| PDB | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 4FIFA | 296 | 589 | 591.0 | ANP:1000 | ATPlike | Active | DFGin | 6.132 | 13.879 | BLAminus | -134.27, -172.64 | 55.78, 65.69 | -91.22, 11.11 | 299.57, 98.92 | -61.37, -20.58 | in-in | in | 7.046 | Saltbr-in | 3.112 | HRD-in | -73.18, -47.2 | 74.11, -8.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.852 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.08, 134.89 | APE9-dihe-na | 136.18, -173.61 | APE8-dihe-in | -102.98, 119.55 | APE8-rot-in | 312.46 | APE67-dihe-in | -69.75, -26.2 | -30.93, -52.34 | APE12-dist-in | 9.318 | APE11-dist-in | 11.709 | APE10-dist-in | 5.875 | APE9-dist-in | 3.299 | None | SEP474 | SEP474 | XRAY | 2.6 | 0.207 | 0.227 | A | 346 | 294 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fif | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIFB | 297 | 589 | 591.0 | ANP:1000 | ATPlike | Active | DFGin | 5.899 | 13.85 | BLAminus | -129.09, -170.37 | 52.27, 68.51 | -93.51, 10.45 | 301.97, 96.23 | -63.09, -15.01 | in-in | in | 7.007 | Saltbr-in | 3.167 | HRD-in | -65.39, -48.9 | 75.1, -7.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.801 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.88, 134.77 | APE9-dihe-na | 136.42, -174.06 | APE8-dihe-in | -101.96, 121.94 | APE8-rot-in | 314.36 | APE67-dihe-in | -72.79, -21.56 | -33.03, -50.98 | APE12-dist-in | 9.238 | APE11-dist-in | 11.712 | APE10-dist-in | 5.886 | APE9-dist-in | 3.335 | None | SEP474 | SEP474 | XRAY | 2.6 | 0.207 | 0.227 | B | 346 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fif | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4JDIA | 300 | 589 | 591.0 | ANP:1000 | ATPlike | Active | DFGin | 6.291 | 14.47 | BLAminus | -134.26, 177.87 | 63.72, 71.58 | -94.6, 13.78 | 289.77, 79.71 | -54.15, -28.77 | in-in | in | 6.959 | Saltbr-in | 2.737 | HRD-in | -72.82, -49.09 | 73.48, 2.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.62, 145.0 | APE9-dihe-na | 130.41, -160.49 | APE8-dihe-in | -120.53, 123.45 | APE8-rot-in | 305.94 | APE67-dihe-in | -63.49, -22.51 | -36.89, -56.07 | APE12-dist-in | 8.769 | APE11-dist-in | 11.535 | APE10-dist-in | 5.874 | APE9-dist-in | 3.327 | None | SEP474 | SEP474 | XRAY | 1.85 | 0.194 | 0.233 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdi | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5UPKB | 300 | 588 | 591.0 | ANP:60600 | ATPlike | Active | DFGin | 6.272 | 14.139 | BLAminus | -132.3, -169.35 | 61.71, 61.5 | -87.86, 7.28 | 293.59, 93.96 | -55.36, -28.3 | in-in | in | 7.077 | Saltbr-in | 3.329 | HRD-in | -65.35, -49.16 | 70.36, 11.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.997 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.55, 149.52 | APE9-dihe-na | 120.09, -163.11 | APE8-dihe-in | -119.51, 121.87 | APE8-rot-in | 313.98 | APE67-dihe-in | -69.89, -18.98 | -32.47, -57.41 | APE12-dist-in | 8.623 | APE11-dist-in | 11.267 | APE10-dist-in | 5.616 | APE9-dist-in | 3.426 | None | SEP474 | SEP474 | XRAY | 2.4 | 0.22 | 0.264 | B | 346 | 289 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5upk | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 7S46A | 300 | 589 | 591.0 | ANP:600 | ATPlike | Active | DFGin | 9.021 | 14.349 | BLAminus | -133.61, -177.07 | 54.75, 76.68 | -92.18, 14.46 | 286.49, 80.35 | -59.04, -19.55 | in-in | in | 7.534 | Saltbr-in | 2.867 | HRD-in | -69.43, -50.5 | 76.76, 2.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.922 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.73, 132.58 | APE9-dihe-na | 145.82, -167.86 | APE8-dihe-in | -110.13, 128.57 | APE8-rot-in | 305.26 | APE67-dihe-in | -70.79, -21.11 | -38.41, -55.32 | APE12-dist-in | 9.02 | APE11-dist-in | 11.537 | APE10-dist-in | 5.793 | APE9-dist-in | 3.286 | D440N,S474E | None | None | XRAY | 2.1 | 0.182 | 0.22 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7s46 | STE_PAK4_HUMAN | STE | 5.5e-87 | 297.4 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 7S47A | 300 | 589 | 591.0 | ANP:600 | ATPlike | Active | DFGin | 9.217 | 14.646 | BLAminus | -126.8, -179.34 | 54.51, 73.91 | -89.97, 15.41 | 285.81, 78.05 | -59.21, -18.99 | in-in | in | 7.79 | Saltbr-in | 2.931 | HRD-in | -66.64, -48.47 | 70.7, 6.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.914 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.53, 138.41 | APE9-dihe-na | 140.72, -164.27 | APE8-dihe-in | -114.61, 124.35 | APE8-rot-in | 304.9 | APE67-dihe-in | -66.22, -20.32 | -36.39, -56.83 | APE12-dist-in | 9.039 | APE11-dist-in | 11.45 | APE10-dist-in | 5.747 | APE9-dist-in | 3.401 | D440N,S474E | None | None | XRAY | 2.0 | 0.196 | 0.237 | A | 383 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7s47 | STE_PAK4_HUMAN | STE | 7.5e-87 | 297.0 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| AF-O96013-K1A | 313 | 580 | 591.0 | No_ligand | No_ligand | Active | DFGin | 5.976 | 13.493 | BLAminus | -130.1, -176.91 | 63.02, 54.98 | -77.11, 5.6 | 302.38, 102.83 | -58.72, -35.23 | in-in | in | 7.715 | Saltbr-in | 2.696 | HRD-in | -71.08, -49.97 | 65.46, 11.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.817 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.24, 162.55 | APE9-dihe-na | 107.8, 178.89 | APE8-dihe-in | -83.65, 126.03 | APE8-rot-in | 303.62 | APE67-dihe-in | -75.87, -21.96 | -48.06, -42.55 | APE12-dist-in | 9.036 | APE11-dist-in | 11.639 | APE10-dist-in | 5.674 | APE9-dist-in | 3.243 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 268 | 268 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | AF-O96013-K1 | STE_PAK4_HUMAN | STE | 1.3e-88 | 302.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| AF-O96013-K3A | 313 | 580 | 591.0 | No_ligand | No_ligand | Active | DFGin | 6.981 | 14.976 | BLAminus | -136.02, -172.75 | 59.27, 53.41 | -76.06, 16.58 | 290.59, 81.49 | -60.1, -26.15 | in-in | in | 8.179 | Saltbr-in | 2.79 | HRD-in | -73.8, -46.38 | 65.56, -0.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.853 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.08, 135.85 | APE9-dihe-na | 132.39, 173.54 | APE8-dihe-in | -86.18, 126.08 | APE8-rot-in | 300.1 | APE67-dihe-in | -76.89, -22.75 | -42.41, -45.98 | APE12-dist-in | 9.021 | APE11-dist-in | 11.486 | APE10-dist-in | 5.617 | APE9-dist-in | 3.125 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 268 | 268 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | AF-O96013-K3 | STE_PAK4_HUMAN | STE | 1.3e-88 | 302.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4L67A | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 10.27 | 14.486 | BLAminus | -151.61, -168.49 | 52.0, 67.37 | -93.33, 11.41 | 289.19, 94.18 | -58.57, -33.07 | in-in | in | 8.3 | Saltbr-in | 3.226 | HRD-in | -102.14, -50.27 | 82.9, -7.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.007 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.16, 134.74 | APE9-dihe-na | 141.36, 174.48 | APE8-dihe-in | -84.97, 121.4 | APE8-rot-in | 323.69 | APE67-dihe-in | -44.13, -27.72 | -31.92, -71.35 | APE12-dist-in | 9.29 | APE11-dist-in | 11.655 | APE10-dist-in | 5.803 | APE9-dist-in | 3.595 | None | SEP474 | SEP474 | XRAY | 2.8 | 0.233 | 0.333 | A | 292 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4l67 | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 2Q0NA | 298 | 591 | 591.0 | No_ligand | No_ligand | Active | DFGin | 7.255 | 14.793 | BLAminus | -133.4, -177.0 | 60.04, 59.83 | -83.03, 16.12 | 284.85, 75.64 | -58.21, -18.8 | in-in | in | 8.517 | Saltbr-in | 2.777 | HRD-in | -73.11, -49.29 | 75.99, 5.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.867 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.34, 142.4 | APE9-dihe-na | 146.55, -148.54 | APE8-dihe-in | -125.26, 117.52 | APE8-rot-in | 303.56 | APE67-dihe-in | -67.05, -21.65 | -33.32, -56.61 | APE12-dist-in | 9.359 | APE11-dist-in | 11.992 | APE10-dist-in | 6.123 | APE9-dist-in | 3.566 | None | SEP474 | SEP474 | XRAY | 1.75 | 0.185 | 0.228 | A | 301 | 294 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2q0n | STE_PAK4_HUMAN | STE | 1.9e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 2J0IA | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 7.46 | 14.626 | BLAminus | -134.36, -165.75 | 58.37, 60.67 | -88.32, 13.39 | 279.76, 75.6 | -62.32, -23.3 | in-in | in | 9.455 | Saltbr-in | 2.627 | HRD-in | -73.73, -49.62 | 71.12, 2.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.899 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.96, 131.78 | APE9-dihe-na | 149.44, -163.72 | APE8-dihe-in | -114.93, 122.79 | APE8-rot-in | 303.47 | APE67-dihe-in | -68.35, -22.9 | -35.96, -56.0 | APE12-dist-in | 9.0 | APE11-dist-in | 11.582 | APE10-dist-in | 5.776 | APE9-dist-in | 3.376 | None | SEP474 | SEP474 | XRAY | 1.6 | 0.174 | 0.215 | A | 303 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2j0i | STE_PAK4_HUMAN | STE | 2e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4JDJA | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.358 | 14.486 | BLAminus | -135.05, -172.77 | 54.02, 73.82 | -92.85, 18.9 | 284.15, 75.9 | -56.84, -29.73 | in-in | in | 7.485 | Saltbr-in | 2.745 | HRD-in | -72.69, -51.05 | 77.52, -2.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.893 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.69, 141.26 | APE9-dihe-na | 128.18, -160.28 | APE8-dihe-in | -117.23, 122.47 | APE8-rot-in | 309.77 | APE67-dihe-in | -61.22, -24.48 | -35.06, -58.78 | APE12-dist-in | 8.557 | APE11-dist-in | 11.313 | APE10-dist-in | 5.753 | APE9-dist-in | 3.513 | F461V | SEP474,TPO562 | SEP474,TPO562 | XRAY | 2.3 | 0.197 | 0.244 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdj | STE_PAK4_HUMAN | STE | 1.4e-88 | 302.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4JDKA | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.298 | 14.327 | BLAminus | -140.41, 175.97 | 54.41, 74.79 | -91.36, 8.02 | 284.28, 75.16 | -60.4, -13.24 | in-in | in | 7.528 | Saltbr-in | 3.384 | HRD-in | -73.1, -44.55 | 68.62, 9.26 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.934 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.09, 153.76 | APE9-dihe-na | 119.82, -165.82 | APE8-dihe-in | -116.32, 129.51 | APE8-rot-in | 313.3 | APE67-dihe-in | -59.03, -26.55 | -44.4, -55.05 | APE12-dist-in | 8.726 | APE11-dist-in | 11.441 | APE10-dist-in | 5.89 | APE9-dist-in | 3.406 | F461V | SEP474,TPO562 | SEP474,TPO562 | XRAY | 2.4 | 0.188 | 0.249 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdk | STE_PAK4_HUMAN | STE | 1.4e-88 | 302.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIHA | 298 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.206 | 14.407 | BLAminus | -135.98, -177.2 | 57.56, 65.31 | -90.69, 14.94 | 285.62, 76.78 | -54.76, -25.38 | in-in | in | 7.578 | Saltbr-in | 2.892 | HRD-in | -76.81, -47.61 | 70.56, 6.