| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK2 | AF-P25098-K1A | P25098 | 183 | 461 | 689.0 | No_ligand | No_ligand | Active | DFGin | 5.5622 | 13.0673 | BLAminus | -119.78, 178.65 | 52.56, 73.94 | -83.8, 16.08 | 278.33, 71.82 | -60.8, -26.56 | in-in | in | 8.5412 | Saltbr-in | 2.5893 | HRD-in | -80.89, -42.45 | 65.72, -2.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8867 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.3, 128.35 | APE9-dihe-na | 142.96, -178.54 | APE8-dihe-in | -87.49, 128.15 | APE8-rot-in | 299.26 | APE67-dihe-inflip | 86.45, 0.9 | -52.52, 136.47 | APE12-dist-in | 10.2338 | APE11-dist-in | 12.0254 | APE10-dist-in | 6.0827 | APE9-dist-in | 3.2902 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P25098-K1 | AGC_GRK2_HUMAN | AGC | 4.6e-78 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | AF-P25098-K3A | P25098 | 183 | 461 | 689.0 | No_ligand | No_ligand | Active | DFGin | 5.32 | 12.8527 | BLAminus | -125.8, 178.57 | 52.64, 62.07 | -71.89, 17.23 | 286.12, 88.29 | -61.97, -25.79 | in-in | in | 8.526 | Saltbr-in | 2.5505 | HRD-in | -86.05, -43.82 | 69.06, 3.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8478 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.98, 153.8 | APE9-dihe-na | 127.94, -163.33 | APE8-dihe-in | -103.05, 123.69 | APE8-rot-in | 298.01 | APE67-dihe-inflip | 89.53, 2.54 | -53.74, 129.56 | APE12-dist-in | 9.0608 | APE11-dist-in | 11.855 | APE10-dist-in | 5.9514 | APE9-dist-in | 3.215 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P25098-K3 | AGC_GRK2_HUMAN | AGC | 4.6e-78 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5UVCA | P25098 | 30 | 536 | 689.0 | 8PV:600 | Type1 | Active | DFGin | 5.6459 | 13.252 | BLAminus | -111.93, -175.1 | 48.95, 84.95 | -96.99, 16.3 | 272.95, 81.76 | -56.56, -35.65 | in-in | in | 8.6666 | Saltbr-in | 2.7965 | HRD-in | -90.5, -43.84 | 74.99, -18.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.796 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.43, 134.46 | APE9-dihe-na | 148.93, -160.88 | APE8-dihe-in | -114.94, 135.94 | APE8-rot-in | 305.71 | APE67-dihe-in | -77.66, 1.58 | -57.71, -38.48 | APE12-dist-in | 10.2466 | APE11-dist-in | 12.0267 | APE10-dist-in | 6.1071 | APE9-dist-in | 3.357 | None | None | None | XRAY | 2.65 | 0.217 | 0.26 | A | 547.0 | 457.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5uvc | AGC_GRK2_HUMAN | AGC | 3.7e-77 | 268.3 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5UKLA | P25098 | 31 | 671 | 689.0 | SIX:702 | Type1 | Active | DFGin | 5.5525 | 13.4547 | BLAminus | -136.15, 162.37 | 65.35, 90.8 | -91.1, 16.16 | 287.26, 80.35 | -44.51, -43.27 | in-in | in | 8.9358 | Saltbr-in | 2.6266 | HRD-in | -76.69, -51.69 | 80.53, -28.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9516 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.59, 119.44 | APE9-dihe-na | 167.03, -154.05 | APE8-dihe-in | -112.97, 140.97 | APE8-rot-in | 300.02 | APE67-dihe-in | -82.52, 9.1 | -61.65, -35.94 | APE12-dist-in | 10.2011 | APE11-dist-in | 11.7419 | APE10-dist-in | 5.8434 | APE9-dist-in | 3.7561 | S670A | None | None | XRAY | 2.15 | 0.184 | 0.228 | A | 642.0 | 630.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5ukl | AGC_GRK2_HUMAN | AGC | 5.4e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5HE1A | P25098 | 29 | 668 | 689.0 | ZS2:701 | Type1 | Active | DFGin | 5.7607 | 13.0739 | BLAminus | -136.45, 161.18 | 63.18, 92.12 | -104.97, 24.32 | 295.58, 61.08 | -54.15, -39.68 | in-in | in | 8.6303 | Saltbr-in | 2.9645 | HRD-in | -75.81, -60.39 | 89.65, -39.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9796 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -121.97, 100.73 | APE9-dihe-na | -165.78, -165.71 | APE8-dihe-in | -91.06, 127.63 | APE8-rot-in | 294.03 | APE67-dihe-inflip | 109.39, -17.56 | -55.26, 129.29 | APE12-dist-in | 10.3336 | APE11-dist-in | 12.1323 | APE10-dist-in | 6.3113 | APE9-dist-in | 3.8934 | S670A | None | None | XRAY | 3.15 | 0.172 | 0.25 | A | 642.0 | 618.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he1 | AGC_GRK2_HUMAN | AGC | 5.4e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 6C2YA | P25098 | 30 | 668 | 689.0 | EJS:701 | Type1 | Active | DFGin | 5.2477 | 13.1313 | BLAminus | -133.84, 169.51 | 63.67, 85.91 | -91.46, 28.99 | 286.98, 69.09 | -62.06, -46.79 | in-in | in | 8.7773 | Saltbr-in | 2.6025 | HRD-in | -71.8, -47.67 | 74.94, -21.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.2292 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -121.32, 147.42 | APE9-dihe-na | 138.79, -162.57 | APE8-dihe-in | -110.7, 130.32 | APE8-rot-in | 292.69 | APE67-dihe-inflip | 102.38, -19.78 | -58.44, 136.12 | APE12-dist-in | 9.5744 | APE11-dist-in | 11.9534 | APE10-dist-in | 5.9756 | APE9-dist-in | 3.4531 | S670A | None | None | XRAY | 2.74 | 0.247 | 0.292 | A | 689.0 | 617.0 | 2 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 6c2y | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 4MK0A | P25098 | 30 | 668 | 689.0 | 29X:60702 | Type1 | Active | DFGin | 5.0222 | 12.5575 | BLAminus | -114.3, 159.32 | 62.47, 95.12 | -99.09, 26.84 | 314.83, 15.76 | -55.23, -46.17 | in-in | in | 8.7964 | Saltbr-in | 3.2929 | HRD-in | -74.82, -46.73 | 65.86, 15.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8054 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.22, 138.8 | APE9-dihe-na | 140.75, -169.47 | APE8-dihe-in | -90.2, 139.3 | APE8-rot-in | 300.61 | APE67-dihe-inflip | 101.57, -12.83 | -69.61, 140.12 | APE12-dist-in | 10.2148 | APE11-dist-in | 12.1548 | APE10-dist-in | 6.4186 | APE9-dist-in | 3.2251 | None | None | None | XRAY | 2.4 | 0.179 | 0.238 | A | 640.0 | 630.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 4mk0 | AGC_GRK2_HUMAN | AGC | 5.3e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 7K7LA | P25098 | 30 | 668 | 689.0 | W4D:702 | Type1 | Active | DFGin | 5.3464 | 13.407 | BLAminus | -120.75, 157.11 | 65.86, 85.74 | -89.44, 20.76 | 269.03, 169.7 | -63.22, -26.35 | in-in | in | 9.0879 | Saltbr-in | 2.7438 | HRD-in | -83.14, -50.8 | 72.46, -22.33 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8171 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.43, 143.89 | APE9-dihe-na | 130.34, -178.78 | APE8-dihe-in | -87.05, 140.86 | APE8-rot-in | 300.91 | APE67-dihe-inflip | 101.09, -17.29 | -67.82, 137.73 | APE12-dist-in | 10.8032 | APE11-dist-in | 12.386 | APE10-dist-in | 6.4429 | APE9-dist-in | 3.6669 | None | None | None | XRAY | 2.539 | 0.203 | 0.244 | A | 640.0 | 616.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 7k7l | AGC_GRK2_HUMAN | AGC | 5.3e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 7K7ZA | P25098 | 30 | 668 | 689.0 | W4G:701 | Type1 | Active | DFGin | 5.2276 | 13.2609 | BLAminus | -131.21, 159.45 | 58.45, 84.74 | -81.51, 17.96 | 273.45, 160.93 | -49.98, -46.53 | in-in | in | 9.1503 | Saltbr-in | 2.6057 | HRD-in | -69.84, -65.83 | 82.28, 6.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8192 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.88, 129.42 | APE9-dihe-na | 151.42, -156.98 | APE8-dihe-in | -108.77, 134.07 | APE8-rot-in | 292.67 | APE67-dihe-inflip | 104.4, -17.1 | -64.98, 131.58 | APE12-dist-in | 12.6858 | APE11-dist-in | 12.3085 | APE10-dist-in | 6.4852 | APE9-dist-in | 3.2799 | None | None | None | XRAY | 2.606 | 0.207 | 0.262 | A | 640.0 | 625.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 7k7z | AGC_GRK2_HUMAN | AGC | 5.3e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 3V5WA | P25098 | 30 | 668 | 689.0 | 8PR:701 | Type1 | Active | DFGin | 5.1567 | 12.9917 | BLAminus | -135.73, 166.74 | 63.47, 84.47 | -90.01, 8.76 | 284.89, 155.02 | -55.83, -32.04 | in-in | in | 8.9278 | Saltbr-in | 2.9291 | HRD-in | -75.87, -48.67 | 77.13, -26.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9163 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.74, 132.09 | APE9-dihe-na | 148.62, -167.37 | APE8-dihe-in | -102.18, 145.22 | APE8-rot-in | 303.37 | APE67-dihe-in | -68.83, -4.06 | -70.22, -32.86 | APE12-dist-in | 10.0001 | APE11-dist-in | 11.8614 | APE10-dist-in | 5.9102 | APE9-dist-in | 3.6888 | None | None | None | XRAY | 2.07 | 0.196 | 0.247 | A | 689.0 | 623.