3KRW

GRK2 (Beta-adrenergic receptor kinase 1)
Group: AGC
Uniprot: ARBK1_HUMAN
Organism: Homo sapiens
Domain boundary: 191 - 453
Resolu: 2.9

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Inactive DFGin None in-in in-in BA1 Type1 30 - 671 0
Representative sequence - Chain A
11 21 31 41
adleavladv sylmameksk atpaarasKK ILLPEPSIRS
51 61 71 81
VMQKYLEDRG EVTFEKIFSQ KLGYLLFRDF CLNHLEEARP
91 101 111 121
LVEFYEEIKK YEKLETEEER VARSREIFDS YIMKELLAcs
131 141 151 161
HPFSKSATEH VQGHLGKKQV PPDLFQPYIE EICQNLRGDV
171 181 191 201
FQKFIESDKF TRFCQWKNVE LNIHLTMNDF SVHRIIGRGG
211 221 231 241
FGEVYGCRKA DTGKMYAMKC LDKKRIKMKQ GETLALNERI
251 261 271 281
MLSLVSTGDC PFIVCMSYAF HTPDKLSFIL DLMNGGDLHY
291 301 311 321
HLSQHGVFSE ADMRFYAAEI ILGLEHMHNR FVVYRDLKPA
331 341 351 361
NILLDEHGHV RISDLGLACD FSKKKPHASV GTHGYMAPEV
371 381 391 401
LQKGVAYDSS ADWFSLGCML FKLLRGHSPF RQHKTKDKHE
411 421 431 441
IDRMTLTMAV ELPDSFSPEL RSLLEGLLQR DVNRRLGCLG
451 461 471 481
RGAQEVKESP FFRSLDWQMV FLQKYPPPLI PPRgevnaad
491 501 511 521
afdigsfdEE DTKGIKLLDS DQELYRNFPL TISERWQQEV
531 541 551 561
AETVFDTINA ETDRLEARKK AKNKQLGHEE DYALGKDCIM
571 581 591 601
HGYMSKMgnp fltqWQRRYF YLFPNRLEWR GEGEAPQSLL
611 621 631 641
TMEEIQSVEE TQIKERKCLL LKIRGGKQFI LQCDSDPELV
651 661 671 681
QWKKELRDAY REAQQLVQRV PKMKNKPRSP vvelskvplv

qrgsangl
Lower-case residues are disordered in structure.
Mutations: None
Phosphorylation: None