 10.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.86 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -166.89, 164.61 | APE9-dihe-na | 124.7, -170.63 | APE8-dihe-in | -100.54, 134.31 | APE8-rot-in | 302.38 | APE67-dihe-in | -67.0, -27.98 | -44.1, -43.89 | APE12-dist-in | 7.941 | APE11-dist-in | 10.713 | APE10-dist-in | 5.308 | APE9-dist-in | 3.712 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | A | 469 | 453 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4t | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4TB | Q13976 | 204 | 671 | 671.0 | PCG:60701,ATP:60702 | Allosteric,ATPlike | Inactive | DFGin | 5.8 | 14.811 | ABAminus | -121.38, -38.76 | -100.76, 117.73 | -112.4, 30.34 | 285.48, 73.71 | -68.75, -29.12 | in-in | in | 9.401 | Saltbr-in | 3.311 | HRD-in | -86.82, -51.68 | 61.52, 10.16 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.853 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -165.5, 164.27 | APE9-dihe-na | 124.32, -169.95 | APE8-dihe-in | -101.18, 134.26 | APE8-rot-in | 302.8 | APE67-dihe-in | -67.54, -26.94 | -44.3, -44.01 | APE12-dist-in | 7.957 | APE11-dist-in | 10.757 | APE10-dist-in | 5.336 | APE9-dist-in | 3.717 | None | TPO517 | TPO517 | XRAY | 2.08 | 0.19 | 0.221 | B | 469 | 453 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4t | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 7T4VA | Q13976 | 205 | 671 | 671.0 | EXZ:69901 | Allosteric | Inactive | DFGin | 6.18 | 14.758 | BLAminus | -117.38, 165.11 | 68.06, 101.28 | -115.37, 45.06 | 282.61, 73.13 | -70.13, -49.07 | in-in | in | 9.838 | Saltbr-in | 2.979 | HRD-in | -86.09, -51.09 | 71.54, -55.93 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.742 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iiio | APE10-dihe-na | -158.12, 169.74 | APE9-dihe-na | 104.56, 162.71 | APE8-dihe-in | -70.69, 125.48 | APE8-rot-in | 298.14 | APE67-dihe-in | -57.19, -28.82 | -42.61, -42.82 | APE12-dist-in | 8.556 | APE11-dist-in | 11.714 | APE10-dist-in | 6.317 | APE9-dist-out | 6.031 | None | TPO517 | TPO517 | XRAY | 2.28 | 0.197 | 0.256 | A | 469 | 467 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 7t4v | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 6.4e-84 | 287.2 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 6BDLA | Q13976 | 337 | 671 | 671.0 | No_ligand | No_ligand | Inactive | DFGin | 5.713 | 14.513 | BLAminus | -122.27, 166.18 | 66.21, 96.03 | -109.78, 28.36 | 280.09, 66.52 | -59.53, -32.57 | in-in | in | 9.565 | Saltbr-in | 2.712 | HRD-in | -93.15, -47.43 | 77.49, -41.85 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.821 | ActLoopCT-out | nonTYR | APEdihe_aaini | APEdist_iiio | APE10-dihe-na | -113.85, 160.0 | APE9-dihe-na | 86.62, 160.7 | APE8-dihe-in | -68.44, 153.87 | APE8-rot-none | 999.0 | APE67-dihe-in | -67.03, -17.86 | -55.61, -25.3 | APE12-dist-in | 7.765 | APE11-dist-in | 11.218 | APE10-dist-in | 5.604 | APE9-dist-out | 6.231 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | A | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bdl | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 6C0TA | Q13976 | 337 | 671 | 671.0 | EE4:701 | Type1.5_Front | Inactive | DFGin | 5.9 | 14.257 | BLAminus | -131.41, 173.3 | 67.52, 81.76 | -101.27, 23.85 | 278.07, 65.63 | -65.26, -23.23 | in-in | in | 8.935 | Saltbr-in | 2.797 | HRD-in | -100.02, -51.71 | 77.78, -11.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.79 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -144.5, 158.55 | APE9-dihe-na | 107.94, 162.3 | APE8-dihe-in | -69.48, 141.18 | APE8-rot-out | 79.81 | APE67-dihe-in | -72.66, -16.0 | -52.58, -33.36 | APE12-dist-in | 7.74 | APE11-dist-in | 11.364 | APE10-dist-in | 5.987 | APE9-dist-in | 4.819 | None | TPO517 | TPO517 | XRAY | 1.98 | 0.21 | 0.244 | A | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6c0t | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| KGP1_HUMAN | 6BDLB | Q13976 | 337 | 671 | 671.0 | No_ligand | No_ligand | None | DFGin | 5.757 | 14.658 | BLAminus | -124.78, 164.72 | 65.46, 95.48 | -109.07, 28.23 | 278.78, 64.61 | -59.31, -33.14 | in-in | in | 9.337 | Saltbr-in | 2.902 | HRD-in | -92.19, -47.19 | 78.26, -40.54 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.877 | ActLoopCT-none | nonTYR | APEdihe_aaini | APEdist_iiii | APE10-dihe-na | -122.13, 167.41 | APE9-dihe-na | 91.21, 161.43 | APE8-dihe-in | -67.63, 145.68 | APE8-rot-none | 999.0 | APE67-dihe-in | -70.27, -17.78 | -60.28, -30.02 | APE12-dist-in | 7.598 | APE11-dist-in | 11.396 | APE10-dist-in | 5.795 | APE9-dist-in | 5.468 | None | TPO517 | TPO517 | XRAY | 1.96 | 0.209 | 0.222 | B | 347 | 335 | 0 | 0 | 0 | 0 | [[360, 619]] | 1.0 | 6bdl | Homo sapiens | AGC_PRKG1_HUMAN | AGC | 2.6e-84 | 288.3 | 1 | 260 | 260 | 501 | 502 | 503 | 505 | 507 | 390 | 409 | 413 | 481 | 483 | 482 | 484 | 540 | 528 | 523 | 522 | 521 | 520 | 519 | 518 | 517 | 439 | cGMP-dependent protein kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|