| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| JAK3-2 | AF-P52333-K2A | P52333 | 814 | 1105 | 1124.0 | No_ligand | No_ligand | Active | DFGin | 6.1026 | 13.7936 | BLAminus | -134.56, -179.19 | 51.31, 75.31 | -82.94, 20.6 | 292.85, 86.33 | -61.55, -30.97 | in-in | in | 8.2483 | Saltbr-in | 2.6953 | HRD-in | -70.59, -43.72 | 65.57, -21.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8552 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -56.42, 123.08 | APE9-dihe-in | -125.57, 135.88 | APE8-dihe-in | -78.86, 68.83 | APE8-rot-na | 34.92 | APE67-dihe-in | -75.13, -6.36 | -53.49, -31.1 | APE12-dist-na | 10.5223 | APE11-dist-na | 9.5286 | APE10-dist-na | 10.1849 | APE9-dist-in | 7.1879 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 292.0 | 292.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | AF-P52333-K2 | TYR_JAK3-2_HUMAN | TYR | 4.6e-81 | 277.9 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | AF-P52333-K4A | P52333 | 814 | 1105 | 1124.0 | No_ligand | No_ligand | Active | DFGin | 6.1108 | 13.7687 | BLAminus | -141.5, -174.59 | 54.28, 75.11 | -88.15, 17.45 | 293.92, 89.95 | -59.55, -34.59 | in-in | in | 8.1169 | Saltbr-in | 2.6779 | HRD-in | -78.79, -45.55 | 61.88, 0.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8819 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -61.64, 120.49 | APE9-dihe-in | -128.67, 141.65 | APE8-dihe-in | -77.57, 68.42 | APE8-rot-na | 36.41 | APE67-dihe-in | -72.34, -8.01 | -50.71, -34.24 | APE12-dist-na | 13.4854 | APE11-dist-na | 9.5574 | APE10-dist-na | 10.1649 | APE9-dist-in | 6.4962 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 292.0 | 292.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | AF-P52333-K4 | TYR_JAK3-2_HUMAN | TYR | 4.6e-81 | 277.9 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6AAKC | P52333 | 814 | 1099 | 1124.0 | 9T6:1201 | Type1 | Active | DFGin | 6.7877 | 14.6346 | BLAminus | -114.47, 172.4 | 69.03, 86.81 | -107.19, 29.58 | 286.76, 78.99 | -58.47, -55.72 | in-in | in | 8.2406 | Saltbr-in | 2.7237 | HRD-in | -89.94, -41.82 | 71.73, -3.81 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7832 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.85, 76.94 | APE9-dihe-in | -171.36, 163.86 | APE8-dihe-in | -58.47, 128.31 | APE8-rot-na | 338.62 | APE67-dihe-in | -73.56, -5.95 | -79.88, -15.99 | APE12-dist-na | 12.9746 | APE11-dist-na | 9.2183 | APE10-dist-na | 10.3986 | APE9-dist-in | 7.7513 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | C | 287.0 | 276.0 | 10 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6aak | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7UYVA | P52333 | 814 | 1100 | 1124.0 | OV5:1201 | Type1 | Active | DFGin | 6.3763 | 14.2869 | BLAminus | -136.33, -178.14 | 60.47, 77.06 | -94.46, 22.49 | 283.21, 76.25 | -61.39, -33.76 | in-in | in | 8.2009 | Saltbr-in | 2.6421 | HRD-in | -69.18, -41.57 | 72.69, -12.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7503 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.18, 82.75 | APE9-dihe-in | -112.58, 159.26 | APE8-dihe-in | -47.72, 129.83 | APE8-rot-na | 329.64 | APE67-dihe-in | -81.57, 1.11 | -69.92, -19.01 | APE12-dist-na | 11.5311 | APE11-dist-na | 8.0482 | APE10-dist-na | 11.6832 | APE9-dist-in | 7.3388 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | A | 291.0 | 278.0 | 9 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7UYVB | P52333 | 814 | 1100 | 1124.0 | OV5:1201 | Type1 | Active | DFGin | 6.2251 | 14.2162 | BLAminus | -136.69, -173.44 | 56.56, 80.52 | -96.27, 21.5 | 284.08, 77.64 | -57.68, -39.3 | in-in | in | 8.1504 | Saltbr-in | 2.6309 | HRD-in | -80.27, -44.25 | 68.81, -0.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7556 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -75.34, 85.59 | APE9-dihe-in | -127.16, 148.54 | APE8-dihe-in | -37.53, 121.21 | APE8-rot-na | 325.53 | APE67-dihe-in | -80.04, -3.68 | -72.05, -16.34 | APE12-dist-na | 11.5779 | APE11-dist-na | 9.1429 | APE10-dist-na | 12.2547 | APE9-dist-in | 7.3873 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | B | 291.0 | 284.0 | 3 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3PJCA | P52333 | 815 | 1104 | 1124.0 | PJC:800 | Type1 | Active | DFGin | 6.6986 | 14.412 | BLAminus | -131.65, -174.74 | 53.97, 85.79 | -100.88, 20.12 | 280.65, 74.1 | -60.63, -24.35 | in-in | in | 8.6962 | Saltbr-in | 2.6139 | HRD-in | -69.63, -48.63 | 77.02, -5.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8226 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.16, 145.45 | APE9-dihe-in | -115.3, 150.0 | APE8-dihe-in | -81.75, 75.29 | APE8-rot-na | 32.65 | APE67-dihe-in | -79.59, -4.38 | -53.88, -28.84 | APE12-dist-na | 13.2005 | APE11-dist-na | 11.5918 | APE10-dist-na | 12.7974 | APE9-dist-in | 7.9845 | None | None | None | XRAY | 2.2 | 0.182 | 0.215 | A | 315.0 | 286.0 | 4 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3pjc | TYR_JAK3-2_HUMAN | TYR | 6.1e-81 | 277.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6GL9A | P52333 | 812 | 1103 | 1124.0 | F3W:1201 | Type1 | Active | DFGin | 6.2475 | 14.0115 | BLAminus | -125.6, -168.17 | 49.24, 81.71 | -98.97, 21.2 | 279.85, 75.03 | -60.06, -26.17 | in-in | in | 7.7934 | Saltbr-in | 2.6834 | HRD-in | -78.49, -49.26 | 75.45, 0.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7882 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.67, 117.53 | APE9-dihe-in | -98.8, 151.13 | APE8-dihe-in | -79.69, 90.74 | APE8-rot-na | 31.23 | APE67-dihe-in | -78.37, -0.16 | -59.8, -32.45 | APE12-dist-na | 9.3301 | APE11-dist-na | 10.7633 | APE10-dist-na | 11.753 | APE9-dist-in | 6.9787 | None | None | None | XRAY | 1.7 | 0.209 | 0.244 | A | 294.0 | 292.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6gl9 | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6GL9B | P52333 | 813 | 1103 | 1124.0 | F3W:1201 | Type1 | Active | DFGin | 6.21 | 14.019 | BLAminus | -123.31, -164.34 | 42.61, 83.03 | -97.02, 22.96 | 280.36, 70.4 | -63.87, -26.0 | in-in | in | 7.7595 | Saltbr-in | 2.667 | HRD-in | -78.77, -47.46 | 73.56, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7746 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.72, 116.63 | APE9-dihe-in | -97.44, 150.89 | APE8-dihe-in | -77.79, 91.0 | APE8-rot-na | 32.15 | APE67-dihe-in | -73.22, -2.71 | -60.01, -35.33 | APE12-dist-na | 9.3264 | APE11-dist-na | 10.7827 | APE10-dist-na | 11.7277 | APE9-dist-in | 6.9767 | None | None | None | XRAY | 1.7 | 0.209 | 0.244 | B | 294.0 | 291.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6gl9 | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7C3NA | P52333 | 814 | 1102 | 1124.0 | FHX:9000 | Type1 | Inactive | DFGin | 6.068 | 13.3862 | ABAminus | -140.24, 14.21 | -145.02, 134.62 | -131.29, 32.79 | 294.67, 80.18 | -64.88, -27.68 | in-in | in | 8.233 | Saltbr-in | 2.7822 | HRD-in | -78.6, -47.11 | 71.84, 1.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8064 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.04, 126.4 | APE9-dihe-in | -81.7, 145.46 | APE8-dihe-in | -77.41, 71.31 | APE8-rot-na | 31.38 | APE67-dihe-in | -79.88, -2.49 | -60.07, -26.59 | APE12-dist-na | 11.7358 | APE11-dist-na | 10.4538 | APE10-dist-na | 12.3096 | APE9-dist-in | 7.2655 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 1.98 | 0.17 | 0.194 | A | 315.0 | 289.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7c3n | TYR_JAK3-2_HUMAN | TYR | 6.1e-81 | 277.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3LXKA | P52333 | 815 | 1098 | 1124.0 | MI1:1125 | Type1 | Inactive | DFGin | 6.0647 | 13.0171 | ABAminus | -128.16, 7.24 | -148.97, 145.15 | -138.77, 31.19 | 300.52, 88.17 | -60.03, -27.75 | in-in | in | 8.251 | Saltbr-in | 2.7565 | HRD-in | -78.64, -46.72 | 70.97, -5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8402 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -118.3, 17.09 | APE9-dihe-in | -92.59, 156.17 | APE8-dihe-in | -54.3, 131.46 | APE8-rot-na | 335.17 | APE67-dihe-in | -82.42, -7.27 | -71.07, -8.83 | APE12-dist-na | 14.2685 | APE11-dist-na | 9.9216 | APE10-dist-na | 10.5049 | APE9-dist-in | 7.209 | C1048S | None | None | XRAY | 2.0 | 0.205 | 0.265 | A | 327.0 | 279.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3lxk | TYR_JAK3-2_HUMAN | TYR | 3.2e-81 | 278.4 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5W86A | P52333 | 814 | 1098 | 1124.0 | 9YV:4000 | Type1 | Inactive | DFGin | 6.508 | 14.2333 | BLAminus | -130.78, -178.04 | 55.33, 86.29 | -99.45, 24.99 | 285.64, 80.91 | -59.45, -36.09 | in-in | in | 8.3613 | Saltbr-in | 2.7197 | HRD-in | -61.74, -49.91 | 79.02, -19.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8338 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -62.63 | APE8-dihe-in | -73.09, 69.06 | APE8-rot-na | 28.5 | APE67-dihe-in | -76.22, -6.14 | -68.16, -24.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.3257 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | A | 287.0 | 271.0 | 14 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5W86D | P52333 | 814 | 1099 | 1124.0 | 9YV:4000 | Type1 | Inactive | DFGin | 6.5614 | 14.2551 | BLAminus | -130.88, -178.77 | 56.18, 85.97 | -99.02, 25.19 | 285.73, 80.24 | -59.91, -34.36 | in-in | in | 8.1827 | Saltbr-in | 2.7569 | HRD-in | -62.59, -49.55 | 78.85, -19.41 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.814 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -64.08 | APE8-dihe-in | -73.59, 57.74 | APE8-rot-na | 27.09 | APE67-dihe-in | -73.08, -10.82 | -59.31, -28.98 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.2414 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | D | 287.0 | 274.0 | 12 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6AAKA | P52333 | 815 | 1098 | 1124.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.4258 | 14.4877 | BLAminus | -141.28, -175.48 | 60.31, 80.99 | -97.75, 30.98 | 284.74, 77.33 | -61.02, -46.05 | in-in | in | 8.5254 | Saltbr-in | 2.67 | HRD-in | -75.62, -45.99 | 77.6, -18.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7362 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.2, -11.07 | APE9-dihe-in | -68.95, 155.07 | APE8-dihe-in | -47.57, 131.1 | APE8-rot-na | 329.72 | APE67-dihe-in | -73.4, -26.9 | -66.76, -22.48 | APE12-dist-na | 11.9929 | APE11-dist-na | 8.6734 | APE10-dist-na | 11.3981 | APE9-dist-in | 7.4704 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | A | 287.0 | 277.0 | 7 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6aak | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6AAKB | P52333 | 815 | 1100 | 1124.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.549 | 14.3135 | BLAminus | -132.57, -171.05 | 56.03, 83.09 | -98.42, 24.6 | 281.38, 75.24 | -63.47, -40.11 | in-in | in | 8.0358 | Saltbr-in | 2.7546 | HRD-in | -65.5, -48.18 | 78.33, -13.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9074 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.61, -28.55 | APE9-dihe-in | -64.46, 151.35 | APE8-dihe-in | -40.19, 130.42 | APE8-rot-na | 326.93 | APE67-dihe-in | -77.17, -14.56 | -72.74, -10.57 | APE12-dist-na | 13.1081 | APE11-dist-na | 9.526 | APE10-dist-na | 10.0845 | APE9-dist-in | 7.2029 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | B | 287.0 | 285.0 | 1 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6aak | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZC6A | P52333 | 814 | 1100 | 1124.0 | VFC:2103 | Type1 | Inactive | DFGin | 6.3992 | 14.249 | BLAminus | -132.73, -176.21 | 56.45, 83.25 | -97.56, 22.77 | 285.82, 73.7 | -62.6, -27.55 | in-in | in | 8.2919 | Saltbr-in | 2.8022 | HRD-in | -72.44, -47.03 | 73.15, -6.