Ligand: BI4

Total number of chains: 5
Active chains: 1
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 5 100.0% 3OTUA

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AGC PDPK1 PDPK1_HUMAN 3ORZA O15530 74 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.622 14.605 BLAminus -134.96, -167.36 70.2, 66.13 -101.26, 0.99 293.7, 88.7 -61.05, -29.24 in-in in 8.215 Saltbr-in 2.81 HRD-in -65.12, -49.46 75.7, -10.07 in-in-out SNCiio in-out ActLoopNT-in 2.833 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -134.38, 111.86 APE9-dihe-na -60.27, -174.97 APE8-dihe-in -55.74, 132.42 APE8-rot-in 303.15 APE67-dihe-in -56.98, -32.17 -55.27, -42.37 APE12-dist-in 11.549 APE11-dist-out 6.544 APE10-dist-out 10.866 APE9-dist-in 4.117 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 A 316 277 9 0 0 9 [[82, 342]] 1.0 3orz AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3ORZB O15530 73 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.648 14.776 BLAminus -139.38, -168.66 74.13, 69.92 -111.18, 3.04 284.6, 93.64 -63.39, -24.83 in-in in 8.292 Saltbr-in 2.759 HRD-in -64.66, -48.81 76.86, -10.42 in-in-out SNCiio in-out ActLoopNT-in 2.866 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -131.43, 114.97 APE9-dihe-na -62.67, -167.65 APE8-dihe-in -63.67, 131.38 APE8-rot-in 299.84 APE67-dihe-in -54.64, -32.97 -56.45, -39.98 APE12-dist-in 11.638 APE11-dist-out 6.397 APE10-dist-out 10.787 APE9-dist-in 4.087 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 B 316 279 8 0 0 8 [[82, 342]] 1.0 3orz AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3ORZC O15530 74 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.667 14.679 BLAminus -134.07, -170.51 76.79, 69.39 -110.34, 1.38 287.93, 89.81 -56.71, -30.43 in-in in 8.225 Saltbr-in 2.804 HRD-in -64.4, -49.76 78.61, -9.94 in-in-out SNCiio in-out ActLoopNT-in 2.805 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -134.53, 111.0 APE9-dihe-na -58.83, -174.56 APE8-dihe-in -56.66, 132.63 APE8-rot-in 302.29 APE67-dihe-in -56.84, -32.58 -55.43, -42.03 APE12-dist-in 11.731 APE11-dist-out 6.55 APE10-dist-out 10.875 APE9-dist-in 4.082 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 C 316 277 9 0 0 9 [[82, 342]] 1.0 3orz AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3ORZD O15530 73 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.649 14.774 BLAminus -139.63, -168.42 74.39, 69.06 -110.33, 3.29 285.32, 93.06 -63.48, -24.84 in-in in 8.31 Saltbr-in 2.754 HRD-in -64.65, -47.43 73.97, -9.52 in-in-out SNCiio in-out ActLoopNT-in 2.877 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -126.78, 121.12 APE9-dihe-na -63.33, -166.44 APE8-dihe-in -63.66, 131.18 APE8-rot-in 301.29 APE67-dihe-in -54.43, -33.46 -55.31, -40.36 APE12-dist-in 11.584 APE11-dist-out 6.406 APE10-dist-out 10.842 APE9-dist-in 4.04 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 D 316 279 8 0 0 8 [[82, 342]] 1.0 3orz AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3OTUA O15530 77 359 556.0 J30:1,BI4:360 Allosteric,Type1.5_Front Active DFGin 6.407 14.986 BLAminus -147.19, -166.49 62.44, 61.65 -95.64, 10.19 290.91, 105.88 -63.28, -24.6 in-in in 8.37 Saltbr-in 3.337 HRD-in -67.23, -53.13 82.11, -16.93 in-in-in SNCiii in-in ActLoopNT-in 2.795 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.97, 157.81 APE9-dihe-na 151.4, -176.81 APE8-dihe-in -123.26, 126.19 APE8-rot-in 294.94 APE67-dihe-in -53.95, -30.51 -40.25, -53.87 APE12-dist-in 7.712 APE11-dist-in 10.329 APE10-dist-in 5.244 APE9-dist-in 4.13 T148C SEP241 SEP241 XRAY 2.101 0.197 0.24 A 316 277 6 0 0 5 [[82, 342]] 1.0 3otu AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1

Ligand: BI4

Total number of chains: 7
Active chains: 2
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 6 85.7% 1SZMA
DFGin ABAminus 1 14.3% 1SZMB

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AGC PRKACA KAPCA_BOVIN 1SZMB P00517 15 351 351.0 BI4:60351 Type1 Inactive DFGin 6.916 16.017 ABAminus -124.67, -37.03 -119.38, 110.7 -112.86, 23.01 290.52, 94.06 -59.96, -45.74 out-out out 10.618 Saltbr-out 4.666 HRD-in -70.48, -44.14 31.9, 37.49 out-in-in SNCoii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.49, 166.21 APE9-dihe-na 109.44, 164.47 APE8-dihe-in -71.29, 133.53 APE8-rot-in 294.81 APE67-dihe-in -63.33, -24.2 -45.0, -46.86 APE12-dist-in 8.346 APE11-dist-in 11.522 APE10-dist-in 5.985 APE9-dist-in 4.445 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 B 350 323 0 0 0 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_BOVIN 1SZMA P00517 16 351 351.0 BI4:60351 Type1 Active DFGin 6.318 15.368 BLAminus -125.27, 171.81 65.17, 99.61 -108.03, 19.56 272.67, 80.44 -58.01, -35.62 in-in in 9.492 Saltbr-in 2.574 HRD-in -86.5, -61.07 68.65, 7.7 in-in-in SNCiii in-in ActLoopNT-in 3.003 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 163.31 APE9-dihe-na 107.11, 170.89 APE8-dihe-in -74.89, 129.09 APE8-rot-in 328.61 APE67-dihe-in -51.73, -30.1 -54.41, -49.2 APE12-dist-in 8.04 APE11-dist-in 11.33 APE10-dist-in 5.763 APE9-dist-in 3.806 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 A 350 320 0 0 0 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PDPK1 PDPK1_HUMAN 3ORZA O15530 74 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.622 14.605 BLAminus -134.96, -167.36 70.2, 66.13 -101.26, 0.99 293.7, 88.7 -61.05, -29.24 in-in in 8.215 Saltbr-in 2.81 HRD-in -65.12, -49.46 75.7, -10.07 in-in-out SNCiio in-out ActLoopNT-in 2.833 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -134.38, 111.86 APE9-dihe-na -60.27, -174.97 APE8-dihe-in -55.74, 132.42 APE8-rot-in 303.15 APE67-dihe-in -56.98, -32.17 -55.27, -42.37 APE12-dist-in 11.549 APE11-dist-out 6.544 APE10-dist-out 10.866 APE9-dist-in 4.117 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 A 316 277 9 0 0 9 [[82, 342]] 1.0 3orz Homo sapiens AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3ORZB O15530 73 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.648 14.776 BLAminus -139.38, -168.66 74.13, 69.92 -111.18, 3.04 284.6, 93.64 -63.39, -24.83 in-in in 8.292 Saltbr-in 2.759 HRD-in -64.66, -48.81 76.86, -10.42 in-in-out SNCiio in-out ActLoopNT-in 2.866 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -131.43, 114.97 APE9-dihe-na -62.67, -167.65 APE8-dihe-in -63.67, 131.38 APE8-rot-in 299.84 APE67-dihe-in -54.64, -32.97 -56.45, -39.98 APE12-dist-in 11.638 APE11-dist-out 6.397 APE10-dist-out 10.787 APE9-dist-in 4.087 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 B 316 279 8 0 0 8 [[82, 342]] 1.0 3orz Homo sapiens AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3ORZC O15530 74 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.667 14.679 BLAminus -134.07, -170.51 76.79, 69.39 -110.34, 1.38 287.93, 89.81 -56.71, -30.43 in-in in 8.225 Saltbr-in 2.804 HRD-in -64.4, -49.76 78.61, -9.94 in-in-out SNCiio in-out ActLoopNT-in 2.805 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -134.53, 111.0 APE9-dihe-na -58.83, -174.56 APE8-dihe-in -56.66, 132.63 APE8-rot-in 302.29 APE67-dihe-in -56.84, -32.58 -55.43, -42.03 APE12-dist-in 11.731 APE11-dist-out 6.55 APE10-dist-out 10.875 APE9-dist-in 4.082 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 C 316 277 9 0 0 9 [[82, 342]] 1.0 3orz Homo sapiens AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3ORZD O15530 73 359 556.0 2A2:1,BI4:360 Allosteric,Type1 Inactive DFGin 6.649 14.774 BLAminus -139.63, -168.42 74.39, 69.06 -110.33, 3.29 285.32, 93.06 -63.48, -24.84 in-in in 8.31 Saltbr-in 2.754 HRD-in -64.65, -47.43 73.97, -9.52 in-in-out SNCiio in-out ActLoopNT-in 2.877 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_iooi APE10-dihe-na -126.78, 121.12 APE9-dihe-na -63.33, -166.44 APE8-dihe-in -63.66, 131.18 APE8-rot-in 301.29 APE67-dihe-in -54.43, -33.46 -55.31, -40.36 APE12-dist-in 11.584 APE11-dist-out 6.406 APE10-dist-out 10.842 APE9-dist-in 4.04 T148C SEP241 SEP241 XRAY 2.0 0.22 0.265 D 316 279 8 0 0 8 [[82, 342]] 1.0 3orz Homo sapiens AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1
AGC PDPK1 PDPK1_HUMAN 3OTUA O15530 77 359 556.0 J30:1,BI4:360 Allosteric,Type1.5_Front Active DFGin 6.407 14.986 BLAminus -147.19, -166.49 62.44, 61.65 -95.64, 10.19 290.91, 105.88 -63.28, -24.6 in-in in 8.37 Saltbr-in 3.337 HRD-in -67.23, -53.13 82.11, -16.93 in-in-in SNCiii in-in ActLoopNT-in 2.795 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -141.97, 157.81 APE9-dihe-na 151.4, -176.81 APE8-dihe-in -123.26, 126.19 APE8-rot-in 294.94 APE67-dihe-in -53.95, -30.51 -40.25, -53.87 APE12-dist-in 7.712 APE11-dist-in 10.329 APE10-dist-in 5.244 APE9-dist-in 4.13 T148C SEP241 SEP241 XRAY 2.101 0.197 0.24 A 316 277 6 0 0 5 [[82, 342]] 1.0 3otu Homo sapiens AGC_PDPK1_HUMAN AGC 7.9e-85 290.0 1 260 260 222 223 224 226 228 111 130 134 202 204 203 205 264 252 247 246 245 244 243 242 241 160 3-phosphoinositide-dependent protein kinase 1

Ligand: BI4

Total number of chains: 2
Active chains: 1
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 1 50.0% 1SZMB
DFGin BLAminus 1 50.0% 1SZMA

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AGC PRKACA KAPCA_BOVIN 1SZMB P00517 15 351 351.0 BI4:60351 Type1 Inactive DFGin 6.916 16.017 ABAminus -124.67, -37.03 -119.38, 110.7 -112.86, 23.01 290.52, 94.06 -59.96, -45.74 out-out out 10.618 Saltbr-out 4.666 HRD-in -70.48, -44.14 31.9, 37.49 out-in-in SNCoii in-in ActLoopNT-in 3.019 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -137.49, 166.21 APE9-dihe-na 109.44, 164.47 APE8-dihe-in -71.29, 133.53 APE8-rot-in 294.81 APE67-dihe-in -63.33, -24.2 -45.0, -46.86 APE12-dist-in 8.346 APE11-dist-in 11.522 APE10-dist-in 5.985 APE9-dist-in 4.445 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 B 350 323 0 0 0 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha
AGC PRKACA KAPCA_BOVIN 1SZMA P00517 16 351 351.0 BI4:60351 Type1 Active DFGin 6.318 15.368 BLAminus -125.27, 171.81 65.17, 99.61 -108.03, 19.56 272.67, 80.44 -58.01, -35.62 in-in in 9.492 Saltbr-in 2.574 HRD-in -86.5, -61.07 68.65, 7.7 in-in-in SNCiii in-in ActLoopNT-in 3.003 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.54, 163.31 APE9-dihe-na 107.11, 170.89 APE8-dihe-in -74.89, 129.09 APE8-rot-in 328.61 APE67-dihe-in -51.73, -30.1 -54.41, -49.2 APE12-dist-in 8.04 APE11-dist-in 11.33 APE10-dist-in 5.763 APE9-dist-in 3.806 V124A,L174M,Q182K SEP140,TPO198,SEP339 SEP140,TPO198,SEP339 XRAY 2.5 0.234 0.289 A 350 320 0 0 0 0 [[44, 298]] 1.0 1szm Bos taurus AGC_PRKACA_BOVIN AGC 1.6e-94 321.9 1 260 260 184 185 186 188 190 73 92 96 164 166 165 167 221 209 204 203 202 201 200 199 198 122 cAMP-dependent protein kinase catalytic subunit alpha