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3v5w | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 4PNKA | P25098 | 30 | 668 | 689.0 | KZQ:701 | Type1 | Active | DFGin | 5.6956 | 13.3098 | BLAminus | -131.92, 150.67 | 73.23, 94.18 | -104.4, 20.24 | 276.38, 72.07 | -49.27, -48.99 | in-in | in | 8.8686 | Saltbr-in | 2.8918 | HRD-in | -75.55, -46.99 | 79.65, -28.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0292 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.99, 151.18 | APE9-dihe-na | 153.42, -170.47 | APE8-dihe-in | -97.49, 139.43 | APE8-rot-in | 296.18 | APE67-dihe-inflip | 99.83, -0.25 | -68.24, 133.65 | APE12-dist-in | 10.1099 | APE11-dist-in | 11.7313 | APE10-dist-in | 5.9401 | APE9-dist-in | 3.5973 | None | None | None | XRAY | 2.56 | 0.194 | 0.259 | A | 689.0 | 625.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 4pnk | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5WG3A | P25098 | 30 | 668 | 689.0 | AFM:701 | Type1 | Active | DFGin | 5.2508 | 12.6657 | BLAminus | -140.32, 170.95 | 56.45, 82.96 | -87.3, 21.74 | 311.79, 174.31 | -59.6, -38.71 | in-in | in | 8.9483 | Saltbr-in | 2.8469 | HRD-in | -82.02, -43.09 | 42.08, 25.46 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.2573 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.78, 131.07 | APE9-dihe-na | 153.01, -166.14 | APE8-dihe-in | -107.02, 132.83 | APE8-rot-in | 302.54 | APE67-dihe-inflip | 106.87, -20.46 | -62.02, 131.15 | APE12-dist-in | 10.4276 | APE11-dist-in | 11.7933 | APE10-dist-in | 5.9015 | APE9-dist-in | 3.3586 | None | None | None | XRAY | 2.896 | 0.201 | 0.248 | A | 689.0 | 618.0 | 5 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5wg3 | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5WG4A | P25098 | 31 | 668 | 689.0 | AFV:701 | Type1 | Active | DFGin | 5.3057 | 12.6907 | BLAminus | -133.5, 178.66 | 54.05, 81.87 | -91.99, 21.58 | 286.03, 73.35 | -64.61, -41.57 | in-in | in | 8.5477 | Saltbr-in | 3.1343 | HRD-in | -85.74, -45.07 | 68.56, -11.01 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1518 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.91, 129.47 | APE9-dihe-na | 146.73, -166.55 | APE8-dihe-in | -108.67, 131.04 | APE8-rot-in | 299.39 | APE67-dihe-inflip | 106.48, -11.49 | -60.32, 128.85 | APE12-dist-in | 10.344 | APE11-dist-in | 11.9796 | APE10-dist-in | 6.1426 | APE9-dist-in | 3.4618 | None | None | None | XRAY | 2.31 | 0.235 | 0.279 | A | 689.0 | 621.0 | 2 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5wg4 | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5WG5A | P25098 | 30 | 668 | 689.0 | ZSO:701 | Type1 | Active | DFGin | 5.4509 | 13.0103 | BLAminus | -128.14, 171.88 | 56.74, 83.28 | -91.88, 32.75 | 279.7, 68.89 | -65.05, -47.67 | in-in | in | 8.625 | Saltbr-in | 2.6505 | HRD-in | -77.29, -47.13 | 67.77, -1.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9921 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.64, 131.79 | APE9-dihe-na | 147.8, -171.59 | APE8-dihe-in | -95.05, 124.52 | APE8-rot-in | 297.6 | APE67-dihe-inflip | 97.31, -8.85 | -62.05, 143.11 | APE12-dist-in | 10.4905 | APE11-dist-in | 12.0444 | APE10-dist-in | 6.1933 | APE9-dist-in | 3.3918 | None | None | None | XRAY | 3.1 | 0.19 | 0.232 | A | 689.0 | 617.0 | 3 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5wg5 | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5UUUA | P25098 | 31 | 538 | 689.0 | QRW:601 | Type1.5_Front | Active | DFGin | 5.4075 | 13.1234 | BLAminus | -119.49, 148.71 | 76.08, 97.29 | -99.15, 18.56 | 280.12, 88.0 | -55.68, -33.52 | in-in | in | 8.3995 | Saltbr-in | 2.9715 | HRD-in | -81.09, -44.67 | 78.9, -27.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1511 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.83, 137.94 | APE9-dihe-na | 132.21, -156.97 | APE8-dihe-in | -118.83, 132.35 | APE8-rot-in | 311.27 | APE67-dihe-inflip | 94.82, -15.58 | -63.39, 132.05 | APE12-dist-in | 9.9224 | APE11-dist-in | 11.8901 | APE10-dist-in | 5.9307 | APE9-dist-in | 3.5492 | None | None | None | XRAY | 2.7 | 0.215 | 0.257 | A | 547.0 | 414.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5uuu | AGC_GRK2_HUMAN | AGC | 3.7e-77 | 268.3 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 5UKKA | P25098 | 30 | 667 | 689.0 | 8DJ:702 | Type1.5_Front | Active | DFGin | 5.4401 | 12.8485 | BLAminus | -148.52, 179.61 | 57.76, 73.54 | -87.98, 8.97 | 274.06, 69.08 | -60.04, -18.89 | in-in | in | 8.2709 | Saltbr-in | 2.6689 | HRD-in | -76.24, -37.94 | 75.49, -51.75 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9425 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.39, 145.94 | APE9-dihe-na | 143.2, -151.45 | APE8-dihe-in | -131.14, 141.32 | APE8-rot-in | 299.97 | APE67-dihe-in | -67.12, -33.98 | -48.24, -30.82 | APE12-dist-in | 9.6352 | APE11-dist-in | 11.8188 | APE10-dist-in | 5.8456 | APE9-dist-in | 4.1568 | S670A | None | None | XRAY | 2.6 | 0.224 | 0.281 | A | 642.0 | 613.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5ukk | AGC_GRK2_HUMAN | AGC | 5.4e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 6U7CA | P25098 | 30 | 669 | 689.0 | Q1Y:701 | Type1.5_Front | Active | DFGin | 5.0615 | 12.4543 | BLAminus | -136.54, 170.55 | 57.52, 81.77 | -86.77, 20.22 | 308.16, 7.53 | -58.1, -34.47 | in-in | in | 9.0498 | Saltbr-in | 2.5429 | HRD-in | -72.35, -46.72 | 70.07, -13.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.3699 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.84, 132.95 | APE9-dihe-na | 147.35, -168.5 | APE8-dihe-in | -105.63, 128.22 | APE8-rot-in | 297.44 | APE67-dihe-inflip | 124.86, -14.55 | -55.92, 113.23 | APE12-dist-in | 10.2056 | APE11-dist-in | 12.016 | APE10-dist-in | 6.0719 | APE9-dist-in | 3.4845 | None | None | None | XRAY | 2.44 | 0.237 | 0.262 | A | 689.0 | 631.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 6u7c | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 3CIKA | P25098 | 29 | 669 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2003 | 12.94 | None | -113.38, -84.39 | -77.41, 106.5 | -85.28, 5.55 | 272.59, 132.44 | -54.41, -34.31 | in-in | in | 8.589 | Saltbr-in | 2.8304 | HRD-in | -65.15, -43.87 | 69.81, -16.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8246 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.98, 126.35 | APE9-dihe-na | 141.75, -159.25 | APE8-dihe-in | -111.86, 146.5 | APE8-rot-in | 310.14 | APE67-dihe-in | -81.13, 3.2 | -68.81, -30.14 | APE12-dist-in | 10.9775 | APE11-dist-in | 12.0726 | APE10-dist-in | 6.4171 | APE9-dist-in | 3.5873 | None | None | None | XRAY | 2.75 | 0.208 | 0.269 | A | 689.0 | 619.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3cik | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 7PWDA | P25098 | 27 | 668 | 689.0 | 8DS:701 | Type1 | Inactive | DFGin | 5.2813 | 12.9593 | None | -103.27, -91.53 | -83.38, 120.45 | -98.95, 11.01 | 295.2, 164.91 | -62.17, -28.84 | in-in | in | 8.7988 | Saltbr-in | 2.8227 | HRD-in | -68.27, -51.69 | 76.81, -22.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8256 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.66, 145.62 | APE9-dihe-na | 123.25, -162.48 | APE8-dihe-in | -110.04, 138.42 | APE8-rot-in | 305.66 | APE67-dihe-inflip | 98.02, -22.76 | -65.28, 137.62 | APE12-dist-in | 10.312 | APE11-dist-in | 11.9263 | APE10-dist-in | 6.0194 | APE9-dist-in | 3.3652 | S670A | None | None | XRAY | 2.6 | 0.192 | 0.23 | A | 697.0 | 621.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 7pwd | AGC_GRK2_HUMAN | AGC | 6.4e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 3KRWA | P25098 | 30 | 671 | 689.0 | BA1:690 | Type1 | Inactive | DFGin | 5.4431 | 12.512 | None | -124.43, -69.99 | -70.72, 103.06 | -103.15, 18.82 | 281.61, 154.56 | -63.74, -46.79 | in-in | in | 8.9073 | Saltbr-in | 2.6208 | HRD-in | -80.35, -50.37 | 71.38, -3.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7506 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -91.68, 135.05 | APE9-dihe-na | 136.51, -178.33 | APE8-dihe-in | -97.44, 143.34 | APE8-rot-in | 311.93 | APE67-dihe-in | -81.84, -17.98 | -65.75, -16.48 | APE12-dist-in | 9.7737 | APE11-dist-in | 11.7182 | APE10-dist-in | 5.7635 | APE9-dist-in | 3.2649 | None | None | None | XRAY | 2.9 | 0.216 | 0.265 | A | 688.0 | 618.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3krw | AGC_GRK2_HUMAN | AGC | 6.2e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | 3KRXA | P25098 | 30 | 671 | 689.0 | BA1:690 | Type1 | Inactive | DFGin | 5.4192 | 12.8449 | None | -125.39, -77.94 | -69.67, 105.65 | -105.64, 33.0 | 281.38, 161.16 | -76.22, -41.07 | in-in | in | 9.1809 | Saltbr-in | 2.9453 | HRD-in | -81.43, -47.09 | 70.32, -0.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7468 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.75, 134.45 | APE9-dihe-na | 144.08, -171.31 | APE8-dihe-in | -102.11, 138.21 | APE8-rot-in | 300.04 | APE67-dihe-in | -91.64, -15.37 | -61.65, -13.24 | APE12-dist-in | 9.2638 | APE11-dist-in | 11.5714 | APE10-dist-in | 5.62 | APE9-dist-in | 3.2776 | None | None | None | XRAY | 3.1 | 0.232 | 0.27 | A | 688.0 | 618.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3krx | AGC_GRK2_HUMAN | AGC | 6.2e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK2 | ARBK1_BOVIN | 5HE0A | P21146 | 30 | 668 | 689.0 | 453:701 | Type1 | Active | DFGin | 5.2592 | 13.1171 | BLAminus | -137.72, 161.16 | 67.72, 86.34 | -84.98, 14.88 | 287.85, 80.12 | -42.13, -60.12 | in-in | in | 8.4671 | Saltbr-in | 2.8678 | HRD-in | -68.65, -49.34 | 77.87, -29.18 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8588 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.25, 120.14 | APE9-dihe-na | 171.2, -142.82 | APE8-dihe-in | -122.87, 132.42 | APE8-rot-in | 285.63 | APE67-dihe-inflip | 113.92, -33.46 | -57.37, 128.9 | APE12-dist-in | 10.1735 | APE11-dist-in | 11.7707 | APE10-dist-in | 5.8798 | APE9-dist-in | 3.5488 | S670A | None | None | XRAY | 2.56 | 0.205 | 0.264 | A | 641.0 | 621.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he0 | Bos taurus | AGC_GRK2_BOVIN | AGC | 5.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 5HE2A | P21146 | 30 | 668 | 689.0 | F0S:701 | Type1 | Active | DFGin | 5.2664 | 13.4322 | BLAminus | -127.84, 162.02 | 76.97, 74.62 | -82.13, 19.63 | 285.89, 54.35 | -44.91, -55.91 | in-in | in | 8.6986 | Saltbr-in | 2.6713 | HRD-in | -87.07, -48.72 | 79.5, -27.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.886 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.3, 135.41 | APE9-dihe-na | 128.88, -173.45 | APE8-dihe-in | -85.86, 172.32 | APE8-rot-in | 301.72 | APE67-dihe-in | -88.54, 16.07 | -85.52, -45.68 | APE12-dist-in | 10.698 | APE11-dist-in | 11.9311 | APE10-dist-in | 5.9928 | APE9-dist-in | 3.7816 | S670A | None | None | XRAY | 2.79 | 0.202 | 0.277 | A | 641.0 | 628.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he2 | Bos taurus | AGC_GRK2_BOVIN | AGC | 5.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 5HE3A | P21146 | 30 | 670 | 689.0 | FF1:702 | Type1 | Active | DFGin | 5.4706 | 13.1124 | BLAminus | -130.61, 154.77 | 82.75, 74.09 | -80.19, 15.36 | 283.76, 73.33 | -31.6, -75.24 | in-in | in | 8.613 | Saltbr-in | 2.7525 | HRD-in | -66.32, -31.89 | 63.86, -19.84 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9166 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.68, 142.9 | APE9-dihe-na | 127.74, 174.69 | APE8-dihe-in | -90.13, 145.29 | APE8-rot-in | 301.32 | APE67-dihe-inflip | 112.74, -14.85 | -68.46, 126.13 | APE12-dist-in | 10.205 | APE11-dist-in | 11.7078 | APE10-dist-in | 5.915 | APE9-dist-in | 3.371 | None | None | None | XRAY | 2.74 | 0.198 | 0.257 | A | 641.0 | 623.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he3 | Bos taurus | AGC_GRK2_BOVIN | AGC | 5.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 5UKMA | P21146 | 31 | 669 | 689.0 | T0E:701 | Type1 | Active | DFGin | 5.5585 | 13.1317 | BLAminus | -130.36, 150.32 | 61.48, 90.2 | -96.51, 21.64 | 296.35, 62.89 | -55.13, -59.92 | in-in | in | 9.0172 | Saltbr-in | 2.7861 | HRD-in | -71.89, -48.96 | 73.51, -73.8 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1669 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.94, 135.34 | APE9-dihe-na | 121.47, 173.74 | APE8-dihe-in | -77.03, 143.73 | APE8-rot-in | 316.68 | APE67-dihe-in | -68.91, -23.51 | -68.56, -33.79 | APE12-dist-in | 10.3025 | APE11-dist-in | 11.6096 | APE10-dist-in | 5.8336 | APE9-dist-in | 5.3132 | S670A | None | None | XRAY | 3.03 | 0.2 | 0.252 | A | 695.0 | 621.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5ukm | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7B | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1989 | 12.4485 | ABAminus | -130.8, -59.92 | -98.26, 108.63 | -91.58, -9.04 | 306.19, 95.69 | -36.4, -48.74 | in-out | in | 8.8033 | Saltbr-out | 4.6419 | HRD-in | -77.09, -44.3 | 73.62, -27.39 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7591 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.17, 125.32 | APE9-dihe-na | 152.82, 174.56 | APE8-dihe-in | -87.32, 142.62 | APE8-rot-in | 313.75 | APE67-dihe-in | -64.86, -36.54 | -62.56, -29.46 | APE12-dist-in | 9.8182 | APE11-dist-in | 11.5603 | APE10-dist-in | 5.5731 | APE9-dist-in | 4.0361 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | B | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 8JPBG | P21146 | 2 | 659 | 689.0 | STU:701 | Type1 | Inactive | DFGin | 5.5082 | 12.2136 | ABAminus | -113.28, -56.44 | -93.74, 100.06 | -93.25, 26.0 | 307.53, 3.55 | -63.32, -43.2 | in-out | in | 8.9334 | Saltbr-out | 4.2174 | HRD-out | -93.17, 87.64 | -73.74, -9.71 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7258 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.15, 142.89 | APE9-dihe-na | 142.59, -152.8 | APE8-dihe-in | -124.3, 137.48 | APE8-rot-in | 299.05 | APE67-dihe-inflip | 90.41, -8.27 | -58.8, 137.88 | APE12-dist-in | 9.9025 | APE11-dist-in | 12.0099 | APE10-dist-in | 6.0986 | APE9-dist-in | 3.6298 | A292P,R295I,S455D | None | None | EM | 3.07 | 999.0 | 999.0 | G | 688.0 | 658.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 8jpb | Bos taurus | AGC_GRK2_BOVIN | AGC | 1.7e-76 | 267.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 8JPCG | P21146 | 2 | 659 | 689.0 | STU:701 | Type1 | Inactive | DFGin | 5.385 | 12.1571 | ABAminus | -113.22, -56.58 | -93.6, 101.44 | -93.44, 27.48 | 306.81, 9.79 | -63.79, -45.14 | in-out | in | 8.9895 | Saltbr-out | 4.6535 | HRD-out | -92.62, 94.67 | -75.66, -35.58 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.6526 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.27, 130.92 | APE9-dihe-na | 162.84, -151.71 | APE8-dihe-in | -129.7, 130.81 | APE8-rot-in | 302.62 | APE67-dihe-inflip | 97.48, -17.5 | -57.09, 134.46 | APE12-dist-in | 9.7132 | APE11-dist-in | 11.9892 | APE10-dist-in | 5.9887 | APE9-dist-in | 4.3163 | A292P,R295I,S455D | None | None | EM | 3.07 | 999.0 | 999.0 | G | 688.0 | 658.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 8jpc | Bos taurus | AGC_GRK2_BOVIN | AGC | 1.7e-76 | 267.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 8JPDG | P21146 | 2 | 659 | 689.0 | STU:701 | Type1 | Inactive | DFGin | 5.3847 | 12.1571 | ABAminus | -113.24, -56.55 | -93.57, 101.39 | -93.42, 27.53 | 306.84, 9.79 | -63.78, -45.12 | in-out | in | 8.9895 | Saltbr-out | 4.6534 | HRD-out | -92.61, 94.65 | -75.65, -35.58 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.6534 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.32, 130.92 | APE9-dihe-na | 162.83, -151.7 | APE8-dihe-in | -129.72, 130.82 | APE8-rot-in | 302.58 | APE67-dihe-inflip | 97.48, -17.49 | -57.11, 134.43 | APE12-dist-in | 9.7137 | APE11-dist-in | 11.9887 | APE10-dist-in | 5.9885 | APE9-dist-in | 4.3171 | A292P,R295I,S455D | None | None | EM | 2.81 | 999.0 | 999.0 | G | 688.0 | 658.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 8jpd | Bos taurus | AGC_GRK2_BOVIN | AGC | 1.7e-76 | 267.