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7419 | ActLoopCT-out | TYR | APEdihe_noiai | APEdist_aaai | APE10-dihe-none | 999.0, 118.21 | APE9-dihe-out | -83.58, -179.01 | APE8-dihe-in | -60.9, 137.23 | APE8-rot-na | 332.96 | APE67-dihe-in | -76.45, -9.26 | -65.3, -16.84 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 9.5354 | APE9-dist-in | 5.9074 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | A | 288.0 | 279.0 | 8 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZC6C | P52333 | 814 | 1100 | 1124.0 | VFC:2103 | Type1 | Inactive | DFGin | 6.2807 | 14.0027 | BLAminus | -123.64, -177.74 | 61.16, 80.91 | -97.9, 27.04 | 288.23, 77.53 | -66.72, -26.1 | in-in | in | 8.1905 | Saltbr-in | 2.6842 | HRD-in | -72.21, -46.31 | 77.05, -24.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7606 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -54.85 | APE8-dihe-in | -77.18, 80.1 | APE8-rot-na | 33.09 | APE67-dihe-in | -76.9, -10.93 | -67.13, -29.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.1774 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | C | 288.0 | 277.0 | 10 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZEPA | P52333 | 814 | 1098 | 1124.0 | 1NX:2099 | Type1 | Inactive | DFGin | 6.4201 | 14.3445 | BLAminus | -139.2, 179.6 | 58.57, 83.63 | -103.43, 28.82 | 290.46, 79.48 | -67.26, -39.4 | in-in | in | 8.1983 | Saltbr-in | 2.7236 | HRD-in | -72.97, -44.84 | 72.81, -0.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7642 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -90.83, 0.53 | APE9-dihe-in | -141.71, 168.37 | APE8-dihe-in | -61.5, 133.7 | APE8-rot-na | 333.46 | APE67-dihe-in | -72.33, -1.68 | -64.6, -21.71 | APE12-dist-na | 13.4306 | APE11-dist-na | 10.6555 | APE10-dist-na | 6.8245 | APE9-dist-in | 6.4001 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | A | 288.0 | 276.0 | 9 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3zep | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7UYVC | P52333 | 812 | 1100 | 1124.0 | OV5:1201 | Type1 | Inactive | DFGin | 6.5497 | 14.2474 | BLAminus | -139.0, -178.89 | 62.41, 84.96 | -102.47, 24.54 | 285.05, 80.61 | -63.66, -34.31 | in-in | in | 8.1764 | Saltbr-in | 2.7239 | HRD-in | -72.48, -47.02 | 76.02, -14.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.6962 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -72.04, 75.71 | APE9-dihe-in | -159.34, 174.75 | APE8-dihe-in | -55.7, 114.03 | APE8-rot-na | 331.85 | APE67-dihe-in | -81.89, -1.84 | -68.05, -12.84 | APE12-dist-na | 12.9994 | APE11-dist-na | 8.9457 | APE10-dist-na | 10.9307 | APE9-dist-out | 8.0032 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | C | 291.0 | 281.0 | 8 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4RIOA | P52333 | 815 | 1099 | 1124.0 | 3QX:4000 | Type1 | Inactive | DFGin | 6.3935 | 13.5705 | BLAminus | -146.26, -172.55 | 60.58, 82.0 | -101.14, 19.19 | 286.89, 85.95 | -65.85, -24.53 | in-in | in | 7.6666 | Saltbr-in | 2.8105 | HRD-in | -70.94, -43.53 | 62.59, 2.86 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9783 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -135.63, 27.38 | APE9-dihe-in | -118.75, 159.28 | APE8-dihe-in | -55.16, 127.94 | APE8-rot-na | 333.58 | APE67-dihe-in | -76.1, -3.72 | -64.2, -13.91 | APE12-dist-na | 12.5847 | APE11-dist-na | 9.8864 | APE10-dist-na | 9.9276 | APE9-dist-in | 7.1524 | C811S,C1040S,C1048S | None | None | XRAY | 2.69 | 0.218 | 0.281 | A | 293.0 | 285.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4rio | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5WFJA | P52333 | 817 | 1099 | 1124.0 | 9Z4:4000 | Type1 | Inactive | DFGin | 6.5811 | 13.8338 | BLAminus | -136.44, -170.83 | 58.73, 75.78 | -96.48, 23.06 | 286.97, 86.34 | -64.05, -24.53 | in-in | in | 7.6299 | Saltbr-in | 2.8738 | HRD-in | -76.6, -46.72 | 68.06, 1.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9182 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.32, 20.43 | APE9-dihe-in | -103.33, 153.28 | APE8-dihe-in | -50.05, 126.35 | APE8-rot-na | 333.7 | APE67-dihe-in | -76.71, 0.96 | -65.58, -12.14 | APE12-dist-na | 13.631 | APE11-dist-na | 9.8634 | APE10-dist-na | 10.1142 | APE9-dist-in | 7.0412 | C811S,C1040S,C1048S | None | None | XRAY | 2.48 | 0.205 | 0.255 | A | 293.0 | 265.0 | 18 | 31 | 29 | 2 | [[521, 779], [822, 1097]] | 2.0 | 5wfj | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4HVDA | P52333 | 815 | 1101 | 1124.0 | 933:1202 | Type1 | Inactive | DFGin | 6.5272 | 14.0171 | BLAminus | -128.55, -166.42 | 58.39, 76.56 | -98.5, 22.97 | 288.27, 78.76 | -65.56, -24.6 | in-in | in | 8.047 | Saltbr-in | 2.8425 | HRD-in | -70.62, -50.61 | 83.01, -13.8 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8441 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -120.35, 6.88 | APE9-dihe-in | -87.79, 153.51 | APE8-dihe-in | -47.35, 128.71 | APE8-rot-na | 328.03 | APE67-dihe-in | -81.29, -0.66 | -70.05, -11.78 | APE12-dist-na | 13.6702 | APE11-dist-na | 9.8379 | APE10-dist-na | 10.1082 | APE9-dist-in | 7.3252 | C1040S,C1048S | None | None | XRAY | 1.85 | 0.225 | 0.259 | A | 314.0 | 276.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvd | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4HVGA | P52333 | 814 | 1103 | 1124.0 | 19Q:1201 | Type1 | Inactive | DFGin | 6.3691 | 14.0706 | BLAminus | -130.41, -171.25 | 53.38, 75.08 | -85.23, 20.51 | 289.87, 75.57 | -58.89, -29.62 | in-in | in | 8.256 | Saltbr-in | 2.8006 | HRD-in | -81.72, -46.13 | 83.55, -16.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9723 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -135.6, 18.04 | APE9-dihe-in | -102.46, 155.94 | APE8-dihe-in | -50.03, 129.65 | APE8-rot-na | 326.24 | APE67-dihe-in | -77.88, -2.28 | -61.37, -21.51 | APE12-dist-na | 13.6391 | APE11-dist-na | 9.8591 | APE10-dist-na | 10.1069 | APE9-dist-in | 7.4421 | C1040S,C1048S | None | None | XRAY | 2.75 | 0.214 | 0.274 | A | 314.0 | 281.0 | 9 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvg | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4HVHA | P52333 | 814 | 1102 | 1124.0 | 19R:1201 | Type1 | Inactive | DFGin | 6.4361 | 14.1039 | BLAminus | -140.81, -174.18 | 54.94, 86.96 | -103.32, 27.47 | 289.17, 75.35 | -59.86, -26.99 | in-in | in | 8.1031 | Saltbr-in | 2.73 | HRD-in | -70.65, -47.69 | 79.95, -7.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8656 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -125.66, 18.79 | APE9-dihe-in | -103.72, 157.23 | APE8-dihe-in | -46.25, 127.99 | APE8-rot-na | 329.23 | APE67-dihe-in | -82.32, 1.96 | -65.92, -16.55 | APE12-dist-na | 13.6054 | APE11-dist-na | 9.7978 | APE10-dist-na | 10.0657 | APE9-dist-in | 7.3949 | C1040S,C1048S | None | None | XRAY | 2.3 | 0.23 | 0.283 | A | 314.0 | 278.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvh | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4HVIA | P52333 | 815 | 1101 | 1124.0 | 19S:1201 | Type1 | Inactive | DFGin | 6.4427 | 13.9006 | BLAminus | -133.13, -169.35 | 58.25, 80.79 | -103.46, 21.02 | 290.11, 82.66 | -64.8, -24.06 | in-in | in | 8.1481 | Saltbr-in | 2.7134 | HRD-in | -70.83, -44.69 | 73.14, -9.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0118 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.42, 8.91 | APE9-dihe-in | -93.49, 161.0 | APE8-dihe-in | -50.05, 128.83 | APE8-rot-na | 327.89 | APE67-dihe-in | -77.81, -4.37 | -61.08, -19.7 | APE12-dist-na | 13.3068 | APE11-dist-na | 9.5384 | APE10-dist-na | 9.8434 | APE9-dist-in | 7.267 | C1040S,C1048S | None | None | XRAY | 2.4 | 0.238 | 0.303 | A | 314.0 | 274.0 | 13 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvi | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4I6QA | P52333 | 815 | 1102 | 1124.0 | 1DT:1202 | Type1 | Inactive | DFGin | 6.5477 | 13.8797 | BLAminus | -122.27, -166.37 | 58.65, 80.25 | -102.66, 18.99 | 282.73, 92.38 | -63.16, -27.69 | in-in | in | 8.1701 | Saltbr-in | 2.6678 | HRD-in | -82.65, -46.76 | 80.12, -11.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8258 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.82, 1.26 | APE9-dihe-in | -88.25, 159.4 | APE8-dihe-in | -50.29, 130.77 | APE8-rot-na | 324.04 | APE67-dihe-in | -86.64, 4.17 | -68.93, -13.66 | APE12-dist-na | 13.7233 | APE11-dist-na | 9.8721 | APE10-dist-na | 9.9493 | APE9-dist-in | 7.3231 | C1040S,C1048S | None | None | XRAY | 1.85 | 0.198 | 0.245 | A | 314.0 | 277.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4i6q | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4QT1A | P52333 | 814 | 1102 | 1124.0 | 3C9:1201 | Type1 | Inactive | DFGin | 6.6492 | 13.9762 | BLAminus | -139.02, 177.24 | 52.6, 80.83 | -91.99, 24.19 | 292.74, 76.91 | -57.05, -27.61 | in-in | in | 7.854 | Saltbr-in | 2.8081 | HRD-in | -76.1, -42.64 | 74.06, 0.56 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8439 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.55, 16.0 | APE9-dihe-in | -104.71, 155.27 | APE8-dihe-in | -51.8, 130.25 | APE8-rot-na | 330.69 | APE67-dihe-in | -80.61, -3.03 | -68.8, -13.83 | APE12-dist-na | 13.5093 | APE11-dist-na | 9.8141 | APE10-dist-na | 9.9829 | APE9-dist-in | 7.1611 | C1040S,C1048S | None | None | XRAY | 2.4 | 0.21 | 0.273 | A | 314.0 | 277.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4qt1 | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5TOZA | P52333 | 815 | 1100 | 1124.0 | 7H4:1201 | Type1 | Inactive | DFGin | 6.4346 | 14.1797 | BLAminus | -132.42, -172.67 | 55.17, 83.47 | -97.89, 23.39 | 288.4, 75.31 | -59.42, -27.52 | in-in | in | 8.0531 | Saltbr-in | 2.7698 | HRD-in | -70.7, -45.74 | 70.21, -7.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8052 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.82, 11.45 | APE9-dihe-in | -93.23, 156.46 | APE8-dihe-in | -46.82, 125.7 | APE8-rot-na | 327.47 | APE67-dihe-in | -74.64, -1.89 | -65.68, -15.53 | APE12-dist-na | 13.7154 | APE11-dist-na | 9.6672 | APE10-dist-na | 10.1541 | APE9-dist-in | 7.336 | None | None | None | XRAY | 1.98 | 0.184 | 0.215 | A | 321.0 | 278.0 | 8 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5toz | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5TTSA | P52333 | 814 | 1100 | 1124.0 | 7KU:4000 | Type1 | Inactive | DFGin | 6.4256 | 14.158 | BLAminus | -129.0, -169.11 | 47.63, 82.34 | -97.79, 20.5 | 281.57, 83.57 | -59.54, -22.32 | in-in | in | 7.8793 | Saltbr-in | 2.727 | HRD-in | -71.68, -45.64 | 72.69, -11.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8295 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -120.94, 5.03 | APE9-dihe-in | -92.95, 155.15 | APE8-dihe-in | -50.68, 128.91 | APE8-rot-na | 333.75 | APE67-dihe-in | -73.89, 0.34 | -64.16, -15.93 | APE12-dist-na | 13.6385 | APE11-dist-na | 9.8268 | APE10-dist-na | 9.9629 | APE9-dist-in | 7.3964 | C1048S | None | None | XRAY | 2.34 | 0.205 | 0.263 | A | 321.0 | 274.0 | 13 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5tts | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5TTUA | P52333 | 815 | 1099 | 1124.0 | 7KV:1201 | Type1 | Inactive | DFGin | 6.5073 | 14.2203 | BLAminus | -134.44, -163.93 | 59.24, 64.07 | -87.63, 14.18 | 281.02, 85.09 | -61.33, -21.77 | in-in | in | 8.1783 | Saltbr-in | 2.6873 | HRD-in | -74.44, -46.15 | 74.73, -11.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.934 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.51, 0.99 | APE9-dihe-in | -84.97, 156.58 | APE8-dihe-in | -52.23, 128.18 | APE8-rot-na | 331.46 | APE67-dihe-in | -73.87, -5.17 | -63.29, -14.0 | APE12-dist-na | 13.6239 | APE11-dist-na | 9.6774 | APE10-dist-na | 9.9919 | APE9-dist-in | 7.2843 | C1048S | None | None | XRAY | 1.72 | 0.193 | 0.212 | A | 321.0 | 271.0 | 14 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5ttu | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5TTVA | P52333 | 814 | 1100 | 1124.0 | 7KX:4000 | Type1 | Inactive | DFGin | 6.389 | 13.9545 | BLAminus | -134.13, -173.38 | 47.72, 81.12 | -99.64, 24.47 | 284.98, 81.27 | -61.89, -30.49 | in-in | in | 7.571 | Saltbr-in | 2.7566 | HRD-in | -68.58, -49.94 | 77.2, -11.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.887 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.83, -8.71 | APE9-dihe-in | -81.68, 166.25 | APE8-dihe-in | -54.83, 134.34 | APE8-rot-na | 333.98 | APE67-dihe-in | -68.58, -14.21 | -64.91, -25.89 | APE12-dist-na | 13.454 | APE11-dist-na | 10.1045 | APE10-dist-na | 9.8444 | APE9-dist-in | 7.0476 | C1048S | None | None | XRAY | 1.93 | 0.195 | 0.25 | A | 321.0 | 280.0 | 7 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5ttv | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6DA4A | P52333 | 815 | 1099 | 1124.0 | G4V:1201 | Type1 | Inactive | DFGin | 6.3399 | 14.1592 | BLAminus | -125.34, -166.51 | 46.1, 93.47 | -106.56, 19.65 | 286.03, 81.95 | -61.5, -24.21 | in-in | in | 8.0349 | Saltbr-in | 2.8116 | HRD-in | -66.39, -43.11 | 68.24, -5.72 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8446 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -76.16, 17.06 | APE9-dihe-in | -99.01, 151.3 | APE8-dihe-in | -54.06, 116.09 | APE8-rot-na | 335.02 | APE67-dihe-in | -66.76, -9.61 | -46.02, -19.91 | APE12-dist-na | 13.2424 | APE11-dist-na | 9.376 | APE10-dist-na | 10.3711 | APE9-dist-in | 7.2615 | C1048S | None | None | XRAY | 2.9 | 0.229 | 0.263 | A | 321.0 | 281.0 | 4 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6da4 | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6DB3A | P52333 | 814 | 1100 | 1124.0 | G54:4000 | Type1 | Inactive | DFGin | 6.286 | 13.9012 | BLAminus | -131.89, -177.11 | 58.86, 88.06 | -99.15, 20.97 | 289.91, 81.31 | -57.3, -32.4 | in-in | in | 8.2338 | Saltbr-in | 2.6892 | HRD-in | -69.32, -44.77 | 72.88, -9.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7455 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.94, 10.67 | APE9-dihe-in | -91.58, 152.91 | APE8-dihe-in | -48.92, 124.78 | APE8-rot-na | 329.3 | APE67-dihe-in | -70.97, -6.33 | -60.73, -15.87 | APE12-dist-na | 13.7116 | APE11-dist-na | 9.5497 | APE10-dist-na | 10.1421 | APE9-dist-in | 7.3914 | C1048S | None | None | XRAY | 1.97 | 0.19 | 0.224 | A | 321.0 | 275.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6db3 | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6DB4A | P52333 | 814 | 1100 | 1124.0 | G4Y:4000 | Type1 | Inactive | DFGin | 6.3293 | 13.8866 | BLAminus | -129.96, -177.19 | 65.04, 85.51 | -102.45, 21.04 | 283.09, 83.98 | -63.09, -23.83 | in-in | in | 8.1031 | Saltbr-in | 2.6779 | HRD-in | -75.95, -47.04 | 72.28, -5.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.844 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.18, 10.26 | APE9-dihe-in | -87.73, 153.8 | APE8-dihe-in | -51.18, 129.01 | APE8-rot-na | 329.23 | APE67-dihe-in | -72.48, -3.98 | -65.43, -15.27 | APE12-dist-na | 14.0574 | APE11-dist-na | 9.8642 | APE10-dist-na | 10.2997 | APE9-dist-in | 7.1511 | C1048S | None | None | XRAY | 1.662 | 0.187 | 0.216 | A | 321.0 | 276.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6db4 | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6DUDA | P52333 | 814 | 1100 | 1124.0 | HB4:1201 | Type1 | Inactive | DFGin | 6.3774 | 14.08 | BLAminus | -130.37, -174.96 | 58.79, 79.77 | -94.85, 21.4 | 284.9, 80.47 | -61.75, -24.01 | in-in | in | 7.8751 | Saltbr-in | 2.7643 | HRD-in | -71.12, -48.96 | 73.72, -5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.844 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.73, 7.91 | APE9-dihe-in | -89.0, 155.98 | APE8-dihe-in | -50.13, 125.96 | APE8-rot-na | 330.56 | APE67-dihe-in | -75.78, -4.72 | -64.96, -12.29 | APE12-dist-na | 14.024 | APE11-dist-na | 9.7788 | APE10-dist-na | 10.0218 | APE9-dist-in | 7.0938 | C1048S | None | None | XRAY | 1.66 | 0.185 | 0.215 | A | 321.0 | 272.0 | 15 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6dud | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7Q6HAAA | P52333 | 814 | 1100 | 1124.0 | 934:1201 | Type1 | Inactive | DFGin | 6.4415 | 13.9124 | BLAminus | -128.11, -171.29 | 67.58, 71.88 | -97.45, 20.62 | 287.7, 81.42 | -64.43, -23.85 | in-in | in | 7.9084 | Saltbr-in | 2.684 | HRD-in | -72.1, -52.28 | 82.4, -12.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.789 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.93, 11.02 | APE9-dihe-in | -86.89, 152.23 | APE8-dihe-in | -44.63, 129.97 | APE8-rot-na | 328.93 | APE67-dihe-in | -80.65, 0.41 | -70.73, -15.65 | APE12-dist-na | 13.7773 | APE11-dist-na | 9.7373 | APE10-dist-na | 10.3425 | APE9-dist-in | 7.2322 | None | None | None | XRAY | 1.749 | 0.185 | 0.22 | AAA | 327.0 | 282.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7q6h | TYR_JAK3-2_HUMAN | TYR | 3.1e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3LXLA | P52333 | 814 | 1098 | 1124.0 | IZA:1 | Type1 | Inactive | DFGin | 6.3563 | 13.9832 | BLAminus | -131.21, -163.1 | 63.94, 61.73 | -90.52, 13.42 | 287.27, 88.72 | -63.24, -20.77 | in-in | in | 7.8734 | Saltbr-in | 2.759 | HRD-in | -76.94, -49.02 | 80.12, -11.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8049 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -131.67, 15.09 | APE9-dihe-in | -90.67, 156.23 | APE8-dihe-in | -48.41, 132.69 | APE8-rot-na | 328.44 | APE67-dihe-in | -80.87, -3.57 | -71.39, -11.92 | APE12-dist-na | 13.8943 | APE11-dist-na | 9.8069 | APE10-dist-na | 10.408 | APE9-dist-in | 7.3708 | C1048S | None | None | XRAY | 1.74 | 0.195 | 0.227 | A | 327.0 | 281.0 | 4 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3lxl | TYR_JAK3-2_HUMAN | TYR | 3.2e-81 | 278.4 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 1YVJA | P52333 | 814 | 1103 | 1124.0 | 4ST:2000 | Type1 | Inactive | DFGin | 6.5054 | 14.0048 | BLAminus | -117.35, -176.34 | 48.83, 98.04 | -113.48, 29.61 | 287.79, 84.73 | -71.88, -20.61 | in-in | in | 8.6181 | Saltbr-in | 2.8369 | HRD-in | -75.54, -39.16 | 74.88, -34.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8318 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -96.81, -5.63 | APE9-dihe-in | -95.15, 159.49 | APE8-dihe-in | -47.0, 152.52 | APE8-rot-na | 325.56 | APE67-dihe-in | -77.97, 4.18 | -53.16, -16.76 | APE12-dist-na | 9.8059 | APE11-dist-na | 6.854 | APE10-dist-na | 8.7777 | APE9-dist-out | 8.1995 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.55 | 0.204 | 0.254 | A | 290.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 1yvj | TYR_JAK3-2_HUMAN | TYR | 5.4e-81 | 277.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4Z16B | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | Inactive | DFGin | 6.6659 | 14.5322 | BLAminus | -124.7, -170.19 | 45.77, 83.37 | -100.74, 26.17 | 289.95, 82.89 | -68.35, -28.49 | in-in | in | 8.3877 | Saltbr-in | 2.8503 | HRD-in | -66.49, -45.94 | 73.56, -20.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8618 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -56.65, -6.62 | APE9-dihe-in | -78.46, 132.64 | APE8-dihe-in | -45.17, 131.02 | APE8-rot-na | 5.36 | APE67-dihe-in | -79.95, -14.25 | -79.37, 1.19 | APE12-dist-na | 12.5366 | APE11-dist-na | 9.232 | APE10-dist-na | 10.615 | APE9-dist-in | 7.017 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | B | 316.0 | 278.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4QPSC | P52333 | 814 | 1102 | 1124.0 | 37Q:1201 | Type1 | Inactive | DFGin | 6.7747 | 14.2003 | BLAminus | -137.32, -176.14 | 60.46, 91.64 | -108.44, 19.09 | 284.35, 76.96 | -56.92, -26.19 | in-in | in | 8.5021 | Saltbr-in | 2.8029 | HRD-in | -82.86, -44.58 | 73.92, -46.68 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8214 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 132.79 | APE8-dihe-in | -74.25, 110.88 | APE8-rot-na | 352.69 | APE67-dihe-in | -70.61, -6.19 | -68.78, -23.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.9914 | D949A,C1040S,C1048S | None | None | XRAY | 1.8 | 0.21 | 0.251 | C | 293.0 | 276.0 | 13 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4qps | TYR_JAK3-2_HUMAN | TYR | 3.9e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5LWMA | P52333 | 814 | 1103 | 1124.0 | 79T:1201 | Type1 | Inactive | DFGin | 6.1807 | 14.0847 | BLAminus | -127.82, -164.11 | 50.78, 78.32 | -96.87, 23.57 | 279.03, 70.69 | -64.42, -25.51 | in-in | in | 7.8434 | Saltbr-in | 2.7715 | HRD-in | -83.79, -41.29 | 73.45, -47.71 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8732 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -137.31, 98.87 | APE9-dihe-in | -108.79, 137.75 | APE8-dihe-in | -66.78, 85.64 | APE8-rot-na | 29.56 | APE67-dihe-in | -76.19, -3.82 | -62.47, -28.25 | APE12-dist-na | 10.173 | APE11-dist-na | 13.4615 | APE10-dist-na | 12.5843 | APE9-dist-out | 8.869 | None | None | None | XRAY | 1.55 | 0.166 | 0.204 | A | 294.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5lwm | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7APFA | P52333 | 814 | 1103 | 1124.0 | RQZ:1201 | Type1 | Inactive | DFGin | 6.1423 | 14.108 | BLAminus | -125.02, -164.76 | 52.74, 82.07 | -99.72, 24.14 | 279.87, 69.9 | -58.8, -33.19 | in-in | in | 8.0164 | Saltbr-in | 2.735 | HRD-in | -77.19, -45.73 | 75.08, -49.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8014 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -141.26, 128.28 | APE9-dihe-in | -143.67, 157.99 | APE8-dihe-in | -81.92, 93.49 | APE8-rot-na | 7.76 | APE67-dihe-in | -79.55, -5.28 | -69.3, -23.78 | APE12-dist-na | 10.1511 | APE11-dist-na | 13.6863 | APE10-dist-na | 13.2698 | APE9-dist-out | 9.0224 | None | None | None | XRAY | 1.95 | 0.206 | 0.255 | A | 294.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apf | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7APFB | P52333 | 814 | 1103 | 1124.0 | RQZ:1201 | Type1 | Inactive | DFGin | 6.2636 | 13.9552 | BLAminus | -125.48, -163.38 | 48.35, 84.73 | -99.0, 25.48 | 280.41, 70.13 | -63.69, -28.85 | in-in | in | 8.0989 | Saltbr-in | 2.7319 | HRD-in | -80.63, -44.7 | 74.93, -48.31 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7771 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -141.78, 126.08 | APE9-dihe-in | -146.46, 155.19 | APE8-dihe-in | -90.31, 98.72 | APE8-rot-na | 9.96 | APE67-dihe-in | -78.0, -2.22 | -75.31, -23.81 | APE12-dist-na | 9.6188 | APE11-dist-na | 13.0285 | APE10-dist-na | 12.5423 | APE9-dist-out | 9.1313 | None | None | None | XRAY | 1.95 | 0.206 | 0.255 | B | 294.0 | 285.