4CT1

PDPK1 (3-phosphoinositide-dependent protein kinase 1)
Group: AGC
Uniprot: PDPK1_HUMAN
Organism: Homo sapiens
Domain boundary: 82 - 342
Resolu: 1.85

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A None DFGin BLAminus in-none in-in ATP 31S Type1 Allosteric 76 - 359 0
Representative sequence - Chain A
58 68 78 88
gamdgtaaep rpgagslqha qpppqprKKR PEDFKFGKIL
98 108 118 128
GEGSFSTVVL ARELATSREY AIKIVEKRHV HKENKIPYVQ
138 148 158 168
REKDVMSRLD HPFFVKLYFC FQDDEKLYLG LSYAKNGELL
178 188 198 208
KYIRKIGSFD ETCTRFYTAE IVSALEYLHG KGIIHRDLKP
218 228 238 248
ENILLNEDMH IQITDFGTAK VLSPESKQAR ANSFVGTAQY
258 268 278 288
VSPELLTEKS ACKSSDLWAL GCIIYQLVAG LPPFRAGNEG
298 308 318 328
LIFAKIIKLE YDFPEKFFPK ARDLVEKLLV LDATKRLGCE
338 348 358
EMEGYGPLKA HPFFESVTWE NLHQQTPPKL T
Lower-case residues are disordered in structure.
Mutations: L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A
Phosphorylation: X241