AF-P25098-K1

GRK2 (Beta-adrenergic receptor kinase 1)
Group: AGC
Uniprot: ARBK1_HUMAN
Organism: Homo sapiens
Domain boundary: 191 - 453
Resolu: -1.0

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in No_ligand No_ligand 183 - 461 0
Representative sequence - Chain A
192 202 212 222
NIHLTMNDFS VHRIIGRGGF GEVYGCRKAD TGKMYAMKCL
232 242 252 262
DKKRIKMKQG ETLALNERIM LSLVSTGDCP FIVCMSYAFH
272 282 292 302
TPDKLSFILD LMNGGDLHYH LSQHGVFSEA DMRFYAAEII
312 322 332 342
LGLEHMHNRF VVYRDLKPAN ILLDEHGHVR ISDLGLACDF
352 362 372 382
SKKKPHASVG THGYMAPEVL QKGVAYDSSA DWFSLGCMLF
392 402 412 422
KLLRGHSPFR QHKTKDKHEI DRMTLTMAVE LPDSFSPELR
432 442 452
SLLEGLLQRD VNRRLGCLGR GAQEVKESPF FRSLDWQMV
Lower-case residues are disordered in structure.
Mutations: None
Phosphorylation: None