Ligand: VSE

Total number of chains: 9
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLBplus 9 100.0% 5ZJ6A

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Family Gene UniprotID PDB Resolution Activity_label Spatial_Dihedral_labels ChelixSaltbr_label ActLoopNT-ActLoopCT APEtype APEdihe_label APEdist_label Ligand Ligand_type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
TYR FGR FGR_HUMAN 7UY0A 2.55 Inactive DFGin‑BLBplus out-out out-in TYR APEdihe_iiiai APEdist_aaai VSE Type1.5_Back 80 - 527 0 PTR523 Q524E,P525E,G526I,D527P Tyrosine-protein kinase Fgr
TYR FGR FGR_HUMAN 7UY0B 2.55 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_iiiai APEdist_aaao VSE Type1.5_Back 80 - 527 0 PTR523 Q524E,P525E,G526I,D527P Tyrosine-protein kinase Fgr
TYR HCK HCK_HUMAN 5ZJ6A 1.696 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_oiiai APEdist_aaai VSE Type1 248 - 518 0 None None Tyrosine-protein kinase HCK
TYR HCK HCK_HUMAN 5ZJ6B 1.696 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_oiiai APEdist_aaai VSE Type1.5_Back 249 - 518 0 None None Tyrosine-protein kinase HCK
TYR HCK HCK_HUMAN 9BYJA 1.8 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_oiiai APEdist_aaai VSE Type1.5_Back 81 - 526 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK
TYR HCK HCK_HUMAN 3VS3A 2.17 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_nniai APEdist_aaao VSE Type1.5_Back 81 - 526 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK
TYR HCK HCK_HUMAN 3VS3B 2.17 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_niiai APEdist_aaao VSE Type1.5_Back 81 - 526 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK
TYR HCK HCK_HUMAN 4LUEA 3.04 Inactive DFGin‑BLBplus out-out out-none TYR APEdihe_nnnai APEdist_aaan VSE Type1.5_Back 81 - 525 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK
TYR HCK HCK_HUMAN 4LUEB 3.04 Inactive DFGin‑BLBplus out-out out-none TYR APEdihe_nnnai APEdist_aaan VSE Type1.5_Back 81 - 525 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK

Ligand: VSE

Total number of chains: 9
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLBplus 9 100.0% 5ZJ6A

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Family Gene UniprotID PDB Resolution Activity_label Spatial_Dihedral_labels ChelixSaltbr_label ActLoopNT-ActLoopCT APEtype APEdihe_label APEdist_label Ligand Ligand_type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
TYR FGR FGR_HUMAN 7UY0A 2.55 Inactive DFGin‑BLBplus out-out out-in TYR APEdihe_iiiai APEdist_aaai VSE Type1.5_Back 80 - 527 0 PTR523 Q524E,P525E,G526I,D527P Tyrosine-protein kinase Fgr Homo sapiens
TYR FGR FGR_HUMAN 7UY0B 2.55 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_iiiai APEdist_aaao VSE Type1.5_Back 80 - 527 0 PTR523 Q524E,P525E,G526I,D527P Tyrosine-protein kinase Fgr Homo sapiens
TYR HCK HCK_HUMAN 5ZJ6A 1.696 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_oiiai APEdist_aaai VSE Type1 248 - 518 0 None None Tyrosine-protein kinase HCK Homo sapiens
TYR HCK HCK_HUMAN 5ZJ6B 1.696 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_oiiai APEdist_aaai VSE Type1.5_Back 249 - 518 0 None None Tyrosine-protein kinase HCK Homo sapiens
TYR HCK HCK_HUMAN 9BYJA 1.8 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_oiiai APEdist_aaai VSE Type1.5_Back 81 - 526 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK Homo sapiens
TYR HCK HCK_HUMAN 3VS3A 2.17 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_nniai APEdist_aaao VSE Type1.5_Back 81 - 526 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK Homo sapiens
TYR HCK HCK_HUMAN 3VS3B 2.17 Inactive DFGin‑BLBplus out-out out-out TYR APEdihe_niiai APEdist_aaao VSE Type1.5_Back 81 - 526 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK Homo sapiens
TYR HCK HCK_HUMAN 4LUEA 3.04 Inactive DFGin‑BLBplus out-out out-none TYR APEdihe_nnnai APEdist_aaan VSE Type1.5_Back 81 - 525 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK Homo sapiens
TYR HCK HCK_HUMAN 4LUEB 3.04 Inactive DFGin‑BLBplus out-out out-none TYR APEdihe_nnnai APEdist_aaan VSE Type1.5_Back 81 - 525 0 PTR522 Q523E,Q524E,Q525I Tyrosine-protein kinase HCK Homo sapiens

Ligand: VSE

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Family Gene UniprotID PDB Resolution Activity_label Spatial_Dihedral_labels ChelixSaltbr_label ActLoopNT-ActLoopCT APEtype APEdihe_label APEdist_label Ligand Ligand_type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism