| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK5 | 4TNDA | P34947 | 15 | 543 | 590.0 | ANP:601 | ATPlike | Active | DFGin | 5.282 | 13.1718 | BLAminus | -119.9, 173.82 | 59.88, 73.64 | -89.53, 7.87 | 278.21, 112.8 | -54.71, -33.69 | in-in | in | 9.1929 | Saltbr-in | 3.0526 | HRD-in | -67.8, -56.87 | 74.64, -6.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.25, 150.21 | APE9-dihe-na | 143.02, -165.26 | APE8-dihe-in | -107.11, 142.28 | APE8-rot-in | 314.69 | APE67-dihe-inflip | 92.64, -22.22 | -59.58, 132.94 | APE12-dist-in | 10.3015 | APE11-dist-in | 12.0563 | APE10-dist-in | 6.2302 | APE9-dist-in | 4.2553 | None | None | None | XRAY | 1.802 | 0.174 | 0.205 | A | 590.0 | 529.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 4tnd | AGC_GRK5_HUMAN | AGC | 1.1e-83 | 286.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9CKRA | P34947 | 25 | 542 | 590.0 | ATP:603 | ATPlike | Active | DFGin | 6.1719 | 12.8672 | BLAminus | -123.04, 159.77 | 67.48, 80.75 | -99.52, 5.04 | 278.7, 83.61 | -52.63, -21.44 | in-in | in | 8.5891 | Saltbr-in | 3.447 | HRD-in | -94.88, -52.49 | 68.7, 5.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9677 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.66, 167.59 | APE9-dihe-na | 129.66, -152.54 | APE8-dihe-in | -119.66, 138.17 | APE8-rot-in | 320.31 | APE67-dihe-inflip | 80.19, -6.12 | -54.38, 134.58 | APE12-dist-in | 9.8722 | APE11-dist-in | 12.2584 | APE10-dist-in | 6.5289 | APE9-dist-in | 4.1807 | D311N | None | None | XRAY | 2.8 | 0.239 | 0.286 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9ckr | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9CKSA | P34947 | 25 | 542 | 590.0 | ATP:603 | ATPlike | Active | DFGin | 6.0382 | 13.0612 | BLAminus | -123.04, 167.6 | 79.98, 56.79 | -87.17, 17.84 | 285.5, 62.72 | -70.38, -31.79 | in-in | in | 9.2222 | Saltbr-in | 2.6724 | HRD-in | -92.29, -53.7 | 68.73, 3.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9627 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.24, 151.24 | APE9-dihe-na | 138.17, -158.29 | APE8-dihe-in | -117.35, 145.2 | APE8-rot-in | 310.61 | APE67-dihe-inflip | 85.98, -22.04 | -53.6, 135.84 | APE12-dist-in | 10.6156 | APE11-dist-in | 12.4068 | APE10-dist-in | 6.5628 | APE9-dist-in | 4.2067 | D311N | None | None | XRAY | 3.08 | 0.228 | 0.28 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9cks | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | AF-P34947-K1A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 5.488 | 12.6736 | BLAminus | -115.97, -177.38 | 48.25, 67.07 | -77.66, 16.16 | 284.97, 107.27 | -63.58, -32.29 | in-in | in | 8.9664 | Saltbr-in | 2.674 | HRD-in | -81.4, -44.95 | 66.95, -1.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.35, 159.3 | APE9-dihe-na | 118.39, -174.52 | APE8-dihe-in | -94.59, 137.57 | APE8-rot-in | 303.09 | APE67-dihe-inflip | 95.72, -15.07 | -56.34, 127.54 | APE12-dist-in | 10.5047 | APE11-dist-in | 12.2476 | APE10-dist-in | 6.2146 | APE9-dist-in | 3.7811 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K1 | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | AF-P34947-K3A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 6.0217 | 12.0992 | BLAminus | -130.04, 178.69 | 50.56, 62.08 | -71.61, 20.06 | 306.44, 6.94 | -60.07, -35.44 | in-in | in | 8.5425 | Saltbr-in | 2.6154 | HRD-in | -88.42, -48.64 | 68.04, 5.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9566 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.09, 156.11 | APE9-dihe-na | 120.9, -174.14 | APE8-dihe-in | -94.05, 138.77 | APE8-rot-in | 297.52 | APE67-dihe-inflip | 92.74, -12.69 | -58.9, 127.55 | APE12-dist-in | 10.5409 | APE11-dist-in | 11.9762 | APE10-dist-in | 5.9613 | APE9-dist-in | 3.3122 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K3 | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9CKQA | P34947 | 25 | 542 | 590.0 | No_ligand | No_ligand | Active | DFGin | 6.0358 | 12.8495 | BLAminus | -128.35, 170.36 | 62.76, 74.57 | -90.62, 17.1 | 285.99, 91.78 | -58.04, -33.82 | in-in | in | 9.1056 | Saltbr-in | 2.9331 | HRD-in | -93.54, -52.56 | 67.97, 1.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9462 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.01, 171.06 | APE9-dihe-na | 118.15, -151.5 | APE8-dihe-in | -127.65, 146.62 | APE8-rot-in | 290.59 | APE67-dihe-inflip | 92.51, -30.74 | -57.11, 135.04 | APE12-dist-in | 9.7791 | APE11-dist-in | 12.0232 | APE10-dist-in | 6.1634 | APE9-dist-in | 4.1157 | D311N | None | None | XRAY | 2.7 | 0.239 | 0.294 | A | 597.0 | 490.0 | 11 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9ckq | AGC_GRK5_HUMAN | AGC | 7.5e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 4TNBA | P34947 | 15 | 543 | 590.0 | SGV:601 | Type1 | Active | DFGin | 5.1347 | 12.7402 | BLAminus | -123.5, 176.17 | 54.54, 74.38 | -84.69, 6.5 | 286.26, 112.63 | -51.75, -34.18 | in-in | in | 9.0014 | Saltbr-in | 2.528 | HRD-in | -77.08, -45.38 | 66.65, 0.7 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9615 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.74, 150.87 | APE9-dihe-na | 143.24, -163.75 | APE8-dihe-in | -110.5, 150.66 | APE8-rot-in | 315.23 | APE67-dihe-inflip | 90.86, -23.2 | -67.3, 136.98 | APE12-dist-in | 10.7387 | APE11-dist-in | 11.8747 | APE10-dist-in | 5.9463 | APE9-dist-in | 4.1118 | None | None | None | XRAY | 2.113 | 0.175 | 0.232 | A | 590.0 | 529.