5HE1

GRK2 (Beta-adrenergic receptor kinase 1)
Group: AGC
Uniprot: ARBK1_HUMAN
Organism: Homo sapiens
Domain boundary: 191 - 453
Resolu: 3.15

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in ZS2 Type1 29 - 668 0
Representative sequence - Chain A
38 48 58 68
SKKILLPEPS IRSVMQKYLE DRGEVTFEKI FSQKLGYLLF
78 88 98 108
RDFCLNHLEE ARPLVEFYEE IKKYEKLETE EERVARSREI
118 128 138 148
FDSYIMKELL ACSHPFSKSA TEHVQGHLGK KQVPPDLFQP
158 168 178 188
YIEEICQNLR GDVFQKFIES DKFTRFCQWK NVELNIHLTM
198 208 218 228
NDFSVHRIIG RGGFGEVYGC RKADTGKMYA MKCLDKKRIK
238 248 258 268
MKQGETLALN ERIMLSLVST GDCPFIVCMS YAFHTPDKLS
278 288 298 308
FILDLMNGGD LHYHLSQHGV FSEADMRFYA AEIILGLEHM
318 328 338 348
HNRFVVYRDL KPANILLDEH GHVRISDLGL ACDFSKKKPH
358 368 378 388
ASVGTHGYMA PEVLQKGVAY DSSADWFSLG CMLFKLLRGH
398 408 418 428
SPFRQHKTKD KHEIDRMTLT MAVELPDSFS PELRSLLEGL
438 448 458 468
LQRDVNRRLG CLGRGAQEVK ESPFFRSLDW QMVFLQKYPP
478 488 498 508
PLIPPrgevn aadafdigsf deedTKGIKL LDSDQELYRN
518 528 538 548
FPLTISERWQ QEVAETVFDT INAETDRLEA RKKAKNKqlg
558 568 578 588
HEEDYALGKD CIMHGYMSKM GNPFLTQWQR RYFYLFPNRL
598 608 618 628
EWRGEGEAPQ SLLTMEEIQS VEETQIKERK CLLLKIRGGK
638 648 658 668
QFILQCDSDP ELVQWKKELR DAYREAQQLV QRVPKMKNKP

ra
Lower-case residues are disordered in structure.
Mutations: S670A
Phosphorylation: None