| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| FLT3 | AF-P36888-K1A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 6.9519 | 14.1313 | BLAminus | -143.23, 178.77 | 67.08, 55.14 | -77.02, 14.59 | 286.19, 76.14 | -61.49, -31.53 | in-in | in | 7.4793 | Saltbr-in | 2.6983 | HRD-in | -78.74, -43.23 | 66.6, -14.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9188 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.73, 89.83 | APE9-dihe-in | -111.39, 151.17 | APE8-dihe-in | -77.59, 83.68 | APE8-rot-na | 35.47 | APE67-dihe-in | -70.07, -16.26 | -43.63, -37.27 | APE12-dist-na | 14.2956 | APE11-dist-na | 8.2372 | APE10-dist-na | 9.8964 | APE9-dist-in | 6.0185 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K1 | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | AF-P36888-K3A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 7.2842 | 13.5426 | BLAminus | -131.51, -179.63 | 57.0, 62.49 | -72.98, 8.43 | 287.44, 96.64 | -61.83, -29.79 | in-in | in | 7.8544 | Saltbr-in | 2.7853 | HRD-in | -79.97, -43.81 | 68.78, -8.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8992 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.33, 109.47 | APE9-dihe-in | -88.85, 151.32 | APE8-dihe-in | -79.53, 61.94 | APE8-rot-na | 36.79 | APE67-dihe-in | -68.95, -18.44 | -45.43, -42.99 | APE12-dist-na | 14.4475 | APE11-dist-na | 8.7996 | APE10-dist-na | 12.3215 | APE9-dist-in | 7.3936 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K3 | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 4XUFA | P36888 | 600 | 947 | 993.0 | P30:1001 | Type2 | Inactive | DFGout | 16.0329 | 10.199 | BBAminus | -143.0, -176.09 | -145.89, 109.83 | -79.74, 65.35 | 291.29, 82.28 | -88.07, 125.53 | in-in | in | 7.6772 | Saltbr-in | 3.1306 | HRD-out | -82.56, 115.59 | -72.64, -20.56 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5483 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.53, 147.84 | APE9-dihe-in | -146.85, 149.22 | APE8-dihe-in | -75.18, 95.57 | APE8-rot-na | 28.09 | APE67-dihe-in | -79.56, 0.39 | -65.83, -40.86 | APE12-dist-na | 17.0014 | APE11-dist-na | 12.6753 | APE10-dist-na | 12.5 | APE9-dist-in | 7.1567 | None | None | None | XRAY | 3.2 | 0.299 | 0.32 | A | 297.0 | 270.0 | 27 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 4xuf | TYR_FLT3_HUMAN | TYR | 5.8e-103 | 349.6 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 4XUFB | P36888 | 600 | 946 | 993.0 | P30:1001 | Type2 | Inactive | DFGout | 15.6204 | 10.1033 | BBAminus | -144.31, -175.77 | -146.27, 108.35 | -80.93, 70.68 | 293.11, 82.52 | -83.4, -47.41 | in-in | in | 7.8934 | Saltbr-in | 2.6077 | HRD-out | -84.03, 114.48 | -73.98, -19.45 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5393 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -85.34, 144.93 | APE9-dihe-in | -152.45, 148.59 | APE8-dihe-in | -76.73, 96.39 | APE8-rot-na | 28.9 | APE67-dihe-in | -79.15, 1.24 | -66.13, -41.05 | APE12-dist-na | 17.7249 | APE11-dist-na | 13.5149 | APE10-dist-na | 12.373 | APE9-dist-in | 7.5793 | None | None | None | XRAY | 3.2 | 0.299 | 0.32 | B | 297.0 | 274.0 | 22 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 4xuf | TYR_FLT3_HUMAN | TYR | 5.8e-103 | 349.6 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 4RT7A | P36888 | 599 | 950 | 993.0 | P30:1001 | Type2 | Inactive | DFGout | 16.2803 | 10.6907 | BBAminus | -148.52, -175.77 | -147.58, 109.4 | -60.96, -39.74 | 289.53, 78.87 | 49.01, -101.54 | in-in | in | 7.6415 | Saltbr-in | 2.9875 | HRD-out | -100.49, 123.78 | -88.21, -0.63 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.567 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -124.24, 104.7 | APE9-dihe-in | -116.44, 148.12 | APE8-dihe-in | -77.95, 71.82 | APE8-rot-na | 30.09 | APE67-dihe-in | -65.85, -17.18 | -55.85, -43.14 | APE12-dist-na | 17.729 | APE11-dist-na | 14.0524 | APE10-dist-na | 12.022 | APE9-dist-in | 7.4427 | None | None | None | XRAY | 3.1 | 0.224 | 0.268 | A | 415.0 | 274.0 | 78 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 4rt7 | TYR_FLT3_HUMAN | TYR | 7.6e-102 | 346.1 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 1RJBA | P36888 | 572 | 947 | 993.0 | No_ligand | No_ligand | Inactive | DFGout | 15.6842 | 8.3625 | None | -155.78, -170.12 | -125.78, 107.33 | -104.31, 21.16 | 225.91, 48.71 | -54.59, -36.41 | in-in | in | 7.8172 | Saltbr-in | 2.5929 | HRD-out | -115.43, 117.74 | -85.28, 1.33 | in-out-in | SNCioi | out-in | ActLoopNT-out | 18.0296 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -130.87, 97.23 | APE9-dihe-in | -99.06, 130.66 | APE8-dihe-in | -82.4, 63.28 | APE8-rot-na | 34.53 | APE67-dihe-in | -68.25, -12.12 | -43.78, -45.7 | APE12-dist-na | 16.7583 | APE11-dist-na | 16.1469 | APE10-dist-na | 11.9453 | APE9-dist-in | 7.2982 | None | None | None | XRAY | 2.1 | 0.23 | 0.248 | A | 344.0 | 298.0 | 27 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 1rjb | TYR_FLT3_HUMAN | TYR | 9.9e-103 | 348.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 6JQRA | P36888 | 571 | 951 | 993.0 | C6F:1001 | Type1 | Inactive | DFGout | 15.3937 | 10.8847 | None | -119.73, 157.71 | -104.23, 115.68 | 77.2, 999.0 | 255.94, 91.42 | 999.0, 999.0 | in-in | in | 8.3262 | Saltbr-in | 2.8041 | HRD-out | -98.26, 117.82 | -85.48, 11.47 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.05, 100.76 | APE9-dihe-in | -103.87, 123.04 | APE8-dihe-in | -78.74, 70.62 | APE8-rot-na | 34.5 | APE67-dihe-in | -69.1, -11.06 | -54.04, -46.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.223 | None | None | None | XRAY | 2.2 | 0.181 | 0.213 | A | 330.0 | 301.0 | 29 | 30 | 24 | 6 | [[610, 945]] | 1.0 | 6jqr | TYR_FLT3_HUMAN | TYR | 8.5e-103 | 349.1 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 8XB1A | P36888 | 573 | 950 | 993.0 | ZX3:1001 | Type1 | Inactive | DFGout | 16.7849 | 8.5029 | None | -137.58, 174.85 | -120.11, 128.8 | 51.2, 999.0 | 176.42, 95.47 | 999.0, 999.0 | in-in | in | 8.4654 | Saltbr-in | 3.2549 | HRD-out | -103.79, 107.3 | -84.06, 13.74 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.92, 110.72 | APE9-dihe-in | -112.36, 129.93 | APE8-dihe-in | -83.81, 80.36 | APE8-rot-na | 31.64 | APE67-dihe-in | -69.59, -10.43 | -56.56, -46.35 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.9566 | None | None | None | XRAY | 2.85 | 0.236 | 0.287 | A | 346.0 | 304.0 | 23 | 30 | 24 | 6 | [[610, 945]] | 1.0 | 8xb1 | TYR_FLT3_HUMAN | TYR | 1e-102 | 348.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 5X02A | P36888 | 573 | 947 | 993.0 | F6M:61001 | Type1 | Inactive | DFGout | 16.5131 | 10.7389 | None | -127.36, 175.28 | -155.15, 109.24 | -131.05, 124.01 | 44.79, 98.96 | -130.39, -30.78 | in-in | in | 8.3837 | Saltbr-in | 2.7312 | HRD-out | -116.89, 102.0 | -82.02, 12.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.2417 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -122.0, 95.48 | APE9-dihe-in | -95.25, 120.88 | APE8-dihe-in | -74.85, 69.27 | APE8-rot-na | 28.28 | APE67-dihe-in | -69.28, -8.01 | -53.09, -46.19 | APE12-dist-na | 13.3264 | APE11-dist-na | 13.8141 | APE10-dist-na | 9.9433 | APE9-dist-in | 7.0561 | None | None | None | XRAY | 2.401 | 0.236 | 0.277 | A | 347.0 | 305.0 | 19 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 5x02 | TYR_FLT3_HUMAN | TYR | 1e-102 | 348.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | 6IL3A | P36888 | 569 | 947 | 993.0 | A9R:1001 | Type1 | Inactive | DFGout | 18.0662 | 9.9905 | None | -137.72, 178.19 | -114.58, 103.78 | -95.53, 10.02 | 188.73, 81.27 | -62.27, -30.79 | in-in | in | 7.9045 | Saltbr-in | 2.6619 | HRD-out | -112.71, 117.58 | -85.2, 6.2 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.3179 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -132.53, 103.3 | APE9-dihe-in | -108.39, 121.39 | APE8-dihe-in | -81.48, 71.82 | APE8-rot-na | 34.93 | APE67-dihe-in | -74.41, -7.85 | -52.12, -42.1 | APE12-dist-na | 15.6858 | APE11-dist-na | 15.4496 | APE10-dist-na | 11.1607 | APE9-dist-in | 7.2327 | None | None | None | XRAY | 2.5 | 0.185 | 0.219 | A | 370.0 | 310.0 | 18 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 6il3 | TYR_FLT3_HUMAN | TYR | 1.3e-102 | 348.6 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| FLT3 | FLT3_HUMAN | AF-P36888-K1A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 6.9519 | 14.1313 | BLAminus | -143.23, 178.77 | 67.08, 55.14 | -77.02, 14.59 | 286.19, 76.14 | -61.49, -31.53 | in-in | in | 7.4793 | Saltbr-in | 2.6983 | HRD-in | -78.74, -43.23 | 66.6, -14.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9188 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.73, 89.83 | APE9-dihe-in | -111.39, 151.17 | APE8-dihe-in | -77.59, 83.68 | APE8-rot-na | 35.47 | APE67-dihe-in | -70.07, -16.26 | -43.63, -37.27 | APE12-dist-na | 14.2956 | APE11-dist-na | 8.2372 | APE10-dist-na | 9.8964 | APE9-dist-in | 6.0185 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K1 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | AF-P36888-K3A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 7.2842 | 13.5426 | BLAminus | -131.51, -179.63 | 57.0, 62.49 | -72.98, 8.43 | 287.44, 96.64 | -61.83, -29.79 | in-in | in | 7.8544 | Saltbr-in | 2.7853 | HRD-in | -79.97, -43.81 | 68.78, -8.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8992 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.33, 109.47 | APE9-dihe-in | -88.85, 151.32 | APE8-dihe-in | -79.53, 61.94 | APE8-rot-na | 36.79 | APE67-dihe-in | -68.95, -18.44 | -45.43, -42.99 | APE12-dist-na | 14.4475 | APE11-dist-na | 8.7996 | APE10-dist-na | 12.3215 | APE9-dist-in | 7.3936 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K3 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 4XUFA | P36888 | 600 | 947 | 993.0 | P30:1001 | Type2 | Inactive | DFGout | 16.0329 | 10.199 | BBAminus | -143.0, -176.09 | -145.89, 109.83 | -79.74, 65.35 | 291.29, 82.28 | -88.07, 125.53 | in-in | in | 7.6772 | Saltbr-in | 3.1306 | HRD-out | -82.56, 115.59 | -72.64, -20.56 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5483 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.53, 147.84 | APE9-dihe-in | -146.85, 149.22 | APE8-dihe-in | -75.18, 95.57 | APE8-rot-na | 28.09 | APE67-dihe-in | -79.56, 0.39 | -65.83, -40.86 | APE12-dist-na | 17.0014 | APE11-dist-na | 12.6753 | APE10-dist-na | 12.5 | APE9-dist-in | 7.1567 | None | None | None | XRAY | 3.2 | 0.299 | 0.32 | A | 297.0 | 270.0 | 27 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 4xuf | Homo sapiens | TYR_FLT3_HUMAN | TYR | 5.8e-103 | 349.6 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 4XUFB | P36888 | 600 | 946 | 993.0 | P30:1001 | Type2 | Inactive | DFGout | 15.6204 | 10.1033 | BBAminus | -144.31, -175.77 | -146.27, 108.35 | -80.93, 70.68 | 293.11, 82.52 | -83.4, -47.41 | in-in | in | 7.8934 | Saltbr-in | 2.6077 | HRD-out | -84.03, 114.48 | -73.98, -19.45 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.5393 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -85.34, 144.93 | APE9-dihe-in | -152.45, 148.59 | APE8-dihe-in | -76.73, 96.39 | APE8-rot-na | 28.9 | APE67-dihe-in | -79.15, 1.24 | -66.13, -41.05 | APE12-dist-na | 17.7249 | APE11-dist-na | 13.5149 | APE10-dist-na | 12.373 | APE9-dist-in | 7.5793 | None | None | None | XRAY | 3.2 | 0.299 | 0.32 | B | 297.0 | 274.0 | 22 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 4xuf | Homo sapiens | TYR_FLT3_HUMAN | TYR | 5.8e-103 | 349.6 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 4RT7A | P36888 | 599 | 950 | 993.0 | P30:1001 | Type2 | Inactive | DFGout | 16.2803 | 10.6907 | BBAminus | -148.52, -175.77 | -147.58, 109.4 | -60.96, -39.74 | 289.53, 78.87 | 49.01, -101.54 | in-in | in | 7.6415 | Saltbr-in | 2.9875 | HRD-out | -100.49, 123.78 | -88.21, -0.63 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.567 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -124.24, 104.7 | APE9-dihe-in | -116.44, 148.12 | APE8-dihe-in | -77.95, 71.82 | APE8-rot-na | 30.09 | APE67-dihe-in | -65.85, -17.18 | -55.85, -43.14 | APE12-dist-na | 17.729 | APE11-dist-na | 14.0524 | APE10-dist-na | 12.022 | APE9-dist-in | 7.4427 | None | None | None | XRAY | 3.1 | 0.224 | 0.268 | A | 415.0 | 274.0 | 78 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 4rt7 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 7.6e-102 | 346.1 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 1RJBA | P36888 | 572 | 947 | 993.0 | No_ligand | No_ligand | Inactive | DFGout | 15.6842 | 8.3625 | None | -155.78, -170.12 | -125.78, 107.33 | -104.31, 21.16 | 225.91, 48.71 | -54.59, -36.41 | in-in | in | 7.8172 | Saltbr-in | 2.5929 | HRD-out | -115.43, 117.74 | -85.28, 1.33 | in-out-in | SNCioi | out-in | ActLoopNT-out | 18.0296 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -130.87, 97.23 | APE9-dihe-in | -99.06, 130.66 | APE8-dihe-in | -82.4, 63.28 | APE8-rot-na | 34.53 | APE67-dihe-in | -68.25, -12.12 | -43.78, -45.7 | APE12-dist-na | 16.7583 | APE11-dist-na | 16.1469 | APE10-dist-na | 11.9453 | APE9-dist-in | 7.2982 | None | None | None | XRAY | 2.1 | 0.23 | 0.248 | A | 344.0 | 298.0 | 27 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 1rjb | Homo sapiens | TYR_FLT3_HUMAN | TYR | 9.9e-103 | 348.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 6JQRA | P36888 | 571 | 951 | 993.0 | C6F:1001 | Type1 | Inactive | DFGout | 15.3937 | 10.8847 | None | -119.73, 157.71 | -104.23, 115.68 | 77.2, 999.0 | 255.94, 91.42 | 999.0, 999.0 | in-in | in | 8.3262 | Saltbr-in | 2.8041 | HRD-out | -98.26, 117.82 | -85.48, 11.47 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -131.05, 100.76 | APE9-dihe-in | -103.87, 123.04 | APE8-dihe-in | -78.74, 70.62 | APE8-rot-na | 34.5 | APE67-dihe-in | -69.1, -11.06 | -54.04, -46.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.223 | None | None | None | XRAY | 2.2 | 0.181 | 0.213 | A | 330.0 | 301.0 | 29 | 30 | 24 | 6 | [[610, 945]] | 1.0 | 6jqr | Homo sapiens | TYR_FLT3_HUMAN | TYR | 8.5e-103 | 349.1 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 8XB1A | P36888 | 573 | 950 | 993.0 | ZX3:1001 | Type1 | Inactive | DFGout | 16.7849 | 8.5029 | None | -137.58, 174.85 | -120.11, 128.8 | 51.2, 999.0 | 176.42, 95.47 | 999.0, 999.0 | in-in | in | 8.4654 | Saltbr-in | 3.2549 | HRD-out | -103.79, 107.3 | -84.06, 13.74 | in-none-in | SNCini | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.92, 110.72 | APE9-dihe-in | -112.36, 129.93 | APE8-dihe-in | -83.81, 80.36 | APE8-rot-na | 31.64 | APE67-dihe-in | -69.59, -10.43 | -56.56, -46.35 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.9566 | None | None | None | XRAY | 2.85 | 0.236 | 0.287 | A | 346.0 | 304.0 | 23 | 30 | 24 | 6 | [[610, 945]] | 1.0 | 8xb1 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 1e-102 | 348.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 5X02A | P36888 | 573 | 947 | 993.0 | F6M:61001 | Type1 | Inactive | DFGout | 16.5131 | 10.7389 | None | -127.36, 175.28 | -155.15, 109.24 | -131.05, 124.01 | 44.79, 98.96 | -130.39, -30.78 | in-in | in | 8.3837 | Saltbr-in | 2.7312 | HRD-out | -116.89, 102.0 | -82.02, 12.69 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.2417 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -122.0, 95.48 | APE9-dihe-in | -95.25, 120.88 | APE8-dihe-in | -74.85, 69.27 | APE8-rot-na | 28.28 | APE67-dihe-in | -69.28, -8.01 | -53.09, -46.19 | APE12-dist-na | 13.3264 | APE11-dist-na | 13.8141 | APE10-dist-na | 9.9433 | APE9-dist-in | 7.0561 | None | None | None | XRAY | 2.401 | 0.236 | 0.277 | A | 347.0 | 305.0 | 19 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 5x02 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 1e-102 | 348.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| FLT3 | FLT3_HUMAN | 6IL3A | P36888 | 569 | 947 | 993.0 | A9R:1001 | Type1 | Inactive | DFGout | 18.0662 | 9.9905 | None | -137.72, 178.19 | -114.58, 103.78 | -95.53, 10.02 | 188.73, 81.27 | -62.27, -30.79 | in-in | in | 7.9045 | Saltbr-in | 2.6619 | HRD-out | -112.71, 117.58 | -85.2, 6.2 | in-out-in | SNCioi | out-in | ActLoopNT-out | 17.3179 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -132.53, 103.3 | APE9-dihe-in | -108.39, 121.39 | APE8-dihe-in | -81.48, 71.82 | APE8-rot-na | 34.93 | APE67-dihe-in | -74.41, -7.85 | -52.12, -42.1 | APE12-dist-na | 15.6858 | APE11-dist-na | 15.4496 | APE10-dist-na | 11.1607 | APE9-dist-in | 7.2327 | None | None | None | XRAY | 2.5 | 0.185 | 0.219 | A | 370.0 | 310.0 | 18 | 30 | 30 | 0 | [[610, 945]] | 1.0 | 6il3 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 1.3e-102 | 348.6 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|