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 4tnb | AGC_GRK5_HUMAN | AGC | 1.1e-83 | 286.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 8UAPA | P34947 | 25 | 542 | 590.0 | W2T:601 | Type1 | Active | DFGin | 5.9519 | 12.6688 | BLAminus | -132.18, -179.7 | 52.11, 79.03 | -91.08, 7.0 | 281.21, 78.18 | -55.19, -15.59 | in-in | in | 8.933 | Saltbr-in | 2.3194 | HRD-in | -89.52, -55.99 | 69.41, 4.8 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0747 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.72, 157.14 | APE9-dihe-na | 134.87, -160.65 | APE8-dihe-in | -105.62, 143.33 | APE8-rot-in | 315.67 | APE67-dihe-inflip | 91.84, -13.85 | -56.42, 130.69 | APE12-dist-in | 10.2424 | APE11-dist-in | 12.3294 | APE10-dist-in | 6.4983 | APE9-dist-in | 4.0827 | D311N | None | None | XRAY | 2.5 | 0.229 | 0.267 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 8uap | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BREA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Active | DFGin | 6.1758 | 12.5641 | BLAminus | -128.67, 172.15 | 57.35, 77.75 | -93.22, 24.8 | 286.17, 72.14 | -63.15, -21.99 | in-in | in | 8.8006 | Saltbr-in | 2.4578 | HRD-in | -88.2, -51.09 | 67.29, 13.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1273 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.49, 165.19 | APE9-dihe-na | 125.58, -150.88 | APE8-dihe-in | -124.55, 138.39 | APE8-rot-in | 312.36 | APE67-dihe-inflip | 92.11, -16.19 | -53.44, 132.83 | APE12-dist-in | 9.9432 | APE11-dist-in | 12.1314 | APE10-dist-in | 6.3367 | APE9-dist-in | 4.1222 | D311N | None | None | XRAY | 2.8 | 0.215 | 0.26 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9bre | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRGA | P34947 | 25 | 542 | 590.0 | A1AQ6:601 | Type1 | Active | DFGin | 5.8882 | 12.7443 | BLAminus | -127.15, 171.02 | 61.76, 75.85 | -94.14, 20.1 | 287.82, 78.85 | -68.02, -19.4 | in-in | in | 9.0433 | Saltbr-in | 2.3465 | HRD-in | -85.19, -53.81 | 70.34, 12.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1046 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.02, 160.56 | APE9-dihe-na | 125.86, -158.84 | APE8-dihe-in | -113.45, 141.13 | APE8-rot-in | 318.14 | APE67-dihe-inflip | 91.69, -20.41 | -53.6, 133.88 | APE12-dist-in | 9.7697 | APE11-dist-in | 12.0735 | APE10-dist-in | 6.2186 | APE9-dist-in | 4.0834 | D311N | None | None | XRAY | 2.7 | 0.242 | 0.277 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brg | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRHA | P34947 | 25 | 542 | 590.0 | A1AQ7:601 | Type1 | Active | DFGin | 6.2132 | 12.9978 | BLAminus | -137.89, -178.33 | 53.87, 65.42 | -85.04, 16.09 | 287.04, 75.14 | -57.93, -30.07 | in-in | in | 9.3637 | Saltbr-in | 2.7875 | HRD-in | -82.45, -56.04 | 70.11, 8.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0985 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.58, 168.01 | APE9-dihe-na | 127.33, -166.12 | APE8-dihe-in | -113.88, 147.37 | APE8-rot-in | 307.37 | APE67-dihe-inflip | 89.75, -29.49 | -53.29, 136.77 | APE12-dist-in | 10.3639 | APE11-dist-in | 12.0679 | APE10-dist-in | 6.1363 | APE9-dist-in | 4.1188 | D311N | None | None | XRAY | 3.69 | 0.2 | 0.244 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brh | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRMA | P34947 | 25 | 542 | 590.0 | A1ARC:601 | Type1 | Active | DFGin | 5.9298 | 12.3198 | BLAminus | -129.54, 170.53 | 64.08, 75.97 | -94.87, 21.89 | 289.68, 68.45 | -68.62, -20.59 | in-in | in | 8.6269 | Saltbr-in | 2.5804 | HRD-in | -82.68, -56.6 | 72.77, 4.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0386 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.28, 165.33 | APE9-dihe-na | 123.74, -150.01 | APE8-dihe-in | -120.92, 138.81 | APE8-rot-in | 302.36 | APE67-dihe-inflip | 99.67, -19.1 | -52.94, 128.15 | APE12-dist-in | 9.8026 | APE11-dist-in | 12.0589 | APE10-dist-in | 6.2126 | APE9-dist-in | 4.1567 | D311N | None | None | XRAY | 2.73 | 0.234 | 0.278 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brm | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRNA | P34947 | 25 | 542 | 590.0 | A1ARD:601 | Type1 | Active | DFGin | 5.9016 | 12.7251 | BLAminus | -139.33, 159.94 | 74.16, 72.44 | -89.41, 22.16 | 291.23, 67.98 | -67.08, -25.78 | in-in | in | 8.9931 | Saltbr-in | 2.4388 | HRD-in | -78.87, -49.6 | 65.54, 8.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9886 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.44, 151.94 | APE9-dihe-na | 136.85, -155.43 | APE8-dihe-in | -118.42, 144.51 | APE8-rot-in | 301.29 | APE67-dihe-inflip | 92.21, -11.38 | -55.67, 128.36 | APE12-dist-in | 9.8088 | APE11-dist-in | 11.9957 | APE10-dist-in | 6.0938 | APE9-dist-in | 4.2745 | D311N | None | None | XRAY | 2.9 | 0.209 | 0.256 | A | 598.0 | 502.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brn | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BROA | P34947 | 25 | 542 | 590.0 | A1ARE:601 | Type1 | Active | DFGin | 5.9636 | 12.5715 | BLAminus | -128.27, -178.6 | 50.36, 73.78 | -90.4, 21.64 | 280.73, 75.17 | -69.22, -25.34 | in-in | in | 8.9064 | Saltbr-in | 2.3898 | HRD-in | -93.36, -59.82 | 68.46, 12.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8302 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.17, 167.74 | APE9-dihe-na | 123.28, -154.67 | APE8-dihe-in | -122.1, 138.71 | APE8-rot-in | 314.65 | APE67-dihe-inflip | 102.22, -12.34 | -51.46, 123.36 | APE12-dist-in | 10.2765 | APE11-dist-in | 12.3372 | APE10-dist-in | 6.4064 | APE9-dist-in | 4.0502 | D311N | None | None | XRAY | 2.8 | 0.221 | 0.271 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9bro | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9CKPA | P34947 | 1 | 542 | 590.0 | SGV:602 | Type1 | Active | DFGin | 5.3856 | 11.9802 | BLAminus | -132.87, 164.94 | 63.45, 71.08 | -85.64, 18.91 | 320.14, 3.39 | -67.22, -15.79 | in-in | in | 8.9749 | Saltbr-in | 3.5693 | HRD-in | -105.81, -54.45 | 67.93, 0.86 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.2698 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.75, 161.15 | APE9-dihe-na | 132.47, 178.17 | APE8-dihe-in | -105.33, 153.16 | APE8-rot-in | 325.98 | APE67-dihe-inflip | 78.63, 4.41 | -62.29, 127.28 | APE12-dist-in | 10.0337 | APE11-dist-in | 12.2231 | APE10-dist-in | 6.3492 | APE9-dist-in | 4.1919 | D311N | None | None | XRAY | 2.6 | 0.236 | 0.27 | A | 598.0 | 538.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9ckp | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9CKOA | P34947 | 1 | 542 | 590.0 | SGV:602 | Type1 | Inactive | DFGin | 5.808 | 12.4965 | ABAminus | -119.73, -59.76 | -93.86, 94.44 | -93.46, 16.21 | 299.92, 79.42 | -62.04, -34.62 | in-in | in | 8.4255 | Saltbr-in | 2.5213 | HRD-in | -104.67, -57.7 | 74.0, 4.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8204 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.51, 140.14 | APE9-dihe-na | 146.41, -176.34 | APE8-dihe-in | -106.42, 130.54 | APE8-rot-in | 306.78 | APE67-dihe-inflip | 81.24, -12.9 | -51.64, 146.1 | APE12-dist-in | 10.4519 | APE11-dist-in | 12.1181 | APE10-dist-in | 6.1554 | APE9-dist-in | 3.7174 | None | None | None | XRAY | 2.8 | 0.243 | 0.28 | A | 598.0 | 540.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9cko | AGC_GRK5_HUMAN | AGC | 5.9e-84 | 287.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRKA | P34947 | 25 | 542 | 590.0 | A1ARA:601 | Type1 | Inactive | DFGin | 5.9989 | 12.7247 | ABAminus | -113.29, -59.28 | -86.52, 97.64 | -98.22, 23.89 | 284.55, 73.36 | -66.95, -28.05 | in-in | in | 8.8856 | Saltbr-in | 2.3562 | HRD-in | -84.62, -58.9 | 74.96, -0.86 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0603 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.94, 168.36 | APE9-dihe-na | 122.17, -155.18 | APE8-dihe-in | -114.33, 143.85 | APE8-rot-in | 306.85 | APE67-dihe-inflip | 94.43, -16.31 | -58.15, 132.79 | APE12-dist-in | 9.6664 | APE11-dist-in | 11.7296 | APE10-dist-in | 6.0615 | APE9-dist-in | 4.128 | D311N | None | None | XRAY | 2.7 | 0.223 | 0.276 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brk | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRLA | P34947 | 25 | 542 | 590.0 | A1ARB:601 | Type1 | Inactive | DFGin | 5.6912 | 12.0225 | ABAminus | -103.25, -52.89 | -74.4, 160.18 | -158.5, 11.72 | 277.51, 97.57 | -69.39, -26.51 | in-in | in | 8.8365 | Saltbr-in | 2.3539 | HRD-in | -84.95, -56.21 | 70.99, 10.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0078 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.81, 162.58 | APE9-dihe-na | 130.63, -156.95 | APE8-dihe-in | -113.5, 144.35 | APE8-rot-in | 307.43 | APE67-dihe-inflip | 83.43, -12.88 | -53.97, 135.79 | APE12-dist-in | 9.7136 | APE11-dist-in | 11.8747 | APE10-dist-in | 6.0426 | APE9-dist-in | 4.2235 | D311N | None | None | XRAY | 2.73 | 0.231 | 0.275 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brl | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRPA | P34947 | 25 | 542 | 590.0 | A1ARF:601 | Type1 | Inactive | DFGin | 6.2535 | 12.4795 | ABAminus | -116.3, -61.02 | -91.04, 101.81 | -97.25, 10.66 | 289.92, 84.11 | -59.57, -18.7 | in-in | in | 8.9098 | Saltbr-in | 3.0371 | HRD-in | -85.07, -56.86 | 71.89, 13.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1048 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.18, 177.63 | APE9-dihe-na | 122.23, -155.28 | APE8-dihe-in | -122.73, 136.27 | APE8-rot-in | 286.0 | APE67-dihe-inflip | 100.9, -21.88 | -54.82, 128.22 | APE12-dist-in | 9.574 | APE11-dist-in | 11.9322 | APE10-dist-in | 6.253 | APE9-dist-in | 4.143 | D311N | None | None | XRAY | 2.8 | 0.245 | 0.283 | A | 598.0 | 502.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brp | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9MX2A | P34947 | 1 | 542 | 590.0 | SGV:60601 | Type1 | Inactive | DFGin | 5.5284 | 11.483 | BLAminus | -134.92, 166.93 | 57.12, 70.75 | -87.84, 20.9 | 322.36, 5.46 | -68.95, -14.98 | in-out | in | 8.3529 | Saltbr-out | 3.6263 | HRD-in | -110.96, -57.41 | 68.72, 2.93 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.3639 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.2, 161.4 | APE9-dihe-na | 129.58, 177.82 | APE8-dihe-in | -100.27, 150.38 | APE8-rot-in | 311.4 | APE67-dihe-inflip | 86.26, -1.66 | -66.59, 129.67 | APE12-dist-in | 10.1545 | APE11-dist-in | 12.3907 | APE10-dist-in | 6.5105 | APE9-dist-in | 4.1735 | D311N | None | None | XRAY | 3.9 | 0.284 | 0.346 | A | 599.0 | 538.