| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK2 | ARBK1_BOVIN | 1YM7B | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1989 | 12.4485 | ABAminus | -130.8, -59.92 | -98.26, 108.63 | -91.58, -9.04 | 306.19, 95.69 | -36.4, -48.74 | in-out | in | 8.8033 | Saltbr-out | 4.6419 | HRD-in | -77.09, -44.3 | 73.62, -27.39 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7591 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.17, 125.32 | APE9-dihe-na | 152.82, 174.56 | APE8-dihe-in | -87.32, 142.62 | APE8-rot-in | 313.75 | APE67-dihe-in | -64.86, -36.54 | -62.56, -29.46 | APE12-dist-in | 9.8182 | APE11-dist-in | 11.5603 | APE10-dist-in | 5.5731 | APE9-dist-in | 4.0361 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | B | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| AGC | GRK2 | ARBK1_BOVIN | 1YM7A | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2239 | 12.3565 | None | -125.66, -66.29 | -94.21, 107.11 | -86.73, -10.11 | 307.87, 97.53 | -38.26, -47.46 | in-out | in | 8.8531 | Saltbr-out | 4.6372 | HRD-in | -74.94, -45.18 | 74.24, -26.22 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7715 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.74, 123.21 | APE9-dihe-na | 155.55, 174.57 | APE8-dihe-in | -86.11, 141.22 | APE8-rot-in | 314.43 | APE67-dihe-in | -66.31, -34.76 | -64.21, -27.3 | APE12-dist-in | 9.8313 | APE11-dist-in | 11.5432 | APE10-dist-in | 5.5926 | APE9-dist-in | 3.9926 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | A | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| AGC | GRK2 | ARBK1_BOVIN | 1YM7C | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2163 | 12.2674 | None | -130.34, -66.38 | -92.79, 106.85 | -85.97, -13.2 | 309.12, 95.06 | -35.96, -48.47 | in-out | in | 8.8136 | Saltbr-out | 4.7358 | HRD-in | -75.86, -48.89 | 75.97, -29.41 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.721 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.29, 128.8 | APE9-dihe-na | 145.96, 173.8 | APE8-dihe-in | -87.44, 141.12 | APE8-rot-in | 314.72 | APE67-dihe-in | -67.09, -36.43 | -60.22, -25.52 | APE12-dist-in | 9.7747 | APE11-dist-in | 11.5691 | APE10-dist-in | 5.6074 | APE9-dist-in | 4.0582 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | C | 689.0 | 607.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| AGC | GRK2 | ARBK1_BOVIN | 1YM7D | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2341 | 12.3436 | None | -128.88, -67.33 | -92.65, 105.41 | -87.88, -10.71 | 307.83, 96.53 | -37.49, -49.46 | in-out | in | 8.801 | Saltbr-out | 4.7459 | HRD-in | -72.13, -45.13 | 72.62, -27.86 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7633 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.27, 125.22 | APE9-dihe-na | 149.39, 173.11 | APE8-dihe-in | -84.5, 141.69 | APE8-rot-in | 315.18 | APE67-dihe-in | -66.11, -35.98 | -62.26, -27.83 | APE12-dist-in | 9.7362 | APE11-dist-in | 11.4974 | APE10-dist-in | 5.5333 | APE9-dist-in | 4.0286 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | D | 689.0 | 599.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK2 | ARBK1_BOVIN | 1YM7B | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1989 | 12.4485 | ABAminus | -130.8, -59.92 | -98.26, 108.63 | -91.58, -9.04 | 306.19, 95.69 | -36.4, -48.74 | in-out | in | 8.8033 | Saltbr-out | 4.6419 | HRD-in | -77.09, -44.3 | 73.62, -27.39 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7591 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.17, 125.32 | APE9-dihe-na | 152.82, 174.56 | APE8-dihe-in | -87.32, 142.62 | APE8-rot-in | 313.75 | APE67-dihe-in | -64.86, -36.54 | -62.56, -29.46 | APE12-dist-in | 9.8182 | APE11-dist-in | 11.5603 | APE10-dist-in | 5.5731 | APE9-dist-in | 4.0361 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | B | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| AGC | GRK2 | ARBK1_BOVIN | 1YM7A | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2239 | 12.3565 | None | -125.66, -66.29 | -94.21, 107.11 | -86.73, -10.11 | 307.87, 97.53 | -38.26, -47.46 | in-out | in | 8.8531 | Saltbr-out | 4.6372 | HRD-in | -74.94, -45.18 | 74.24, -26.22 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7715 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.74, 123.21 | APE9-dihe-na | 155.55, 174.57 | APE8-dihe-in | -86.11, 141.22 | APE8-rot-in | 314.43 | APE67-dihe-in | -66.31, -34.76 | -64.21, -27.3 | APE12-dist-in | 9.8313 | APE11-dist-in | 11.5432 | APE10-dist-in | 5.5926 | APE9-dist-in | 3.9926 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | A | 689.0 | 608.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| AGC | GRK2 | ARBK1_BOVIN | 1YM7C | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2163 | 12.2674 | None | -130.34, -66.38 | -92.79, 106.85 | -85.97, -13.2 | 309.12, 95.06 | -35.96, -48.47 | in-out | in | 8.8136 | Saltbr-out | 4.7358 | HRD-in | -75.86, -48.89 | 75.97, -29.41 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.721 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -118.29, 128.8 | APE9-dihe-na | 145.96, 173.8 | APE8-dihe-in | -87.44, 141.12 | APE8-rot-in | 314.72 | APE67-dihe-in | -67.09, -36.43 | -60.22, -25.52 | APE12-dist-in | 9.7747 | APE11-dist-in | 11.5691 | APE10-dist-in | 5.6074 | APE9-dist-in | 4.0582 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | C | 689.0 | 607.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |
| AGC | GRK2 | ARBK1_BOVIN | 1YM7D | P21146 | 29 | 656 | 689.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2341 | 12.3436 | None | -128.88, -67.33 | -92.65, 105.41 | -87.88, -10.71 | 307.83, 96.53 | -37.49, -49.46 | in-out | in | 8.801 | Saltbr-out | 4.7459 | HRD-in | -72.13, -45.13 | 72.62, -27.86 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7633 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -116.27, 125.22 | APE9-dihe-na | 149.39, 173.11 | APE8-dihe-in | -84.5, 141.69 | APE8-rot-in | 315.18 | APE67-dihe-in | -66.11, -35.98 | -62.26, -27.83 | APE12-dist-in | 9.7362 | APE11-dist-in | 11.4974 | APE10-dist-in | 5.5333 | APE9-dist-in | 4.0286 | S670A | None | None | XRAY | 4.5 | 0.226 | 0.279 | D | 689.0 | 599.0 | 0 | 26 | 26 | 0 | [[191, 453]] | 1.0 | 1ym7 | Bos taurus | AGC_GRK2_BOVIN | AGC | 6.3e-77 | 268.8 | 1.0 | 260.0 | 260.0 | 334 | 335 | 336 | 338 | 340 | 220 | 239 | 243 | 314 | 316 | 315 | 317.0 | 373 | 360 | 355 | 354 | 353 | 352 | 351 | 350 | 349 | 272 | Beta-adrenergic receptor kinase 1 |