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.845 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.25, 153.53 | APE9-dihe-na | 122.35, -158.41 | APE8-dihe-in | -122.77, 125.62 | APE8-rot-in | 308.66 | APE67-dihe-in | -66.29, -20.2 | -45.47, -47.52 | APE12-dist-in | 8.616 | APE11-dist-in | 11.303 | APE10-dist-in | 5.566 | APE9-dist-in | 3.307 | None | SEP474 | SEP474 | XRAY | 1.97 | 0.181 | 0.225 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fih | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIIA | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.073 | 14.201 | BLAminus | -132.45, 178.79 | 60.3, 61.71 | -80.38, 12.79 | 288.68, 79.5 | -61.8, -21.84 | in-in | in | 7.306 | Saltbr-in | 2.72 | HRD-in | -76.29, -44.67 | 66.21, 4.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.897 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.33, 143.29 | APE9-dihe-na | 138.12, -155.84 | APE8-dihe-in | -121.98, 122.0 | APE8-rot-in | 307.09 | APE67-dihe-in | -73.04, -19.21 | -34.75, -51.15 | APE12-dist-in | 8.727 | APE11-dist-in | 11.467 | APE10-dist-in | 5.694 | APE9-dist-in | 3.357 | None | SEP474 | SEP474 | XRAY | 2.0 | 0.203 | 0.24 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fii | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIJA | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.292 | 14.118 | BLAminus | -121.84, -176.7 | 65.31, 67.51 | -99.57, 14.75 | 281.79, 80.65 | -61.33, -22.97 | in-in | in | 7.674 | Saltbr-in | 3.269 | HRD-in | -67.47, -53.79 | 82.69, -7.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.902 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.15, 145.87 | APE9-dihe-na | 132.39, -161.12 | APE8-dihe-in | -117.16, 124.28 | APE8-rot-in | 306.73 | APE67-dihe-in | -60.5, -24.88 | -30.89, -62.08 | APE12-dist-in | 8.634 | APE11-dist-in | 11.233 | APE10-dist-in | 5.492 | APE9-dist-in | 3.441 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.21 | 0.271 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fij | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4JDHA | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.213 | 14.456 | BLAminus | -133.94, -173.46 | 58.56, 59.99 | -88.47, 17.74 | 285.35, 78.93 | -64.25, -20.67 | in-in | in | 7.641 | Saltbr-in | 3.319 | HRD-in | -69.0, -48.43 | 71.31, 1.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.884 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.94, 132.78 | APE9-dihe-na | 145.26, -171.34 | APE8-dihe-in | -107.31, 123.45 | APE8-rot-in | 307.6 | APE67-dihe-in | -61.34, -23.1 | -36.34, -56.17 | APE12-dist-in | 8.85 | APE11-dist-in | 11.633 | APE10-dist-in | 5.92 | APE9-dist-in | 3.451 | None | SEP474 | SEP474 | XRAY | 2.0 | 0.185 | 0.224 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdh | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 6WLXA | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.201 | 14.18 | BLAminus | -131.59, -176.89 | 52.24, 74.82 | -93.47, 12.81 | 286.48, 76.04 | -60.21, -15.65 | in-in | in | 7.465 | Saltbr-in | 3.141 | HRD-in | -75.87, -52.52 | 76.84, 4.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.82 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.58, 142.68 | APE9-dihe-na | 133.42, -162.48 | APE8-dihe-in | -119.0, 127.34 | APE8-rot-in | 308.13 | APE67-dihe-in | -62.55, -20.45 | -37.98, -61.18 | APE12-dist-in | 8.684 | APE11-dist-in | 11.422 | APE10-dist-in | 5.762 | APE9-dist-in | 3.399 | None | SEP474 | SEP474 | XRAY | 2.2 | 0.198 | 0.229 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 6wlx | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 6WLYA | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.224 | 14.295 | BLAminus | -137.23, -173.74 | 57.81, 67.07 | -89.26, 13.37 | 287.97, 80.51 | -62.01, -15.87 | in-in | in | 7.533 | Saltbr-in | 3.048 | HRD-in | -73.43, -48.63 | 72.76, 3.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.868 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.41, 131.81 | APE9-dihe-na | 146.78, -170.14 | APE8-dihe-in | -112.43, 122.77 | APE8-rot-in | 308.27 | APE67-dihe-in | -64.63, -20.86 | -40.07, -54.5 | APE12-dist-in | 9.032 | APE11-dist-in | 11.625 | APE10-dist-in | 5.893 | APE9-dist-in | 3.458 | None | SEP474 | SEP474 | XRAY | 1.9 | 0.187 | 0.205 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 6wly | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 7S48A | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.263 | 14.359 | BLAminus | -132.18, -176.07 | 57.15, 66.61 | -90.62, 13.14 | 283.96, 77.99 | -58.72, -23.33 | in-in | in | 7.568 | Saltbr-in | 3.013 | HRD-in | -68.6, -50.0 | 72.97, 5.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.95, 147.83 | APE9-dihe-na | 129.62, -155.85 | APE8-dihe-in | -124.91, 120.05 | APE8-rot-in | 304.0 | APE67-dihe-in | -65.8, -21.35 | -34.95, -54.24 | APE12-dist-in | 8.739 | APE11-dist-in | 11.41 | APE10-dist-in | 5.72 | APE9-dist-in | 3.359 | None | SEP474 | SEP474 | XRAY | 1.9 | 0.182 | 0.222 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7s48 | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5UPLA | 299 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 6.912 | 14.21 | BLAminus | -163.39, -166.4 | 59.78, 65.71 | -85.27, 8.4 | 284.5, 105.17 | -65.55, -24.21 | in-in | in | 7.153 | Saltbr-in | 3.45 | HRD-in | -74.32, -54.24 | 91.8, -11.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.896 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.47, 142.27 | APE9-dihe-na | 127.52, -177.54 | APE8-dihe-in | -94.03, 129.74 | APE8-rot-in | 310.33 | APE67-dihe-in | -74.72, -26.02 | -36.97, -49.73 | APE12-dist-in | 9.097 | APE11-dist-in | 11.606 | APE10-dist-in | 5.991 | APE9-dist-in | 3.47 | None | SEP474 | SEP474 | XRAY | 3.003 | 0.259 | 0.31 | A | 453 | 291 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5upl | STE_PAK4_HUMAN | STE | 6.8e-88 | 300.4 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5XVFA | 300 | 588 | 591.0 | 8FR:60601 | Type1 | Active | DFGin | 6.41 | 13.597 | BLAminus | -139.57, -167.28 | 48.68, 69.67 | -90.45, 14.2 | 300.76, 102.19 | -49.74, -29.58 | in-in | in | 6.835 | Saltbr-in | 2.694 | HRD-in | -68.54, -55.23 | 77.68, 6.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.909 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.25, 148.38 | APE9-dihe-na | 130.46, 176.96 | APE8-dihe-in | -94.44, 129.78 | APE8-rot-in | 311.81 | APE67-dihe-in | -56.47, -21.8 | -39.65, -64.54 | APE12-dist-in | 9.78 | APE11-dist-in | 11.712 | APE10-dist-in | 6.021 | APE9-dist-in | 3.115 | None | SEP474 | SEP474 | XRAY | 2.655 | 0.197 | 0.251 | A | 290 | 289 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5xvf | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.3 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5XVAA | 300 | 591 | 591.0 | 8FU:60601 | Type1 | Active | DFGin | 7.292 | 14.678 | BLAminus | -136.68, -167.04 | 56.18, 61.77 | -88.8, 17.56 | 283.16, 73.25 | -67.91, -15.71 | in-in | in | 9.132 | Saltbr-in | 3.092 | HRD-in | -72.82, -52.08 | 71.15, 6.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.857 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.16, 135.82 | APE9-dihe-na | 145.24, -159.73 | APE8-dihe-in | -113.25, 122.53 | APE8-rot-in | 304.59 | APE67-dihe-in | -66.13, -21.23 | -41.05, -53.04 | APE12-dist-in | 9.038 | APE11-dist-in | 11.494 | APE10-dist-in | 5.663 | APE9-dist-in | 3.454 | None | SEP474 | SEP474 | XRAY | 1.847 | 0.17 | 0.209 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5xva | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5XVGA | 300 | 591 | 591.0 | 8FX:60601 | Type1 | Active | DFGin | 7.024 | 14.57 | BLAminus | -144.25, -166.15 | 65.18, 60.23 | -89.33, 20.04 | 283.56, 74.99 | -67.07, -12.05 | in-in | in | 8.826 | Saltbr-in | 2.764 | HRD-in | -73.13, -52.27 | 72.69, 11.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.915 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.8, 143.35 | APE9-dihe-na | 134.84, -159.43 | APE8-dihe-in | -114.76, 122.91 | APE8-rot-in | 304.21 | APE67-dihe-in | -67.25, -18.32 | -47.47, -47.2 | APE12-dist-in | 8.974 | APE11-dist-in | 11.481 | APE10-dist-in | 5.603 | APE9-dist-in | 3.372 | None | SEP474 | SEP474 | XRAY | 2.1 | 0.184 | 0.235 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5xvg | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5ZJWA | 300 | 591 | 591.0 | 9EO:60601 | Type1 | Active | DFGin | 7.467 | 14.64 | BLAminus | -132.98, -163.71 | 63.14, 51.92 | -88.51, 14.85 | 280.26, 75.04 | -63.71, -21.2 | in-in | in | 8.86 | Saltbr-in | 2.964 | HRD-in | -75.73, -49.33 | 70.25, 5.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.833 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.08, 137.6 | APE9-dihe-na | 143.8, -159.07 | APE8-dihe-in | -117.35, 122.21 | APE8-rot-in | 300.48 | APE67-dihe-in | -67.39, -19.86 | -42.33, -52.03 | APE12-dist-in | 8.996 | APE11-dist-in | 11.569 | APE10-dist-in | 5.792 | APE9-dist-in | 3.463 | None | SEP474 | SEP474 | XRAY | 1.798 | 0.171 | 0.215 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5zjw | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 9D52A | 300 | 589 | 591.0 | A1A2R:601 | Type1 | Active | DFGin | 5.845 | 13.851 | BLAminus | -137.59, -174.27 | 58.3, 72.52 | -97.57, 11.47 | 297.67, 101.1 | -60.39, -21.88 | in-in | in | 7.298 | Saltbr-in | 3.091 | HRD-in | -68.35, -60.99 | 83.79, -1.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.19, 138.88 | APE9-dihe-na | 146.77, -167.01 | APE8-dihe-in | -103.22, 122.41 | APE8-rot-in | 308.06 | APE67-dihe-in | -66.75, -19.09 | -36.2, -56.16 | APE12-dist-in | 9.053 | APE11-dist-in | 11.768 | APE10-dist-in | 5.918 | APE9-dist-in | 3.302 | None | SEP474 | SEP474 | XRAY | 2.449 | 0.205 | 0.287 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 9d52 | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 9D53A | 300 | 591 | 591.0 | A1A2P:601 | Type1 | Active | DFGin | 7.419 | 14.388 | BLAminus | -130.46, -168.1 | 66.3, 64.12 | -97.32, 16.28 | 284.99, 83.03 | -56.88, -20.45 | in-in | in | 8.429 | Saltbr-in | 3.039 | HRD-in | -68.67, -55.34 | 70.78, 15.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.701 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.76, 128.71 | APE9-dihe-na | 154.97, -168.87 | APE8-dihe-in | -101.14, 120.06 | APE8-rot-in | 318.43 | APE67-dihe-in | -66.45, -26.26 | -33.54, -52.96 | APE12-dist-in | 9.874 | APE11-dist-in | 11.678 | APE10-dist-in | 5.88 | APE9-dist-in | 3.4 | None | SEP474 | SEP474 | XRAY | 2.468 | 0.19 | 0.263 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 9d53 | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5BMSA | 300 | 589 | 591.0 | 4T6:60601 | Type1 | Active | DFGin | 5.882 | 13.769 | BLAminus | -127.85, -156.82 | 35.49, 78.34 | -98.96, 8.42 | 299.27, 100.83 | -63.09, -11.52 | in-in | in | 7.312 | Saltbr-in | 3.075 | HRD-in | -77.22, -46.32 | 67.96, 4.24 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.832 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.5, 139.88 | APE9-dihe-na | 129.41, -167.55 | APE8-dihe-in | -107.17, 120.88 | APE8-rot-in | 315.49 | APE67-dihe-in | -62.73, -29.26 | -33.47, -61.67 | APE12-dist-in | 9.996 | APE11-dist-in | 11.617 | APE10-dist-in | 5.891 | APE9-dist-in | 3.222 | None | SEP474 | SEP474 | XRAY | 2.903 | 0.176 | 0.23 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5bms | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 2X4ZA | 299 | 590 | 591.0 | 7KC:1593 | Type1 | Active | DFGin | 7.175 | 15.683 | BLAminus | -132.06, -173.98 | 55.27, 65.86 | -89.03, 22.48 | 286.31, 71.15 | -56.55, -18.72 | out-in | out | 10.093 | Saltbr-in | 3.353 | HRD-in | -64.34, -55.81 | 75.26, 4.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.874 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.15, 164.59 | APE9-dihe-na | 116.46, -153.03 | APE8-dihe-in | -123.41, 117.02 | APE8-rot-in | 305.72 | APE67-dihe-in | -61.08, -22.54 | -22.19, -62.41 | APE12-dist-in | 8.425 | APE11-dist-in | 11.116 | APE10-dist-in | 5.211 | APE9-dist-in | 3.362 | P296G,Q297S,R298H,V299M | SEP474 | SEP474 | XRAY | 2.1 | 0.2 | 0.262 | A | 296 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2x4z | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4APPA | 300 | 591 | 591.0 | N53:60601 | Type1 | Active | DFGin | 7.373 | 15.543 | BLAminus | -133.61, -169.75 | 57.81, 63.69 | -88.94, 22.51 | 284.15, 66.92 | -58.72, -20.97 | out-in | out | 10.218 | Saltbr-in | 2.879 | HRD-in | -73.06, -52.18 | 73.4, 4.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.997 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.88, 162.5 | APE9-dihe-na | 116.5, -157.47 | APE8-dihe-in | -119.99, 123.77 | APE8-rot-in | 310.26 | APE67-dihe-in | -55.32, -22.24 | -23.87, -72.11 | APE12-dist-in | 8.564 | APE11-dist-in | 11.028 | APE10-dist-in | 5.227 | APE9-dist-in | 3.3 | None | SEP474 | SEP474 | XRAY | 2.2 | 0.188 | 0.229 | A | 296 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4app | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4NJDA | 300 | 589 | 591.0 | NJD:60600 | Type1 | Active | DFGin | 7.55 | 14.534 | BLAminus | -137.61, -170.79 | 59.81, 63.86 | -89.24, 10.26 | 288.33, 68.78 | -51.39, -35.62 | in-in | in | 8.832 | Saltbr-in | 2.774 | HRD-in | -64.48, -51.46 | 71.88, -2.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.827 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.47, 156.67 | APE9-dihe-na | 134.13, -165.38 | APE8-dihe-in | -113.07, 115.38 | APE8-rot-in | 315.39 | APE67-dihe-in | -65.56, -7.99 | -27.21, -63.29 | APE12-dist-in | 9.033 | APE11-dist-in | 11.457 | APE10-dist-in | 5.589 | APE9-dist-in | 3.292 | None | SEP474 | SEP474 | XRAY | 2.5 | 0.239 | 0.321 | A | 296 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4njd | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5I0BA | 301 | 589 | 591.0 | 67U:601 | Type1 | Active | DFGin | 7.442 | 14.009 | BLAminus | -124.94, -168.52 | 59.76, 54.09 | -85.49, 7.58 | 290.32, 78.2 | -49.18, -28.77 | in-in | in | 8.386 | Saltbr-in | 2.784 | HRD-in | -62.72, -43.63 | 65.0, -1.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.79 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -124.17, -174.46 | APE9-dihe-na | 97.06, -178.26 | APE8-dihe-in | -118.11, 136.57 | APE8-rot-in | 266.84 | APE67-dihe-in | -62.52, -33.2 | -59.08, -48.11 | APE12-dist-in | 9.53 | APE11-dist-in | 11.272 | APE10-dist-in | 5.32 | APE9-dist-in | 2.849 | None | SEP474 | SEP474 | XRAY | 3.09 | 0.199 | 0.269 | A | 296 | 289 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5i0b | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 8AHGA | 300 | 591 | 591.0 | M4I:60601 | Type1 | Active | DFGin | 9.274 | 14.621 | BLAminus | -140.7, -178.52 | 59.09, 59.79 | -84.52, 9.62 | 282.61, 76.91 | -57.19, -25.15 | in-in | in | 7.783 | Saltbr-in | 3.0 | HRD-in | -68.05, -53.29 | 75.32, 3.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.88 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.99, 144.76 | APE9-dihe-na | 133.62, -152.42 | APE8-dihe-in | -126.55, 119.92 | APE8-rot-in | 307.01 | APE67-dihe-in | -70.16, -19.98 | -38.25, -51.28 | APE12-dist-in | 8.713 | APE11-dist-in | 11.311 | APE10-dist-in | 5.642 | APE9-dist-in | 3.378 | L310A | SEP474 | SEP474 | XRAY | 1.885 | 0.181 | 0.227 | A | 297 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8ahg | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 8AHHA | 300 | 591 | 591.0 | M4X:60601 | Type1 | Active | DFGin | 9.202 | 14.302 | BLAminus | -140.1, -178.26 | 56.12, 62.98 | -87.16, 10.59 | 287.77, 78.02 | -51.14, -27.59 | in-in | in | 7.613 | Saltbr-in | 3.166 | HRD-in | -71.92, -49.28 | 69.03, 2.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.883 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.71, 139.6 | APE9-dihe-na | 140.63, -152.77 | APE8-dihe-in | -124.55, 121.97 | APE8-rot-in | 311.5 | APE67-dihe-in | -69.72, -19.91 | -39.05, -51.53 | APE12-dist-in | 8.885 | APE11-dist-in | 11.313 | APE10-dist-in | 5.683 | APE9-dist-in | 3.346 | L310A | SEP474 | SEP474 | XRAY | 2.037 | 0.188 | 0.25 | A | 297 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8ahh | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 2CDZA | 299 | 590 | 591.0 | 23D:1591 | Type1 | Active | DFGin | 6.851 | 14.239 | BLAminus | -131.93, -172.68 | 60.56, 61.36 | -89.92, 17.05 | 286.34, 82.19 | -67.68, -14.12 | in-in | in | 8.413 | Saltbr-in | 2.548 | HRD-in | -67.95, -51.01 | 69.05, 1.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.912 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.41, 141.72 | APE9-dihe-na | 145.87, -158.12 | APE8-dihe-in | -124.24, 119.58 | APE8-rot-in | 305.81 | APE67-dihe-in | -67.53, -21.67 | -30.06, -59.48 | APE12-dist-in | 9.103 | APE11-dist-in | 11.374 | APE10-dist-in | 5.44 | APE9-dist-in | 3.375 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.202 | 0.248 | A | 303 | 290 | 2 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2cdz | STE_PAK4_HUMAN | STE | 2e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5VEFA | 300 | 589 | 591.0 | M77:601 | Type1 | Active | DFGin | 9.346 | 14.591 | BLAminus | -136.52, -176.88 | 59.47, 65.15 | -89.64, 13.99 | 283.23, 80.94 | -61.13, -20.52 | in-in | in | 7.74 | Saltbr-in | 3.421 | HRD-in | -69.98, -53.91 | 75.95, 7.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.864 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.13, 146.51 | APE9-dihe-na | 127.95, -160.54 | APE8-dihe-in | -118.96, 120.95 | APE8-rot-in | 302.31 | APE67-dihe-in | -69.34, -18.53 | -36.63, -52.05 | APE12-dist-in | 8.781 | APE11-dist-in | 11.284 | APE10-dist-in | 5.646 | APE9-dist-in | 3.383 | None | SEP474 | SEP474 | XRAY | 1.752 | 0.202 | 0.239 | A | 319 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5vef | STE_PAK4_HUMAN | STE | 2.4e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 7CP3A | 300 | 589 | 591.0 | GC6:601 | Type1.5_Back | Active | DFGin | 7.425 | 14.516 | BLAminus | -143.23, -161.44 | 54.49, 56.58 | -84.68, 17.45 | 283.38, 69.37 | -57.63, -18.5 | in-in | in | 8.25 | Saltbr-in | 2.97 | HRD-in | -75.52, -44.49 | 67.1, 5.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.046 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.2, 132.66 | APE9-dihe-na | 144.26, -150.95 | APE8-dihe-in | -112.54, 134.18 | APE8-rot-in | 306.62 | APE67-dihe-in | -71.08, -11.39 | -57.8, -50.41 | APE12-dist-in | 8.889 | APE11-dist-in | 11.521 | APE10-dist-in | 5.733 | APE9-dist-in | 3.741 | None | SEP474 | SEP474 | XRAY | 2.9 | 0.245 | 0.267 | A | 292 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7cp3 | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 7CP4A | 300 | 591 | 591.0 | GCC:601 | Type1.5_Back | Active | DFGin | 7.635 | 14.952 | BLAminus | -133.21, 179.04 | 59.99, 67.29 | -90.26, 23.6 | 285.11, 67.74 | -63.22, -23.85 | in-in | in | 9.553 | Saltbr-in | 3.29 | HRD-in | -66.61, -55.01 | 72.71, 4.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.906 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.28, 137.07 | APE9-dihe-na | 140.56, -171.81 | APE8-dihe-in | -103.14, 125.77 | APE8-rot-in | 309.43 | APE67-dihe-in | -72.75, -28.29 | -48.05, -39.75 | APE12-dist-in | 8.651 | APE11-dist-in | 11.228 | APE10-dist-in | 5.429 | APE9-dist-in | 3.361 | None | SEP474 | SEP474 | XRAY | 2.5 | 0.199 | 0.252 | A | 292 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7cp4 | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 7CMBA | 300 | 589 | 591.0 | G5X:60601 | Type1.5_Back | Active | DFGin | 7.29 | 14.864 | BLAminus | -144.05, 179.08 | 58.57, 70.68 | -90.04, 21.82 | 285.98, 71.77 | -65.95, -9.86 | in-in | in | 8.729 | Saltbr-in | 2.802 | HRD-in | -64.8, -46.41 | 64.06, 19.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -114.38, 168.28 | APE9-dihe-na | 114.24, -179.32 | APE8-dihe-in | -97.31, 129.92 | APE8-rot-in | 316.69 | APE67-dihe-in | -69.15, -20.09 | -50.08, -47.79 | APE12-dist-in | 8.971 | APE11-dist-in | 11.233 | APE10-dist-in | 5.229 | APE9-dist-in | 3.486 | None | SEP474 | SEP474 | XRAY | 2.592 | 0.208 | 0.251 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7cmb | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4O0VA | 300 | 589 | 591.0 | 2OL:60601 | Type1.5_Back | Active | DFGin | 7.72 | 14.855 | BLAminus | -129.91, -179.13 | 52.93, 70.48 | -91.0, 31.77 | 289.31, 80.54 | -68.79, -11.49 | in-in | in | 9.386 | Saltbr-in | 2.715 | HRD-in | -63.47, -48.3 | 66.54, 12.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.98 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.31, 136.62 | APE9-dihe-na | 128.1, -161.84 | APE8-dihe-in | -105.46, 125.26 | APE8-rot-in | 314.65 | APE67-dihe-in | -70.36, -25.33 | -37.86, -50.41 | APE12-dist-in | 9.483 | APE11-dist-in | 11.399 | APE10-dist-in | 5.692 | APE9-dist-in | 3.35 | None | SEP474 | SEP474 | XRAY | 2.8 | 0.204 | 0.253 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4o0v | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4O0XA | 300 | 589 | 591.0 | 2OQ:60601 | Type1.5_Back | Active | DFGin | 7.686 | 14.42 | BLAminus | -143.48, 175.23 | 50.73, 80.07 | -96.8, 29.16 | 288.57, 62.64 | -65.03, -22.79 | in-in | in | 7.841 | Saltbr-in | 2.524 | HRD-in | -64.27, -54.17 | 74.62, 7.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.044 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.91, 146.7 | APE9-dihe-na | 131.01, -164.91 | APE8-dihe-in | -110.0, 119.08 | APE8-rot-in | 309.56 | APE67-dihe-in | -57.87, -20.38 | -32.76, -63.35 | APE12-dist-in | 9.115 | APE11-dist-in | 11.502 | APE10-dist-in | 5.674 | APE9-dist-in | 3.39 | None | SEP474 | SEP474 | XRAY | 2.483 | 0.242 | 0.242 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4o0x | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4O0YA | 300 | 589 | 591.0 | 2OO:60601 | Type1.5_Back | Active | DFGin | 7.439 | 13.922 | BLAminus | -135.18, 176.5 | 49.39, 78.85 | -92.46, 20.76 | 288.83, 77.11 | -54.08, -29.88 | in-in | in | 7.462 | Saltbr-in | 2.628 | HRD-in | -74.32, -48.56 | 73.38, 6.1 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -124.29, 136.66 | APE9-dihe-na | 144.79, -161.28 | APE8-dihe-in | -119.15, 122.67 | APE8-rot-in | 309.1 | APE67-dihe-in | -63.4, -19.31 | -38.26, -57.11 | APE12-dist-in | 9.651 | APE11-dist-in | 11.689 | APE10-dist-in | 5.96 | APE9-dist-in | 3.34 | None | SEP474 | SEP474 | XRAY | 2.2 | 0.2 | 0.238 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4o0y | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4XBRA | 177 | 589 | 591.0 | ATP:60601 | ATPlike | Inactive | DFGin | 5.852 | 14.061 | ABAminus | -142.04, -22.23 | -111.42, 72.59 | -86.56, 10.51 | 310.81, 99.4 | -46.84, -40.66 | in-in | in | 7.009 | Saltbr-in | 3.158 | HRD-in | -84.11, -33.57 | 58.48, -1.