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9mx2 | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 6PJXA | P34947 | 1 | 542 | 590.0 | SGV:60601 | Type1 | Inactive | DFGin | 5.2367 | 11.8767 | None | -101.92, -82.66 | -75.73, 114.06 | -96.27, 14.0 | 297.14, 3.15 | -60.02, -23.28 | in-in | in | 8.7999 | Saltbr-in | 2.3601 | HRD-in | -81.73, -51.04 | 76.16, -8.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8132 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.38, 158.39 | APE9-dihe-na | 127.63, -164.44 | APE8-dihe-in | -112.45, 140.59 | APE8-rot-in | 303.57 | APE67-dihe-inflip | 81.94, -9.46 | -52.3, 137.55 | APE12-dist-in | 9.8463 | APE11-dist-in | 11.9422 | APE10-dist-in | 6.1145 | APE9-dist-in | 4.4639 | E104K,R304H,G438E | None | None | XRAY | 1.96 | 0.197 | 0.23 | A | 591.0 | 542.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 6pjx | AGC_GRK5_HUMAN | AGC | 1.1e-83 | 286.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 8UAQA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Inactive | DFGin | 6.0198 | 12.8412 | None | -112.48, -65.82 | -86.97, 96.33 | -93.06, 17.75 | 286.66, 70.13 | -64.2, -19.76 | in-in | in | 9.3335 | Saltbr-in | 3.3688 | HRD-in | -90.24, -57.5 | 70.99, -0.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0372 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.56, 170.13 | APE9-dihe-na | 119.68, -157.85 | APE8-dihe-in | -112.7, 143.6 | APE8-rot-in | 314.4 | APE67-dihe-inflip | 89.64, -4.73 | -59.54, 131.81 | APE12-dist-in | 9.916 | APE11-dist-in | 12.1019 | APE10-dist-in | 6.3064 | APE9-dist-in | 4.1737 | D311N | None | None | XRAY | 2.8 | 0.232 | 0.277 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 8uaq | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRFA | P34947 | 25 | 542 | 590.0 | A1AQ5:601 | Type1 | Inactive | DFGin | 6.2131 | 12.8852 | None | -116.13, -75.08 | -76.38, 97.42 | -93.08, 20.96 | 275.91, 78.29 | -67.65, -17.42 | in-in | in | 9.0758 | Saltbr-in | 2.4746 | HRD-in | -89.29, -49.76 | 68.56, 5.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0583 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.67, 152.28 | APE9-dihe-na | 135.63, -159.61 | APE8-dihe-in | -113.28, 137.14 | APE8-rot-in | 304.0 | APE67-dihe-inflip | 86.51, -10.19 | -50.9, 134.51 | APE12-dist-in | 9.9844 | APE11-dist-in | 12.0653 | APE10-dist-in | 6.2254 | APE9-dist-in | 4.1192 | D311N | None | None | XRAY | 2.84 | 0.224 | 0.277 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brf | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRIA | P34947 | 25 | 542 | 590.0 | A1AQ8:601 | Type1 | Inactive | DFGin | 5.7901 | 12.7141 | None | -118.56, -79.42 | -70.93, 91.99 | -85.99, 18.72 | 271.5, 67.77 | -66.54, -25.08 | in-in | in | 8.8021 | Saltbr-in | 2.6488 | HRD-in | -85.77, -46.41 | 67.52, 4.46 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1673 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.68, 145.74 | APE9-dihe-na | 145.19, -146.92 | APE8-dihe-in | -122.56, 141.77 | APE8-rot-in | 306.39 | APE67-dihe-inflip | 92.75, -9.14 | -56.37, 130.7 | APE12-dist-in | 10.1331 | APE11-dist-in | 12.2149 | APE10-dist-in | 6.5714 | APE9-dist-in | 4.2246 | D311N | None | None | XRAY | 2.9 | 0.217 | 0.26 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9bri | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | 9BRJA | P34947 | 25 | 542 | 590.0 | A1AQ9:601 | Type1 | Inactive | DFGin | 5.7352 | 12.6187 | None | -115.77, -57.96 | -84.12, 93.88 | -92.94, 12.58 | 279.31, 72.41 | -59.97, -23.3 | in-in | in | 9.0567 | Saltbr-in | 2.377 | HRD-in | -83.8, -57.51 | 72.28, 3.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1163 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.79, 160.14 | APE9-dihe-na | 133.68, -150.07 | APE8-dihe-in | -119.54, 137.2 | APE8-rot-in | 310.18 | APE67-dihe-inflip | 98.77, -19.66 | -54.34, 129.82 | APE12-dist-in | 9.7235 | APE11-dist-in | 12.1088 | APE10-dist-in | 6.4144 | APE9-dist-in | 4.1673 | D311N | None | None | XRAY | 2.8 | 0.239 | 0.273 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brj | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK5 | GRK5_BOVIN | 4WNKA | P43249 | 24 | 541 | 590.0 | 453:60701 | Type1.5_Front | Inactive | DFGin | 6.2666 | 12.7972 | ABAminus | -122.04, -4.62 | -137.77, 133.15 | -132.09, 26.08 | 277.95, 69.95 | -56.52, -33.29 | in-in | in | 8.4843 | Saltbr-in | 2.7813 | HRD-in | -75.83, -57.19 | 76.27, -3.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0303 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.86, 160.08 | APE9-dihe-na | 138.36, -161.11 | APE8-dihe-in | -117.24, 138.85 | APE8-rot-in | 306.21 | APE67-dihe-inflip | 84.72, -13.63 | -52.7, 138.28 | APE12-dist-in | 10.076 | APE11-dist-in | 11.9507 | APE10-dist-in | 6.1011 | APE9-dist-in | 3.9199 | None | None | None | XRAY | 2.42 | 0.196 | 0.243 | A | 598.0 | 499.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 4wnk | Bos taurus | AGC_GRK5_BOVIN | AGC | 2.2e-84 | 288.8 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 4TNDA | P34947 | 15 | 543 | 590.0 | ANP:601 | ATPlike | Active | DFGin | 5.282 | 13.1718 | BLAminus | -119.9, 173.82 | 59.88, 73.64 | -89.53, 7.87 | 278.21, 112.8 | -54.71, -33.69 | in-in | in | 9.1929 | Saltbr-in | 3.0526 | HRD-in | -67.8, -56.87 | 74.64, -6.