TKL_BMPR2 (Bone morphogenetic protein receptor type-2)

Total number of chains: 6
Active chains: 5
Uniprot: BMPR2_HUMAN
Kinase Domain Residues: 203 - 503
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 6 100.0% AF-Q13873-K1A

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
BMPR2 3G2FA Q13873 197 510 1038.0 ADP:900 ATPlike Active DFGin 6.9573 13.9443 BLAminus -131.62, -179.2 66.08, 79.87 -102.79, 27.43 304.26, 96.52 -59.99, -25.3 in-in in 8.1073 Saltbr-in 2.7568 HRD-in -69.81, -50.66 82.19, -10.63 in-in-in SNCiii in-in ActLoopNT-in 2.9811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.1, -22.11 APE9-dihe-na -73.96, -168.61 APE8-dihe-in -80.16, 127.03 APE8-rot-in 308.56 APE67-dihe-in -65.91, -22.58 -59.75, -41.5 APE12-dist-in 11.4026 APE11-dist-in 12.6299 APE10-dist-in 7.0259 APE9-dist-in 4.0326 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 A 336.0 305.0 9 36 27 9 [[202, 503]] 1.0 3g2f TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 3G2FB Q13873 198 513 1038.0 ADP:900 ATPlike Active DFGin 6.9679 14.0082 BLAminus -149.7, 179.95 61.07, 87.18 -102.54, 11.93 293.8, 112.47 -56.7, -17.91 in-in in 8.0646 Saltbr-in 2.7316 HRD-in -73.22, -52.25 87.7, -10.0 in-in-in SNCiii in-in ActLoopNT-in 2.9139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.94, -26.41 APE9-dihe-na -71.73, -175.39 APE8-dihe-in -71.07, 133.08 APE8-rot-in 315.55 APE67-dihe-in -68.07, -13.93 -56.75, -42.89 APE12-dist-in 11.1939 APE11-dist-in 12.1078 APE10-dist-in 6.494 APE9-dist-in 3.7222 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 B 336.0 303.0 13 36 23 13 [[202, 503]] 1.0 3g2f TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 6UNPB Q13873 197 509 1038.0 ADP:601 ATPlike Active DFGin 6.9166 14.0508 BLAminus -140.56, 176.5 63.35, 76.41 -96.26, 25.8 302.12, 104.12 -61.08, -20.73 in-in in 7.9042 Saltbr-in 2.8646 HRD-in -75.95, -48.17 78.17, -6.91 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.29, -9.38 APE9-dihe-na -69.43, -161.26 APE8-dihe-in -89.59, 127.34 APE8-rot-in 301.19 APE67-dihe-in -48.39, -33.11 -62.11, -43.63 APE12-dist-in 12.0086 APE11-dist-in 12.508 APE10-dist-in 7.0989 APE9-dist-in 4.016 D485G None CAS288,CAS397,CAS496 XRAY 2.3 0.19 0.211 B 363.0 303.0 10 36 28 8 [[202, 503]] 1.0 6unp TKL_BMPR2_HUMAN TKL 1.1e-74 257.3 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 AF-Q13873-K1A Q13873 195 511 1038.0 No_ligand No_ligand Active DFGin 6.8747 13.8799 BLAminus -141.81, 174.26 66.05, 62.15 -80.12, 19.48 303.5, 100.88 -62.94, -18.22 in-in in 7.7734 Saltbr-in 2.7229 HRD-in -74.25, -44.66 69.23, -7.61 in-in-in SNCiii in-in ActLoopNT-in 2.9211 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.76, 161.84 APE9-dihe-na 90.67, 173.58 APE8-dihe-in -87.87, 115.69 APE8-rot-in 299.44 APE67-dihe-in -57.12, -29.27 -45.32, -43.89 APE12-dist-in 13.9416 APE11-dist-in 10.9778 APE10-dist-in 6.25 APE9-dist-in 3.8086 None None None AF2 -1.0 1.0 1.0 A 317.0 317.0 0 36 36 0 [[202, 503]] 1.0 AF-Q13873-K1 TKL_BMPR2_HUMAN TKL 1.2e-75 260.5 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 AF-Q13873-K3A Q13873 195 511 1038.0 No_ligand No_ligand Active DFGin 7.0122 13.9069 BLAminus -141.79, 177.72 65.01, 59.4 -77.77, 17.3 300.16, 94.71 -64.36, -23.28 in-in in 7.8749 Saltbr-in 2.7367 HRD-in -79.43, -45.87 64.01, 9.98 in-in-in SNCiii in-in ActLoopNT-in 2.9308 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.99, 157.3 APE9-dihe-na 117.25, -171.77 APE8-dihe-in -83.43, 113.58 APE8-rot-in 297.45 APE67-dihe-in -59.95, -28.51 -41.61, -44.44 APE12-dist-in 12.3047 APE11-dist-in 11.8227 APE10-dist-in 5.9764 APE9-dist-in 3.3599 None None None AF2 -1.0 1.0 1.0 A 317.0 317.0 0 36 36 0 [[202, 503]] 1.0 AF-Q13873-K3 TKL_BMPR2_HUMAN TKL 1.2e-75 260.5 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 6UNPA Q13873 199 509 1038.0 ADP:601,ADP:602 ATPlike,Allosteric None DFGin 7.015 14.0658 BLAminus -140.5, 177.86 62.51, 75.21 -94.82, 26.77 301.08, 104.11 -62.66, -20.97 in-in in 7.9826 Saltbr-in 2.8316 HRD-in -73.31, -49.03 80.8, -8.07 in-in-none SNCiin in-none ActLoopNT-in 2.9199 ActLoopCT-none nonTYR APEdihe_aaiii APEdist_niii APE10-dihe-na -134.35, -10.44 APE9-dihe-na -70.57, -158.87 APE8-dihe-in -91.29, 127.64 APE8-rot-in 299.54 APE67-dihe-in -49.77, -33.71 -61.84, -45.11 APE12-dist-none 999.0 APE11-dist-in 12.7405 APE10-dist-in 7.2841 APE9-dist-in 4.0925 D485G None CAS288,CAS397,CAS496 XRAY 2.3 0.19 0.211 A 363.0 302.0 9 36 27 9 [[202, 503]] 1.0 6unp TKL_BMPR2_HUMAN TKL 1.1e-74 257.3 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2

TKL_BMPR2 (Bone morphogenetic protein receptor type-2)

Total number of chains: 6
Active chains: 5
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 6 100.0% AF-Q13873-K1A

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
BMPR2 BMPR2_HUMAN 3G2FA Q13873 197 510 1038.0 ADP:900 ATPlike Active DFGin 6.9573 13.9443 BLAminus -131.62, -179.2 66.08, 79.87 -102.79, 27.43 304.26, 96.52 -59.99, -25.3 in-in in 8.1073 Saltbr-in 2.7568 HRD-in -69.81, -50.66 82.19, -10.63 in-in-in SNCiii in-in ActLoopNT-in 2.9811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.1, -22.11 APE9-dihe-na -73.96, -168.61 APE8-dihe-in -80.16, 127.03 APE8-rot-in 308.56 APE67-dihe-in -65.91, -22.58 -59.75, -41.5 APE12-dist-in 11.4026 APE11-dist-in 12.6299 APE10-dist-in 7.0259 APE9-dist-in 4.0326 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 A 336.0 305.0 9 36 27 9 [[202, 503]] 1.0 3g2f Homo sapiens TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 BMPR2_HUMAN 3G2FB Q13873 198 513 1038.0 ADP:900 ATPlike Active DFGin 6.9679 14.0082 BLAminus -149.7, 179.95 61.07, 87.18 -102.54, 11.93 293.8, 112.47 -56.7, -17.91 in-in in 8.0646 Saltbr-in 2.7316 HRD-in -73.22, -52.25 87.7, -10.0 in-in-in SNCiii in-in ActLoopNT-in 2.9139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.94, -26.41 APE9-dihe-na -71.73, -175.39 APE8-dihe-in -71.07, 133.08 APE8-rot-in 315.55 APE67-dihe-in -68.07, -13.93 -56.75, -42.89 APE12-dist-in 11.1939 APE11-dist-in 12.1078 APE10-dist-in 6.494 APE9-dist-in 3.7222 None None CAS288,CAS397,CAS496 XRAY 2.35 0.21 0.246 B 336.0 303.0 13 36 23 13 [[202, 503]] 1.0 3g2f Homo sapiens TKL_BMPR2_HUMAN TKL 1.4e-75 260.2 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 BMPR2_HUMAN 6UNPB Q13873 197 509 1038.0 ADP:601 ATPlike Active DFGin 6.9166 14.0508 BLAminus -140.56, 176.5 63.35, 76.41 -96.26, 25.8 302.12, 104.12 -61.08, -20.73 in-in in 7.9042 Saltbr-in 2.8646 HRD-in -75.95, -48.17 78.17, -6.91 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.29, -9.38 APE9-dihe-na -69.43, -161.26 APE8-dihe-in -89.59, 127.34 APE8-rot-in 301.19 APE67-dihe-in -48.39, -33.11 -62.11, -43.63 APE12-dist-in 12.0086 APE11-dist-in 12.508 APE10-dist-in 7.0989 APE9-dist-in 4.016 D485G None CAS288,CAS397,CAS496 XRAY 2.3 0.19 0.211 B 363.0 303.0 10 36 28 8 [[202, 503]] 1.0 6unp Homo sapiens TKL_BMPR2_HUMAN TKL 1.1e-74 257.3 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 BMPR2_HUMAN AF-Q13873-K1A Q13873 195 511 1038.0 No_ligand No_ligand Active DFGin 6.8747 13.8799 BLAminus -141.81, 174.26 66.05, 62.15 -80.12, 19.48 303.5, 100.88 -62.94, -18.22 in-in in 7.7734 Saltbr-in 2.7229 HRD-in -74.25, -44.66 69.23, -7.61 in-in-in SNCiii in-in ActLoopNT-in 2.9211 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -123.76, 161.84 APE9-dihe-na 90.67, 173.58 APE8-dihe-in -87.87, 115.69 APE8-rot-in 299.44 APE67-dihe-in -57.12, -29.27 -45.32, -43.89 APE12-dist-in 13.9416 APE11-dist-in 10.9778 APE10-dist-in 6.25 APE9-dist-in 3.8086 None None None AF2 -1.0 1.0 1.0 A 317.0 317.0 0 36 36 0 [[202, 503]] 1.0 AF-Q13873-K1 Homo sapiens TKL_BMPR2_HUMAN TKL 1.2e-75 260.5 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 BMPR2_HUMAN AF-Q13873-K3A Q13873 195 511 1038.0 No_ligand No_ligand Active DFGin 7.0122 13.9069 BLAminus -141.79, 177.72 65.01, 59.4 -77.77, 17.3 300.16, 94.71 -64.36, -23.28 in-in in 7.8749 Saltbr-in 2.7367 HRD-in -79.43, -45.87 64.01, 9.98 in-in-in SNCiii in-in ActLoopNT-in 2.9308 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.99, 157.3 APE9-dihe-na 117.25, -171.77 APE8-dihe-in -83.43, 113.58 APE8-rot-in 297.45 APE67-dihe-in -59.95, -28.51 -41.61, -44.44 APE12-dist-in 12.3047 APE11-dist-in 11.8227 APE10-dist-in 5.9764 APE9-dist-in 3.3599 None None None AF2 -1.0 1.0 1.0 A 317.0 317.0 0 36 36 0 [[202, 503]] 1.0 AF-Q13873-K3 Homo sapiens TKL_BMPR2_HUMAN TKL 1.2e-75 260.5 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2
BMPR2 BMPR2_HUMAN 6UNPA Q13873 199 509 1038.0 ADP:601,ADP:602 ATPlike,Allosteric None DFGin 7.015 14.0658 BLAminus -140.5, 177.86 62.51, 75.21 -94.82, 26.77 301.08, 104.11 -62.66, -20.97 in-in in 7.9826 Saltbr-in 2.8316 HRD-in -73.31, -49.03 80.8, -8.07 in-in-none SNCiin in-none ActLoopNT-in 2.9199 ActLoopCT-none nonTYR APEdihe_aaiii APEdist_niii APE10-dihe-na -134.35, -10.44 APE9-dihe-na -70.57, -158.87 APE8-dihe-in -91.29, 127.64 APE8-rot-in 299.54 APE67-dihe-in -49.77, -33.71 -61.84, -45.11 APE12-dist-none 999.0 APE11-dist-in 12.7405 APE10-dist-in 7.2841 APE9-dist-in 4.0925 D485G None CAS288,CAS397,CAS496 XRAY 2.3 0.19 0.211 A 363.0 302.0 9 36 27 9 [[202, 503]] 1.0 6unp Homo sapiens TKL_BMPR2_HUMAN TKL 1.1e-74 257.3 2.0 266.0 265.0 350 351 352 354 356 230 243 247 330 332 331 333.0 405 386 381 380 379 378 377 376 375 280 Bone morphogenetic protein receptor type-2

TKL_BMPR2 (Bone morphogenetic protein receptor type-2)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help.

Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name