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.974 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.96, 132.02 | APE9-dihe-na | 150.85, -176.82 | APE8-dihe-in | -102.34, 122.5 | APE8-rot-in | 312.14 | APE67-dihe-in | -59.91, -25.15 | -35.82, -60.88 | APE12-dist-in | 9.335 | APE11-dist-in | 11.927 | APE10-dist-in | 6.05 | APE9-dist-in | 3.396 | None | SEP474 | SEP474 | XRAY | 2.94 | 0.191 | 0.23 | A | 366 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4xbr | STE_PAK4_HUMAN | STE | 3.7e-88 | 301.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIGA | 298 | 590 | 591.0 | ANP:1001 | ATPlike | Inactive | DFGin | 5.976 | 13.995 | BLAminus | -134.45, -166.25 | 59.06, 57.3 | -88.34, 9.13 | 298.9, 106.14 | -61.58, -20.66 | in-in | in | 7.133 | Saltbr-in | 3.168 | HRD-in | -77.25, -46.66 | 72.07, -3.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.86 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.47, 161.1 | APE9-dihe-na | 110.61, 163.55 | APE8-dihe-in | -79.54, 130.34 | APE8-rot-out | 29.96 | APE67-dihe-in | -76.38, -28.34 | -35.31, -49.63 | APE12-dist-in | 9.418 | APE11-dist-in | 11.569 | APE10-dist-in | 5.635 | APE9-dist-in | 3.369 | None | SEP474 | SEP474 | XRAY | 3.01 | 0.197 | 0.221 | A | 346 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fig | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIEA | 49 | 590 | 591.0 | ANP:1001 | ATPlike | Inactive | DFGin | 6.278 | 14.03 | BLAminus | -142.71, -177.86 | 63.75, 67.7 | -92.97, 13.53 | 295.29, 98.36 | -64.15, -7.0 | in-out | in | 6.991 | Saltbr-out | 3.974 | HRD-in | -74.78, -36.69 | 67.65, -13.13 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.856 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -135.98, 139.97 | APE9-dihe-na | 123.6, -177.34 | APE8-dihe-in | -84.44, 139.76 | APE8-rot-out | 19.51 | APE67-dihe-in | -74.38, -37.99 | -51.24, -48.18 | APE12-dist-in | 9.515 | APE11-dist-in | 11.685 | APE10-dist-in | 5.909 | APE9-dist-in | 3.508 | None | SEP474 | SEP474 | XRAY | 3.11 | 0.257 | 0.276 | A | 423 | 301 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fie | STE_PAK4_HUMAN | STE | 5.6e-88 | 300.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIEB | 49 | 590 | 591.0 | ANP:1001 | ATPlike | Inactive | DFGin | 6.278 | 14.031 | BLAminus | -142.24, -177.62 | 63.59, 67.55 | -92.7, 13.49 | 295.33, 98.22 | -64.04, -7.21 | in-out | in | 6.989 | Saltbr-out | 3.957 | HRD-in | -74.95, -36.21 | 66.97, -12.74 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.857 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.0, 139.86 | APE9-dihe-na | 123.6, -177.41 | APE8-dihe-in | -84.57, 139.76 | APE8-rot-out | 19.62 | APE67-dihe-in | -74.42, -37.89 | -51.19, -48.15 | APE12-dist-in | 9.515 | APE11-dist-in | 11.689 | APE10-dist-in | 5.912 | APE9-dist-in | 3.51 | None | SEP474 | SEP474 | XRAY | 3.11 | 0.257 | 0.276 | B | 423 | 301 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fie | STE_PAK4_HUMAN | STE | 5.6e-88 | 300.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 2BVAA | 300 | 587 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 7.438 | 16.475 | BLAminus | -117.27, -176.72 | 56.65, 71.44 | -91.27, 35.1 | 289.21, 80.8 | -69.61, -2.94 | out-out | out | 10.481 | Saltbr-out | 4.02 | HRD-in | -57.52, -60.13 | 72.86, 5.02 | out-out-in | SNCooi | out-in | ActLoopNT-out | 3.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.79, 153.17 | APE9-dihe-na | 127.58, -141.52 | APE8-dihe-in | -136.11, 111.21 | APE8-rot-in | 333.57 | APE67-dihe-in | -60.96, -14.16 | -40.33, -50.6 | APE12-dist-in | 8.848 | APE11-dist-in | 11.484 | APE10-dist-in | 5.83 | APE9-dist-in | 3.471 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.192 | 0.269 | A | 292 | 273 | 15 | 0 | 0 | 2 | [[321, 572]] | 1.0 | 2bva | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 2BVAB | 301 | 587 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 7.572 | 17.238 | BLAminus | -131.91, -158.23 | 65.58, 44.26 | -84.57, 26.99 | 293.34, 56.33 | -60.85, -21.66 | out-out | out | 11.675 | Saltbr-out | 7.148 | HRD-in | -60.3, -59.82 | 75.14, 24.4 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.499 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.93, 163.72 | APE9-dihe-na | 104.79, -155.19 | APE8-dihe-in | -112.34, 124.37 | APE8-rot-in | 319.0 | APE67-dihe-in | -73.92, -14.55 | -41.39, -45.76 | APE12-dist-in | 8.588 | APE11-dist-in | 11.399 | APE10-dist-in | 5.909 | APE9-dist-in | 3.197 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.192 | 0.269 | B | 292 | 275 | 12 | 0 | 0 | 2 | [[321, 572]] | 1.0 | 2bva | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 8YHKA | 298 | 591 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 6.394 | 13.95 | BLAminus | -144.78, -174.84 | 60.87, 52.46 | -74.27, -7.16 | 291.41, 99.22 | -44.42, -31.64 | in-out | in | 7.212 | Saltbr-out | 5.663 | HRD-out | -76.82, 93.99 | -85.26, 6.82 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.734 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.02, 139.67 | APE9-dihe-na | 131.69, -172.38 | APE8-dihe-in | -96.54, 118.36 | APE8-rot-in | 308.12 | APE67-dihe-in | -79.25, -37.48 | -34.17, -42.18 | APE12-dist-in | 9.944 | APE11-dist-in | 11.39 | APE10-dist-in | 5.545 | APE9-dist-in | 3.243 | None | None | None | XRAY | 3.3 | 0.253 | 0.319 | A | 301 | 294 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8yhk | STE_PAK4_HUMAN | STE | 1.9e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4XBUA | 297 | 589 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 7.426 | 14.345 | BLAminus | -134.76, -171.38 | 58.13, 68.14 | -90.95, 10.75 | 282.43, 88.09 | -57.4, -26.1 | in-out | in | 8.875 | Saltbr-out | 4.505 | HRD-in | -80.19, -49.71 | 68.99, 2.54 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.842 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.64, 133.45 | APE9-dihe-na | 156.19, -154.61 | APE8-dihe-in | -123.57, 122.27 | APE8-rot-in | 305.74 | APE67-dihe-in | -70.59, -15.2 | -40.43, -52.25 | APE12-dist-in | 8.806 | APE11-dist-in | 11.559 | APE10-dist-in | 5.875 | APE9-dist-in | 3.518 | None | SEP474 | SEP474 | XRAY | 2.06 | 0.201 | 0.243 | A | 326 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4xbu | STE_PAK4_HUMAN | STE | 2.5e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 8AHIA | 300 | 591 | 591.0 | M56:601 | Type1 | Inactive | DFGin | 9.181 | 14.38 | BLAminus | -137.45, -173.93 | 55.91, 63.31 | -90.54, 16.67 | 287.37, 76.55 | -61.73, -19.34 | in-out | in | 7.694 | Saltbr-out | 3.645 | HRD-in | -78.82, -49.15 | 74.56, 0.81 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.882 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.24, 128.69 | APE9-dihe-na | 143.74, -151.59 | APE8-dihe-in | -115.17, 123.77 | APE8-rot-in | 313.27 | APE67-dihe-in | -68.11, -27.23 | -45.23, -43.93 | APE12-dist-in | 8.803 | APE11-dist-in | 11.358 | APE10-dist-in | 5.796 | APE9-dist-in | 3.534 | L310A | SEP474 | SEP474 | XRAY | 2.69 | 0.16 | 0.249 | A | 297 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8ahi | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5VEDA | 300 | 589 | 591.0 | STU:601 | Type1 | Inactive | DFGin | 7.591 | 14.871 | BLAminus | -137.67, -169.84 | 57.61, 74.14 | -100.29, 38.24 | 286.21, 78.54 | -72.3, -31.74 | in-out | in | 8.771 | Saltbr-out | 5.279 | HRD-in | -70.67, -47.26 | 60.82, 22.3 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.978 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.74, 169.93 | APE9-dihe-na | 110.0, -167.24 | APE8-dihe-in | -107.4, 122.99 | APE8-rot-in | 313.49 | APE67-dihe-in | -72.02, -18.93 | -37.81, -47.81 | APE12-dist-in | 8.493 | APE11-dist-in | 11.13 | APE10-dist-in | 5.271 | APE9-dist-in | 3.412 | None | SEP474 | SEP474 | XRAY | 2.301 | 0.231 | 0.277 | A | 319 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5ved | STE_PAK4_HUMAN | STE | 2.4e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 5VEEA | 300 | 589 | 591.0 | 981:601 | Type1 | Inactive | DFGin | 6.832 | 15.436 | BLAminus | -149.85, -166.61 | 63.61, 64.4 | -91.35, 12.72 | 287.99, 79.38 | -42.54, -35.66 | in-out | in | 8.369 | Saltbr-out | 6.665 | HRD-in | -63.93, -45.62 | 68.7, 8.17 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.12 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.59, 147.54 | APE9-dihe-na | 146.37, -170.93 | APE8-dihe-in | -104.03, 125.68 | APE8-rot-in | 311.71 | APE67-dihe-in | -46.67, -33.8 | -40.96, -66.37 | APE12-dist-in | 9.09 | APE11-dist-in | 11.607 | APE10-dist-in | 5.815 | APE9-dist-in | 3.64 | None | SEP474 | SEP474 | XRAY | 2.5 | 0.231 | 0.276 | A | 319 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5vee | STE_PAK4_HUMAN | STE | 2.4e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| 4FIGB | 298 | 590 | 591.0 | ANP:602 | ATPlike | Inactive | DFGin | 5.979 | 13.845 | None | -136.1, -40.27 | -82.41, 70.29 | -85.54, 12.48 | 305.29, 106.7 | -66.77, -24.27 | in-in | in | 7.007 | Saltbr-in | 3.047 | HRD-in | -63.37, -48.9 | 73.21, -4.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.929 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.8, 141.64 | APE9-dihe-na | 130.69, -165.45 | APE8-dihe-in | -110.43, 122.9 | APE8-rot-in | 324.7 | APE67-dihe-in | -77.33, -31.89 | -29.23, -51.11 | APE12-dist-in | 9.706 | APE11-dist-in | 11.743 | APE10-dist-in | 5.92 | APE9-dist-in | 3.386 | None | SEP474 | SEP474 | XRAY | 3.01 | 0.197 | 0.221 | B | 346 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fig | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| PAK4_HUMAN | 4FIFA | O96013 | 296 | 589 | 591.0 | ANP:1000 | ATPlike | Active | DFGin | 6.132 | 13.879 | BLAminus | -134.27, -172.64 | 55.78, 65.69 | -91.22, 11.11 | 299.57, 98.92 | -61.37, -20.58 | in-in | in | 7.046 | Saltbr-in | 3.112 | HRD-in | -73.18, -47.2 | 74.11, -8.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.852 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -136.08, 134.89 | APE9-dihe-na | 136.18, -173.61 | APE8-dihe-in | -102.98, 119.55 | APE8-rot-in | 312.46 | APE67-dihe-in | -69.75, -26.2 | -30.93, -52.34 | APE12-dist-in | 9.318 | APE11-dist-in | 11.709 | APE10-dist-in | 5.875 | APE9-dist-in | 3.299 | None | SEP474 | SEP474 | XRAY | 2.6 | 0.207 | 0.227 | A | 346 | 294 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fif | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIFB | O96013 | 297 | 589 | 591.0 | ANP:1000 | ATPlike | Active | DFGin | 5.899 | 13.85 | BLAminus | -129.09, -170.37 | 52.27, 68.51 | -93.51, 10.45 | 301.97, 96.23 | -63.09, -15.01 | in-in | in | 7.007 | Saltbr-in | 3.167 | HRD-in | -65.39, -48.9 | 75.1, -7.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.801 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.88, 134.77 | APE9-dihe-na | 136.42, -174.06 | APE8-dihe-in | -101.96, 121.94 | APE8-rot-in | 314.36 | APE67-dihe-in | -72.79, -21.56 | -33.03, -50.98 | APE12-dist-in | 9.238 | APE11-dist-in | 11.712 | APE10-dist-in | 5.886 | APE9-dist-in | 3.335 | None | SEP474 | SEP474 | XRAY | 2.6 | 0.207 | 0.227 | B | 346 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fif | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4JDIA | O96013 | 300 | 589 | 591.0 | ANP:1000 | ATPlike | Active | DFGin | 6.291 | 14.47 | BLAminus | -134.26, 177.87 | 63.72, 71.58 | -94.6, 13.78 | 289.77, 79.71 | -54.15, -28.77 | in-in | in | 6.959 | Saltbr-in | 2.737 | HRD-in | -72.82, -49.09 | 73.48, 2.76 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.829 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.62, 145.0 | APE9-dihe-na | 130.41, -160.49 | APE8-dihe-in | -120.53, 123.45 | APE8-rot-in | 305.94 | APE67-dihe-in | -63.49, -22.51 | -36.89, -56.07 | APE12-dist-in | 8.769 | APE11-dist-in | 11.535 | APE10-dist-in | 5.874 | APE9-dist-in | 3.327 | None | SEP474 | SEP474 | XRAY | 1.85 | 0.194 | 0.233 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdi | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5UPKB | O96013 | 300 | 588 | 591.0 | ANP:60600 | ATPlike | Active | DFGin | 6.272 | 14.139 | BLAminus | -132.3, -169.35 | 61.71, 61.5 | -87.86, 7.28 | 293.59, 93.96 | -55.36, -28.3 | in-in | in | 7.077 | Saltbr-in | 3.329 | HRD-in | -65.35, -49.16 | 70.36, 11.54 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.997 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.55, 149.52 | APE9-dihe-na | 120.09, -163.11 | APE8-dihe-in | -119.51, 121.87 | APE8-rot-in | 313.98 | APE67-dihe-in | -69.89, -18.98 | -32.47, -57.41 | APE12-dist-in | 8.623 | APE11-dist-in | 11.267 | APE10-dist-in | 5.616 | APE9-dist-in | 3.426 | None | SEP474 | SEP474 | XRAY | 2.4 | 0.22 | 0.264 | B | 346 | 289 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5upk | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 7S46A | O96013 | 300 | 589 | 591.0 | ANP:600 | ATPlike | Active | DFGin | 9.021 | 14.349 | BLAminus | -133.61, -177.07 | 54.75, 76.68 | -92.18, 14.46 | 286.49, 80.35 | -59.04, -19.55 | in-in | in | 7.534 | Saltbr-in | 2.867 | HRD-in | -69.43, -50.5 | 76.76, 2.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.922 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.73, 132.58 | APE9-dihe-na | 145.82, -167.86 | APE8-dihe-in | -110.13, 128.57 | APE8-rot-in | 305.26 | APE67-dihe-in | -70.79, -21.11 | -38.41, -55.32 | APE12-dist-in | 9.02 | APE11-dist-in | 11.537 | APE10-dist-in | 5.793 | APE9-dist-in | 3.286 | D440N,S474E | None | None | XRAY | 2.1 | 0.182 | 0.22 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7s46 | Homo sapiens | STE_PAK4_HUMAN | STE | 5.5e-87 | 297.4 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 7S47A | O96013 | 300 | 589 | 591.0 | ANP:600 | ATPlike | Active | DFGin | 9.217 | 14.646 | BLAminus | -126.8, -179.34 | 54.51, 73.91 | -89.97, 15.41 | 285.81, 78.05 | -59.21, -18.99 | in-in | in | 7.79 | Saltbr-in | 2.931 | HRD-in | -66.64, -48.47 | 70.7, 6.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.914 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.53, 138.41 | APE9-dihe-na | 140.72, -164.27 | APE8-dihe-in | -114.61, 124.35 | APE8-rot-in | 304.9 | APE67-dihe-in | -66.22, -20.32 | -36.39, -56.83 | APE12-dist-in | 9.039 | APE11-dist-in | 11.45 | APE10-dist-in | 5.747 | APE9-dist-in | 3.401 | D440N,S474E | None | None | XRAY | 2.0 | 0.196 | 0.237 | A | 383 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7s47 | Homo sapiens | STE_PAK4_HUMAN | STE | 7.5e-87 | 297.0 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | AF-O96013-K1A | O96013 | 313 | 580 | 591.0 | No_ligand | No_ligand | Active | DFGin | 5.976 | 13.493 | BLAminus | -130.1, -176.91 | 63.02, 54.98 | -77.11, 5.6 | 302.38, 102.83 | -58.72, -35.23 | in-in | in | 7.715 | Saltbr-in | 2.696 | HRD-in | -71.08, -49.97 | 65.46, 11.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.817 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.24, 162.55 | APE9-dihe-na | 107.8, 178.89 | APE8-dihe-in | -83.65, 126.03 | APE8-rot-in | 303.62 | APE67-dihe-in | -75.87, -21.96 | -48.06, -42.55 | APE12-dist-in | 9.036 | APE11-dist-in | 11.639 | APE10-dist-in | 5.674 | APE9-dist-in | 3.243 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 268 | 268 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | AF-O96013-K1 | Homo sapiens | STE_PAK4_HUMAN | STE | 1.3e-88 | 302.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | AF-O96013-K3A | O96013 | 313 | 580 | 591.0 | No_ligand | No_ligand | Active | DFGin | 6.981 | 14.976 | BLAminus | -136.02, -172.75 | 59.27, 53.41 | -76.06, 16.58 | 290.59, 81.49 | -60.1, -26.15 | in-in | in | 8.179 | Saltbr-in | 2.79 | HRD-in | -73.8, -46.38 | 65.56, -0.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.853 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.08, 135.85 | APE9-dihe-na | 132.39, 173.54 | APE8-dihe-in | -86.18, 126.08 | APE8-rot-in | 300.1 | APE67-dihe-in | -76.89, -22.75 | -42.41, -45.98 | APE12-dist-in | 9.021 | APE11-dist-in | 11.486 | APE10-dist-in | 5.617 | APE9-dist-in | 3.125 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 268 | 268 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | AF-O96013-K3 | Homo sapiens | STE_PAK4_HUMAN | STE | 1.3e-88 | 302.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4L67A | O96013 | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 10.27 | 14.486 | BLAminus | -151.61, -168.49 | 52.0, 67.37 | -93.33, 11.41 | 289.19, 94.18 | -58.57, -33.07 | in-in | in | 8.3 | Saltbr-in | 3.226 | HRD-in | -102.14, -50.27 | 82.9, -7.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.007 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.16, 134.74 | APE9-dihe-na | 141.36, 174.48 | APE8-dihe-in | -84.97, 121.4 | APE8-rot-in | 323.69 | APE67-dihe-in | -44.13, -27.72 | -31.92, -71.35 | APE12-dist-in | 9.29 | APE11-dist-in | 11.655 | APE10-dist-in | 5.803 | APE9-dist-in | 3.595 | None | SEP474 | SEP474 | XRAY | 2.8 | 0.233 | 0.333 | A | 292 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4l67 | Homo sapiens | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 2Q0NA | O96013 | 298 | 591 | 591.0 | No_ligand | No_ligand | Active | DFGin | 7.255 | 14.793 | BLAminus | -133.4, -177.0 | 60.04, 59.83 | -83.03, 16.12 | 284.85, 75.64 | -58.21, -18.8 | in-in | in | 8.517 | Saltbr-in | 2.777 | HRD-in | -73.11, -49.29 | 75.99, 5.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.867 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.34, 142.4 | APE9-dihe-na | 146.55, -148.54 | APE8-dihe-in | -125.26, 117.52 | APE8-rot-in | 303.56 | APE67-dihe-in | -67.05, -21.65 | -33.32, -56.61 | APE12-dist-in | 9.359 | APE11-dist-in | 11.992 | APE10-dist-in | 6.123 | APE9-dist-in | 3.566 | None | SEP474 | SEP474 | XRAY | 1.75 | 0.185 | 0.228 | A | 301 | 294 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2q0n | Homo sapiens | STE_PAK4_HUMAN | STE | 1.9e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 2J0IA | O96013 | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 7.46 | 14.626 | BLAminus | -134.36, -165.75 | 58.37, 60.67 | -88.32, 13.39 | 279.76, 75.6 | -62.32, -23.3 | in-in | in | 9.455 | Saltbr-in | 2.627 | HRD-in | -73.73, -49.62 | 71.12, 2.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.899 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.96, 131.78 | APE9-dihe-na | 149.44, -163.72 | APE8-dihe-in | -114.93, 122.79 | APE8-rot-in | 303.47 | APE67-dihe-in | -68.35, -22.9 | -35.96, -56.0 | APE12-dist-in | 9.0 | APE11-dist-in | 11.582 | APE10-dist-in | 5.776 | APE9-dist-in | 3.376 | None | SEP474 | SEP474 | XRAY | 1.6 | 0.174 | 0.215 | A | 303 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2j0i | Homo sapiens | STE_PAK4_HUMAN | STE | 2e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4JDJA | O96013 | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.358 | 14.486 | BLAminus | -135.05, -172.77 | 54.02, 73.82 | -92.85, 18.9 | 284.15, 75.9 | -56.84, -29.73 | in-in | in | 7.485 | Saltbr-in | 2.745 | HRD-in | -72.69, -51.05 | 77.52, -2.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.893 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.69, 141.26 | APE9-dihe-na | 128.18, -160.28 | APE8-dihe-in | -117.23, 122.47 | APE8-rot-in | 309.77 | APE67-dihe-in | -61.22, -24.48 | -35.06, -58.78 | APE12-dist-in | 8.557 | APE11-dist-in | 11.313 | APE10-dist-in | 5.753 | APE9-dist-in | 3.513 | F461V | SEP474,TPO562 | SEP474,TPO562 | XRAY | 2.3 | 0.197 | 0.244 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdj | Homo sapiens | STE_PAK4_HUMAN | STE | 1.4e-88 | 302.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4JDKA | O96013 | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.298 | 14.327 | BLAminus | -140.41, 175.97 | 54.41, 74.79 | -91.36, 8.02 | 284.28, 75.16 | -60.4, -13.24 | in-in | in | 7.528 | Saltbr-in | 3.384 | HRD-in | -73.1, -44.55 | 68.62, 9.26 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.934 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.09, 153.76 | APE9-dihe-na | 119.82, -165.82 | APE8-dihe-in | -116.32, 129.51 | APE8-rot-in | 313.3 | APE67-dihe-in | -59.03, -26.55 | -44.4, -55.05 | APE12-dist-in | 8.726 | APE11-dist-in | 11.441 | APE10-dist-in | 5.89 | APE9-dist-in | 3.406 | F461V | SEP474,TPO562 | SEP474,TPO562 | XRAY | 2.4 | 0.188 | 0.249 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdk | Homo sapiens | STE_PAK4_HUMAN | STE | 1.4e-88 | 302.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIHA | O96013 | 298 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.206 | 14.407 | BLAminus | -135.98, -177.2 | 57.56, 65.31 | -90.69, 14.94 | 285.62, 76.78 | -54.76, -25.38 | in-in | in | 7.578 | Saltbr-in | 2.892 | HRD-in | -76.81, -47.61 | 70.56, 6.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.845 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.25, 153.53 | APE9-dihe-na | 122.35, -158.41 | APE8-dihe-in | -122.77, 125.62 | APE8-rot-in | 308.66 | APE67-dihe-in | -66.29, -20.2 | -45.47, -47.52 | APE12-dist-in | 8.616 | APE11-dist-in | 11.303 | APE10-dist-in | 5.566 | APE9-dist-in | 3.307 | None | SEP474 | SEP474 | XRAY | 1.97 | 0.181 | 0.225 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fih | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIIA | O96013 | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.073 | 14.201 | BLAminus | -132.45, 178.79 | 60.3, 61.71 | -80.38, 12.79 | 288.68, 79.5 | -61.8, -21.84 | in-in | in | 7.306 | Saltbr-in | 2.72 | HRD-in | -76.29, -44.67 | 66.21, 4.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.897 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -147.33, 143.29 | APE9-dihe-na | 138.12, -155.84 | APE8-dihe-in | -121.98, 122.0 | APE8-rot-in | 307.09 | APE67-dihe-in | -73.04, -19.21 | -34.75, -51.15 | APE12-dist-in | 8.727 | APE11-dist-in | 11.467 | APE10-dist-in | 5.694 | APE9-dist-in | 3.357 | None | SEP474 | SEP474 | XRAY | 2.0 | 0.203 | 0.24 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fii | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIJA | O96013 | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.292 | 14.118 | BLAminus | -121.84, -176.7 | 65.31, 67.51 | -99.57, 14.75 | 281.79, 80.65 | -61.33, -22.97 | in-in | in | 7.674 | Saltbr-in | 3.269 | HRD-in | -67.47, -53.79 | 82.69, -7.78 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.902 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.15, 145.87 | APE9-dihe-na | 132.39, -161.12 | APE8-dihe-in | -117.16, 124.28 | APE8-rot-in | 306.73 | APE67-dihe-in | -60.5, -24.88 | -30.89, -62.08 | APE12-dist-in | 8.634 | APE11-dist-in | 11.233 | APE10-dist-in | 5.492 | APE9-dist-in | 3.441 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.21 | 0.271 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fij | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4JDHA | O96013 | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.213 | 14.456 | BLAminus | -133.94, -173.46 | 58.56, 59.99 | -88.47, 17.74 | 285.35, 78.93 | -64.25, -20.67 | in-in | in | 7.641 | Saltbr-in | 3.319 | HRD-in | -69.0, -48.43 | 71.31, 1.52 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.884 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.94, 132.78 | APE9-dihe-na | 145.26, -171.34 | APE8-dihe-in | -107.31, 123.45 | APE8-rot-in | 307.6 | APE67-dihe-in | -61.34, -23.1 | -36.34, -56.17 | APE12-dist-in | 8.85 | APE11-dist-in | 11.633 | APE10-dist-in | 5.92 | APE9-dist-in | 3.451 | None | SEP474 | SEP474 | XRAY | 2.0 | 0.185 | 0.224 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4jdh | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 6WLXA | O96013 | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.201 | 14.18 | BLAminus | -131.59, -176.89 | 52.24, 74.82 | -93.47, 12.81 | 286.48, 76.04 | -60.21, -15.65 | in-in | in | 7.465 | Saltbr-in | 3.141 | HRD-in | -75.87, -52.52 | 76.84, 4.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.82 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.58, 142.68 | APE9-dihe-na | 133.42, -162.48 | APE8-dihe-in | -119.0, 127.34 | APE8-rot-in | 308.13 | APE67-dihe-in | -62.55, -20.45 | -37.98, -61.18 | APE12-dist-in | 8.684 | APE11-dist-in | 11.422 | APE10-dist-in | 5.762 | APE9-dist-in | 3.399 | None | SEP474 | SEP474 | XRAY | 2.2 | 0.198 | 0.229 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 6wlx | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 6WLYA | O96013 | 299 | 590 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.224 | 14.295 | BLAminus | -137.23, -173.74 | 57.81, 67.07 | -89.26, 13.37 | 287.97, 80.51 | -62.01, -15.87 | in-in | in | 7.533 | Saltbr-in | 3.048 | HRD-in | -73.43, -48.63 | 72.76, 3.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.868 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -142.41, 131.81 | APE9-dihe-na | 146.78, -170.14 | APE8-dihe-in | -112.43, 122.77 | APE8-rot-in | 308.27 | APE67-dihe-in | -64.63, -20.86 | -40.07, -54.5 | APE12-dist-in | 9.032 | APE11-dist-in | 11.625 | APE10-dist-in | 5.893 | APE9-dist-in | 3.458 | None | SEP474 | SEP474 | XRAY | 1.9 | 0.187 | 0.205 | A | 346 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 6wly | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 7S48A | O96013 | 300 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 9.263 | 14.359 | BLAminus | -132.18, -176.07 | 57.15, 66.61 | -90.62, 13.14 | 283.96, 77.99 | -58.72, -23.33 | in-in | in | 7.568 | Saltbr-in | 3.013 | HRD-in | -68.6, -50.0 | 72.97, 5.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.95, 147.83 | APE9-dihe-na | 129.62, -155.85 | APE8-dihe-in | -124.91, 120.05 | APE8-rot-in | 304.0 | APE67-dihe-in | -65.8, -21.35 | -34.95, -54.24 | APE12-dist-in | 8.739 | APE11-dist-in | 11.41 | APE10-dist-in | 5.72 | APE9-dist-in | 3.359 | None | SEP474 | SEP474 | XRAY | 1.9 | 0.182 | 0.222 | A | 346 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7s48 | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5UPLA | O96013 | 299 | 589 | 591.0 | No_ligand | No_ligand | Active | DFGin | 6.912 | 14.21 | BLAminus | -163.39, -166.4 | 59.78, 65.71 | -85.27, 8.4 | 284.5, 105.17 | -65.55, -24.21 | in-in | in | 7.153 | Saltbr-in | 3.45 | HRD-in | -74.32, -54.24 | 91.8, -11.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.896 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.47, 142.27 | APE9-dihe-na | 127.52, -177.54 | APE8-dihe-in | -94.03, 129.74 | APE8-rot-in | 310.33 | APE67-dihe-in | -74.72, -26.02 | -36.97, -49.73 | APE12-dist-in | 9.097 | APE11-dist-in | 11.606 | APE10-dist-in | 5.991 | APE9-dist-in | 3.47 | None | SEP474 | SEP474 | XRAY | 3.003 | 0.259 | 0.31 | A | 453 | 291 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5upl | Homo sapiens | STE_PAK4_HUMAN | STE | 6.8e-88 | 300.4 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5XVFA | O96013 | 300 | 588 | 591.0 | 8FR:60601 | Type1 | Active | DFGin | 6.41 | 13.597 | BLAminus | -139.57, -167.28 | 48.68, 69.67 | -90.45, 14.2 | 300.76, 102.19 | -49.74, -29.58 | in-in | in | 6.835 | Saltbr-in | 2.694 | HRD-in | -68.54, -55.23 | 77.68, 6.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.909 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.25, 148.38 | APE9-dihe-na | 130.46, 176.96 | APE8-dihe-in | -94.44, 129.78 | APE8-rot-in | 311.81 | APE67-dihe-in | -56.47, -21.8 | -39.65, -64.54 | APE12-dist-in | 9.78 | APE11-dist-in | 11.712 | APE10-dist-in | 6.021 | APE9-dist-in | 3.115 | None | SEP474 | SEP474 | XRAY | 2.655 | 0.197 | 0.251 | A | 290 | 289 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5xvf | Homo sapiens | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.3 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5XVAA | O96013 | 300 | 591 | 591.0 | 8FU:60601 | Type1 | Active | DFGin | 7.292 | 14.678 | BLAminus | -136.68, -167.04 | 56.18, 61.77 | -88.8, 17.56 | 283.16, 73.25 | -67.91, -15.71 | in-in | in | 9.132 | Saltbr-in | 3.092 | HRD-in | -72.82, -52.08 | 71.15, 6.91 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.857 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.16, 135.82 | APE9-dihe-na | 145.24, -159.73 | APE8-dihe-in | -113.25, 122.53 | APE8-rot-in | 304.59 | APE67-dihe-in | -66.13, -21.23 | -41.05, -53.04 | APE12-dist-in | 9.038 | APE11-dist-in | 11.494 | APE10-dist-in | 5.663 | APE9-dist-in | 3.454 | None | SEP474 | SEP474 | XRAY | 1.847 | 0.17 | 0.209 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5xva | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5XVGA | O96013 | 300 | 591 | 591.0 | 8FX:60601 | Type1 | Active | DFGin | 7.024 | 14.57 | BLAminus | -144.25, -166.15 | 65.18, 60.23 | -89.33, 20.04 | 283.56, 74.99 | -67.07, -12.05 | in-in | in | 8.826 | Saltbr-in | 2.764 | HRD-in | -73.13, -52.27 | 72.69, 11.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.915 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.8, 143.35 | APE9-dihe-na | 134.84, -159.43 | APE8-dihe-in | -114.76, 122.91 | APE8-rot-in | 304.21 | APE67-dihe-in | -67.25, -18.32 | -47.47, -47.2 | APE12-dist-in | 8.974 | APE11-dist-in | 11.481 | APE10-dist-in | 5.603 | APE9-dist-in | 3.372 | None | SEP474 | SEP474 | XRAY | 2.1 | 0.184 | 0.235 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5xvg | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5ZJWA | O96013 | 300 | 591 | 591.0 | 9EO:60601 | Type1 | Active | DFGin | 7.467 | 14.64 | BLAminus | -132.98, -163.71 | 63.14, 51.92 | -88.51, 14.85 | 280.26, 75.04 | -63.71, -21.2 | in-in | in | 8.86 | Saltbr-in | 2.964 | HRD-in | -75.73, -49.33 | 70.25, 5.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.833 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.08, 137.6 | APE9-dihe-na | 143.8, -159.07 | APE8-dihe-in | -117.35, 122.21 | APE8-rot-in | 300.48 | APE67-dihe-in | -67.39, -19.86 | -42.33, -52.03 | APE12-dist-in | 8.996 | APE11-dist-in | 11.569 | APE10-dist-in | 5.792 | APE9-dist-in | 3.463 | None | SEP474 | SEP474 | XRAY | 1.798 | 0.171 | 0.215 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5zjw | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 9D52A | O96013 | 300 | 589 | 591.0 | A1A2R:601 | Type1 | Active | DFGin | 5.845 | 13.851 | BLAminus | -137.59, -174.27 | 58.3, 72.52 | -97.57, 11.47 | 297.67, 101.1 | -60.39, -21.88 | in-in | in | 7.298 | Saltbr-in | 3.091 | HRD-in | -68.35, -60.99 | 83.79, -1.35 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.19, 138.88 | APE9-dihe-na | 146.77, -167.01 | APE8-dihe-in | -103.22, 122.41 | APE8-rot-in | 308.06 | APE67-dihe-in | -66.75, -19.09 | -36.2, -56.16 | APE12-dist-in | 9.053 | APE11-dist-in | 11.768 | APE10-dist-in | 5.918 | APE9-dist-in | 3.302 | None | SEP474 | SEP474 | XRAY | 2.449 | 0.205 | 0.287 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 9d52 | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 9D53A | O96013 | 300 | 591 | 591.0 | A1A2P:601 | Type1 | Active | DFGin | 7.419 | 14.388 | BLAminus | -130.46, -168.1 | 66.3, 64.12 | -97.32, 16.28 | 284.99, 83.03 | -56.88, -20.45 | in-in | in | 8.429 | Saltbr-in | 3.039 | HRD-in | -68.67, -55.34 | 70.78, 15.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.701 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.76, 128.71 | APE9-dihe-na | 154.97, -168.87 | APE8-dihe-in | -101.14, 120.06 | APE8-rot-in | 318.43 | APE67-dihe-in | -66.45, -26.26 | -33.54, -52.96 | APE12-dist-in | 9.874 | APE11-dist-in | 11.678 | APE10-dist-in | 5.88 | APE9-dist-in | 3.4 | None | SEP474 | SEP474 | XRAY | 2.468 | 0.19 | 0.263 | A | 293 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 9d53 | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5BMSA | O96013 | 300 | 589 | 591.0 | 4T6:60601 | Type1 | Active | DFGin | 5.882 | 13.769 | BLAminus | -127.85, -156.82 | 35.49, 78.34 | -98.96, 8.42 | 299.27, 100.83 | -63.09, -11.52 | in-in | in | 7.312 | Saltbr-in | 3.075 | HRD-in | -77.22, -46.32 | 67.96, 4.24 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.832 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.5, 139.88 | APE9-dihe-na | 129.41, -167.55 | APE8-dihe-in | -107.17, 120.88 | APE8-rot-in | 315.49 | APE67-dihe-in | -62.73, -29.26 | -33.47, -61.67 | APE12-dist-in | 9.996 | APE11-dist-in | 11.617 | APE10-dist-in | 5.891 | APE9-dist-in | 3.222 | None | SEP474 | SEP474 | XRAY | 2.903 | 0.176 | 0.23 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5bms | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 2X4ZA | O96013 | 299 | 590 | 591.0 | 7KC:1593 | Type1 | Active | DFGin | 7.175 | 15.683 | BLAminus | -132.06, -173.98 | 55.27, 65.86 | -89.03, 22.48 | 286.31, 71.15 | -56.55, -18.72 | out-in | out | 10.093 | Saltbr-in | 3.353 | HRD-in | -64.34, -55.81 | 75.26, 4.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.874 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.15, 164.59 | APE9-dihe-na | 116.46, -153.03 | APE8-dihe-in | -123.41, 117.02 | APE8-rot-in | 305.72 | APE67-dihe-in | -61.08, -22.54 | -22.19, -62.41 | APE12-dist-in | 8.425 | APE11-dist-in | 11.116 | APE10-dist-in | 5.211 | APE9-dist-in | 3.362 | P296G,Q297S,R298H,V299M | SEP474 | SEP474 | XRAY | 2.1 | 0.2 | 0.262 | A | 296 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2x4z | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4APPA | O96013 | 300 | 591 | 591.0 | N53:60601 | Type1 | Active | DFGin | 7.373 | 15.543 | BLAminus | -133.61, -169.75 | 57.81, 63.69 | -88.94, 22.51 | 284.15, 66.92 | -58.72, -20.97 | out-in | out | 10.218 | Saltbr-in | 2.879 | HRD-in | -73.06, -52.18 | 73.4, 4.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.997 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.88, 162.5 | APE9-dihe-na | 116.5, -157.47 | APE8-dihe-in | -119.99, 123.77 | APE8-rot-in | 310.26 | APE67-dihe-in | -55.32, -22.24 | -23.87, -72.11 | APE12-dist-in | 8.564 | APE11-dist-in | 11.028 | APE10-dist-in | 5.227 | APE9-dist-in | 3.3 | None | SEP474 | SEP474 | XRAY | 2.2 | 0.188 | 0.229 | A | 296 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4app | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4NJDA | O96013 | 300 | 589 | 591.0 | NJD:60600 | Type1 | Active | DFGin | 7.55 | 14.534 | BLAminus | -137.61, -170.79 | 59.81, 63.86 | -89.24, 10.26 | 288.33, 68.78 | -51.39, -35.62 | in-in | in | 8.832 | Saltbr-in | 2.774 | HRD-in | -64.48, -51.46 | 71.88, -2.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.827 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.47, 156.67 | APE9-dihe-na | 134.13, -165.38 | APE8-dihe-in | -113.07, 115.38 | APE8-rot-in | 315.39 | APE67-dihe-in | -65.56, -7.99 | -27.21, -63.29 | APE12-dist-in | 9.033 | APE11-dist-in | 11.457 | APE10-dist-in | 5.589 | APE9-dist-in | 3.292 | None | SEP474 | SEP474 | XRAY | 2.5 | 0.239 | 0.321 | A | 296 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4njd | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5I0BA | O96013 | 301 | 589 | 591.0 | 67U:601 | Type1 | Active | DFGin | 7.442 | 14.009 | BLAminus | -124.94, -168.52 | 59.76, 54.09 | -85.49, 7.58 | 290.32, 78.2 | -49.18, -28.77 | in-in | in | 8.386 | Saltbr-in | 2.784 | HRD-in | -62.72, -43.63 | 65.0, -1.19 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.79 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -124.17, -174.46 | APE9-dihe-na | 97.06, -178.26 | APE8-dihe-in | -118.11, 136.57 | APE8-rot-in | 266.84 | APE67-dihe-in | -62.52, -33.2 | -59.08, -48.11 | APE12-dist-in | 9.53 | APE11-dist-in | 11.272 | APE10-dist-in | 5.32 | APE9-dist-in | 2.849 | None | SEP474 | SEP474 | XRAY | 3.09 | 0.199 | 0.269 | A | 296 | 289 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5i0b | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 8AHGA | O96013 | 300 | 591 | 591.0 | M4I:60601 | Type1 | Active | DFGin | 9.274 | 14.621 | BLAminus | -140.7, -178.52 | 59.09, 59.79 | -84.52, 9.62 | 282.61, 76.91 | -57.19, -25.15 | in-in | in | 7.783 | Saltbr-in | 3.0 | HRD-in | -68.05, -53.29 | 75.32, 3.61 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.88 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.99, 144.76 | APE9-dihe-na | 133.62, -152.42 | APE8-dihe-in | -126.55, 119.92 | APE8-rot-in | 307.01 | APE67-dihe-in | -70.16, -19.98 | -38.25, -51.28 | APE12-dist-in | 8.713 | APE11-dist-in | 11.311 | APE10-dist-in | 5.642 | APE9-dist-in | 3.378 | L310A | SEP474 | SEP474 | XRAY | 1.885 | 0.181 | 0.227 | A | 297 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8ahg | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 8AHHA | O96013 | 300 | 591 | 591.0 | M4X:60601 | Type1 | Active | DFGin | 9.202 | 14.302 | BLAminus | -140.1, -178.26 | 56.12, 62.98 | -87.16, 10.59 | 287.77, 78.02 | -51.14, -27.59 | in-in | in | 7.613 | Saltbr-in | 3.166 | HRD-in | -71.92, -49.28 | 69.03, 2.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.883 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.71, 139.6 | APE9-dihe-na | 140.63, -152.77 | APE8-dihe-in | -124.55, 121.97 | APE8-rot-in | 311.5 | APE67-dihe-in | -69.72, -19.91 | -39.05, -51.53 | APE12-dist-in | 8.885 | APE11-dist-in | 11.313 | APE10-dist-in | 5.683 | APE9-dist-in | 3.346 | L310A | SEP474 | SEP474 | XRAY | 2.037 | 0.188 | 0.25 | A | 297 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8ahh | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 2CDZA | O96013 | 299 | 590 | 591.0 | 23D:1591 | Type1 | Active | DFGin | 6.851 | 14.239 | BLAminus | -131.93, -172.68 | 60.56, 61.36 | -89.92, 17.05 | 286.34, 82.19 | -67.68, -14.12 | in-in | in | 8.413 | Saltbr-in | 2.548 | HRD-in | -67.95, -51.01 | 69.05, 1.71 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.912 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.41, 141.72 | APE9-dihe-na | 145.87, -158.12 | APE8-dihe-in | -124.24, 119.58 | APE8-rot-in | 305.81 | APE67-dihe-in | -67.53, -21.67 | -30.06, -59.48 | APE12-dist-in | 9.103 | APE11-dist-in | 11.374 | APE10-dist-in | 5.44 | APE9-dist-in | 3.375 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.202 | 0.248 | A | 303 | 290 | 2 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 2cdz | Homo sapiens | STE_PAK4_HUMAN | STE | 2e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5VEFA | O96013 | 300 | 589 | 591.0 | M77:601 | Type1 | Active | DFGin | 9.346 | 14.591 | BLAminus | -136.52, -176.88 | 59.47, 65.15 | -89.64, 13.99 | 283.23, 80.94 | -61.13, -20.52 | in-in | in | 7.74 | Saltbr-in | 3.421 | HRD-in | -69.98, -53.91 | 75.95, 7.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.864 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.13, 146.51 | APE9-dihe-na | 127.95, -160.54 | APE8-dihe-in | -118.96, 120.95 | APE8-rot-in | 302.31 | APE67-dihe-in | -69.34, -18.53 | -36.63, -52.05 | APE12-dist-in | 8.781 | APE11-dist-in | 11.284 | APE10-dist-in | 5.646 | APE9-dist-in | 3.383 | None | SEP474 | SEP474 | XRAY | 1.752 | 0.202 | 0.239 | A | 319 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5vef | Homo sapiens | STE_PAK4_HUMAN | STE | 2.4e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 7CP3A | O96013 | 300 | 589 | 591.0 | GC6:601 | Type1.5_Back | Active | DFGin | 7.425 | 14.516 | BLAminus | -143.23, -161.44 | 54.49, 56.58 | -84.68, 17.45 | 283.38, 69.37 | -57.63, -18.5 | in-in | in | 8.25 | Saltbr-in | 2.97 | HRD-in | -75.52, -44.49 | 67.1, 5.14 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.046 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.2, 132.66 | APE9-dihe-na | 144.26, -150.95 | APE8-dihe-in | -112.54, 134.18 | APE8-rot-in | 306.62 | APE67-dihe-in | -71.08, -11.39 | -57.8, -50.41 | APE12-dist-in | 8.889 | APE11-dist-in | 11.521 | APE10-dist-in | 5.733 | APE9-dist-in | 3.741 | None | SEP474 | SEP474 | XRAY | 2.9 | 0.245 | 0.267 | A | 292 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7cp3 | Homo sapiens | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 7CP4A | O96013 | 300 | 591 | 591.0 | GCC:601 | Type1.5_Back | Active | DFGin | 7.635 | 14.952 | BLAminus | -133.21, 179.04 | 59.99, 67.29 | -90.26, 23.6 | 285.11, 67.74 | -63.22, -23.85 | in-in | in | 9.553 | Saltbr-in | 3.29 | HRD-in | -66.61, -55.01 | 72.71, 4.31 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.906 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.28, 137.07 | APE9-dihe-na | 140.56, -171.81 | APE8-dihe-in | -103.14, 125.77 | APE8-rot-in | 309.43 | APE67-dihe-in | -72.75, -28.29 | -48.05, -39.75 | APE12-dist-in | 8.651 | APE11-dist-in | 11.228 | APE10-dist-in | 5.429 | APE9-dist-in | 3.361 | None | SEP474 | SEP474 | XRAY | 2.5 | 0.199 | 0.252 | A | 292 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7cp4 | Homo sapiens | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 7CMBA | O96013 | 300 | 589 | 591.0 | G5X:60601 | Type1.5_Back | Active | DFGin | 7.29 | 14.864 | BLAminus | -144.05, 179.08 | 58.57, 70.68 | -90.04, 21.82 | 285.98, 71.77 | -65.95, -9.86 | in-in | in | 8.729 | Saltbr-in | 2.802 | HRD-in | -64.8, -46.41 | 64.06, 19.25 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.943 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -114.38, 168.28 | APE9-dihe-na | 114.24, -179.32 | APE8-dihe-in | -97.31, 129.92 | APE8-rot-in | 316.69 | APE67-dihe-in | -69.15, -20.09 | -50.08, -47.79 | APE12-dist-in | 8.971 | APE11-dist-in | 11.233 | APE10-dist-in | 5.229 | APE9-dist-in | 3.486 | None | SEP474 | SEP474 | XRAY | 2.592 | 0.208 | 0.251 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 7cmb | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4O0VA | O96013 | 300 | 589 | 591.0 | 2OL:60601 | Type1.5_Back | Active | DFGin | 7.72 | 14.855 | BLAminus | -129.91, -179.13 | 52.93, 70.48 | -91.0, 31.77 | 289.31, 80.54 | -68.79, -11.49 | in-in | in | 9.386 | Saltbr-in | 2.715 | HRD-in | -63.47, -48.3 | 66.54, 12.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.98 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.31, 136.62 | APE9-dihe-na | 128.1, -161.84 | APE8-dihe-in | -105.46, 125.26 | APE8-rot-in | 314.65 | APE67-dihe-in | -70.36, -25.33 | -37.86, -50.41 | APE12-dist-in | 9.483 | APE11-dist-in | 11.399 | APE10-dist-in | 5.692 | APE9-dist-in | 3.35 | None | SEP474 | SEP474 | XRAY | 2.8 | 0.204 | 0.253 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4o0v | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4O0XA | O96013 | 300 | 589 | 591.0 | 2OQ:60601 | Type1.5_Back | Active | DFGin | 7.686 | 14.42 | BLAminus | -143.48, 175.23 | 50.73, 80.07 | -96.8, 29.16 | 288.57, 62.64 | -65.03, -22.79 | in-in | in | 7.841 | Saltbr-in | 2.524 | HRD-in | -64.27, -54.17 | 74.62, 7.89 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.044 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.91, 146.7 | APE9-dihe-na | 131.01, -164.91 | APE8-dihe-in | -110.0, 119.08 | APE8-rot-in | 309.56 | APE67-dihe-in | -57.87, -20.38 | -32.76, -63.35 | APE12-dist-in | 9.115 | APE11-dist-in | 11.502 | APE10-dist-in | 5.674 | APE9-dist-in | 3.39 | None | SEP474 | SEP474 | XRAY | 2.483 | 0.242 | 0.242 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4o0x | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4O0YA | O96013 | 300 | 589 | 591.0 | 2OO:60601 | Type1.5_Back | Active | DFGin | 7.439 | 13.922 | BLAminus | -135.18, 176.5 | 49.39, 78.85 | -92.46, 20.76 | 288.83, 77.11 | -54.08, -29.88 | in-in | in | 7.462 | Saltbr-in | 2.628 | HRD-in | -74.32, -48.56 | 73.38, 6.1 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.855 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -124.29, 136.66 | APE9-dihe-na | 144.79, -161.28 | APE8-dihe-in | -119.15, 122.67 | APE8-rot-in | 309.1 | APE67-dihe-in | -63.4, -19.31 | -38.26, -57.11 | APE12-dist-in | 9.651 | APE11-dist-in | 11.689 | APE10-dist-in | 5.96 | APE9-dist-in | 3.34 | None | SEP474 | SEP474 | XRAY | 2.2 | 0.2 | 0.238 | A | 293 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4o0y | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4XBRA | O96013 | 177 | 589 | 591.0 | ATP:60601 | ATPlike | Inactive | DFGin | 5.852 | 14.061 | ABAminus | -142.04, -22.23 | -111.42, 72.59 | -86.56, 10.51 | 310.81, 99.4 | -46.84, -40.66 | in-in | in | 7.009 | Saltbr-in | 3.158 | HRD-in | -84.11, -33.57 | 58.48, -1.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.974 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.96, 132.02 | APE9-dihe-na | 150.85, -176.82 | APE8-dihe-in | -102.34, 122.5 | APE8-rot-in | 312.14 | APE67-dihe-in | -59.91, -25.15 | -35.82, -60.88 | APE12-dist-in | 9.335 | APE11-dist-in | 11.927 | APE10-dist-in | 6.05 | APE9-dist-in | 3.396 | None | SEP474 | SEP474 | XRAY | 2.94 | 0.191 | 0.23 | A | 366 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4xbr | Homo sapiens | STE_PAK4_HUMAN | STE | 3.7e-88 | 301.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIGA | O96013 | 298 | 590 | 591.0 | ANP:1001 | ATPlike | Inactive | DFGin | 5.976 | 13.995 | BLAminus | -134.45, -166.25 | 59.06, 57.3 | -88.34, 9.13 | 298.9, 106.14 | -61.58, -20.66 | in-in | in | 7.133 | Saltbr-in | 3.168 | HRD-in | -77.25, -46.66 | 72.07, -3.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.86 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -129.47, 161.1 | APE9-dihe-na | 110.61, 163.55 | APE8-dihe-in | -79.54, 130.34 | APE8-rot-out | 29.96 | APE67-dihe-in | -76.38, -28.34 | -35.31, -49.63 | APE12-dist-in | 9.418 | APE11-dist-in | 11.569 | APE10-dist-in | 5.635 | APE9-dist-in | 3.369 | None | SEP474 | SEP474 | XRAY | 3.01 | 0.197 | 0.221 | A | 346 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fig | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIEA | O96013 | 49 | 590 | 591.0 | ANP:1001 | ATPlike | Inactive | DFGin | 6.278 | 14.03 | BLAminus | -142.71, -177.86 | 63.75, 67.7 | -92.97, 13.53 | 295.29, 98.36 | -64.15, -7.0 | in-out | in | 6.991 | Saltbr-out | 3.974 | HRD-in | -74.78, -36.69 | 67.65, -13.13 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.856 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -135.98, 139.97 | APE9-dihe-na | 123.6, -177.34 | APE8-dihe-in | -84.44, 139.76 | APE8-rot-out | 19.51 | APE67-dihe-in | -74.38, -37.99 | -51.24, -48.18 | APE12-dist-in | 9.515 | APE11-dist-in | 11.685 | APE10-dist-in | 5.909 | APE9-dist-in | 3.508 | None | SEP474 | SEP474 | XRAY | 3.11 | 0.257 | 0.276 | A | 423 | 301 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fie | Homo sapiens | STE_PAK4_HUMAN | STE | 5.6e-88 | 300.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIEB | O96013 | 49 | 590 | 591.0 | ANP:1001 | ATPlike | Inactive | DFGin | 6.278 | 14.031 | BLAminus | -142.24, -177.62 | 63.59, 67.55 | -92.7, 13.49 | 295.33, 98.22 | -64.04, -7.21 | in-out | in | 6.989 | Saltbr-out | 3.957 | HRD-in | -74.95, -36.21 | 66.97, -12.74 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.857 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.0, 139.86 | APE9-dihe-na | 123.6, -177.41 | APE8-dihe-in | -84.57, 139.76 | APE8-rot-out | 19.62 | APE67-dihe-in | -74.42, -37.89 | -51.19, -48.15 | APE12-dist-in | 9.515 | APE11-dist-in | 11.689 | APE10-dist-in | 5.912 | APE9-dist-in | 3.51 | None | SEP474 | SEP474 | XRAY | 3.11 | 0.257 | 0.276 | B | 423 | 301 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fie | Homo sapiens | STE_PAK4_HUMAN | STE | 5.6e-88 | 300.6 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 2BVAA | O96013 | 300 | 587 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 7.438 | 16.475 | BLAminus | -117.27, -176.72 | 56.65, 71.44 | -91.27, 35.1 | 289.21, 80.8 | -69.61, -2.94 | out-out | out | 10.481 | Saltbr-out | 4.02 | HRD-in | -57.52, -60.13 | 72.86, 5.02 | out-out-in | SNCooi | out-in | ActLoopNT-out | 3.877 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.79, 153.17 | APE9-dihe-na | 127.58, -141.52 | APE8-dihe-in | -136.11, 111.21 | APE8-rot-in | 333.57 | APE67-dihe-in | -60.96, -14.16 | -40.33, -50.6 | APE12-dist-in | 8.848 | APE11-dist-in | 11.484 | APE10-dist-in | 5.83 | APE9-dist-in | 3.471 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.192 | 0.269 | A | 292 | 273 | 15 | 0 | 0 | 2 | [[321, 572]] | 1.0 | 2bva | Homo sapiens | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 2BVAB | O96013 | 301 | 587 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 7.572 | 17.238 | BLAminus | -131.91, -158.23 | 65.58, 44.26 | -84.57, 26.99 | 293.34, 56.33 | -60.85, -21.66 | out-out | out | 11.675 | Saltbr-out | 7.148 | HRD-in | -60.3, -59.82 | 75.14, 24.4 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.499 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.93, 163.72 | APE9-dihe-na | 104.79, -155.19 | APE8-dihe-in | -112.34, 124.37 | APE8-rot-in | 319.0 | APE67-dihe-in | -73.92, -14.55 | -41.39, -45.76 | APE12-dist-in | 8.588 | APE11-dist-in | 11.399 | APE10-dist-in | 5.909 | APE9-dist-in | 3.197 | None | SEP474 | SEP474 | XRAY | 2.3 | 0.192 | 0.269 | B | 292 | 275 | 12 | 0 | 0 | 2 | [[321, 572]] | 1.0 | 2bva | Homo sapiens | STE_PAK4_HUMAN | STE | 1.7e-88 | 302.2 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 8YHKA | O96013 | 298 | 591 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 6.394 | 13.95 | BLAminus | -144.78, -174.84 | 60.87, 52.46 | -74.27, -7.16 | 291.41, 99.22 | -44.42, -31.64 | in-out | in | 7.212 | Saltbr-out | 5.663 | HRD-out | -76.82, 93.99 | -85.26, 6.82 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.734 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.02, 139.67 | APE9-dihe-na | 131.69, -172.38 | APE8-dihe-in | -96.54, 118.36 | APE8-rot-in | 308.12 | APE67-dihe-in | -79.25, -37.48 | -34.17, -42.18 | APE12-dist-in | 9.944 | APE11-dist-in | 11.39 | APE10-dist-in | 5.545 | APE9-dist-in | 3.243 | None | None | None | XRAY | 3.3 | 0.253 | 0.319 | A | 301 | 294 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8yhk | Homo sapiens | STE_PAK4_HUMAN | STE | 1.9e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4XBUA | O96013 | 297 | 589 | 591.0 | No_ligand | No_ligand | Inactive | DFGin | 7.426 | 14.345 | BLAminus | -134.76, -171.38 | 58.13, 68.14 | -90.95, 10.75 | 282.43, 88.09 | -57.4, -26.1 | in-out | in | 8.875 | Saltbr-out | 4.505 | HRD-in | -80.19, -49.71 | 68.99, 2.54 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.842 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.64, 133.45 | APE9-dihe-na | 156.19, -154.61 | APE8-dihe-in | -123.57, 122.27 | APE8-rot-in | 305.74 | APE67-dihe-in | -70.59, -15.2 | -40.43, -52.25 | APE12-dist-in | 8.806 | APE11-dist-in | 11.559 | APE10-dist-in | 5.875 | APE9-dist-in | 3.518 | None | SEP474 | SEP474 | XRAY | 2.06 | 0.201 | 0.243 | A | 326 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4xbu | Homo sapiens | STE_PAK4_HUMAN | STE | 2.5e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 8AHIA | O96013 | 300 | 591 | 591.0 | M56:601 | Type1 | Inactive | DFGin | 9.181 | 14.38 | BLAminus | -137.45, -173.93 | 55.91, 63.31 | -90.54, 16.67 | 287.37, 76.55 | -61.73, -19.34 | in-out | in | 7.694 | Saltbr-out | 3.645 | HRD-in | -78.82, -49.15 | 74.56, 0.81 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.882 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.24, 128.69 | APE9-dihe-na | 143.74, -151.59 | APE8-dihe-in | -115.17, 123.77 | APE8-rot-in | 313.27 | APE67-dihe-in | -68.11, -27.23 | -45.23, -43.93 | APE12-dist-in | 8.803 | APE11-dist-in | 11.358 | APE10-dist-in | 5.796 | APE9-dist-in | 3.534 | L310A | SEP474 | SEP474 | XRAY | 2.69 | 0.16 | 0.249 | A | 297 | 292 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 8ahi | Homo sapiens | STE_PAK4_HUMAN | STE | 1.8e-88 | 302.1 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5VEDA | O96013 | 300 | 589 | 591.0 | STU:601 | Type1 | Inactive | DFGin | 7.591 | 14.871 | BLAminus | -137.67, -169.84 | 57.61, 74.14 | -100.29, 38.24 | 286.21, 78.54 | -72.3, -31.74 | in-out | in | 8.771 | Saltbr-out | 5.279 | HRD-in | -70.67, -47.26 | 60.82, 22.3 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.978 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.74, 169.93 | APE9-dihe-na | 110.0, -167.24 | APE8-dihe-in | -107.4, 122.99 | APE8-rot-in | 313.49 | APE67-dihe-in | -72.02, -18.93 | -37.81, -47.81 | APE12-dist-in | 8.493 | APE11-dist-in | 11.13 | APE10-dist-in | 5.271 | APE9-dist-in | 3.412 | None | SEP474 | SEP474 | XRAY | 2.301 | 0.231 | 0.277 | A | 319 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5ved | Homo sapiens | STE_PAK4_HUMAN | STE | 2.4e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 5VEEA | O96013 | 300 | 589 | 591.0 | 981:601 | Type1 | Inactive | DFGin | 6.832 | 15.436 | BLAminus | -149.85, -166.61 | 63.61, 64.4 | -91.35, 12.72 | 287.99, 79.38 | -42.54, -35.66 | in-out | in | 8.369 | Saltbr-out | 6.665 | HRD-in | -63.93, -45.62 | 68.7, 8.17 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.12 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.59, 147.54 | APE9-dihe-na | 146.37, -170.93 | APE8-dihe-in | -104.03, 125.68 | APE8-rot-in | 311.71 | APE67-dihe-in | -46.67, -33.8 | -40.96, -66.37 | APE12-dist-in | 9.09 | APE11-dist-in | 11.607 | APE10-dist-in | 5.815 | APE9-dist-in | 3.64 | None | SEP474 | SEP474 | XRAY | 2.5 | 0.231 | 0.276 | A | 319 | 290 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 5vee | Homo sapiens | STE_PAK4_HUMAN | STE | 2.4e-88 | 301.8 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| PAK4_HUMAN | 4FIGB | O96013 | 298 | 590 | 591.0 | ANP:602 | ATPlike | Inactive | DFGin | 5.979 | 13.845 | None | -136.1, -40.27 | -82.41, 70.29 | -85.54, 12.48 | 305.29, 106.7 | -66.77, -24.27 | in-in | in | 7.007 | Saltbr-in | 3.047 | HRD-in | -63.37, -48.9 | 73.21, -4.05 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.929 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -134.8, 141.64 | APE9-dihe-na | 130.69, -165.45 | APE8-dihe-in | -110.43, 122.9 | APE8-rot-in | 324.7 | APE67-dihe-in | -77.33, -31.89 | -29.23, -51.11 | APE12-dist-in | 9.706 | APE11-dist-in | 11.743 | APE10-dist-in | 5.92 | APE9-dist-in | 3.386 | None | SEP474 | SEP474 | XRAY | 3.01 | 0.197 | 0.221 | B | 346 | 293 | 0 | 0 | 0 | 0 | [[321, 572]] | 1.0 | 4fig | Homo sapiens | STE_PAK4_HUMAN | STE | 3.1e-88 | 301.5 | 5 | 257 | 253 | 457 | 458 | 459 | 461 | 463 | 350 | 366 | 370 | 437 | 439 | 438 | 440 | 497 | 485 | 480 | 479 | 478 | 477 | 476 | 475 | 474 | 396 | Serine/threonine-protein kinase PAK 4 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|