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.944 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.25, 150.21 | APE9-dihe-na | 143.02, -165.26 | APE8-dihe-in | -107.11, 142.28 | APE8-rot-in | 314.69 | APE67-dihe-inflip | 92.64, -22.22 | -59.58, 132.94 | APE12-dist-in | 10.3015 | APE11-dist-in | 12.0563 | APE10-dist-in | 6.2302 | APE9-dist-in | 4.2553 | None | None | None | XRAY | 1.802 | 0.174 | 0.205 | A | 590.0 | 529.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 4tnd | Homo sapiens | AGC_GRK5_HUMAN | AGC | 1.1e-83 | 286.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9CKRA | P34947 | 25 | 542 | 590.0 | ATP:603 | ATPlike | Active | DFGin | 6.1719 | 12.8672 | BLAminus | -123.04, 159.77 | 67.48, 80.75 | -99.52, 5.04 | 278.7, 83.61 | -52.63, -21.44 | in-in | in | 8.5891 | Saltbr-in | 3.447 | HRD-in | -94.88, -52.49 | 68.7, 5.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9677 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.66, 167.59 | APE9-dihe-na | 129.66, -152.54 | APE8-dihe-in | -119.66, 138.17 | APE8-rot-in | 320.31 | APE67-dihe-inflip | 80.19, -6.12 | -54.38, 134.58 | APE12-dist-in | 9.8722 | APE11-dist-in | 12.2584 | APE10-dist-in | 6.5289 | APE9-dist-in | 4.1807 | D311N | None | None | XRAY | 2.8 | 0.239 | 0.286 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9ckr | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9CKSA | P34947 | 25 | 542 | 590.0 | ATP:603 | ATPlike | Active | DFGin | 6.0382 | 13.0612 | BLAminus | -123.04, 167.6 | 79.98, 56.79 | -87.17, 17.84 | 285.5, 62.72 | -70.38, -31.79 | in-in | in | 9.2222 | Saltbr-in | 2.6724 | HRD-in | -92.29, -53.7 | 68.73, 3.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9627 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.24, 151.24 | APE9-dihe-na | 138.17, -158.29 | APE8-dihe-in | -117.35, 145.2 | APE8-rot-in | 310.61 | APE67-dihe-inflip | 85.98, -22.04 | -53.6, 135.84 | APE12-dist-in | 10.6156 | APE11-dist-in | 12.4068 | APE10-dist-in | 6.5628 | APE9-dist-in | 4.2067 | D311N | None | None | XRAY | 3.08 | 0.228 | 0.28 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9cks | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | AF-P34947-K1A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 5.488 | 12.6736 | BLAminus | -115.97, -177.38 | 48.25, 67.07 | -77.66, 16.16 | 284.97, 107.27 | -63.58, -32.29 | in-in | in | 8.9664 | Saltbr-in | 2.674 | HRD-in | -81.4, -44.95 | 66.95, -1.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.35, 159.3 | APE9-dihe-na | 118.39, -174.52 | APE8-dihe-in | -94.59, 137.57 | APE8-rot-in | 303.09 | APE67-dihe-inflip | 95.72, -15.07 | -56.34, 127.54 | APE12-dist-in | 10.5047 | APE11-dist-in | 12.2476 | APE10-dist-in | 6.2146 | APE9-dist-in | 3.7811 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K1 | Homo sapiens | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | AF-P34947-K3A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 6.0217 | 12.0992 | BLAminus | -130.04, 178.69 | 50.56, 62.08 | -71.61, 20.06 | 306.44, 6.94 | -60.07, -35.44 | in-in | in | 8.5425 | Saltbr-in | 2.6154 | HRD-in | -88.42, -48.64 | 68.04, 5.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9566 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.09, 156.11 | APE9-dihe-na | 120.9, -174.14 | APE8-dihe-in | -94.05, 138.77 | APE8-rot-in | 297.52 | APE67-dihe-inflip | 92.74, -12.69 | -58.9, 127.55 | APE12-dist-in | 10.5409 | APE11-dist-in | 11.9762 | APE10-dist-in | 5.9613 | APE9-dist-in | 3.3122 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K3 | Homo sapiens | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9CKQA | P34947 | 25 | 542 | 590.0 | No_ligand | No_ligand | Active | DFGin | 6.0358 | 12.8495 | BLAminus | -128.35, 170.36 | 62.76, 74.57 | -90.62, 17.1 | 285.99, 91.78 | -58.04, -33.82 | in-in | in | 9.1056 | Saltbr-in | 2.9331 | HRD-in | -93.54, -52.56 | 67.97, 1.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9462 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.01, 171.06 | APE9-dihe-na | 118.15, -151.5 | APE8-dihe-in | -127.65, 146.62 | APE8-rot-in | 290.59 | APE67-dihe-inflip | 92.51, -30.74 | -57.11, 135.04 | APE12-dist-in | 9.7791 | APE11-dist-in | 12.0232 | APE10-dist-in | 6.1634 | APE9-dist-in | 4.1157 | D311N | None | None | XRAY | 2.7 | 0.239 | 0.294 | A | 597.0 | 490.0 | 11 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9ckq | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.5e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 4TNBA | P34947 | 15 | 543 | 590.0 | SGV:601 | Type1 | Active | DFGin | 5.1347 | 12.7402 | BLAminus | -123.5, 176.17 | 54.54, 74.38 | -84.69, 6.5 | 286.26, 112.63 | -51.75, -34.18 | in-in | in | 9.0014 | Saltbr-in | 2.528 | HRD-in | -77.08, -45.38 | 66.65, 0.7 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9615 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.74, 150.87 | APE9-dihe-na | 143.24, -163.75 | APE8-dihe-in | -110.5, 150.66 | APE8-rot-in | 315.23 | APE67-dihe-inflip | 90.86, -23.2 | -67.3, 136.98 | APE12-dist-in | 10.7387 | APE11-dist-in | 11.8747 | APE10-dist-in | 5.9463 | APE9-dist-in | 4.1118 | None | None | None | XRAY | 2.113 | 0.175 | 0.232 | A | 590.0 | 529.