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apf | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7APGA | P52333 | 813 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0309 | 13.9524 | BLAminus | -145.19, -172.66 | 53.39, 85.17 | -97.7, 25.99 | 284.4, 73.93 | -62.87, -25.47 | in-in | in | 8.4915 | Saltbr-in | 3.0886 | HRD-in | -83.97, -50.23 | 79.99, -46.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9125 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -120.14, 50.45 | APE9-dihe-in | -76.86, 156.83 | APE8-dihe-in | -73.67, 136.77 | APE8-rot-na | 351.29 | APE67-dihe-in | -81.27, -2.59 | -94.73, -13.37 | APE12-dist-na | 10.6785 | APE11-dist-na | 10.8995 | APE10-dist-na | 13.6012 | APE9-dist-out | 8.9847 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | A | 294.0 | 279.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7APGB | P52333 | 814 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0387 | 14.0695 | BLAminus | -144.05, -171.58 | 55.33, 84.79 | -97.11, 25.47 | 284.03, 75.74 | -64.12, -25.92 | in-in | in | 8.44 | Saltbr-in | 3.0791 | HRD-in | -83.8, -49.69 | 80.24, -45.58 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9057 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -121.16, 48.46 | APE9-dihe-in | -74.89, 156.25 | APE8-dihe-in | -72.87, 137.28 | APE8-rot-na | 354.01 | APE67-dihe-in | -82.99, -1.84 | -93.81, -9.25 | APE12-dist-na | 10.8058 | APE11-dist-na | 10.8121 | APE10-dist-na | 13.4192 | APE9-dist-out | 8.9175 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | B | 294.0 | 278.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7APGC | P52333 | 812 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0574 | 14.0501 | BLAminus | -143.35, -172.89 | 56.23, 84.96 | -97.07, 24.64 | 284.44, 74.77 | -64.51, -25.55 | in-in | in | 8.468 | Saltbr-in | 3.0668 | HRD-in | -82.68, -50.65 | 80.68, -46.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9124 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -120.01, 55.65 | APE9-dihe-in | -74.89, 157.1 | APE8-dihe-in | -74.45, 136.81 | APE8-rot-na | 351.06 | APE67-dihe-in | -81.76, -1.91 | -93.74, -14.98 | APE12-dist-na | 10.5477 | APE11-dist-na | 11.1621 | APE10-dist-na | 13.9629 | APE9-dist-out | 8.9485 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | C | 294.0 | 287.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7APGD | P52333 | 815 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0092 | 14.041 | BLAminus | -143.73, -171.03 | 51.78, 85.49 | -96.62, 26.59 | 283.85, 72.76 | -64.13, -26.23 | in-in | in | 8.434 | Saltbr-in | 3.0873 | HRD-in | -83.66, -49.57 | 81.52, -47.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9154 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -120.66, 45.43 | APE9-dihe-in | -76.74, 156.2 | APE8-dihe-in | -73.01, 137.72 | APE8-rot-na | 354.08 | APE67-dihe-in | -79.85, -1.41 | -95.44, -12.08 | APE12-dist-na | 10.8366 | APE11-dist-na | 10.5366 | APE10-dist-na | 13.2359 | APE9-dist-out | 8.9582 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | D | 294.0 | 277.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5LWNA | P52333 | 814 | 1103 | 1124.0 | 79R:1208,79S:1209 | Type1,Type1 | Inactive | DFGin | 6.1459 | 14.132 | BLAminus | -129.49, -162.36 | 48.02, 73.73 | -88.01, 20.06 | 281.83, 72.86 | -61.77, -25.11 | in-in | in | 7.8172 | Saltbr-in | 2.7083 | HRD-in | -84.52, -44.16 | 75.64, -46.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8251 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -141.38, 98.08 | APE9-dihe-in | -113.86, 140.78 | APE8-dihe-in | -73.27, 87.08 | APE8-rot-na | 29.33 | APE67-dihe-in | -77.95, -2.97 | -61.74, -27.63 | APE12-dist-na | 10.0824 | APE11-dist-na | 13.4052 | APE10-dist-na | 12.4459 | APE9-dist-out | 8.904 | None | None | None | XRAY | 1.6 | 0.169 | 0.209 | A | 294.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5lwn | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6HZVA | P52333 | 815 | 1098 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.4293 | 14.257 | BLAminus | -133.87, 178.6 | 61.51, 90.4 | -109.85, 28.17 | 289.99, 77.52 | -67.6, -31.52 | in-in | in | 8.3241 | Saltbr-in | 2.9312 | HRD-in | -62.66, -43.13 | 71.32, -8.68 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7324 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 119.68 | APE8-rot-na | 14.07 | APE67-dihe-in | -79.55, -1.3 | -80.03, -13.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | A | 285.0 | 266.0 | 18 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6HZVB | P52333 | 815 | 1099 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.1943 | 14.2143 | BLAminus | -135.38, 176.48 | 64.47, 86.88 | -105.43, 20.89 | 286.69, 85.17 | -66.35, -29.51 | in-in | in | 8.1494 | Saltbr-in | 2.8265 | HRD-in | -61.18, -44.44 | 71.7, 4.93 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.6907 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 129.11 | APE8-rot-na | 330.57 | APE67-dihe-in | -79.98, -2.63 | -77.74, -18.2 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | B | 285.0 | 269.0 | 16 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6HZVC | P52333 | 815 | 1098 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.477 | 14.2719 | BLAminus | -130.86, 179.06 | 58.44, 90.28 | -109.09, 23.07 | 290.05, 84.12 | -62.59, -33.96 | in-in | in | 8.0905 | Saltbr-in | 2.8088 | HRD-in | -69.82, -48.24 | 78.15, -8.29 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.6892 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -41.25 | APE8-dihe-in | -66.72, 131.5 | APE8-rot-na | 341.69 | APE67-dihe-in | -75.5, -7.29 | -73.63, -18.87 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.346 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | C | 285.0 | 265.0 | 19 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6HZVD | P52333 | 815 | 1098 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.418 | 14.1518 | BLAminus | -133.07, -178.12 | 58.66, 85.08 | -104.02, 25.84 | 292.67, 81.24 | -61.98, -32.78 | in-in | in | 8.1402 | Saltbr-in | 2.7701 | HRD-in | -71.74, -43.92 | 75.22, -14.51 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7079 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -35.5 | APE8-dihe-in | -66.27, 131.93 | APE8-rot-na | 340.52 | APE67-dihe-in | -79.97, 1.1 | -77.2, -17.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.6337 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | D | 285.0 | 259.0 | 25 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5W86B | P52333 | 816 | 1098 | 1124.0 | 9YV:4000 | Type1 | None | DFGin | 6.5719 | 14.1258 | BLAminus | -130.89, -177.7 | 55.33, 86.59 | -98.74, 23.53 | 285.65, 80.73 | -58.36, -36.34 | in-in | in | 8.1755 | Saltbr-in | 2.7815 | HRD-in | -61.09, -43.56 | 75.39, -22.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8266 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-in | -98.06, 144.28 | APE8-rot-na | 28.22 | APE67-dihe-in | -84.46, -5.87 | -122.29, -17.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.7561 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | B | 287.0 | 269.0 | 14 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5W86C | P52333 | 814 | 1099 | 1124.0 | 9YV:4000 | Type1 | None | DFGin | 6.5069 | 14.1113 | BLAminus | -131.5, -178.51 | 55.57, 86.1 | -97.59, 23.31 | 285.7, 80.13 | -57.67, -36.43 | in-in | in | 8.1655 | Saltbr-in | 2.9403 | HRD-in | -62.63, -48.44 | 77.31, -20.33 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8223 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -67.29 | APE8-rot-na | 15.79 | APE67-dihe-in | -70.13, -18.29 | -58.03, -20.5 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | C | 287.0 | 275.0 | 11 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6AAKD | P52333 | 814 | 1098 | 1124.0 | 9T6:1201 | Type1 | None | DFGin | 6.3309 | 14.1383 | BLAminus | -145.03, 168.99 | 56.55, 97.11 | -103.75, 32.24 | 293.47, 81.71 | -62.01, -33.71 | in-in | in | 8.0179 | Saltbr-in | 2.8556 | HRD-in | -76.49, -42.81 | 76.74, -36.27 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7662 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 72.65 | APE8-dihe-in | -50.29, 134.06 | APE8-rot-na | 332.19 | APE67-dihe-in | -63.85, -16.03 | -70.13, -20.9 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.3842 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | D | 287.0 | 268.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6aak | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZC6B | P52333 | 813 | 1100 | 1124.0 | VFC:2103 | Type1 | None | DFGin | 6.2181 | 14.0462 | BLAminus | -128.88, -176.96 | 59.69, 81.97 | -99.61, 22.0 | 289.18, 82.46 | -63.53, -20.72 | in-in | in | 8.2087 | Saltbr-in | 2.7991 | HRD-in | -71.31, -49.71 | 79.31, 3.34 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7475 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 25.15 | APE9-dihe-in | -99.95, 171.81 | APE8-dihe-in | -50.02, 112.29 | APE8-rot-na | 325.04 | APE67-dihe-in | -73.29, -4.3 | -58.87, -25.22 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.4818 | APE9-dist-in | 6.8402 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | B | 288.0 | 278.0 | 10 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZC6D | P52333 | 814 | 1100 | 1124.0 | VFC:2103 | Type1 | None | DFGin | 6.3147 | 14.132 | BLAminus | -134.59, -176.68 | 59.2, 81.95 | -97.58, 24.75 | 285.45, 76.49 | -66.73, -25.04 | in-in | in | 8.057 | Saltbr-in | 2.7416 | HRD-in | -74.86, -52.02 | 77.99, -12.75 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7303 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 79.2 | APE8-rot-na | 32.25 | APE67-dihe-in | -80.63, -5.09 | -78.85, -21.32 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | D | 288.0 | 269.0 | 18 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZEPB | P52333 | 814 | 1100 | 1124.0 | 1NX:2101 | Type1 | None | DFGin | 6.3528 | 14.2219 | BLAminus | -142.2, 177.46 | 62.39, 84.45 | -101.38, 32.38 | 292.96, 77.07 | -73.1, -37.75 | in-in | in | 8.2407 | Saltbr-in | 2.735 | HRD-in | -71.3, -45.86 | 73.98, -5.89 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7688 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 174.81 | APE8-dihe-in | -59.17, 141.04 | APE8-rot-na | 332.8 | APE67-dihe-in | -80.76, -5.98 | -67.68, -15.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.4769 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | B | 288.0 | 270.0 | 17 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zep | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZEPC | P52333 | 814 | 1100 | 1124.0 | 1NX:2101 | Type1 | None | DFGin | 6.2667 | 14.2845 | BLAminus | -143.3, 179.56 | 63.59, 86.35 | -106.32, 31.56 | 290.45, 75.82 | -68.82, -32.0 | in-in | in | 8.1744 | Saltbr-in | 2.7545 | HRD-in | -76.43, -48.0 | 76.34, -21.16 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7144 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 45.01 | APE9-dihe-in | -93.38, 161.79 | APE8-dihe-in | -56.5, 116.98 | APE8-rot-na | 326.42 | APE67-dihe-in | -74.98, -4.7 | -72.25, -13.12 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.7287 | APE9-dist-in | 6.8497 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | C | 288.0 | 278.0 | 9 | 31 | 29 | 2 | [[521, 779], [822, 1097]] | 2.0 | 3zep | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 3ZEPD | P52333 | 814 | 1099 | 1124.0 | 1NX:2100 | Type1 | None | DFGin | 6.5755 | 14.572 | BLAminus | -134.12, 176.57 | 59.25, 80.73 | -100.38, 28.57 | 291.24, 76.13 | -63.83, -42.01 | in-in | in | 8.3615 | Saltbr-in | 2.6719 | HRD-in | -72.39, -47.07 | 79.2, -13.88 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7779 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 161.47 | APE8-dihe-in | -52.69, 138.76 | APE8-rot-na | 329.47 | APE67-dihe-in | -77.9, -7.22 | -77.25, -13.54 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.5559 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | D | 288.0 | 274.0 | 12 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 3zep | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 7UYVD | P52333 | 814 | 1100 | 1124.0 | OV5:1201 | Type1 | None | DFGin | 6.4207 | 14.2582 | BLAminus | -133.29, -179.06 | 58.4, 83.86 | -99.71, 22.65 | 285.23, 81.71 | -62.49, -28.09 | in-in | in | 8.2976 | Saltbr-in | 2.6722 | HRD-in | -64.99, -48.29 | 76.96, -0.25 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7457 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 163.98 | APE8-dihe-in | -58.27, 129.89 | APE8-rot-na | 335.93 | APE67-dihe-in | -80.69, -3.3 | -71.81, -12.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4681 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | D | 291.0 | 272.0 | 15 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 5VO6A | P52333 | 815 | 1099 | 1124.0 | 9J4:4000 | Type1 | None | DFGin | 6.5587 | 13.7482 | BLAminus | -128.78, -173.97 | 61.05, 89.09 | -107.4, 19.66 | 285.17, 86.8 | -68.24, -28.8 | in-in | in | 7.5123 | Saltbr-in | 2.9107 | HRD-in | -75.3, -50.06 | 76.72, -16.95 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9825 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 135.66 | APE8-rot-na | 332.57 | APE67-dihe-in | -81.44, -5.82 | -70.82, -9.6 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1040S,C1048S | None | None | XRAY | 2.65 | 0.215 | 0.284 | A | 293.0 | 271.0 | 14 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 5vo6 | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6NY4A | P52333 | 815 | 1099 | 1124.0 | Z3A:4000 | Type1 | None | DFGin | 6.4319 | 13.7522 | BLAminus | -130.0, -166.41 | 50.15, 85.44 | -100.28, 21.12 | 284.91, 84.56 | -64.41, -23.36 | in-in | in | 7.6903 | Saltbr-in | 2.7769 | HRD-in | -74.4, -47.07 | 70.71, -6.14 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8428 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -0.08 | APE9-dihe-in | -95.23, 160.07 | APE8-dihe-in | -49.81, 129.43 | APE8-rot-na | 333.86 | APE67-dihe-in | -73.45, 2.08 | -64.08, -16.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 9.7064 | APE9-dist-in | 7.0951 | C811S,C1040S,C1048S | None | None | XRAY | 2.33 | 0.216 | 0.241 | A | 293.0 | 277.0 | 8 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 6ny4 | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4V0GB | P52333 | 816 | 1098 | 1124.0 | G9B:2099 | Type1 | None | DFGin | 6.202 | 14.6329 | BLAminus | -137.8, -174.69 | 52.03, 76.68 | -96.09, 37.57 | 296.46, 78.81 | -70.34, -40.16 | in-in | in | 8.7004 | Saltbr-in | 2.629 | HRD-in | -75.76, -37.0 | 67.95, -17.09 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8243 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -54.69 | APE8-rot-na | 331.57 | APE67-dihe-in | -77.98, -0.68 | -62.56, -42.14 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 3.0 | 0.254 | 0.295 | B | 283.0 | 274.0 | 9 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4v0g | TYR_JAK3-2_HUMAN | TYR | 2.3e-81 | 278.9 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4V0GA | P52333 | 817 | 1098 | 1124.0 | G9B:2099 | Type1 | None | DFGin | 6.198 | 14.7166 | BLAminus | -144.75, -176.45 | 39.25, 85.88 | -90.52, 22.25 | 286.27, 74.42 | -61.38, -18.98 | in-in | in | 8.3521 | Saltbr-in | 2.7066 | HRD-in | -65.46, -44.14 | 69.1, 4.41 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8503 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -33.75 | APE8-rot-na | 330.77 | APE67-dihe-in | -73.45, -1.83 | -68.02, -39.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 3.0 | 0.254 | 0.295 | A | 283.0 | 269.0 | 13 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 4v0g | TYR_JAK3-2_HUMAN | TYR | 2.3e-81 | 278.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4Z16A | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | None | DFGin | 6.693 | 14.5354 | BLAminus | -125.11, -170.67 | 46.31, 83.09 | -100.98, 26.25 | 290.17, 83.28 | -67.99, -29.42 | in-in | in | 8.3468 | Saltbr-in | 2.8339 | HRD-in | -67.29, -45.59 | 73.41, -19.17 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8291 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 77.57 | APE8-rot-na | 328.09 | APE67-dihe-in | -74.64, -13.67 | -80.93, -12.04 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | A | 316.0 | 273.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4Z16C | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | None | DFGin | 6.724 | 14.5409 | BLAminus | -124.89, -171.04 | 46.95, 83.36 | -101.0, 25.74 | 290.21, 83.17 | -68.15, -28.94 | in-in | in | 8.3723 | Saltbr-in | 2.8403 | HRD-in | -67.03, -45.78 | 73.53, -19.66 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7882 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 38.92 | APE8-rot-na | 335.43 | APE67-dihe-in | -76.63, -13.6 | -68.45, -18.81 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | C | 316.0 | 273.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4Z16D | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | None | DFGin | 6.6883 | 14.5667 | BLAminus | -124.04, -170.5 | 45.94, 82.68 | -99.35, 24.89 | 290.17, 82.54 | -66.47, -27.42 | in-in | in | 8.3931 | Saltbr-in | 2.8748 | HRD-in | -67.23, -45.45 | 73.09, -20.62 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7942 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 52.48 | APE8-rot-na | 345.61 | APE67-dihe-in | -77.91, -13.97 | -72.79, -6.5 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | D | 316.0 | 273.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 4QPSA | P52333 | 814 | 1100 | 1124.0 | 37Q:1201 | Type1 | None | DFGin | 6.8957 | 14.0909 | BLAminus | -130.94, -174.49 | 64.52, 86.82 | -104.86, 15.71 | 281.27, 81.21 | -57.28, -32.23 | in-in | in | 8.5879 | Saltbr-in | 2.8637 | HRD-in | -78.56, -46.33 | 74.55, -53.21 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.801 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 149.07 | APE8-rot-na | 18.94 | APE67-dihe-in | -69.31, -9.6 | -100.11, -5.26 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | D949A,C1040S,C1048S | None | None | XRAY | 1.8 | 0.21 | 0.251 | A | 293.0 | 270.0 | 17 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 4qps | TYR_JAK3-2_HUMAN | TYR | 3.9e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6GLAA | P52333 | 813 | 1103 | 1124.0 | F4B:1201 | Type1 | None | DFGin | 6.1255 | 14.0661 | BLAminus | -126.69, -163.69 | 45.61, 84.37 | -97.16, 18.74 | 276.14, 73.33 | -60.39, -30.05 | in-in | in | 7.8334 | Saltbr-in | 2.6744 | HRD-in | -80.36, -50.35 | 74.06, -4.7 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7495 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 115.39 | APE9-dihe-in | -100.65, 143.31 | APE8-dihe-in | -75.22, 92.35 | APE8-rot-na | 30.49 | APE67-dihe-in | -81.25, -0.82 | -60.88, -31.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.6793 | APE9-dist-in | 7.0014 | None | None | None | XRAY | 1.92 | 0.228 | 0.273 | A | 294.0 | 288.0 | 3 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6gla | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6GLAB | P52333 | 813 | 1103 | 1124.0 | F4B:1201 | Type1 | None | DFGin | 6.1346 | 14.0372 | BLAminus | -126.98, -166.17 | 47.87, 84.06 | -100.26, 19.16 | 275.64, 73.52 | -60.46, -30.51 | in-in | in | 7.8307 | Saltbr-in | 2.6702 | HRD-in | -83.39, -49.56 | 74.28, -3.93 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7748 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 114.52 | APE9-dihe-in | -101.31, 145.02 | APE8-dihe-in | -77.95, 91.55 | APE8-rot-na | 29.11 | APE67-dihe-in | -79.72, -1.04 | -62.76, -29.93 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.7449 | APE9-dist-in | 6.9663 | None | None | None | XRAY | 1.92 | 0.228 | 0.273 | B | 294.0 | 286.0 | 5 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6gla | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6GLBA | P52333 | 813 | 1103 | 1124.0 | F48:1201 | Type1 | None | DFGin | 6.0868 | 14.0047 | BLAminus | -127.29, -165.11 | 42.2, 80.94 | -98.99, 18.18 | 281.6, 72.22 | -46.91, -40.63 | in-in | in | 7.5761 | Saltbr-in | 2.7125 | HRD-in | -78.7, -52.76 | 77.75, 9.6 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7344 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 129.22 | APE9-dihe-in | -106.96, 151.72 | APE8-dihe-in | -79.63, 91.52 | APE8-rot-na | 32.17 | APE67-dihe-in | -74.91, -5.23 | -62.01, -34.09 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.734 | APE9-dist-in | 6.7274 | None | None | None | XRAY | 2.0 | 0.236 | 0.29 | A | 294.0 | 288.0 | 3 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6glb | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 6GLBB | P52333 | 813 | 1103 | 1124.0 | F48:1201 | Type1 | None | DFGin | 6.117 | 14.0249 | BLAminus | -125.81, -165.95 | 42.86, 80.87 | -97.87, 18.6 | 282.22, 74.99 | -51.1, -37.8 | in-in | in | 7.5451 | Saltbr-in | 2.7085 | HRD-in | -76.97, -51.62 | 77.21, 8.56 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7568 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 130.97 | APE9-dihe-in | -105.16, 150.45 | APE8-dihe-in | -79.13, 89.35 | APE8-rot-na | 33.14 | APE67-dihe-in | -76.14, -3.82 | -57.76, -35.85 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.6293 | APE9-dist-in | 6.7039 | None | None | None | XRAY | 2.0 | 0.236 | 0.29 | B | 294.0 | 288.0 | 3 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6glb | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 9R5ZA | P52333 | 822 | 1101 | 1124.0 | A1JJU:60301 | Type1 | None | DFGin | 6.1324 | 14.0012 | BLAminus | -127.52, -161.85 | 48.17, 81.61 | -92.0, 24.85 | 277.91, 73.75 | -73.44, -23.7 | in-in | in | 7.6679 | Saltbr-in | 2.7676 | HRD-in | -79.16, -47.46 | 79.61, -35.13 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8804 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 92.63 | APE8-rot-na | 20.77 | APE67-dihe-in | -76.47, -3.83 | -62.4, -34.74 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.8 | 0.239 | 0.289 | A | 294.0 | 258.0 | 22 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 9r5z | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | 9R5ZB | P52333 | 816 | 1101 | 1124.0 | A1JJU:60301 | Type1 | None | DFGin | 6.2264 | 14.1304 | BLAminus | -127.35, -164.41 | 49.32, 77.12 | -91.09, 23.07 | 281.2, 72.28 | -62.52, -23.26 | in-in | in | 7.8816 | Saltbr-in | 2.8186 | HRD-in | -86.18, -46.89 | 79.27, -42.6 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8747 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 79.25 | APE8-rot-na | 31.77 | APE67-dihe-in | -82.31, -0.99 | -65.94, -24.16 | APE12-dist-na | 11.0451 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.8 | 0.239 | 0.289 | B | 294.0 | 275.0 | 11 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 9r5z | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| JAK3-2 | JAK3_HUMAN | AF-P52333-K2A | P52333 | 814 | 1105 | 1124.0 | No_ligand | No_ligand | Active | DFGin | 6.1026 | 13.7936 | BLAminus | -134.56, -179.19 | 51.31, 75.31 | -82.94, 20.6 | 292.85, 86.33 | -61.55, -30.97 | in-in | in | 8.2483 | Saltbr-in | 2.6953 | HRD-in | -70.59, -43.72 | 65.57, -21.68 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8552 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -56.42, 123.08 | APE9-dihe-in | -125.57, 135.88 | APE8-dihe-in | -78.86, 68.83 | APE8-rot-na | 34.92 | APE67-dihe-in | -75.13, -6.36 | -53.49, -31.1 | APE12-dist-na | 10.5223 | APE11-dist-na | 9.5286 | APE10-dist-na | 10.1849 | APE9-dist-in | 7.1879 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 292.0 | 292.