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1OMWA | P21146 | 29 | 668 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.448 | 13.0685 | None | -112.27, -91.9 | -67.18, 126.78 | -99.0, 7.24 | 286.96, 109.41 | -44.09, -46.49 | in-in | in | 8.9372 | Saltbr-in | 3.4107 | HRD-in | -73.22, -52.41 | 80.02, -28.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8622 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.71, 128.56 | APE9-dihe-na | 124.77, -168.54 | APE8-dihe-in | -89.28, 150.91 | APE8-rot-in | 295.71 | APE67-dihe-in | -77.59, -9.92 | -72.81, -27.02 | APE12-dist-in | 10.5885 | APE11-dist-in | 11.8774 | APE10-dist-in | 6.1942 | APE9-dist-in | 3.5029 | S670A | None | None | XRAY | 2.5 | 0.216 | 0.252 | A | 689.0 | 614.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1omw | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7A | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2239 | 12.3565 | None | -125.66, -66.29 | -94.21, 107.11 | -86.73, -10.11 | 307.87, 97.53 | -38.26, -47.46 | in-out | in | 8.8531 | Saltbr-out | 4.6372 | HRD-in | -74.94, -45.18 | 74.24, -26.22 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7715 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.74, 123.21 | APE9-dihe-na | 155.55, 174.57 | APE8-dihe-in | -86.11, 141.22 | APE8-rot-in | 314.43 | APE67-dihe-in | -66.31, -34.76 | -64.21, -27.3 | APE12-dist-in | 9.8313 | APE11-dist-in | 11.5432 | APE10-dist-in | 5.5926 | APE9-dist-in | 3.9926 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | A | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7C | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2163 | 12.2674 | None | -130.34, -66.38 | -92.79, 106.85 | -85.97, -13.2 | 309.12, 95.06 | -35.96, -48.47 | in-out | in | 8.8136 | Saltbr-out | 4.7358 | HRD-in | -75.86, -48.89 | 75.97, -29.41 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.721 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.29, 128.8 | APE9-dihe-na | 145.96, 173.8 | APE8-dihe-in | -87.44, 141.12 | APE8-rot-in | 314.72 | APE67-dihe-in | -67.09, -36.43 | -60.22, -25.52 | APE12-dist-in | 9.7747 | APE11-dist-in | 11.5691 | APE10-dist-in | 5.6074 | APE9-dist-in | 4.0582 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | C | 689.0 | 607.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7D | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2341 | 12.3436 | None | -128.88, -67.33 | -92.65, 105.41 | -87.88, -10.71 | 307.83, 96.53 | -37.49, -49.46 | in-out | in | 8.801 | Saltbr-out | 4.7459 | HRD-in | -72.13, -45.13 | 72.62, -27.86 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7633 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.27, 125.22 | APE9-dihe-na | 149.39, 173.11 | APE8-dihe-in | -84.5, 141.69 | APE8-rot-in | 315.18 | APE67-dihe-in | -66.11, -35.98 | -62.26, -27.83 | APE12-dist-in | 9.7362 | APE11-dist-in | 11.4974 | APE10-dist-in | 5.5333 | APE9-dist-in | 4.0286 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | D | 689.0 | 599.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 2BCJA | P21146 | 28 | 667 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1531 | 12.3754 | None | -114.23, -125.71 | -23.26, 91.28 | -81.33, 0.62 | 275.63, 158.44 | -51.51, -42.54 | in-in | in | 8.6198 | Saltbr-in | 2.6334 | HRD-in | -86.19, -45.87 | 70.94, -23.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7186 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.73, 137.19 | APE9-dihe-na | 118.03, -177.98 | APE8-dihe-in | -75.0, 121.63 | APE8-rot-in | 302.92 | APE67-dihe-in | -97.57, -19.7 | -76.89, 19.37 | APE12-dist-in | 11.0395 | APE11-dist-in | 11.9406 | APE10-dist-in | 6.0057 | APE9-dist-in | 3.715 | S670A | None | None | XRAY | 3.061 | 0.236 | 0.292 | A | 689.0 | 624.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 2bcj | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3UZSA | P21146 | 29 | 671 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.731 | 11.1485 | None | -107.21, -110.21 | -68.72, 97.64 | -52.38, -56.06 | 299.08, 3.09 | 42.56, -75.63 | in-out | in | 9.0047 | Saltbr-out | 3.9207 | HRD-in | -77.33, -41.02 | 60.69, 32.77 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.5286 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -98.18, 142.14 | APE9-dihe-na | 139.16, 169.96 | APE8-dihe-in | -74.03, 124.78 | APE8-rot-in | 315.02 | APE67-dihe-out | 166.07, -43.85 | -59.08, 78.84 | APE12-dist-in | 10.2386 | APE11-dist-in | 12.0969 | APE10-dist-in | 6.31 | APE9-dist-in | 3.5138 | S670A | None | None | XRAY | 4.52 | 0.188 | 0.268 | A | 689.0 | 609.0 | 20 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3uzs | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3UZTA | P21146 | 30 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.216 | 12.499 | None | -94.28, -95.77 | -83.37, 90.84 | -54.75, -37.85 | 271.69, 47.64 | -2.65, -69.38 | in-out | in | 8.8257 | Saltbr-out | 5.0807 | HRD-in | -72.79, -37.98 | 67.02, -27.54 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.085 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -99.51, 148.65 | APE9-dihe-na | 138.76, 168.6 | APE8-dihe-in | -71.39, 126.55 | APE8-rot-in | 294.92 | APE67-dihe-in | -71.95, -17.71 | -54.34, -25.29 | APE12-dist-in | 9.5328 | APE11-dist-in | 12.0098 | APE10-dist-in | 5.9885 | APE9-dist-in | 3.8685 | S670A | None | None | XRAY | 3.51 | 0.22 | 0.317 | A | 689.0 | 586.0 | 12 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3uzt | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3PSCA | P21146 | 29 | 668 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4842 | 12.8251 | None | -112.1, -116.4 | -50.02, 128.26 | -100.71, 13.15 | 287.53, 88.47 | -45.02, -46.74 | in-in | in | 8.8883 | Saltbr-in | 3.1136 | HRD-in | -73.4, -47.49 | 67.75, 0.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.59, 142.02 | APE9-dihe-na | 121.44, 174.37 | APE8-dihe-in | -79.3, 138.73 | APE8-rot-in | 323.05 | APE67-dihe-in | -80.94, 3.9 | -61.06, -31.71 | APE12-dist-in | 10.1172 | APE11-dist-in | 11.7629 | APE10-dist-in | 5.9289 | APE9-dist-in | 3.1916 | S670A | None | None | XRAY | 2.67 | 0.225 | 0.257 | A | 695.0 | 614.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3psc | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3PVUA | P21146 | 30 | 668 | 689.0 | QRW:800 | Type1 | Inactive | DFGin | 5.4293 | 12.5496 | None | -114.2, -126.97 | -29.78, 116.79 | -95.83, 7.38 | 283.37, 161.7 | -55.56, -22.85 | in-in | in | 8.7486 | Saltbr-in | 2.9863 | HRD-in | -71.34, -46.23 | 80.59, -11.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9271 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -154.26, 142.91 | APE9-dihe-na | 117.3, -165.9 | APE8-dihe-in | -102.62, 148.45 | APE8-rot-in | 314.0 | APE67-dihe-in | -77.54, 11.33 | -67.23, -35.08 | APE12-dist-in | 10.2837 | APE11-dist-in | 11.8902 | APE10-dist-in | 6.1863 | APE9-dist-in | 3.4202 | S670A | None | None | XRAY | 2.48 | 0.229 | 0.274 | A | 695.0 | 609.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3pvu | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3PVWA | P21146 | 29 | 668 | 689.0 | QRX:800 | Type1 | Inactive | DFGin | 5.249 | 12.3972 | None | -104.93, -94.33 | -60.0, 121.61 | -95.37, 6.96 | 285.31, 4.38 | -65.85, -19.47 | in-in | in | 8.7495 | Saltbr-in | 3.07 | HRD-in | -69.01, -52.71 | 78.6, -13.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9188 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.25, 142.6 | APE9-dihe-na | 127.77, 176.65 | APE8-dihe-in | -84.9, 148.79 | APE8-rot-in | 327.3 | APE67-dihe-in | -77.16, 13.46 | -65.86, -42.83 | APE12-dist-in | 10.7375 | APE11-dist-in | 12.1865 | APE10-dist-in | 6.4122 | APE9-dist-in | 3.337 | S670A | None | None | XRAY | 2.49 | 0.239 | 0.285 | A | 695.0 | 613.