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 4tnb | Homo sapiens | AGC_GRK5_HUMAN | AGC | 1.1e-83 | 286.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 8UAPA | P34947 | 25 | 542 | 590.0 | W2T:601 | Type1 | Active | DFGin | 5.9519 | 12.6688 | BLAminus | -132.18, -179.7 | 52.11, 79.03 | -91.08, 7.0 | 281.21, 78.18 | -55.19, -15.59 | in-in | in | 8.933 | Saltbr-in | 2.3194 | HRD-in | -89.52, -55.99 | 69.41, 4.8 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0747 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.72, 157.14 | APE9-dihe-na | 134.87, -160.65 | APE8-dihe-in | -105.62, 143.33 | APE8-rot-in | 315.67 | APE67-dihe-inflip | 91.84, -13.85 | -56.42, 130.69 | APE12-dist-in | 10.2424 | APE11-dist-in | 12.3294 | APE10-dist-in | 6.4983 | APE9-dist-in | 4.0827 | D311N | None | None | XRAY | 2.5 | 0.229 | 0.267 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 8uap | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BREA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Active | DFGin | 6.1758 | 12.5641 | BLAminus | -128.67, 172.15 | 57.35, 77.75 | -93.22, 24.8 | 286.17, 72.14 | -63.15, -21.99 | in-in | in | 8.8006 | Saltbr-in | 2.4578 | HRD-in | -88.2, -51.09 | 67.29, 13.94 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1273 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.49, 165.19 | APE9-dihe-na | 125.58, -150.88 | APE8-dihe-in | -124.55, 138.39 | APE8-rot-in | 312.36 | APE67-dihe-inflip | 92.11, -16.19 | -53.44, 132.83 | APE12-dist-in | 9.9432 | APE11-dist-in | 12.1314 | APE10-dist-in | 6.3367 | APE9-dist-in | 4.1222 | D311N | None | None | XRAY | 2.8 | 0.215 | 0.26 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9bre | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRGA | P34947 | 25 | 542 | 590.0 | A1AQ6:601 | Type1 | Active | DFGin | 5.8882 | 12.7443 | BLAminus | -127.15, 171.02 | 61.76, 75.85 | -94.14, 20.1 | 287.82, 78.85 | -68.02, -19.4 | in-in | in | 9.0433 | Saltbr-in | 2.3465 | HRD-in | -85.19, -53.81 | 70.34, 12.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1046 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.02, 160.56 | APE9-dihe-na | 125.86, -158.84 | APE8-dihe-in | -113.45, 141.13 | APE8-rot-in | 318.14 | APE67-dihe-inflip | 91.69, -20.41 | -53.6, 133.88 | APE12-dist-in | 9.7697 | APE11-dist-in | 12.0735 | APE10-dist-in | 6.2186 | APE9-dist-in | 4.0834 | D311N | None | None | XRAY | 2.7 | 0.242 | 0.277 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brg | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRHA | P34947 | 25 | 542 | 590.0 | A1AQ7:601 | Type1 | Active | DFGin | 6.2132 | 12.9978 | BLAminus | -137.89, -178.33 | 53.87, 65.42 | -85.04, 16.09 | 287.04, 75.14 | -57.93, -30.07 | in-in | in | 9.3637 | Saltbr-in | 2.7875 | HRD-in | -82.45, -56.04 | 70.11, 8.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0985 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -104.58, 168.01 | APE9-dihe-na | 127.33, -166.12 | APE8-dihe-in | -113.88, 147.37 | APE8-rot-in | 307.37 | APE67-dihe-inflip | 89.75, -29.49 | -53.29, 136.77 | APE12-dist-in | 10.3639 | APE11-dist-in | 12.0679 | APE10-dist-in | 6.1363 | APE9-dist-in | 4.1188 | D311N | None | None | XRAY | 3.69 | 0.2 | 0.244 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brh | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRMA | P34947 | 25 | 542 | 590.0 | A1ARC:601 | Type1 | Active | DFGin | 5.9298 | 12.3198 | BLAminus | -129.54, 170.53 | 64.08, 75.97 | -94.87, 21.89 | 289.68, 68.45 | -68.62, -20.59 | in-in | in | 8.6269 | Saltbr-in | 2.5804 | HRD-in | -82.68, -56.6 | 72.77, 4.07 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0386 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.28, 165.33 | APE9-dihe-na | 123.74, -150.01 | APE8-dihe-in | -120.92, 138.81 | APE8-rot-in | 302.36 | APE67-dihe-inflip | 99.67, -19.1 | -52.94, 128.15 | APE12-dist-in | 9.8026 | APE11-dist-in | 12.0589 | APE10-dist-in | 6.2126 | APE9-dist-in | 4.1567 | D311N | None | None | XRAY | 2.73 | 0.234 | 0.278 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brm | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRNA | P34947 | 25 | 542 | 590.0 | A1ARD:601 | Type1 | Active | DFGin | 5.9016 | 12.7251 | BLAminus | -139.33, 159.94 | 74.16, 72.44 | -89.41, 22.16 | 291.23, 67.98 | -67.08, -25.78 | in-in | in | 8.9931 | Saltbr-in | 2.4388 | HRD-in | -78.87, -49.6 | 65.54, 8.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9886 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.44, 151.94 | APE9-dihe-na | 136.85, -155.43 | APE8-dihe-in | -118.42, 144.51 | APE8-rot-in | 301.29 | APE67-dihe-inflip | 92.21, -11.38 | -55.67, 128.36 | APE12-dist-in | 9.8088 | APE11-dist-in | 11.9957 | APE10-dist-in | 6.0938 | APE9-dist-in | 4.2745 | D311N | None | None | XRAY | 2.9 | 0.209 | 0.256 | A | 598.0 | 502.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brn | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BROA | P34947 | 25 | 542 | 590.0 | A1ARE:601 | Type1 | Active | DFGin | 5.9636 | 12.5715 | BLAminus | -128.27, -178.6 | 50.36, 73.78 | -90.4, 21.64 | 280.73, 75.17 | -69.22, -25.34 | in-in | in | 8.9064 | Saltbr-in | 2.3898 | HRD-in | -93.36, -59.82 | 68.46, 12.