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | AF-P52333-K2 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4.6e-81 | 277.9 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | AF-P52333-K4A | P52333 | 814 | 1105 | 1124.0 | No_ligand | No_ligand | Active | DFGin | 6.1108 | 13.7687 | BLAminus | -141.5, -174.59 | 54.28, 75.11 | -88.15, 17.45 | 293.92, 89.95 | -59.55, -34.59 | in-in | in | 8.1169 | Saltbr-in | 2.6779 | HRD-in | -78.79, -45.55 | 61.88, 0.83 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8819 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -61.64, 120.49 | APE9-dihe-in | -128.67, 141.65 | APE8-dihe-in | -77.57, 68.42 | APE8-rot-na | 36.41 | APE67-dihe-in | -72.34, -8.01 | -50.71, -34.24 | APE12-dist-na | 13.4854 | APE11-dist-na | 9.5574 | APE10-dist-na | 10.1649 | APE9-dist-in | 6.4962 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 292.0 | 292.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | AF-P52333-K4 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4.6e-81 | 277.9 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6AAKC | P52333 | 814 | 1099 | 1124.0 | 9T6:1201 | Type1 | Active | DFGin | 6.7877 | 14.6346 | BLAminus | -114.47, 172.4 | 69.03, 86.81 | -107.19, 29.58 | 286.76, 78.99 | -58.47, -55.72 | in-in | in | 8.2406 | Saltbr-in | 2.7237 | HRD-in | -89.94, -41.82 | 71.73, -3.81 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7832 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -68.85, 76.94 | APE9-dihe-in | -171.36, 163.86 | APE8-dihe-in | -58.47, 128.31 | APE8-rot-na | 338.62 | APE67-dihe-in | -73.56, -5.95 | -79.88, -15.99 | APE12-dist-na | 12.9746 | APE11-dist-na | 9.2183 | APE10-dist-na | 10.3986 | APE9-dist-in | 7.7513 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | C | 287.0 | 276.0 | 10 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6aak | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7UYVA | P52333 | 814 | 1100 | 1124.0 | OV5:1201 | Type1 | Active | DFGin | 6.3763 | 14.2869 | BLAminus | -136.33, -178.14 | 60.47, 77.06 | -94.46, 22.49 | 283.21, 76.25 | -61.39, -33.76 | in-in | in | 8.2009 | Saltbr-in | 2.6421 | HRD-in | -69.18, -41.57 | 72.69, -12.85 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7503 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.18, 82.75 | APE9-dihe-in | -112.58, 159.26 | APE8-dihe-in | -47.72, 129.83 | APE8-rot-na | 329.64 | APE67-dihe-in | -81.57, 1.11 | -69.92, -19.01 | APE12-dist-na | 11.5311 | APE11-dist-na | 8.0482 | APE10-dist-na | 11.6832 | APE9-dist-in | 7.3388 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | A | 291.0 | 278.0 | 9 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7UYVB | P52333 | 814 | 1100 | 1124.0 | OV5:1201 | Type1 | Active | DFGin | 6.2251 | 14.2162 | BLAminus | -136.69, -173.44 | 56.56, 80.52 | -96.27, 21.5 | 284.08, 77.64 | -57.68, -39.3 | in-in | in | 8.1504 | Saltbr-in | 2.6309 | HRD-in | -80.27, -44.25 | 68.81, -0.6 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7556 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -75.34, 85.59 | APE9-dihe-in | -127.16, 148.54 | APE8-dihe-in | -37.53, 121.21 | APE8-rot-na | 325.53 | APE67-dihe-in | -80.04, -3.68 | -72.05, -16.34 | APE12-dist-na | 11.5779 | APE11-dist-na | 9.1429 | APE10-dist-na | 12.2547 | APE9-dist-in | 7.3873 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | B | 291.0 | 284.0 | 3 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3PJCA | P52333 | 815 | 1104 | 1124.0 | PJC:800 | Type1 | Active | DFGin | 6.6986 | 14.412 | BLAminus | -131.65, -174.74 | 53.97, 85.79 | -100.88, 20.12 | 280.65, 74.1 | -60.63, -24.35 | in-in | in | 8.6962 | Saltbr-in | 2.6139 | HRD-in | -69.63, -48.63 | 77.02, -5.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8226 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.16, 145.45 | APE9-dihe-in | -115.3, 150.0 | APE8-dihe-in | -81.75, 75.29 | APE8-rot-na | 32.65 | APE67-dihe-in | -79.59, -4.38 | -53.88, -28.84 | APE12-dist-na | 13.2005 | APE11-dist-na | 11.5918 | APE10-dist-na | 12.7974 | APE9-dist-in | 7.9845 | None | None | None | XRAY | 2.2 | 0.182 | 0.215 | A | 315.0 | 286.0 | 4 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3pjc | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 6.1e-81 | 277.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6GL9A | P52333 | 812 | 1103 | 1124.0 | F3W:1201 | Type1 | Active | DFGin | 6.2475 | 14.0115 | BLAminus | -125.6, -168.17 | 49.24, 81.71 | -98.97, 21.2 | 279.85, 75.03 | -60.06, -26.17 | in-in | in | 7.7934 | Saltbr-in | 2.6834 | HRD-in | -78.49, -49.26 | 75.45, 0.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7882 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.67, 117.53 | APE9-dihe-in | -98.8, 151.13 | APE8-dihe-in | -79.69, 90.74 | APE8-rot-na | 31.23 | APE67-dihe-in | -78.37, -0.16 | -59.8, -32.45 | APE12-dist-na | 9.3301 | APE11-dist-na | 10.7633 | APE10-dist-na | 11.753 | APE9-dist-in | 6.9787 | None | None | None | XRAY | 1.7 | 0.209 | 0.244 | A | 294.0 | 292.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6gl9 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6GL9B | P52333 | 813 | 1103 | 1124.0 | F3W:1201 | Type1 | Active | DFGin | 6.21 | 14.019 | BLAminus | -123.31, -164.34 | 42.61, 83.03 | -97.02, 22.96 | 280.36, 70.4 | -63.87, -26.0 | in-in | in | 7.7595 | Saltbr-in | 2.667 | HRD-in | -78.77, -47.46 | 73.56, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7746 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -76.72, 116.63 | APE9-dihe-in | -97.44, 150.89 | APE8-dihe-in | -77.79, 91.0 | APE8-rot-na | 32.15 | APE67-dihe-in | -73.22, -2.71 | -60.01, -35.33 | APE12-dist-na | 9.3264 | APE11-dist-na | 10.7827 | APE10-dist-na | 11.7277 | APE9-dist-in | 6.9767 | None | None | None | XRAY | 1.7 | 0.209 | 0.244 | B | 294.0 | 291.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6gl9 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7C3NA | P52333 | 814 | 1102 | 1124.0 | FHX:9000 | Type1 | Inactive | DFGin | 6.068 | 13.3862 | ABAminus | -140.24, 14.21 | -145.02, 134.62 | -131.29, 32.79 | 294.67, 80.18 | -64.88, -27.68 | in-in | in | 8.233 | Saltbr-in | 2.7822 | HRD-in | -78.6, -47.11 | 71.84, 1.59 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8064 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.04, 126.4 | APE9-dihe-in | -81.7, 145.46 | APE8-dihe-in | -77.41, 71.31 | APE8-rot-na | 31.38 | APE67-dihe-in | -79.88, -2.49 | -60.07, -26.59 | APE12-dist-na | 11.7358 | APE11-dist-na | 10.4538 | APE10-dist-na | 12.3096 | APE9-dist-in | 7.2655 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 1.98 | 0.17 | 0.194 | A | 315.0 | 289.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7c3n | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 6.1e-81 | 277.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3LXKA | P52333 | 815 | 1098 | 1124.0 | MI1:1125 | Type1 | Inactive | DFGin | 6.0647 | 13.0171 | ABAminus | -128.16, 7.24 | -148.97, 145.15 | -138.77, 31.19 | 300.52, 88.17 | -60.03, -27.75 | in-in | in | 8.251 | Saltbr-in | 2.7565 | HRD-in | -78.64, -46.72 | 70.97, -5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8402 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -118.3, 17.09 | APE9-dihe-in | -92.59, 156.17 | APE8-dihe-in | -54.3, 131.46 | APE8-rot-na | 335.17 | APE67-dihe-in | -82.42, -7.27 | -71.07, -8.83 | APE12-dist-na | 14.2685 | APE11-dist-na | 9.9216 | APE10-dist-na | 10.5049 | APE9-dist-in | 7.209 | C1048S | None | None | XRAY | 2.0 | 0.205 | 0.265 | A | 327.0 | 279.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3lxk | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3.2e-81 | 278.4 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5W86A | P52333 | 814 | 1098 | 1124.0 | 9YV:4000 | Type1 | Inactive | DFGin | 6.508 | 14.2333 | BLAminus | -130.78, -178.04 | 55.33, 86.29 | -99.45, 24.99 | 285.64, 80.91 | -59.45, -36.09 | in-in | in | 8.3613 | Saltbr-in | 2.7197 | HRD-in | -61.74, -49.91 | 79.02, -19.05 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8338 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -62.63 | APE8-dihe-in | -73.09, 69.06 | APE8-rot-na | 28.5 | APE67-dihe-in | -76.22, -6.14 | -68.16, -24.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.3257 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | A | 287.0 | 271.0 | 14 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5W86D | P52333 | 814 | 1099 | 1124.0 | 9YV:4000 | Type1 | Inactive | DFGin | 6.5614 | 14.2551 | BLAminus | -130.88, -178.77 | 56.18, 85.97 | -99.02, 25.19 | 285.73, 80.24 | -59.91, -34.36 | in-in | in | 8.1827 | Saltbr-in | 2.7569 | HRD-in | -62.59, -49.55 | 78.85, -19.41 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.814 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -64.08 | APE8-dihe-in | -73.59, 57.74 | APE8-rot-na | 27.09 | APE67-dihe-in | -73.08, -10.82 | -59.31, -28.98 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.2414 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | D | 287.0 | 274.0 | 12 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6AAKA | P52333 | 815 | 1098 | 1124.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.4258 | 14.4877 | BLAminus | -141.28, -175.48 | 60.31, 80.99 | -97.75, 30.98 | 284.74, 77.33 | -61.02, -46.05 | in-in | in | 8.5254 | Saltbr-in | 2.67 | HRD-in | -75.62, -45.99 | 77.6, -18.1 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7362 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -74.2, -11.07 | APE9-dihe-in | -68.95, 155.07 | APE8-dihe-in | -47.57, 131.1 | APE8-rot-na | 329.72 | APE67-dihe-in | -73.4, -26.9 | -66.76, -22.48 | APE12-dist-na | 11.9929 | APE11-dist-na | 8.6734 | APE10-dist-na | 11.3981 | APE9-dist-in | 7.4704 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | A | 287.0 | 277.0 | 7 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6aak | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6AAKB | P52333 | 815 | 1100 | 1124.0 | 9T6:1201 | Type1 | Inactive | DFGin | 6.549 | 14.3135 | BLAminus | -132.57, -171.05 | 56.03, 83.09 | -98.42, 24.6 | 281.38, 75.24 | -63.47, -40.11 | in-in | in | 8.0358 | Saltbr-in | 2.7546 | HRD-in | -65.5, -48.18 | 78.33, -13.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9074 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.61, -28.55 | APE9-dihe-in | -64.46, 151.35 | APE8-dihe-in | -40.19, 130.42 | APE8-rot-na | 326.93 | APE67-dihe-in | -77.17, -14.56 | -72.74, -10.57 | APE12-dist-na | 13.1081 | APE11-dist-na | 9.526 | APE10-dist-na | 10.0845 | APE9-dist-in | 7.2029 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | B | 287.0 | 285.0 | 1 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6aak | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZC6A | P52333 | 814 | 1100 | 1124.0 | VFC:2103 | Type1 | Inactive | DFGin | 6.3992 | 14.249 | BLAminus | -132.73, -176.21 | 56.45, 83.25 | -97.56, 22.77 | 285.82, 73.7 | -62.6, -27.55 | in-in | in | 8.2919 | Saltbr-in | 2.8022 | HRD-in | -72.44, -47.03 | 73.15, -6.89 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7419 | ActLoopCT-out | TYR | APEdihe_noiai | APEdist_aaai | APE10-dihe-none | 999.0, 118.21 | APE9-dihe-out | -83.58, -179.01 | APE8-dihe-in | -60.9, 137.23 | APE8-rot-na | 332.96 | APE67-dihe-in | -76.45, -9.26 | -65.3, -16.84 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 9.5354 | APE9-dist-in | 5.9074 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | A | 288.0 | 279.0 | 8 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZC6C | P52333 | 814 | 1100 | 1124.0 | VFC:2103 | Type1 | Inactive | DFGin | 6.2807 | 14.0027 | BLAminus | -123.64, -177.74 | 61.16, 80.91 | -97.9, 27.04 | 288.23, 77.53 | -66.72, -26.1 | in-in | in | 8.1905 | Saltbr-in | 2.6842 | HRD-in | -72.21, -46.31 | 77.05, -24.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7606 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -54.85 | APE8-dihe-in | -77.18, 80.1 | APE8-rot-na | 33.09 | APE67-dihe-in | -76.9, -10.93 | -67.13, -29.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.1774 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | C | 288.0 | 277.0 | 10 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZEPA | P52333 | 814 | 1098 | 1124.0 | 1NX:2099 | Type1 | Inactive | DFGin | 6.4201 | 14.3445 | BLAminus | -139.2, 179.6 | 58.57, 83.63 | -103.43, 28.82 | 290.46, 79.48 | -67.26, -39.4 | in-in | in | 8.1983 | Saltbr-in | 2.7236 | HRD-in | -72.97, -44.84 | 72.81, -0.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7642 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -90.83, 0.53 | APE9-dihe-in | -141.71, 168.37 | APE8-dihe-in | -61.5, 133.7 | APE8-rot-na | 333.46 | APE67-dihe-in | -72.33, -1.68 | -64.6, -21.71 | APE12-dist-na | 13.4306 | APE11-dist-na | 10.6555 | APE10-dist-na | 6.8245 | APE9-dist-in | 6.4001 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | A | 288.0 | 276.0 | 9 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3zep | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7UYVC | P52333 | 812 | 1100 | 1124.0 | OV5:1201 | Type1 | Inactive | DFGin | 6.5497 | 14.2474 | BLAminus | -139.0, -178.89 | 62.41, 84.96 | -102.47, 24.54 | 285.05, 80.61 | -63.66, -34.31 | in-in | in | 8.1764 | Saltbr-in | 2.7239 | HRD-in | -72.48, -47.02 | 76.02, -14.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.6962 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -72.04, 75.71 | APE9-dihe-in | -159.34, 174.75 | APE8-dihe-in | -55.7, 114.03 | APE8-rot-na | 331.85 | APE67-dihe-in | -81.89, -1.84 | -68.05, -12.84 | APE12-dist-na | 12.9994 | APE11-dist-na | 8.9457 | APE10-dist-na | 10.9307 | APE9-dist-out | 8.0032 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | C | 291.0 | 281.0 | 8 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4RIOA | P52333 | 815 | 1099 | 1124.0 | 3QX:4000 | Type1 | Inactive | DFGin | 6.3935 | 13.5705 | BLAminus | -146.26, -172.55 | 60.58, 82.0 | -101.14, 19.19 | 286.89, 85.95 | -65.85, -24.53 | in-in | in | 7.6666 | Saltbr-in | 2.8105 | HRD-in | -70.94, -43.53 | 62.59, 2.86 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9783 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -135.63, 27.38 | APE9-dihe-in | -118.75, 159.28 | APE8-dihe-in | -55.16, 127.94 | APE8-rot-na | 333.58 | APE67-dihe-in | -76.1, -3.72 | -64.2, -13.91 | APE12-dist-na | 12.5847 | APE11-dist-na | 9.8864 | APE10-dist-na | 9.9276 | APE9-dist-in | 7.1524 | C811S,C1040S,C1048S | None | None | XRAY | 2.69 | 0.218 | 0.281 | A | 293.0 | 285.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4rio | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5WFJA | P52333 | 817 | 1099 | 1124.0 | 9Z4:4000 | Type1 | Inactive | DFGin | 6.5811 | 13.8338 | BLAminus | -136.44, -170.83 | 58.73, 75.78 | -96.48, 23.06 | 286.97, 86.34 | -64.05, -24.53 | in-in | in | 7.6299 | Saltbr-in | 2.8738 | HRD-in | -76.6, -46.72 | 68.06, 1.53 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9182 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.32, 20.43 | APE9-dihe-in | -103.33, 153.28 | APE8-dihe-in | -50.05, 126.35 | APE8-rot-na | 333.7 | APE67-dihe-in | -76.71, 0.96 | -65.58, -12.14 | APE12-dist-na | 13.631 | APE11-dist-na | 9.8634 | APE10-dist-na | 10.1142 | APE9-dist-in | 7.0412 | C811S,C1040S,C1048S | None | None | XRAY | 2.48 | 0.205 | 0.255 | A | 293.0 | 265.0 | 18 | 31 | 29 | 2 | [[521, 779], [822, 1097]] | 2.0 | 5wfj | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4HVDA | P52333 | 815 | 1101 | 1124.0 | 933:1202 | Type1 | Inactive | DFGin | 6.5272 | 14.0171 | BLAminus | -128.55, -166.42 | 58.39, 76.56 | -98.5, 22.97 | 288.27, 78.76 | -65.56, -24.6 | in-in | in | 8.047 | Saltbr-in | 2.8425 | HRD-in | -70.62, -50.61 | 83.01, -13.8 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8441 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -120.35, 6.88 | APE9-dihe-in | -87.79, 153.51 | APE8-dihe-in | -47.35, 128.71 | APE8-rot-na | 328.03 | APE67-dihe-in | -81.29, -0.66 | -70.05, -11.78 | APE12-dist-na | 13.6702 | APE11-dist-na | 9.8379 | APE10-dist-na | 10.1082 | APE9-dist-in | 7.3252 | C1040S,C1048S | None | None | XRAY | 1.85 | 0.225 | 0.259 | A | 314.0 | 276.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvd | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4HVGA | P52333 | 814 | 1103 | 1124.0 | 19Q:1201 | Type1 | Inactive | DFGin | 6.3691 | 14.0706 | BLAminus | -130.41, -171.25 | 53.38, 75.08 | -85.23, 20.51 | 289.87, 75.57 | -58.89, -29.62 | in-in | in | 8.256 | Saltbr-in | 2.8006 | HRD-in | -81.72, -46.13 | 83.55, -16.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9723 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -135.6, 18.04 | APE9-dihe-in | -102.46, 155.94 | APE8-dihe-in | -50.03, 129.65 | APE8-rot-na | 326.24 | APE67-dihe-in | -77.88, -2.28 | -61.37, -21.51 | APE12-dist-na | 13.6391 | APE11-dist-na | 9.8591 | APE10-dist-na | 10.1069 | APE9-dist-in | 7.4421 | C1040S,C1048S | None | None | XRAY | 2.75 | 0.214 | 0.274 | A | 314.0 | 281.0 | 9 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvg | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4HVHA | P52333 | 814 | 1102 | 1124.0 | 19R:1201 | Type1 | Inactive | DFGin | 6.4361 | 14.1039 | BLAminus | -140.81, -174.18 | 54.94, 86.96 | -103.32, 27.47 | 289.17, 75.35 | -59.86, -26.99 | in-in | in | 8.1031 | Saltbr-in | 2.73 | HRD-in | -70.65, -47.69 | 79.95, -7.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8656 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -125.66, 18.79 | APE9-dihe-in | -103.72, 157.23 | APE8-dihe-in | -46.25, 127.99 | APE8-rot-na | 329.23 | APE67-dihe-in | -82.32, 1.96 | -65.92, -16.55 | APE12-dist-na | 13.6054 | APE11-dist-na | 9.7978 | APE10-dist-na | 10.0657 | APE9-dist-in | 7.3949 | C1040S,C1048S | None | None | XRAY | 2.3 | 0.23 | 0.283 | A | 314.0 | 278.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvh | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4HVIA | P52333 | 815 | 1101 | 1124.0 | 19S:1201 | Type1 | Inactive | DFGin | 6.4427 | 13.9006 | BLAminus | -133.13, -169.35 | 58.25, 80.79 | -103.46, 21.02 | 290.11, 82.66 | -64.8, -24.06 | in-in | in | 8.1481 | Saltbr-in | 2.7134 | HRD-in | -70.83, -44.69 | 73.14, -9.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0118 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.42, 8.91 | APE9-dihe-in | -93.49, 161.0 | APE8-dihe-in | -50.05, 128.83 | APE8-rot-na | 327.89 | APE67-dihe-in | -77.81, -4.37 | -61.08, -19.7 | APE12-dist-na | 13.3068 | APE11-dist-na | 9.5384 | APE10-dist-na | 9.8434 | APE9-dist-in | 7.267 | C1040S,C1048S | None | None | XRAY | 2.4 | 0.238 | 0.303 | A | 314.0 | 274.0 | 13 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4hvi | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4I6QA | P52333 | 815 | 1102 | 1124.0 | 1DT:1202 | Type1 | Inactive | DFGin | 6.5477 | 13.8797 | BLAminus | -122.27, -166.37 | 58.65, 80.25 | -102.66, 18.99 | 282.73, 92.38 | -63.16, -27.69 | in-in | in | 8.1701 | Saltbr-in | 2.6678 | HRD-in | -82.65, -46.76 | 80.12, -11.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8258 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.82, 1.26 | APE9-dihe-in | -88.25, 159.4 | APE8-dihe-in | -50.29, 130.77 | APE8-rot-na | 324.04 | APE67-dihe-in | -86.64, 4.17 | -68.93, -13.66 | APE12-dist-na | 13.7233 | APE11-dist-na | 9.8721 | APE10-dist-na | 9.9493 | APE9-dist-in | 7.3231 | C1040S,C1048S | None | None | XRAY | 1.85 | 0.198 | 0.245 | A | 314.0 | 277.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4i6q | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4QT1A | P52333 | 814 | 1102 | 1124.0 | 3C9:1201 | Type1 | Inactive | DFGin | 6.6492 | 13.9762 | BLAminus | -139.02, 177.24 | 52.6, 80.83 | -91.99, 24.19 | 292.74, 76.91 | -57.05, -27.61 | in-in | in | 7.854 | Saltbr-in | 2.8081 | HRD-in | -76.1, -42.64 | 74.06, 0.56 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8439 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.55, 16.0 | APE9-dihe-in | -104.71, 155.27 | APE8-dihe-in | -51.8, 130.25 | APE8-rot-na | 330.69 | APE67-dihe-in | -80.61, -3.03 | -68.8, -13.83 | APE12-dist-na | 13.5093 | APE11-dist-na | 9.8141 | APE10-dist-na | 9.9829 | APE9-dist-in | 7.1611 | C1040S,C1048S | None | None | XRAY | 2.4 | 0.21 | 0.273 | A | 314.0 | 277.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4qt1 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.7e-81 | 278.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5TOZA | P52333 | 815 | 1100 | 1124.0 | 7H4:1201 | Type1 | Inactive | DFGin | 6.4346 | 14.1797 | BLAminus | -132.42, -172.67 | 55.17, 83.47 | -97.89, 23.39 | 288.4, 75.31 | -59.42, -27.52 | in-in | in | 8.0531 | Saltbr-in | 2.7698 | HRD-in | -70.7, -45.74 | 70.21, -7.