7PWD

GRK2 (Beta-adrenergic receptor kinase 1)
Group: AGC
Uniprot: ARBK1_HUMAN
Organism: Homo sapiens
Domain boundary: 191 - 453
Resolu: 2.6

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Inactive DFGin None in-in in-in 8DS Type1 27 - 668 0
Representative sequence - Chain A
10 20 30 40
madleavlad vsylmameks katpaaRASK KILLPEPSIR
50 60 70 80
SVMQKYLEDR GEVTFEKIFS QKLGYLLFRD FCLNHLEEAR
90 100 110 120
PLVEFYEEIK KYEKLETEEE RVARSREIFD SYIMKELLAC
130 140 150 160
SHPFSKSATE HVQGHLGKKQ VPPDLFQPYI EEICQNLRGD
170 180 190 200
VFQKFIESDK FTRFCQWKNV ELNIHLTMND FSVHRIIGRG
210 220 230 240
GFGEVYGCRK ADTGKMYAMK CLDKKRIKMK QGETLALNER
250 260 270 280
IMLSLVSTGD CPFIVCMSYA FHTPDKLSFI LDLMNGGDLH
290 300 310 320
YHLSQHGVFS EADMRFYAAE IILGLEHMHN RFVVYRDLKP
330 340 350 360
ANILLDEHGH VRISDLGLAC DFSKKKPHAS VGTHGYMAPE
370 380 390 400
VLQKGVAYDS SADWFSLGCM LFKLLRGHSP FRQHKTKDKH
410 420 430 440
EIDRMTLTMA VELPDSFSPE LRSLLEGLLQ RDVNRRLGCL
450 460 470 480
GRGAQEVKES PFFRSLDWQM VFLQKYPPPL IPPRGevnaa
490 500 510 520
dafdigsfde edTKGIKLLD SDQELYRNFP LTISERWQQE
530 540 550 560
VAETVFDTIN AETDRLEARK KAKNKQLGHE EDYALGKDCI
570 580 590 600
MHGYMSKMgn pfLTQWQRRY FYLFPNRLEW RGEGEAPQSL
610 620 630 640
LTMEEIQSVE ETQIKERKCL LLKIRGGKQF ILQCDSDPEL
650 660 670 680
VQWKKELRDA YREAQQLVQR VPKMKNKPra pvvelskvpl
-
vqrgsanglg shhhhhh
Lower-case residues are disordered in structure.
Mutations: S670A
Phosphorylation: None