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8302 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.17, 167.74 | APE9-dihe-na | 123.28, -154.67 | APE8-dihe-in | -122.1, 138.71 | APE8-rot-in | 314.65 | APE67-dihe-inflip | 102.22, -12.34 | -51.46, 123.36 | APE12-dist-in | 10.2765 | APE11-dist-in | 12.3372 | APE10-dist-in | 6.4064 | APE9-dist-in | 4.0502 | D311N | None | None | XRAY | 2.8 | 0.221 | 0.271 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9bro | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9CKPA | P34947 | 1 | 542 | 590.0 | SGV:602 | Type1 | Active | DFGin | 5.3856 | 11.9802 | BLAminus | -132.87, 164.94 | 63.45, 71.08 | -85.64, 18.91 | 320.14, 3.39 | -67.22, -15.79 | in-in | in | 8.9749 | Saltbr-in | 3.5693 | HRD-in | -105.81, -54.45 | 67.93, 0.86 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.2698 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.75, 161.15 | APE9-dihe-na | 132.47, 178.17 | APE8-dihe-in | -105.33, 153.16 | APE8-rot-in | 325.98 | APE67-dihe-inflip | 78.63, 4.41 | -62.29, 127.28 | APE12-dist-in | 10.0337 | APE11-dist-in | 12.2231 | APE10-dist-in | 6.3492 | APE9-dist-in | 4.1919 | D311N | None | None | XRAY | 2.6 | 0.236 | 0.27 | A | 598.0 | 538.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9ckp | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9CKOA | P34947 | 1 | 542 | 590.0 | SGV:602 | Type1 | Inactive | DFGin | 5.808 | 12.4965 | ABAminus | -119.73, -59.76 | -93.86, 94.44 | -93.46, 16.21 | 299.92, 79.42 | -62.04, -34.62 | in-in | in | 8.4255 | Saltbr-in | 2.5213 | HRD-in | -104.67, -57.7 | 74.0, 4.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8204 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.51, 140.14 | APE9-dihe-na | 146.41, -176.34 | APE8-dihe-in | -106.42, 130.54 | APE8-rot-in | 306.78 | APE67-dihe-inflip | 81.24, -12.9 | -51.64, 146.1 | APE12-dist-in | 10.4519 | APE11-dist-in | 12.1181 | APE10-dist-in | 6.1554 | APE9-dist-in | 3.7174 | None | None | None | XRAY | 2.8 | 0.243 | 0.28 | A | 598.0 | 540.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9cko | Homo sapiens | AGC_GRK5_HUMAN | AGC | 5.9e-84 | 287.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRKA | P34947 | 25 | 542 | 590.0 | A1ARA:601 | Type1 | Inactive | DFGin | 5.9989 | 12.7247 | ABAminus | -113.29, -59.28 | -86.52, 97.64 | -98.22, 23.89 | 284.55, 73.36 | -66.95, -28.05 | in-in | in | 8.8856 | Saltbr-in | 2.3562 | HRD-in | -84.62, -58.9 | 74.96, -0.86 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0603 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.94, 168.36 | APE9-dihe-na | 122.17, -155.18 | APE8-dihe-in | -114.33, 143.85 | APE8-rot-in | 306.85 | APE67-dihe-inflip | 94.43, -16.31 | -58.15, 132.79 | APE12-dist-in | 9.6664 | APE11-dist-in | 11.7296 | APE10-dist-in | 6.0615 | APE9-dist-in | 4.128 | D311N | None | None | XRAY | 2.7 | 0.223 | 0.276 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brk | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRLA | P34947 | 25 | 542 | 590.0 | A1ARB:601 | Type1 | Inactive | DFGin | 5.6912 | 12.0225 | ABAminus | -103.25, -52.89 | -74.4, 160.18 | -158.5, 11.72 | 277.51, 97.57 | -69.39, -26.51 | in-in | in | 8.8365 | Saltbr-in | 2.3539 | HRD-in | -84.95, -56.21 | 70.99, 10.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0078 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.81, 162.58 | APE9-dihe-na | 130.63, -156.95 | APE8-dihe-in | -113.5, 144.35 | APE8-rot-in | 307.43 | APE67-dihe-inflip | 83.43, -12.88 | -53.97, 135.79 | APE12-dist-in | 9.7136 | APE11-dist-in | 11.8747 | APE10-dist-in | 6.0426 | APE9-dist-in | 4.2235 | D311N | None | None | XRAY | 2.73 | 0.231 | 0.275 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brl | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRPA | P34947 | 25 | 542 | 590.0 | A1ARF:601 | Type1 | Inactive | DFGin | 6.2535 | 12.4795 | ABAminus | -116.3, -61.02 | -91.04, 101.81 | -97.25, 10.66 | 289.92, 84.11 | -59.57, -18.7 | in-in | in | 8.9098 | Saltbr-in | 3.0371 | HRD-in | -85.07, -56.86 | 71.89, 13.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1048 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.18, 177.63 | APE9-dihe-na | 122.23, -155.28 | APE8-dihe-in | -122.73, 136.27 | APE8-rot-in | 286.0 | APE67-dihe-inflip | 100.9, -21.88 | -54.82, 128.22 | APE12-dist-in | 9.574 | APE11-dist-in | 11.9322 | APE10-dist-in | 6.253 | APE9-dist-in | 4.143 | D311N | None | None | XRAY | 2.8 | 0.245 | 0.283 | A | 598.0 | 502.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brp | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9MX2A | P34947 | 1 | 542 | 590.0 | SGV:60601 | Type1 | Inactive | DFGin | 5.5284 | 11.483 | BLAminus | -134.92, 166.93 | 57.12, 70.75 | -87.84, 20.9 | 322.36, 5.46 | -68.95, -14.98 | in-out | in | 8.3529 | Saltbr-out | 3.6263 | HRD-in | -110.96, -57.41 | 68.72, 2.93 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.3639 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -112.2, 161.4 | APE9-dihe-na | 129.58, 177.82 | APE8-dihe-in | -100.27, 150.38 | APE8-rot-in | 311.4 | APE67-dihe-inflip | 86.26, -1.66 | -66.59, 129.67 | APE12-dist-in | 10.1545 | APE11-dist-in | 12.3907 | APE10-dist-in | 6.5105 | APE9-dist-in | 4.1735 | D311N | None | None | XRAY | 3.9 | 0.284 | 0.346 | A | 599.0 | 538.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9mx2 | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 6PJXA | P34947 | 1 | 542 | 590.0 | SGV:60601 | Type1 | Inactive | DFGin | 5.2367 | 11.8767 | None | -101.92, -82.66 | -75.73, 114.06 | -96.27, 14.0 | 297.14, 3.15 | -60.02, -23.28 | in-in | in | 8.7999 | Saltbr-in | 2.3601 | HRD-in | -81.73, -51.04 | 76.16, -8.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8132 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.38, 158.39 | APE9-dihe-na | 127.63, -164.44 | APE8-dihe-in | -112.45, 140.59 | APE8-rot-in | 303.57 | APE67-dihe-inflip | 81.94, -9.46 | -52.3, 137.55 | APE12-dist-in | 9.8463 | APE11-dist-in | 11.9422 | APE10-dist-in | 6.1145 | APE9-dist-in | 4.4639 | E104K,R304H,G438E | None | None | XRAY | 1.96 | 0.197 | 0.23 | A | 591.0 | 542.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 6pjx | Homo sapiens | AGC_GRK5_HUMAN | AGC | 1.1e-83 | 286.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 8UAQA | P34947 | 25 | 542 | 590.0 | W3F:601 | Type1 | Inactive | DFGin | 6.0198 | 12.8412 | None | -112.48, -65.82 | -86.97, 96.33 | -93.06, 17.75 | 286.66, 70.13 | -64.2, -19.76 | in-in | in | 9.3335 | Saltbr-in | 3.3688 | HRD-in | -90.24, -57.5 | 70.99, -0.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0372 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.56, 170.13 | APE9-dihe-na | 119.68, -157.85 | APE8-dihe-in | -112.7, 143.6 | APE8-rot-in | 314.4 | APE67-dihe-inflip | 89.64, -4.73 | -59.54, 131.81 | APE12-dist-in | 9.916 | APE11-dist-in | 12.1019 | APE10-dist-in | 6.3064 | APE9-dist-in | 4.1737 | D311N | None | None | XRAY | 2.8 | 0.232 | 0.277 | A | 598.0 | 501.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 8uaq | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRFA | P34947 | 25 | 542 | 590.0 | A1AQ5:601 | Type1 | Inactive | DFGin | 6.2131 | 12.8852 | None | -116.13, -75.08 | -76.38, 97.42 | -93.08, 20.96 | 275.91, 78.29 | -67.65, -17.42 | in-in | in | 9.0758 | Saltbr-in | 2.4746 | HRD-in | -89.29, -49.76 | 68.56, 5.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0583 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.67, 152.28 | APE9-dihe-na | 135.63, -159.61 | APE8-dihe-in | -113.28, 137.14 | APE8-rot-in | 304.0 | APE67-dihe-inflip | 86.51, -10.19 | -50.9, 134.51 | APE12-dist-in | 9.9844 | APE11-dist-in | 12.0653 | APE10-dist-in | 6.2254 | APE9-dist-in | 4.1192 | D311N | None | None | XRAY | 2.84 | 0.224 | 0.277 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brf | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRIA | P34947 | 25 | 542 | 590.0 | A1AQ8:601 | Type1 | Inactive | DFGin | 5.7901 | 12.7141 | None | -118.56, -79.42 | -70.93, 91.99 | -85.99, 18.72 | 271.5, 67.77 | -66.54, -25.08 | in-in | in | 8.8021 | Saltbr-in | 2.6488 | HRD-in | -85.77, -46.41 | 67.52, 4.46 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1673 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -151.68, 145.74 | APE9-dihe-na | 145.19, -146.92 | APE8-dihe-in | -122.56, 141.77 | APE8-rot-in | 306.39 | APE67-dihe-inflip | 92.75, -9.14 | -56.37, 130.7 | APE12-dist-in | 10.1331 | APE11-dist-in | 12.2149 | APE10-dist-in | 6.5714 | APE9-dist-in | 4.2246 | D311N | None | None | XRAY | 2.9 | 0.217 | 0.26 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9bri | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| GRK5 | GRK5_HUMAN | 9BRJA | P34947 | 25 | 542 | 590.0 | A1AQ9:601 | Type1 | Inactive | DFGin | 5.7352 | 12.6187 | None | -115.77, -57.96 | -84.12, 93.88 | -92.94, 12.58 | 279.31, 72.41 | -59.97, -23.3 | in-in | in | 9.0567 | Saltbr-in | 2.377 | HRD-in | -83.8, -57.51 | 72.28, 3.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1163 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.79, 160.14 | APE9-dihe-na | 133.68, -150.07 | APE8-dihe-in | -119.54, 137.2 | APE8-rot-in | 310.18 | APE67-dihe-inflip | 98.77, -19.66 | -54.34, 129.82 | APE12-dist-in | 9.7235 | APE11-dist-in | 12.1088 | APE10-dist-in | 6.4144 | APE9-dist-in | 4.1673 | D311N | None | None | XRAY | 2.8 | 0.239 | 0.273 | A | 598.0 | 503.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 9brj | Homo sapiens | AGC_GRK5_HUMAN | AGC | 7.6e-83 | 283.7 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK5 | GRK5_BOVIN | 4WNKA | P43249 | 24 | 541 | 590.0 | 453:60701 | Type1.5_Front | Inactive | DFGin | 6.2666 | 12.7972 | ABAminus | -122.04, -4.62 | -137.77, 133.15 | -132.09, 26.08 | 277.95, 69.95 | -56.52, -33.29 | in-in | in | 8.4843 | Saltbr-in | 2.7813 | HRD-in | -75.83, -57.19 | 76.27, -3.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0303 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.86, 160.08 | APE9-dihe-na | 138.36, -161.11 | APE8-dihe-in | -117.24, 138.85 | APE8-rot-in | 306.21 | APE67-dihe-inflip | 84.72, -13.63 | -52.7, 138.28 | APE12-dist-in | 10.076 | APE11-dist-in | 11.9507 | APE10-dist-in | 6.1011 | APE9-dist-in | 3.9199 | None | None | None | XRAY | 2.42 | 0.196 | 0.243 | A | 598.0 | 499.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 4wnk | Bos taurus | AGC_GRK5_BOVIN | AGC | 2.2e-84 | 288.8 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |