4XX9

PDPK1 (3-phosphoinositide-dependent protein kinase 1)
Group: AGC
Uniprot: PDPK1_HUMAN
Organism: Homo sapiens
Domain boundary: 82 - 342
Resolu: 1.4

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in ATP RF4 RF4 Type1 Allosteric Allosteric 71 - 359 0
Representative sequence - Chain A
59 69 79 89
amdgtaaepr pgagslqhaq pPPQPRKKRP EDFKFGKILG
99 109 119 129
EGSFSTVVLA RELATSREYA IKILEKRHII KENKVPYVTR
139 149 159 169
ERDVMSRLDH PFFVKLYFTF QDDEKLYFGL SYAKNGELLK
179 189 199 209
YIRKIGSFDE TCTRFYTAEI VSALEYLHGK GIIHRDLKPE
219 229 239 249
NILLNEDMHI QITDFGTAKV LSPESKQARA NSFVGTAQYV
259 269 279 289
SPELLTEKSA CKSSDLWALG CIIYQLVAGL PPFRAGNEGL
299 309 319 329
IFAKIIKLEY DFPEKFFPKA RDLVEKLLVL DATKRLGCEE
339 349 359
MEGYGPLKAH PFFESVTWEN LHQQTPPKLT
Lower-case residues are disordered in structure.
Mutations: Y288G,Q292A
Phosphorylation: X241