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3pvw | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | AF-P25098-K1A | P25098 | 183 | 461 | 689.0 | No_ligand | No_ligand | Active | DFGin | 5.5622 | 13.0673 | BLAminus | -119.78, 178.65 | 52.56, 73.94 | -83.8, 16.08 | 278.33, 71.82 | -60.8, -26.56 | in-in | in | 8.5412 | Saltbr-in | 2.5893 | HRD-in | -80.89, -42.45 | 65.72, -2.62 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8867 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.3, 128.35 | APE9-dihe-na | 142.96, -178.54 | APE8-dihe-in | -87.49, 128.15 | APE8-rot-in | 299.26 | APE67-dihe-inflip | 86.45, 0.9 | -52.52, 136.47 | APE12-dist-in | 10.2338 | APE11-dist-in | 12.0254 | APE10-dist-in | 6.0827 | APE9-dist-in | 3.2902 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P25098-K1 | Homo sapiens | AGC_GRK2_HUMAN | AGC | 4.6e-78 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | AF-P25098-K3A | P25098 | 183 | 461 | 689.0 | No_ligand | No_ligand | Active | DFGin | 5.32 | 12.8527 | BLAminus | -125.8, 178.57 | 52.64, 62.07 | -71.89, 17.23 | 286.12, 88.29 | -61.97, -25.79 | in-in | in | 8.526 | Saltbr-in | 2.5505 | HRD-in | -86.05, -43.82 | 69.06, 3.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8478 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.98, 153.8 | APE9-dihe-na | 127.94, -163.33 | APE8-dihe-in | -103.05, 123.69 | APE8-rot-in | 298.01 | APE67-dihe-inflip | 89.53, 2.54 | -53.74, 129.56 | APE12-dist-in | 9.0608 | APE11-dist-in | 11.855 | APE10-dist-in | 5.9514 | APE9-dist-in | 3.215 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | AF-P25098-K3 | Homo sapiens | AGC_GRK2_HUMAN | AGC | 4.6e-78 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5UVCA | P25098 | 30 | 536 | 689.0 | 8PV:600 | Type1 | Active | DFGin | 5.6459 | 13.252 | BLAminus | -111.93, -175.1 | 48.95, 84.95 | -96.99, 16.3 | 272.95, 81.76 | -56.56, -35.65 | in-in | in | 8.6666 | Saltbr-in | 2.7965 | HRD-in | -90.5, -43.84 | 74.99, -18.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.796 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.43, 134.46 | APE9-dihe-na | 148.93, -160.88 | APE8-dihe-in | -114.94, 135.94 | APE8-rot-in | 305.71 | APE67-dihe-in | -77.66, 1.58 | -57.71, -38.48 | APE12-dist-in | 10.2466 | APE11-dist-in | 12.0267 | APE10-dist-in | 6.1071 | APE9-dist-in | 3.357 | None | None | None | XRAY | 2.65 | 0.217 | 0.26 | A | 547.0 | 457.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5uvc | Homo sapiens | AGC_GRK2_HUMAN | AGC | 3.7e-77 | 268.3 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5UKLA | P25098 | 31 | 671 | 689.0 | SIX:702 | Type1 | Active | DFGin | 5.5525 | 13.4547 | BLAminus | -136.15, 162.37 | 65.35, 90.8 | -91.1, 16.16 | 287.26, 80.35 | -44.51, -43.27 | in-in | in | 8.9358 | Saltbr-in | 2.6266 | HRD-in | -76.69, -51.69 | 80.53, -28.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9516 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.59, 119.44 | APE9-dihe-na | 167.03, -154.05 | APE8-dihe-in | -112.97, 140.97 | APE8-rot-in | 300.02 | APE67-dihe-in | -82.52, 9.1 | -61.65, -35.94 | APE12-dist-in | 10.2011 | APE11-dist-in | 11.7419 | APE10-dist-in | 5.8434 | APE9-dist-in | 3.7561 | S670A | None | None | XRAY | 2.15 | 0.184 | 0.228 | A | 642.0 | 630.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5ukl | Homo sapiens | AGC_GRK2_HUMAN | AGC | 5.4e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5HE1A | P25098 | 29 | 668 | 689.0 | ZS2:701 | Type1 | Active | DFGin | 5.7607 | 13.0739 | BLAminus | -136.45, 161.18 | 63.18, 92.12 | -104.97, 24.32 | 295.58, 61.08 | -54.15, -39.68 | in-in | in | 8.6303 | Saltbr-in | 2.9645 | HRD-in | -75.81, -60.39 | 89.65, -39.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9796 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -121.97, 100.73 | APE9-dihe-na | -165.78, -165.71 | APE8-dihe-in | -91.06, 127.63 | APE8-rot-in | 294.03 | APE67-dihe-inflip | 109.39, -17.56 | -55.26, 129.29 | APE12-dist-in | 10.3336 | APE11-dist-in | 12.1323 | APE10-dist-in | 6.3113 | APE9-dist-in | 3.8934 | S670A | None | None | XRAY | 3.15 | 0.172 | 0.25 | A | 642.0 | 618.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he1 | Homo sapiens | AGC_GRK2_HUMAN | AGC | 5.4e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 6C2YA | P25098 | 30 | 668 | 689.0 | EJS:701 | Type1 | Active | DFGin | 5.2477 | 13.1313 | BLAminus | -133.84, 169.51 | 63.67, 85.91 | -91.46, 28.99 | 286.98, 69.09 | -62.06, -46.79 | in-in | in | 8.7773 | Saltbr-in | 2.6025 | HRD-in | -71.8, -47.67 | 74.94, -21.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.2292 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -121.32, 147.42 | APE9-dihe-na | 138.79, -162.57 | APE8-dihe-in | -110.7, 130.32 | APE8-rot-in | 292.69 | APE67-dihe-inflip | 102.38, -19.78 | -58.44, 136.12 | APE12-dist-in | 9.5744 | APE11-dist-in | 11.9534 | APE10-dist-in | 5.9756 | APE9-dist-in | 3.4531 | S670A | None | None | XRAY | 2.74 | 0.247 | 0.292 | A | 689.0 | 617.0 | 2 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 6c2y | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 4MK0A | P25098 | 30 | 668 | 689.0 | 29X:60702 | Type1 | Active | DFGin | 5.0222 | 12.5575 | BLAminus | -114.3, 159.32 | 62.47, 95.12 | -99.09, 26.84 | 314.83, 15.76 | -55.23, -46.17 | in-in | in | 8.7964 | Saltbr-in | 3.2929 | HRD-in | -74.82, -46.73 | 65.86, 15.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8054 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.22, 138.8 | APE9-dihe-na | 140.75, -169.47 | APE8-dihe-in | -90.2, 139.3 | APE8-rot-in | 300.61 | APE67-dihe-inflip | 101.57, -12.83 | -69.61, 140.12 | APE12-dist-in | 10.2148 | APE11-dist-in | 12.1548 | APE10-dist-in | 6.4186 | APE9-dist-in | 3.2251 | None | None | None | XRAY | 2.4 | 0.179 | 0.238 | A | 640.0 | 630.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 4mk0 | Homo sapiens | AGC_GRK2_HUMAN | AGC | 5.3e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 7K7LA | P25098 | 30 | 668 | 689.0 | W4D:702 | Type1 | Active | DFGin | 5.3464 | 13.407 | BLAminus | -120.75, 157.11 | 65.86, 85.74 | -89.44, 20.76 | 269.03, 169.7 | -63.22, -26.35 | in-in | in | 9.0879 | Saltbr-in | 2.7438 | HRD-in | -83.14, -50.8 | 72.46, -22.33 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8171 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.43, 143.89 | APE9-dihe-na | 130.34, -178.78 | APE8-dihe-in | -87.05, 140.86 | APE8-rot-in | 300.91 | APE67-dihe-inflip | 101.09, -17.29 | -67.82, 137.73 | APE12-dist-in | 10.8032 | APE11-dist-in | 12.386 | APE10-dist-in | 6.4429 | APE9-dist-in | 3.6669 | None | None | None | XRAY | 2.539 | 0.203 | 0.244 | A | 640.0 | 616.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 7k7l | Homo sapiens | AGC_GRK2_HUMAN | AGC | 5.3e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 7K7ZA | P25098 | 30 | 668 | 689.0 | W4G:701 | Type1 | Active | DFGin | 5.2276 | 13.2609 | BLAminus | -131.21, 159.45 | 58.45, 84.74 | -81.51, 17.96 | 273.45, 160.93 | -49.98, -46.53 | in-in | in | 9.1503 | Saltbr-in | 2.6057 | HRD-in | -69.84, -65.83 | 82.28, 6.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8192 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.88, 129.42 | APE9-dihe-na | 151.42, -156.98 | APE8-dihe-in | -108.77, 134.07 | APE8-rot-in | 292.67 | APE67-dihe-inflip | 104.4, -17.1 | -64.98, 131.58 | APE12-dist-in | 12.6858 | APE11-dist-in | 12.3085 | APE10-dist-in | 6.4852 | APE9-dist-in | 3.2799 | None | None | None | XRAY | 2.606 | 0.207 | 0.262 | A | 640.0 | 625.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 7k7z | Homo sapiens | AGC_GRK2_HUMAN | AGC | 5.3e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 3V5WA | P25098 | 30 | 668 | 689.0 | 8PR:701 | Type1 | Active | DFGin | 5.1567 | 12.9917 | BLAminus | -135.73, 166.74 | 63.47, 84.47 | -90.01, 8.76 | 284.89, 155.02 | -55.83, -32.04 | in-in | in | 8.9278 | Saltbr-in | 2.9291 | HRD-in | -75.87, -48.67 | 77.13, -26.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9163 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.74, 132.09 | APE9-dihe-na | 148.62, -167.37 | APE8-dihe-in | -102.18, 145.22 | APE8-rot-in | 303.37 | APE67-dihe-in | -68.83, -4.06 | -70.22, -32.86 | APE12-dist-in | 10.0001 | APE11-dist-in | 11.8614 | APE10-dist-in | 5.9102 | APE9-dist-in | 3.6888 | None | None | None | XRAY | 2.07 | 0.196 | 0.247 | A | 689.0 | 623.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3v5w | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 4PNKA | P25098 | 30 | 668 | 689.0 | KZQ:701 | Type1 | Active | DFGin | 5.6956 | 13.3098 | BLAminus | -131.92, 150.67 | 73.23, 94.18 | -104.4, 20.24 | 276.38, 72.07 | -49.27, -48.99 | in-in | in | 8.8686 | Saltbr-in | 2.8918 | HRD-in | -75.55, -46.99 | 79.65, -28.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0292 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.99, 151.18 | APE9-dihe-na | 153.42, -170.47 | APE8-dihe-in | -97.49, 139.43 | APE8-rot-in | 296.18 | APE67-dihe-inflip | 99.83, -0.25 | -68.24, 133.65 | APE12-dist-in | 10.1099 | APE11-dist-in | 11.7313 | APE10-dist-in | 5.9401 | APE9-dist-in | 3.5973 | None | None | None | XRAY | 2.56 | 0.194 | 0.259 | A | 689.0 | 625.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 4pnk | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5WG3A | P25098 | 30 | 668 | 689.0 | AFM:701 | Type1 | Active | DFGin | 5.2508 | 12.6657 | BLAminus | -140.32, 170.95 | 56.45, 82.96 | -87.3, 21.74 | 311.79, 174.31 | -59.6, -38.71 | in-in | in | 8.9483 | Saltbr-in | 2.8469 | HRD-in | -82.02, -43.09 | 42.08, 25.46 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.2573 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.78, 131.07 | APE9-dihe-na | 153.01, -166.14 | APE8-dihe-in | -107.02, 132.83 | APE8-rot-in | 302.54 | APE67-dihe-inflip | 106.87, -20.46 | -62.02, 131.15 | APE12-dist-in | 10.4276 | APE11-dist-in | 11.7933 | APE10-dist-in | 5.9015 | APE9-dist-in | 3.3586 | None | None | None | XRAY | 2.896 | 0.201 | 0.248 | A | 689.0 | 618.0 | 5 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5wg3 | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5WG4A | P25098 | 31 | 668 | 689.0 | AFV:701 | Type1 | Active | DFGin | 5.3057 | 12.6907 | BLAminus | -133.5, 178.66 | 54.05, 81.87 | -91.99, 21.58 | 286.03, 73.35 | -64.61, -41.57 | in-in | in | 8.5477 | Saltbr-in | 3.1343 | HRD-in | -85.74, -45.07 | 68.56, -11.01 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1518 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.91, 129.47 | APE9-dihe-na | 146.73, -166.55 | APE8-dihe-in | -108.67, 131.04 | APE8-rot-in | 299.39 | APE67-dihe-inflip | 106.48, -11.49 | -60.32, 128.85 | APE12-dist-in | 10.344 | APE11-dist-in | 11.9796 | APE10-dist-in | 6.1426 | APE9-dist-in | 3.4618 | None | None | None | XRAY | 2.31 | 0.235 | 0.279 | A | 689.0 | 621.0 | 2 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5wg4 | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5WG5A | P25098 | 30 | 668 | 689.0 | ZSO:701 | Type1 | Active | DFGin | 5.4509 | 13.0103 | BLAminus | -128.14, 171.88 | 56.74, 83.28 | -91.88, 32.75 | 279.7, 68.89 | -65.05, -47.67 | in-in | in | 8.625 | Saltbr-in | 2.6505 | HRD-in | -77.29, -47.13 | 67.77, -1.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9921 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.64, 131.79 | APE9-dihe-na | 147.8, -171.59 | APE8-dihe-in | -95.05, 124.52 | APE8-rot-in | 297.6 | APE67-dihe-inflip | 97.31, -8.85 | -62.05, 143.11 | APE12-dist-in | 10.4905 | APE11-dist-in | 12.0444 | APE10-dist-in | 6.1933 | APE9-dist-in | 3.3918 | None | None | None | XRAY | 3.1 | 0.19 | 0.232 | A | 689.0 | 617.0 | 3 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5wg5 | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5UUUA | P25098 | 31 | 538 | 689.0 | QRW:601 | Type1.5_Front | Active | DFGin | 5.4075 | 13.1234 | BLAminus | -119.49, 148.71 | 76.08, 97.29 | -99.15, 18.56 | 280.12, 88.0 | -55.68, -33.52 | in-in | in | 8.3995 | Saltbr-in | 2.9715 | HRD-in | -81.09, -44.67 | 78.9, -27.11 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1511 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -108.83, 137.94 | APE9-dihe-na | 132.21, -156.97 | APE8-dihe-in | -118.83, 132.35 | APE8-rot-in | 311.27 | APE67-dihe-inflip | 94.82, -15.58 | -63.39, 132.05 | APE12-dist-in | 9.9224 | APE11-dist-in | 11.8901 | APE10-dist-in | 5.9307 | APE9-dist-in | 3.5492 | None | None | None | XRAY | 2.7 | 0.215 | 0.257 | A | 547.0 | 414.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5uuu | Homo sapiens | AGC_GRK2_HUMAN | AGC | 3.7e-77 | 268.3 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 5UKKA | P25098 | 30 | 667 | 689.0 | 8DJ:702 | Type1.5_Front | Active | DFGin | 5.4401 | 12.8485 | BLAminus | -148.52, 179.61 | 57.76, 73.54 | -87.98, 8.97 | 274.06, 69.08 | -60.04, -18.89 | in-in | in | 8.2709 | Saltbr-in | 2.6689 | HRD-in | -76.24, -37.94 | 75.49, -51.75 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9425 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.39, 145.94 | APE9-dihe-na | 143.2, -151.45 | APE8-dihe-in | -131.14, 141.32 | APE8-rot-in | 299.97 | APE67-dihe-in | -67.12, -33.98 | -48.24, -30.82 | APE12-dist-in | 9.6352 | APE11-dist-in | 11.8188 | APE10-dist-in | 5.8456 | APE9-dist-in | 4.1568 | S670A | None | None | XRAY | 2.6 | 0.224 | 0.281 | A | 642.0 | 613.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5ukk | Homo sapiens | AGC_GRK2_HUMAN | AGC | 5.4e-77 | 267.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 6U7CA | P25098 | 30 | 669 | 689.0 | Q1Y:701 | Type1.5_Front | Active | DFGin | 5.0615 | 12.4543 | BLAminus | -136.54, 170.55 | 57.52, 81.77 | -86.77, 20.22 | 308.16, 7.53 | -58.1, -34.47 | in-in | in | 9.0498 | Saltbr-in | 2.5429 | HRD-in | -72.35, -46.72 | 70.07, -13.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.3699 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.84, 132.95 | APE9-dihe-na | 147.35, -168.5 | APE8-dihe-in | -105.63, 128.22 | APE8-rot-in | 297.44 | APE67-dihe-inflip | 124.86, -14.55 | -55.92, 113.23 | APE12-dist-in | 10.2056 | APE11-dist-in | 12.016 | APE10-dist-in | 6.0719 | APE9-dist-in | 3.4845 | None | None | None | XRAY | 2.44 | 0.237 | 0.262 | A | 689.0 | 631.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 6u7c | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 3CIKA | P25098 | 29 | 669 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2003 | 12.94 | None | -113.38, -84.39 | -77.41, 106.5 | -85.28, 5.55 | 272.59, 132.44 | -54.41, -34.31 | in-in | in | 8.589 | Saltbr-in | 2.8304 | HRD-in | -65.15, -43.87 | 69.81, -16.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8246 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.98, 126.35 | APE9-dihe-na | 141.75, -159.25 | APE8-dihe-in | -111.86, 146.5 | APE8-rot-in | 310.14 | APE67-dihe-in | -81.13, 3.2 | -68.81, -30.14 | APE12-dist-in | 10.9775 | APE11-dist-in | 12.0726 | APE10-dist-in | 6.4171 | APE9-dist-in | 3.5873 | None | None | None | XRAY | 2.75 | 0.208 | 0.269 | A | 689.0 | 619.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3cik | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.3e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 7PWDA | P25098 | 27 | 668 | 689.0 | 8DS:701 | Type1 | Inactive | DFGin | 5.2813 | 12.9593 | None | -103.27, -91.53 | -83.38, 120.45 | -98.95, 11.01 | 295.2, 164.91 | -62.17, -28.84 | in-in | in | 8.7988 | Saltbr-in | 2.8227 | HRD-in | -68.27, -51.69 | 76.81, -22.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8256 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.66, 145.62 | APE9-dihe-na | 123.25, -162.48 | APE8-dihe-in | -110.04, 138.42 | APE8-rot-in | 305.66 | APE67-dihe-inflip | 98.02, -22.76 | -65.28, 137.62 | APE12-dist-in | 10.312 | APE11-dist-in | 11.9263 | APE10-dist-in | 6.0194 | APE9-dist-in | 3.3652 | S670A | None | None | XRAY | 2.6 | 0.192 | 0.23 | A | 697.0 | 621.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 7pwd | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.4e-77 | 267.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 3KRWA | P25098 | 30 | 671 | 689.0 | BA1:690 | Type1 | Inactive | DFGin | 5.4431 | 12.512 | None | -124.43, -69.99 | -70.72, 103.06 | -103.15, 18.82 | 281.61, 154.56 | -63.74, -46.79 | in-in | in | 8.9073 | Saltbr-in | 2.6208 | HRD-in | -80.35, -50.37 | 71.38, -3.06 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7506 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -91.68, 135.05 | APE9-dihe-na | 136.51, -178.33 | APE8-dihe-in | -97.44, 143.34 | APE8-rot-in | 311.93 | APE67-dihe-in | -81.84, -17.98 | -65.75, -16.48 | APE12-dist-in | 9.7737 | APE11-dist-in | 11.7182 | APE10-dist-in | 5.7635 | APE9-dist-in | 3.2649 | None | None | None | XRAY | 2.9 | 0.216 | 0.265 | A | 688.0 | 618.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3krw | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.2e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_HUMAN | 3KRXA | P25098 | 30 | 671 | 689.0 | BA1:690 | Type1 | Inactive | DFGin | 5.4192 | 12.8449 | None | -125.39, -77.94 | -69.67, 105.65 | -105.64, 33.0 | 281.38, 161.16 | -76.22, -41.07 | in-in | in | 9.1809 | Saltbr-in | 2.9453 | HRD-in | -81.43, -47.09 | 70.32, -0.2 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7468 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -83.75, 134.45 | APE9-dihe-na | 144.08, -171.31 | APE8-dihe-in | -102.11, 138.21 | APE8-rot-in | 300.04 | APE67-dihe-in | -91.64, -15.37 | -61.65, -13.24 | APE12-dist-in | 9.2638 | APE11-dist-in | 11.5714 | APE10-dist-in | 5.62 | APE9-dist-in | 3.2776 | None | None | None | XRAY | 3.1 | 0.232 | 0.27 | A | 688.0 | 618.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3krx | Homo sapiens | AGC_GRK2_HUMAN | AGC | 6.2e-77 | 267.6 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK2 | ARBK1_BOVIN | 5HE0A | P21146 | 30 | 668 | 689.0 | 453:701 | Type1 | Active | DFGin | 5.2592 | 13.1171 | BLAminus | -137.72, 161.16 | 67.72, 86.34 | -84.98, 14.88 | 287.85, 80.12 | -42.13, -60.12 | in-in | in | 8.4671 | Saltbr-in | 2.8678 | HRD-in | -68.65, -49.34 | 77.87, -29.18 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8588 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.25, 120.14 | APE9-dihe-na | 171.2, -142.82 | APE8-dihe-in | -122.87, 132.42 | APE8-rot-in | 285.63 | APE67-dihe-inflip | 113.92, -33.46 | -57.37, 128.9 | APE12-dist-in | 10.1735 | APE11-dist-in | 11.7707 | APE10-dist-in | 5.8798 | APE9-dist-in | 3.5488 | S670A | None | None | XRAY | 2.56 | 0.205 | 0.264 | A | 641.0 | 621.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he0 | Bos taurus | AGC_GRK2_BOVIN | AGC | 5.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 5HE2A | P21146 | 30 | 668 | 689.0 | F0S:701 | Type1 | Active | DFGin | 5.2664 | 13.4322 | BLAminus | -127.84, 162.02 | 76.97, 74.62 | -82.13, 19.63 | 285.89, 54.35 | -44.91, -55.91 | in-in | in | 8.6986 | Saltbr-in | 2.6713 | HRD-in | -87.07, -48.72 | 79.5, -27.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.886 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.3, 135.41 | APE9-dihe-na | 128.88, -173.45 | APE8-dihe-in | -85.86, 172.32 | APE8-rot-in | 301.72 | APE67-dihe-in | -88.54, 16.07 | -85.52, -45.68 | APE12-dist-in | 10.698 | APE11-dist-in | 11.9311 | APE10-dist-in | 5.9928 | APE9-dist-in | 3.7816 | S670A | None | None | XRAY | 2.79 | 0.202 | 0.277 | A | 641.0 | 628.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he2 | Bos taurus | AGC_GRK2_BOVIN | AGC | 5.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 5HE3A | P21146 | 30 | 670 | 689.0 | FF1:702 | Type1 | Active | DFGin | 5.4706 | 13.1124 | BLAminus | -130.61, 154.77 | 82.75, 74.09 | -80.19, 15.36 | 283.76, 73.33 | -31.6, -75.24 | in-in | in | 8.613 | Saltbr-in | 2.7525 | HRD-in | -66.32, -31.89 | 63.86, -19.84 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9166 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.68, 142.9 | APE9-dihe-na | 127.74, 174.69 | APE8-dihe-in | -90.13, 145.29 | APE8-rot-in | 301.32 | APE67-dihe-inflip | 112.74, -14.85 | -68.46, 126.13 | APE12-dist-in | 10.205 | APE11-dist-in | 11.7078 | APE10-dist-in | 5.915 | APE9-dist-in | 3.371 | None | None | None | XRAY | 2.74 | 0.198 | 0.257 | A | 641.0 | 623.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5he3 | Bos taurus | AGC_GRK2_BOVIN | AGC | 5.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 5UKMA | P21146 | 31 | 669 | 689.0 | T0E:701 | Type1 | Active | DFGin | 5.5585 | 13.1317 | BLAminus | -130.36, 150.32 | 61.48, 90.2 | -96.51, 21.64 | 296.35, 62.89 | -55.13, -59.92 | in-in | in | 9.0172 | Saltbr-in | 2.7861 | HRD-in | -71.89, -48.96 | 73.51, -73.8 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1669 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.94, 135.34 | APE9-dihe-na | 121.47, 173.74 | APE8-dihe-in | -77.03, 143.73 | APE8-rot-in | 316.68 | APE67-dihe-in | -68.91, -23.51 | -68.56, -33.79 | APE12-dist-in | 10.3025 | APE11-dist-in | 11.6096 | APE10-dist-in | 5.8336 | APE9-dist-in | 5.3132 | S670A | None | None | XRAY | 3.03 | 0.2 | 0.252 | A | 695.0 | 621.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 5ukm | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7B | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1989 | 12.4485 | ABAminus | -130.8, -59.92 | -98.26, 108.63 | -91.58, -9.04 | 306.19, 95.69 | -36.4, -48.74 | in-out | in | 8.8033 | Saltbr-out | 4.6419 | HRD-in | -77.09, -44.3 | 73.62, -27.39 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7591 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.17, 125.32 | APE9-dihe-na | 152.82, 174.56 | APE8-dihe-in | -87.32, 142.62 | APE8-rot-in | 313.75 | APE67-dihe-in | -64.86, -36.54 | -62.56, -29.46 | APE12-dist-in | 9.8182 | APE11-dist-in | 11.5603 | APE10-dist-in | 5.5731 | APE9-dist-in | 4.0361 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | B | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 8JPBG | P21146 | 2 | 659 | 689.0 | STU:701 | Type1 | Inactive | DFGin | 5.5082 | 12.2136 | ABAminus | -113.28, -56.44 | -93.74, 100.06 | -93.25, 26.0 | 307.53, 3.55 | -63.32, -43.2 | in-out | in | 8.9334 | Saltbr-out | 4.2174 | HRD-out | -93.17, 87.64 | -73.74, -9.71 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7258 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.15, 142.89 | APE9-dihe-na | 142.59, -152.8 | APE8-dihe-in | -124.3, 137.48 | APE8-rot-in | 299.05 | APE67-dihe-inflip | 90.41, -8.27 | -58.8, 137.88 | APE12-dist-in | 9.9025 | APE11-dist-in | 12.0099 | APE10-dist-in | 6.0986 | APE9-dist-in | 3.6298 | A292P,R295I,S455D | None | None | EM | 3.07 | 999.0 | 999.0 | G | 688.0 | 658.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 8jpb | Bos taurus | AGC_GRK2_BOVIN | AGC | 1.7e-76 | 267.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 8JPCG | P21146 | 2 | 659 | 689.0 | STU:701 | Type1 | Inactive | DFGin | 5.385 | 12.1571 | ABAminus | -113.22, -56.58 | -93.6, 101.44 | -93.44, 27.48 | 306.81, 9.79 | -63.79, -45.14 | in-out | in | 8.9895 | Saltbr-out | 4.6535 | HRD-out | -92.62, 94.67 | -75.66, -35.58 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.6526 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.27, 130.92 | APE9-dihe-na | 162.84, -151.71 | APE8-dihe-in | -129.7, 130.81 | APE8-rot-in | 302.62 | APE67-dihe-inflip | 97.48, -17.5 | -57.09, 134.46 | APE12-dist-in | 9.7132 | APE11-dist-in | 11.9892 | APE10-dist-in | 5.9887 | APE9-dist-in | 4.3163 | A292P,R295I,S455D | None | None | EM | 3.07 | 999.0 | 999.0 | G | 688.0 | 658.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 8jpc | Bos taurus | AGC_GRK2_BOVIN | AGC | 1.7e-76 | 267.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 8JPDG | P21146 | 2 | 659 | 689.0 | STU:701 | Type1 | Inactive | DFGin | 5.3847 | 12.1571 | ABAminus | -113.24, -56.55 | -93.57, 101.39 | -93.42, 27.53 | 306.84, 9.79 | -63.78, -45.12 | in-out | in | 8.9895 | Saltbr-out | 4.6534 | HRD-out | -92.61, 94.65 | -75.65, -35.58 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.6534 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.32, 130.92 | APE9-dihe-na | 162.83, -151.7 | APE8-dihe-in | -129.72, 130.82 | APE8-rot-in | 302.58 | APE67-dihe-inflip | 97.48, -17.49 | -57.11, 134.43 | APE12-dist-in | 9.7137 | APE11-dist-in | 11.9887 | APE10-dist-in | 5.9885 | APE9-dist-in | 4.3171 | A292P,R295I,S455D | None | None | EM | 2.81 | 999.0 | 999.0 | G | 688.0 | 658.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 8jpd | Bos taurus | AGC_GRK2_BOVIN | AGC | 1.7e-76 | 267.2 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1OMWA | P21146 | 29 | 668 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.448 | 13.0685 | None | -112.27, -91.9 | -67.18, 126.78 | -99.0, 7.24 | 286.96, 109.41 | -44.09, -46.49 | in-in | in | 8.9372 | Saltbr-in | 3.4107 | HRD-in | -73.22, -52.41 | 80.02, -28.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8622 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.71, 128.56 | APE9-dihe-na | 124.77, -168.54 | APE8-dihe-in | -89.28, 150.91 | APE8-rot-in | 295.71 | APE67-dihe-in | -77.59, -9.92 | -72.81, -27.02 | APE12-dist-in | 10.5885 | APE11-dist-in | 11.8774 | APE10-dist-in | 6.1942 | APE9-dist-in | 3.5029 | S670A | None | None | XRAY | 2.5 | 0.216 | 0.252 | A | 689.0 | 614.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1omw | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7A | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2239 | 12.3565 | None | -125.66, -66.29 | -94.21, 107.11 | -86.73, -10.11 | 307.87, 97.53 | -38.26, -47.46 | in-out | in | 8.8531 | Saltbr-out | 4.6372 | HRD-in | -74.94, -45.18 | 74.24, -26.22 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7715 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.74, 123.21 | APE9-dihe-na | 155.55, 174.57 | APE8-dihe-in | -86.11, 141.22 | APE8-rot-in | 314.43 | APE67-dihe-in | -66.31, -34.76 | -64.21, -27.3 | APE12-dist-in | 9.8313 | APE11-dist-in | 11.5432 | APE10-dist-in | 5.5926 | APE9-dist-in | 3.9926 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | A | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7C | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2163 | 12.2674 | None | -130.34, -66.38 | -92.79, 106.85 | -85.97, -13.2 | 309.12, 95.06 | -35.96, -48.47 | in-out | in | 8.8136 | Saltbr-out | 4.7358 | HRD-in | -75.86, -48.89 | 75.97, -29.41 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.721 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.29, 128.8 | APE9-dihe-na | 145.96, 173.8 | APE8-dihe-in | -87.44, 141.12 | APE8-rot-in | 314.72 | APE67-dihe-in | -67.09, -36.43 | -60.22, -25.52 | APE12-dist-in | 9.7747 | APE11-dist-in | 11.5691 | APE10-dist-in | 5.6074 | APE9-dist-in | 4.0582 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | C | 689.0 | 607.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 1YM7D | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2341 | 12.3436 | None | -128.88, -67.33 | -92.65, 105.41 | -87.88, -10.71 | 307.83, 96.53 | -37.49, -49.46 | in-out | in | 8.801 | Saltbr-out | 4.7459 | HRD-in | -72.13, -45.13 | 72.62, -27.86 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7633 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.27, 125.22 | APE9-dihe-na | 149.39, 173.11 | APE8-dihe-in | -84.5, 141.69 | APE8-rot-in | 315.18 | APE67-dihe-in | -66.11, -35.98 | -62.26, -27.83 | APE12-dist-in | 9.7362 | APE11-dist-in | 11.4974 | APE10-dist-in | 5.5333 | APE9-dist-in | 4.0286 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | D | 689.0 | 599.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 2BCJA | P21146 | 28 | 667 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1531 | 12.3754 | None | -114.23, -125.71 | -23.26, 91.28 | -81.33, 0.62 | 275.63, 158.44 | -51.51, -42.54 | in-in | in | 8.6198 | Saltbr-in | 2.6334 | HRD-in | -86.19, -45.87 | 70.94, -23.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7186 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -106.73, 137.19 | APE9-dihe-na | 118.03, -177.98 | APE8-dihe-in | -75.0, 121.63 | APE8-rot-in | 302.92 | APE67-dihe-in | -97.57, -19.7 | -76.89, 19.37 | APE12-dist-in | 11.0395 | APE11-dist-in | 11.9406 | APE10-dist-in | 6.0057 | APE9-dist-in | 3.715 | S670A | None | None | XRAY | 3.061 | 0.236 | 0.292 | A | 689.0 | 624.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 2bcj | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3UZSA | P21146 | 29 | 671 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.731 | 11.1485 | None | -107.21, -110.21 | -68.72, 97.64 | -52.38, -56.06 | 299.08, 3.09 | 42.56, -75.63 | in-out | in | 9.0047 | Saltbr-out | 3.9207 | HRD-in | -77.33, -41.02 | 60.69, 32.77 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.5286 | ActLoopCT-out | nonTYR | APEdihe_aaiio | APEdist_iiii | APE10-dihe-na | -98.18, 142.14 | APE9-dihe-na | 139.16, 169.96 | APE8-dihe-in | -74.03, 124.78 | APE8-rot-in | 315.02 | APE67-dihe-out | 166.07, -43.85 | -59.08, 78.84 | APE12-dist-in | 10.2386 | APE11-dist-in | 12.0969 | APE10-dist-in | 6.31 | APE9-dist-in | 3.5138 | S670A | None | None | XRAY | 4.52 | 0.188 | 0.268 | A | 689.0 | 609.0 | 20 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3uzs | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3UZTA | P21146 | 30 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.216 | 12.499 | None | -94.28, -95.77 | -83.37, 90.84 | -54.75, -37.85 | 271.69, 47.64 | -2.65, -69.38 | in-out | in | 8.8257 | Saltbr-out | 5.0807 | HRD-in | -72.79, -37.98 | 67.02, -27.54 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.085 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -99.51, 148.65 | APE9-dihe-na | 138.76, 168.6 | APE8-dihe-in | -71.39, 126.55 | APE8-rot-in | 294.92 | APE67-dihe-in | -71.95, -17.71 | -54.34, -25.29 | APE12-dist-in | 9.5328 | APE11-dist-in | 12.0098 | APE10-dist-in | 5.9885 | APE9-dist-in | 3.8685 | S670A | None | None | XRAY | 3.51 | 0.22 | 0.317 | A | 689.0 | 586.0 | 12 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3uzt | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3PSCA | P21146 | 29 | 668 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.4842 | 12.8251 | None | -112.1, -116.4 | -50.02, 128.26 | -100.71, 13.15 | 287.53, 88.47 | -45.02, -46.74 | in-in | in | 8.8883 | Saltbr-in | 3.1136 | HRD-in | -73.4, -47.49 | 67.75, 0.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.59, 142.02 | APE9-dihe-na | 121.44, 174.37 | APE8-dihe-in | -79.3, 138.73 | APE8-rot-in | 323.05 | APE67-dihe-in | -80.94, 3.9 | -61.06, -31.71 | APE12-dist-in | 10.1172 | APE11-dist-in | 11.7629 | APE10-dist-in | 5.9289 | APE9-dist-in | 3.1916 | S670A | None | None | XRAY | 2.67 | 0.225 | 0.257 | A | 695.0 | 614.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3psc | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3PVUA | P21146 | 30 | 668 | 689.0 | QRW:800 | Type1 | Inactive | DFGin | 5.4293 | 12.5496 | None | -114.2, -126.97 | -29.78, 116.79 | -95.83, 7.38 | 283.37, 161.7 | -55.56, -22.85 | in-in | in | 8.7486 | Saltbr-in | 2.9863 | HRD-in | -71.34, -46.23 | 80.59, -11.92 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9271 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -154.26, 142.91 | APE9-dihe-na | 117.3, -165.9 | APE8-dihe-in | -102.62, 148.45 | APE8-rot-in | 314.0 | APE67-dihe-in | -77.54, 11.33 | -67.23, -35.08 | APE12-dist-in | 10.2837 | APE11-dist-in | 11.8902 | APE10-dist-in | 6.1863 | APE9-dist-in | 3.4202 | S670A | None | None | XRAY | 2.48 | 0.229 | 0.274 | A | 695.0 | 609.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3pvu | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| GRK2 | ARBK1_BOVIN | 3PVWA | P21146 | 29 | 668 | 689.0 | QRX:800 | Type1 | Inactive | DFGin | 5.249 | 12.3972 | None | -104.93, -94.33 | -60.0, 121.61 | -95.37, 6.96 | 285.31, 4.38 | -65.85, -19.47 | in-in | in | 8.7495 | Saltbr-in | 3.07 | HRD-in | -69.01, -52.71 | 78.6, -13.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9188 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.25, 142.6 | APE9-dihe-na | 127.77, 176.65 | APE8-dihe-in | -84.9, 148.79 | APE8-rot-in | 327.3 | APE67-dihe-in | -77.16, 13.46 | -65.86, -42.83 | APE12-dist-in | 10.7375 | APE11-dist-in | 12.1865 | APE10-dist-in | 6.4122 | APE9-dist-in | 3.337 | S670A | None | None | XRAY | 2.49 | 0.239 | 0.285 | A | 695.0 | 613.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 3pvw | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.4e-77 | 268.7 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |