| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| STE | STK3 | STK3_HUMAN | 5DH3B | Q13188 | 18 | 302 | 491.0 | 5BS:401 | Type1 | Inactive | DFGin | 5.7864 | 14.8202 | ABAminus | -107.93, -47.86 | -103.07, 119.05 | -112.25, 18.06 | 290.67, 93.25 | -61.59, -41.21 | out-in | out | 10.1371 | Saltbr-in | 3.2082 | HRD-in | -63.36, -51.22 | 81.92, -5.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7123 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -158.17, 161.15 | APE9-dihe-na | 132.06, -164.99 | APE8-dihe-in | -104.21, 128.47 | APE8-rot-in | 313.02 | APE67-dihe-in | -62.35, -41.65 | -60.99, -39.89 | APE12-dist-in | 8.8777 | APE11-dist-in | 11.4071 | APE10-dist-in | 5.8267 | APE9-dist-in | 3.6653 | None | TPO174,TPO180 | TPO174,TPO180 | XRAY | 2.468 | 0.213 | 0.247 | B | 315.0 | 285.0 | 0 | 28 | 28 | 0 | [[27, 278]] | 1.0 | 5dh3 | STE_STK3_HUMAN | STE | 2.8e-101 | 344.2 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK3 | STK3_HUMAN | 8A66A | Q13188 | 24 | 303 | 491.0 | 5BS:60501 | Type1 | Inactive | DFGin | 6.2317 | 14.6625 | BLAminus | -139.57, 162.57 | 72.11, 84.59 | -98.16, 23.52 | 293.51, 92.3 | -65.59, -22.75 | in-in | in | 9.5593 | Saltbr-in | 2.7359 | HRD-in | -65.32, -44.41 | 72.25, -5.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.838 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -147.11, 158.64 | APE9-dihe-na | 124.6, -157.27 | APE8-dihe-in | -114.81, 122.93 | APE8-rot-out | 43.78 | APE67-dihe-in | -62.92, -24.25 | -35.94, -56.9 | APE12-dist-in | 8.6802 | APE11-dist-in | 11.8235 | APE10-dist-in | 5.9829 | APE9-dist-in | 3.5305 | None | TPO180 | TPO180 | XRAY | 1.901 | 0.22 | 0.258 | A | 298.0 | 275.0 | 5 | 28 | 27 | 1 | [[27, 278]] | 1.0 | 8a66 | STE_STK3_HUMAN | STE | 2.3e-101 | 344.5 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK3 | STK3_HUMAN | 8A66B | Q13188 | 18 | 304 | 491.0 | 5BS:60501 | Type1 | Inactive | DFGin | 6.2293 | 14.4906 | BLAminus | -139.08, 162.57 | 69.6, 85.67 | -96.89, 21.95 | 294.07, 84.34 | -63.47, -19.34 | in-in | in | 9.5136 | Saltbr-in | 2.883 | HRD-in | -65.79, -48.59 | 72.98, -4.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8323 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -146.04, 152.12 | APE9-dihe-na | 134.76, -156.35 | APE8-dihe-in | -108.07, 116.58 | APE8-rot-out | 42.21 | APE67-dihe-in | -60.0, -23.48 | -33.57, -55.3 | APE12-dist-in | 8.6046 | APE11-dist-in | 11.7522 | APE10-dist-in | 5.9813 | APE9-dist-in | 3.4102 | None | TPO174,TPO180,TPO268 | TPO174,TPO180,TPO268 | XRAY | 1.901 | 0.22 | 0.258 | B | 298.0 | 282.0 | 5 | 28 | 28 | 0 | [[27, 278]] | 1.0 | 8a66 | STE_STK3_HUMAN | STE | 2.3e-101 | 344.5 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK3 | STK3_HUMAN | 5DH3A | Q13188 | 19 | 307 | 491.0 | 5BS:401 | Type1 | Inactive | DFGin | 5.9475 | 14.6144 | BLAminus | -145.26, 166.53 | 56.21, 58.22 | -79.02, 55.98 | 309.22, 59.68 | -65.37, -40.98 | out-out | out | 10.1578 | Saltbr-out | 3.8887 | HRD-in | -64.99, -53.25 | 81.51, -5.49 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8183 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -156.11, 158.66 | APE9-dihe-na | 133.82, -164.61 | APE8-dihe-in | -99.88, 125.54 | APE8-rot-in | 317.53 | APE67-dihe-in | -61.6, -38.71 | -57.46, -40.82 | APE12-dist-in | 8.8819 | APE11-dist-in | 11.3596 | APE10-dist-in | 5.7728 | APE9-dist-in | 3.3878 | None | TPO174,TPO180 | TPO174,TPO180 | XRAY | 2.468 | 0.213 | 0.247 | A | 315.0 | 289.0 | 0 | 28 | 28 | 0 | [[27, 278]] | 1.0 | 5dh3 | STE_STK3_HUMAN | STE | 2.8e-101 | 344.2 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK4 | STK4_HUMAN | 8A5JA | Q13043 | 28 | 309 | 487.0 | 5BS:60501 | Type1 | Active | DFGin | 6.1115 | 14.4237 | BLAminus | -137.01, 164.18 | 68.22, 83.42 | -95.37, 24.9 | 295.6, 83.78 | -58.89, -29.18 | in-in | in | 9.5782 | Saltbr-in | 2.6601 | HRD-in | -62.52, -46.35 | 71.81, -5.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.816 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.87, 157.76 | APE9-dihe-na | 133.26, -159.59 | APE8-dihe-in | -112.62, 116.79 | APE8-rot-in | 307.48 | APE67-dihe-in | -60.45, -27.7 | -37.29, -52.56 | APE12-dist-in | 8.4002 | APE11-dist-in | 11.5567 | APE10-dist-in | 5.8785 | APE9-dist-in | 3.3033 | None | TPO177,TPO183 | TPO177,TPO183 | XRAY | 2.123 | 0.243 | 0.248 | A | 282.0 | 279.0 | 3 | 28 | 28 | 0 | [[30, 281]] | 1.0 | 8a5j | STE_STK4_HUMAN | STE | 2.9e-102 | 347.4 | 2.0 | 257.0 | 256.0 | 166 | 167 | 168 | 170 | 172 | 59 | 73 | 77 | 146 | 148 | 147 | 149.0 | 206 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 103 | Serine/threonine-protein kinase 4 |
| STE | STK4 | STK4_HUMAN | 8A5JB | Q13043 | 32 | 309 | 487.0 | 5BS:60501 | Type1 | Inactive | None | 6.1832 | 999.0 | None | -136.98, 164.64 | 68.65, 82.94 | -95.0, 23.57 | 294.73, 84.74 | -56.91, -33.47 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -61.94, -46.75 | 72.95, -3.57 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.7991 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.28, 156.86 | APE9-dihe-na | 133.22, -159.66 | APE8-dihe-in | -113.06, 118.47 | APE8-rot-in | 300.84 | APE67-dihe-in | -66.93, -24.0 | -39.55, -46.8 | APE12-dist-in | 8.294 | APE11-dist-in | 11.5278 | APE10-dist-in | 5.8585 | APE9-dist-in | 3.2972 | None | TPO177,TPO183 | TPO177,TPO183 | XRAY | 2.123 | 0.243 | 0.248 | B | 282.0 | 249.0 | 31 | 28 | 28 | 0 | [[30, 281]] | 1.0 | 8a5j | STE_STK4_HUMAN | STE | 2.9e-102 | 347.4 | 2.0 | 257.0 | 256.0 | 166 | 167 | 168 | 170 | 172 | 59 | 73 | 77 | 146 | 148 | 147 | 149.0 | 206 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 103 | Serine/threonine-protein kinase 4 |
| TYR | JAK2-1 | JAK2_HUMAN | 6BRWA | O60674 | 537 | 808 | 1132.0 | 5BS:901 | Type1 | Pseudo | DFGin | 7.7052 | 13.3794 | None | -93.41, 174.89 | -67.04, 156.04 | -83.01, 0.59 | 33.82, 139.96 | 67.03, -167.12 | in-na | in | 9.6698 | Saltbr-na | 999.0 | HRD-in | -76.15, -62.39 | 95.18, -6.76 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.3464 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -74.9, -35.05 | APE9-dihe-out | -58.77, -25.82 | APE8-dihe-out | -90.17, 2.34 | APE8-rot-na | 284.96 | APE67-dihe-out | -99.82, 21.48 | -62.86, 134.79 | APE12-dist-na | 9.9909 | APE11-dist-na | 11.5633 | APE10-dist-na | 16.1812 | APE9-dist-out | 12.8111 | W659A,W777A,F794H | None | None | XRAY | 2.031 | 0.197 | 0.25 | A | 289.0 | 272.0 | 0 | 24 | 24 | 0 | [[545, 807], [849, 1125]] | 2.0 | 6brw | TYR_JAK2-1_HUMAN | TYR | 1.9e-64 | 223.4 | 2.0 | 260.0 | 259.0 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673.0 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| STE | STK3 | STK3_HUMAN | 5DH3B | Q13188 | 18 | 302 | 491.0 | 5BS:401 | Type1 | Inactive | DFGin | 5.7864 | 14.8202 | ABAminus | -107.93, -47.86 | -103.07, 119.05 | -112.25, 18.06 | 290.67, 93.25 | -61.59, -41.21 | out-in | out | 10.1371 | Saltbr-in | 3.2082 | HRD-in | -63.36, -51.22 | 81.92, -5.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7123 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -158.17, 161.15 | APE9-dihe-na | 132.06, -164.99 | APE8-dihe-in | -104.21, 128.47 | APE8-rot-in | 313.02 | APE67-dihe-in | -62.35, -41.65 | -60.99, -39.89 | APE12-dist-in | 8.8777 | APE11-dist-in | 11.4071 | APE10-dist-in | 5.8267 | APE9-dist-in | 3.6653 | None | TPO174,TPO180 | TPO174,TPO180 | XRAY | 2.468 | 0.213 | 0.247 | B | 315.0 | 285.0 | 0 | 28 | 28 | 0 | [[27, 278]] | 1.0 | 5dh3 | Homo sapiens | STE_STK3_HUMAN | STE | 2.8e-101 | 344.2 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK3 | STK3_HUMAN | 8A66A | Q13188 | 24 | 303 | 491.0 | 5BS:60501 | Type1 | Inactive | DFGin | 6.2317 | 14.6625 | BLAminus | -139.57, 162.57 | 72.11, 84.59 | -98.16, 23.52 | 293.51, 92.3 | -65.59, -22.75 | in-in | in | 9.5593 | Saltbr-in | 2.7359 | HRD-in | -65.32, -44.41 | 72.25, -5.9 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.838 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -147.11, 158.64 | APE9-dihe-na | 124.6, -157.27 | APE8-dihe-in | -114.81, 122.93 | APE8-rot-out | 43.78 | APE67-dihe-in | -62.92, -24.25 | -35.94, -56.9 | APE12-dist-in | 8.6802 | APE11-dist-in | 11.8235 | APE10-dist-in | 5.9829 | APE9-dist-in | 3.5305 | None | TPO180 | TPO180 | XRAY | 1.901 | 0.22 | 0.258 | A | 298.0 | 275.0 | 5 | 28 | 27 | 1 | [[27, 278]] | 1.0 | 8a66 | Homo sapiens | STE_STK3_HUMAN | STE | 2.3e-101 | 344.5 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK3 | STK3_HUMAN | 8A66B | Q13188 | 18 | 304 | 491.0 | 5BS:60501 | Type1 | Inactive | DFGin | 6.2293 | 14.4906 | BLAminus | -139.08, 162.57 | 69.6, 85.67 | -96.89, 21.95 | 294.07, 84.34 | -63.47, -19.34 | in-in | in | 9.5136 | Saltbr-in | 2.883 | HRD-in | -65.79, -48.59 | 72.98, -4.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8323 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -146.04, 152.12 | APE9-dihe-na | 134.76, -156.35 | APE8-dihe-in | -108.07, 116.58 | APE8-rot-out | 42.21 | APE67-dihe-in | -60.0, -23.48 | -33.57, -55.3 | APE12-dist-in | 8.6046 | APE11-dist-in | 11.7522 | APE10-dist-in | 5.9813 | APE9-dist-in | 3.4102 | None | TPO174,TPO180,TPO268 | TPO174,TPO180,TPO268 | XRAY | 1.901 | 0.22 | 0.258 | B | 298.0 | 282.0 | 5 | 28 | 28 | 0 | [[27, 278]] | 1.0 | 8a66 | Homo sapiens | STE_STK3_HUMAN | STE | 2.3e-101 | 344.5 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK3 | STK3_HUMAN | 5DH3A | Q13188 | 19 | 307 | 491.0 | 5BS:401 | Type1 | Inactive | DFGin | 5.9475 | 14.6144 | BLAminus | -145.26, 166.53 | 56.21, 58.22 | -79.02, 55.98 | 309.22, 59.68 | -65.37, -40.98 | out-out | out | 10.1578 | Saltbr-out | 3.8887 | HRD-in | -64.99, -53.25 | 81.51, -5.49 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8183 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -156.11, 158.66 | APE9-dihe-na | 133.82, -164.61 | APE8-dihe-in | -99.88, 125.54 | APE8-rot-in | 317.53 | APE67-dihe-in | -61.6, -38.71 | -57.46, -40.82 | APE12-dist-in | 8.8819 | APE11-dist-in | 11.3596 | APE10-dist-in | 5.7728 | APE9-dist-in | 3.3878 | None | TPO174,TPO180 | TPO174,TPO180 | XRAY | 2.468 | 0.213 | 0.247 | A | 315.0 | 289.0 | 0 | 28 | 28 | 0 | [[27, 278]] | 1.0 | 5dh3 | Homo sapiens | STE_STK3_HUMAN | STE | 2.8e-101 | 344.2 | 2.0 | 257.0 | 256.0 | 163 | 164 | 165 | 167 | 169 | 56 | 70 | 74 | 143 | 145 | 144 | 146.0 | 203 | 191 | 186 | 185 | 184 | 183 | 182 | 181 | 180 | 100 | Serine/threonine-protein kinase 3 |
| STE | STK4 | STK4_HUMAN | 8A5JA | Q13043 | 28 | 309 | 487.0 | 5BS:60501 | Type1 | Active | DFGin | 6.1115 | 14.4237 | BLAminus | -137.01, 164.18 | 68.22, 83.42 | -95.37, 24.9 | 295.6, 83.78 | -58.89, -29.18 | in-in | in | 9.5782 | Saltbr-in | 2.6601 | HRD-in | -62.52, -46.35 | 71.81, -5.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.816 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.87, 157.76 | APE9-dihe-na | 133.26, -159.59 | APE8-dihe-in | -112.62, 116.79 | APE8-rot-in | 307.48 | APE67-dihe-in | -60.45, -27.7 | -37.29, -52.56 | APE12-dist-in | 8.4002 | APE11-dist-in | 11.5567 | APE10-dist-in | 5.8785 | APE9-dist-in | 3.3033 | None | TPO177,TPO183 | TPO177,TPO183 | XRAY | 2.123 | 0.243 | 0.248 | A | 282.0 | 279.0 | 3 | 28 | 28 | 0 | [[30, 281]] | 1.0 | 8a5j | Homo sapiens | STE_STK4_HUMAN | STE | 2.9e-102 | 347.4 | 2.0 | 257.0 | 256.0 | 166 | 167 | 168 | 170 | 172 | 59 | 73 | 77 | 146 | 148 | 147 | 149.0 | 206 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 103 | Serine/threonine-protein kinase 4 |
| STE | STK4 | STK4_HUMAN | 8A5JB | Q13043 | 32 | 309 | 487.0 | 5BS:60501 | Type1 | Inactive | None | 6.1832 | 999.0 | None | -136.98, 164.64 | 68.65, 82.94 | -95.0, 23.57 | 294.73, 84.74 | -56.91, -33.47 | none-none | none | 999.0 | Saltbr-none | 999.0 | HRD-in | -61.94, -46.75 | 72.95, -3.57 | none-in-in | SNCnii | in-in | ActLoopNT-in | 2.7991 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.28, 156.86 | APE9-dihe-na | 133.22, -159.66 | APE8-dihe-in | -113.06, 118.47 | APE8-rot-in | 300.84 | APE67-dihe-in | -66.93, -24.0 | -39.55, -46.8 | APE12-dist-in | 8.294 | APE11-dist-in | 11.5278 | APE10-dist-in | 5.8585 | APE9-dist-in | 3.2972 | None | TPO177,TPO183 | TPO177,TPO183 | XRAY | 2.123 | 0.243 | 0.248 | B | 282.0 | 249.0 | 31 | 28 | 28 | 0 | [[30, 281]] | 1.0 | 8a5j | Homo sapiens | STE_STK4_HUMAN | STE | 2.9e-102 | 347.4 | 2.0 | 257.0 | 256.0 | 166 | 167 | 168 | 170 | 172 | 59 | 73 | 77 | 146 | 148 | 147 | 149.0 | 206 | 194 | 189 | 188 | 187 | 186 | 185 | 184 | 183 | 103 | Serine/threonine-protein kinase 4 |
| TYR | JAK2-1 | JAK2_HUMAN | 6BRWA | O60674 | 537 | 808 | 1132.0 | 5BS:901 | Type1 | Pseudo | DFGin | 7.7052 | 13.3794 | None | -93.41, 174.89 | -67.04, 156.04 | -83.01, 0.59 | 33.82, 139.96 | 67.03, -167.12 | in-na | in | 9.6698 | Saltbr-na | 999.0 | HRD-in | -76.15, -62.39 | 95.18, -6.76 | na-out-out | SNCaoo | out-out | ActLoopNT-out | 9.3464 | ActLoopCT-out | TYR | APEdihe_oooao | APEdist_aaao | APE10-dihe-out | -74.9, -35.05 | APE9-dihe-out | -58.77, -25.82 | APE8-dihe-out | -90.17, 2.34 | APE8-rot-na | 284.96 | APE67-dihe-out | -99.82, 21.48 | -62.86, 134.79 | APE12-dist-na | 9.9909 | APE11-dist-na | 11.5633 | APE10-dist-na | 16.1812 | APE9-dist-out | 12.8111 | W659A,W777A,F794H | None | None | XRAY | 2.031 | 0.197 | 0.25 | A | 289.0 | 272.0 | 0 | 24 | 24 | 0 | [[545, 807], [849, 1125]] | 2.0 | 6brw | Homo sapiens | TYR_JAK2-1_HUMAN | TYR | 1.9e-64 | 223.4 | 2.0 | 260.0 | 259.0 | 698 | 699 | 700 | 702 | 704 | 581 | 597 | 601 | 670 | 672 | 671 | 673.0 | 735 | 722 | 717 | 716 | 715 | 714 | 713 | 712 | 711 | 627 | Tyrosine-protein kinase JAK2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|