| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KDR | VGFR2_HUMAN | 3EFLA | P35968 | 817 | 1171 | 1356.0 | 706:60501 | Type2 | Inactive | DFGout | 16.1802 | 10.559 | BBAminus | -138.71, -172.72 | -156.17, 97.27 | -59.6, -16.87 | 285.84, 75.59 | 69.09, 999.0 | in-in | in | 7.3332 | Saltbr-in | 2.8225 | HRD-in | -65.88, -53.9 | 89.41, -28.23 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 54.05 | APE8-rot-na | 34.8 | APE67-dihe-in | -59.53, -20.45 | -52.35, -30.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | A | 314.0 | 279.0 | 26 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3efl | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| TYR | KDR | VGFR2_HUMAN | 3EFLB | P35968 | 821 | 1165 | 1356.0 | 706:60502 | Type2 | Inactive | DFGout | 16.1133 | 10.2301 | BBAminus | -141.16, -175.15 | -153.12, 108.94 | -69.6, -34.74 | 280.14, 78.23 | 138.83, 999.0 | in-in | in | 7.0963 | Saltbr-in | 3.2421 | HRD-in | -62.3, -53.81 | 81.7, -4.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.71 | APE8-dihe-out | -39.02, -20.75 | APE8-rot-na | 27.77 | APE67-dihe-in | -68.47, -11.11 | -59.68, -39.14 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.8201 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | B | 314.0 | 263.0 | 32 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3efl | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KDR | VGFR2_HUMAN | 3EFLA | P35968 | 817 | 1171 | 1356.0 | 706:60501 | Type2 | Inactive | DFGout | 16.1802 | 10.559 | BBAminus | -138.71, -172.72 | -156.17, 97.27 | -59.6, -16.87 | 285.84, 75.59 | 69.09, 999.0 | in-in | in | 7.3332 | Saltbr-in | 2.8225 | HRD-in | -65.88, -53.9 | 89.41, -28.23 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 54.05 | APE8-rot-na | 34.8 | APE67-dihe-in | -59.53, -20.45 | -52.35, -30.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | A | 314.0 | 279.0 | 26 | 30 | 11 | 19 | [[834, 1162]] | 1.0 | 3efl | Homo sapiens | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| TYR | KDR | VGFR2_HUMAN | 3EFLB | P35968 | 821 | 1165 | 1356.0 | 706:60502 | Type2 | Inactive | DFGout | 16.1133 | 10.2301 | BBAminus | -141.16, -175.15 | -153.12, 108.94 | -69.6, -34.74 | 280.14, 78.23 | 138.83, 999.0 | in-in | in | 7.0963 | Saltbr-in | 3.2421 | HRD-in | -62.3, -53.81 | 81.7, -4.86 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.71 | APE8-dihe-out | -39.02, -20.75 | APE8-rot-na | 27.77 | APE67-dihe-in | -68.47, -11.11 | -59.68, -39.14 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.8201 | C817A,E990V | PTR1054,PTR1059 | PTR1054,PTR1059 | XRAY | 2.2 | 0.23 | 0.264 | B | 314.0 | 263.0 | 32 | 30 | 12 | 18 | [[834, 1162]] | 1.0 | 3efl | Homo sapiens | TYR_KDR_HUMAN | TYR | 4e-100 | 340.4 | 1.0 | 260.0 | 260.0 | 1045 | 1046 | 1047 | 1049 | 1051 | 868 | 885 | 889 | 1025 | 1027 | 1026 | 1028.0 | 1087 | 1075 | 1070 | 1069 | 1068 | 1067 | 1066 | 1065 | 1064 | 917 | Vascular endothelial growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|