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8052 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.82, 11.45 | APE9-dihe-in | -93.23, 156.46 | APE8-dihe-in | -46.82, 125.7 | APE8-rot-na | 327.47 | APE67-dihe-in | -74.64, -1.89 | -65.68, -15.53 | APE12-dist-na | 13.7154 | APE11-dist-na | 9.6672 | APE10-dist-na | 10.1541 | APE9-dist-in | 7.336 | None | None | None | XRAY | 1.98 | 0.184 | 0.215 | A | 321.0 | 278.0 | 8 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5toz | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5TTSA | P52333 | 814 | 1100 | 1124.0 | 7KU:4000 | Type1 | Inactive | DFGin | 6.4256 | 14.158 | BLAminus | -129.0, -169.11 | 47.63, 82.34 | -97.79, 20.5 | 281.57, 83.57 | -59.54, -22.32 | in-in | in | 7.8793 | Saltbr-in | 2.727 | HRD-in | -71.68, -45.64 | 72.69, -11.39 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8295 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -120.94, 5.03 | APE9-dihe-in | -92.95, 155.15 | APE8-dihe-in | -50.68, 128.91 | APE8-rot-na | 333.75 | APE67-dihe-in | -73.89, 0.34 | -64.16, -15.93 | APE12-dist-na | 13.6385 | APE11-dist-na | 9.8268 | APE10-dist-na | 9.9629 | APE9-dist-in | 7.3964 | C1048S | None | None | XRAY | 2.34 | 0.205 | 0.263 | A | 321.0 | 274.0 | 13 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5tts | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5TTUA | P52333 | 815 | 1099 | 1124.0 | 7KV:1201 | Type1 | Inactive | DFGin | 6.5073 | 14.2203 | BLAminus | -134.44, -163.93 | 59.24, 64.07 | -87.63, 14.18 | 281.02, 85.09 | -61.33, -21.77 | in-in | in | 8.1783 | Saltbr-in | 2.6873 | HRD-in | -74.44, -46.15 | 74.73, -11.09 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.934 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -108.51, 0.99 | APE9-dihe-in | -84.97, 156.58 | APE8-dihe-in | -52.23, 128.18 | APE8-rot-na | 331.46 | APE67-dihe-in | -73.87, -5.17 | -63.29, -14.0 | APE12-dist-na | 13.6239 | APE11-dist-na | 9.6774 | APE10-dist-na | 9.9919 | APE9-dist-in | 7.2843 | C1048S | None | None | XRAY | 1.72 | 0.193 | 0.212 | A | 321.0 | 271.0 | 14 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5ttu | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5TTVA | P52333 | 814 | 1100 | 1124.0 | 7KX:4000 | Type1 | Inactive | DFGin | 6.389 | 13.9545 | BLAminus | -134.13, -173.38 | 47.72, 81.12 | -99.64, 24.47 | 284.98, 81.27 | -61.89, -30.49 | in-in | in | 7.571 | Saltbr-in | 2.7566 | HRD-in | -68.58, -49.94 | 77.2, -11.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.887 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.83, -8.71 | APE9-dihe-in | -81.68, 166.25 | APE8-dihe-in | -54.83, 134.34 | APE8-rot-na | 333.98 | APE67-dihe-in | -68.58, -14.21 | -64.91, -25.89 | APE12-dist-na | 13.454 | APE11-dist-na | 10.1045 | APE10-dist-na | 9.8444 | APE9-dist-in | 7.0476 | C1048S | None | None | XRAY | 1.93 | 0.195 | 0.25 | A | 321.0 | 280.0 | 7 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5ttv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6DA4A | P52333 | 815 | 1099 | 1124.0 | G4V:1201 | Type1 | Inactive | DFGin | 6.3399 | 14.1592 | BLAminus | -125.34, -166.51 | 46.1, 93.47 | -106.56, 19.65 | 286.03, 81.95 | -61.5, -24.21 | in-in | in | 8.0349 | Saltbr-in | 2.8116 | HRD-in | -66.39, -43.11 | 68.24, -5.72 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8446 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -76.16, 17.06 | APE9-dihe-in | -99.01, 151.3 | APE8-dihe-in | -54.06, 116.09 | APE8-rot-na | 335.02 | APE67-dihe-in | -66.76, -9.61 | -46.02, -19.91 | APE12-dist-na | 13.2424 | APE11-dist-na | 9.376 | APE10-dist-na | 10.3711 | APE9-dist-in | 7.2615 | C1048S | None | None | XRAY | 2.9 | 0.229 | 0.263 | A | 321.0 | 281.0 | 4 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6da4 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6DB3A | P52333 | 814 | 1100 | 1124.0 | G54:4000 | Type1 | Inactive | DFGin | 6.286 | 13.9012 | BLAminus | -131.89, -177.11 | 58.86, 88.06 | -99.15, 20.97 | 289.91, 81.31 | -57.3, -32.4 | in-in | in | 8.2338 | Saltbr-in | 2.6892 | HRD-in | -69.32, -44.77 | 72.88, -9.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7455 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -107.94, 10.67 | APE9-dihe-in | -91.58, 152.91 | APE8-dihe-in | -48.92, 124.78 | APE8-rot-na | 329.3 | APE67-dihe-in | -70.97, -6.33 | -60.73, -15.87 | APE12-dist-na | 13.7116 | APE11-dist-na | 9.5497 | APE10-dist-na | 10.1421 | APE9-dist-in | 7.3914 | C1048S | None | None | XRAY | 1.97 | 0.19 | 0.224 | A | 321.0 | 275.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6db3 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6DB4A | P52333 | 814 | 1100 | 1124.0 | G4Y:4000 | Type1 | Inactive | DFGin | 6.3293 | 13.8866 | BLAminus | -129.96, -177.19 | 65.04, 85.51 | -102.45, 21.04 | 283.09, 83.98 | -63.09, -23.83 | in-in | in | 8.1031 | Saltbr-in | 2.6779 | HRD-in | -75.95, -47.04 | 72.28, -5.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.844 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.18, 10.26 | APE9-dihe-in | -87.73, 153.8 | APE8-dihe-in | -51.18, 129.01 | APE8-rot-na | 329.23 | APE67-dihe-in | -72.48, -3.98 | -65.43, -15.27 | APE12-dist-na | 14.0574 | APE11-dist-na | 9.8642 | APE10-dist-na | 10.2997 | APE9-dist-in | 7.1511 | C1048S | None | None | XRAY | 1.662 | 0.187 | 0.216 | A | 321.0 | 276.0 | 11 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6db4 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6DUDA | P52333 | 814 | 1100 | 1124.0 | HB4:1201 | Type1 | Inactive | DFGin | 6.3774 | 14.08 | BLAminus | -130.37, -174.96 | 58.79, 79.77 | -94.85, 21.4 | 284.9, 80.47 | -61.75, -24.01 | in-in | in | 7.8751 | Saltbr-in | 2.7643 | HRD-in | -71.12, -48.96 | 73.72, -5.63 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.844 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -109.73, 7.91 | APE9-dihe-in | -89.0, 155.98 | APE8-dihe-in | -50.13, 125.96 | APE8-rot-na | 330.56 | APE67-dihe-in | -75.78, -4.72 | -64.96, -12.29 | APE12-dist-na | 14.024 | APE11-dist-na | 9.7788 | APE10-dist-na | 10.0218 | APE9-dist-in | 7.0938 | C1048S | None | None | XRAY | 1.66 | 0.185 | 0.215 | A | 321.0 | 272.0 | 15 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 6dud | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7Q6HAAA | P52333 | 814 | 1100 | 1124.0 | 934:1201 | Type1 | Inactive | DFGin | 6.4415 | 13.9124 | BLAminus | -128.11, -171.29 | 67.58, 71.88 | -97.45, 20.62 | 287.7, 81.42 | -64.43, -23.85 | in-in | in | 7.9084 | Saltbr-in | 2.684 | HRD-in | -72.1, -52.28 | 82.4, -12.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.789 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.93, 11.02 | APE9-dihe-in | -86.89, 152.23 | APE8-dihe-in | -44.63, 129.97 | APE8-rot-na | 328.93 | APE67-dihe-in | -80.65, 0.41 | -70.73, -15.65 | APE12-dist-na | 13.7773 | APE11-dist-na | 9.7373 | APE10-dist-na | 10.3425 | APE9-dist-in | 7.2322 | None | None | None | XRAY | 1.749 | 0.185 | 0.22 | AAA | 327.0 | 282.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7q6h | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3.1e-81 | 278.5 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3LXLA | P52333 | 814 | 1098 | 1124.0 | IZA:1 | Type1 | Inactive | DFGin | 6.3563 | 13.9832 | BLAminus | -131.21, -163.1 | 63.94, 61.73 | -90.52, 13.42 | 287.27, 88.72 | -63.24, -20.77 | in-in | in | 7.8734 | Saltbr-in | 2.759 | HRD-in | -76.94, -49.02 | 80.12, -11.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8049 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -131.67, 15.09 | APE9-dihe-in | -90.67, 156.23 | APE8-dihe-in | -48.41, 132.69 | APE8-rot-na | 328.44 | APE67-dihe-in | -80.87, -3.57 | -71.39, -11.92 | APE12-dist-na | 13.8943 | APE11-dist-na | 9.8069 | APE10-dist-na | 10.408 | APE9-dist-in | 7.3708 | C1048S | None | None | XRAY | 1.74 | 0.195 | 0.227 | A | 327.0 | 281.0 | 4 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 3lxl | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3.2e-81 | 278.4 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 1YVJA | P52333 | 814 | 1103 | 1124.0 | 4ST:2000 | Type1 | Inactive | DFGin | 6.5054 | 14.0048 | BLAminus | -117.35, -176.34 | 48.83, 98.04 | -113.48, 29.61 | 287.79, 84.73 | -71.88, -20.61 | in-in | in | 8.6181 | Saltbr-in | 2.8369 | HRD-in | -75.54, -39.16 | 74.88, -34.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8318 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -96.81, -5.63 | APE9-dihe-in | -95.15, 159.49 | APE8-dihe-in | -47.0, 152.52 | APE8-rot-na | 325.56 | APE67-dihe-in | -77.97, 4.18 | -53.16, -16.76 | APE12-dist-na | 9.8059 | APE11-dist-na | 6.854 | APE10-dist-na | 8.7777 | APE9-dist-out | 8.1995 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.55 | 0.204 | 0.254 | A | 290.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 1yvj | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 5.4e-81 | 277.7 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4Z16B | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | Inactive | DFGin | 6.6659 | 14.5322 | BLAminus | -124.7, -170.19 | 45.77, 83.37 | -100.74, 26.17 | 289.95, 82.89 | -68.35, -28.49 | in-in | in | 8.3877 | Saltbr-in | 2.8503 | HRD-in | -66.49, -45.94 | 73.56, -20.74 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8618 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -56.65, -6.62 | APE9-dihe-in | -78.46, 132.64 | APE8-dihe-in | -45.17, 131.02 | APE8-rot-na | 5.36 | APE67-dihe-in | -79.95, -14.25 | -79.37, 1.19 | APE12-dist-na | 12.5366 | APE11-dist-na | 9.232 | APE10-dist-na | 10.615 | APE9-dist-in | 7.017 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | B | 316.0 | 278.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4QPSC | P52333 | 814 | 1102 | 1124.0 | 37Q:1201 | Type1 | Inactive | DFGin | 6.7747 | 14.2003 | BLAminus | -137.32, -176.14 | 60.46, 91.64 | -108.44, 19.09 | 284.35, 76.96 | -56.92, -26.19 | in-in | in | 8.5021 | Saltbr-in | 2.8029 | HRD-in | -82.86, -44.58 | 73.92, -46.68 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8214 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 132.79 | APE8-dihe-in | -74.25, 110.88 | APE8-rot-na | 352.69 | APE67-dihe-in | -70.61, -6.19 | -68.78, -23.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.9914 | D949A,C1040S,C1048S | None | None | XRAY | 1.8 | 0.21 | 0.251 | C | 293.0 | 276.0 | 13 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4qps | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3.9e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5LWMA | P52333 | 814 | 1103 | 1124.0 | 79T:1201 | Type1 | Inactive | DFGin | 6.1807 | 14.0847 | BLAminus | -127.82, -164.11 | 50.78, 78.32 | -96.87, 23.57 | 279.03, 70.69 | -64.42, -25.51 | in-in | in | 7.8434 | Saltbr-in | 2.7715 | HRD-in | -83.79, -41.29 | 73.45, -47.71 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8732 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -137.31, 98.87 | APE9-dihe-in | -108.79, 137.75 | APE8-dihe-in | -66.78, 85.64 | APE8-rot-na | 29.56 | APE67-dihe-in | -76.19, -3.82 | -62.47, -28.25 | APE12-dist-na | 10.173 | APE11-dist-na | 13.4615 | APE10-dist-na | 12.5843 | APE9-dist-out | 8.869 | None | None | None | XRAY | 1.55 | 0.166 | 0.204 | A | 294.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5lwm | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7APFA | P52333 | 814 | 1103 | 1124.0 | RQZ:1201 | Type1 | Inactive | DFGin | 6.1423 | 14.108 | BLAminus | -125.02, -164.76 | 52.74, 82.07 | -99.72, 24.14 | 279.87, 69.9 | -58.8, -33.19 | in-in | in | 8.0164 | Saltbr-in | 2.735 | HRD-in | -77.19, -45.73 | 75.08, -49.11 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8014 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -141.26, 128.28 | APE9-dihe-in | -143.67, 157.99 | APE8-dihe-in | -81.92, 93.49 | APE8-rot-na | 7.76 | APE67-dihe-in | -79.55, -5.28 | -69.3, -23.78 | APE12-dist-na | 10.1511 | APE11-dist-na | 13.6863 | APE10-dist-na | 13.2698 | APE9-dist-out | 9.0224 | None | None | None | XRAY | 1.95 | 0.206 | 0.255 | A | 294.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apf | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7APFB | P52333 | 814 | 1103 | 1124.0 | RQZ:1201 | Type1 | Inactive | DFGin | 6.2636 | 13.9552 | BLAminus | -125.48, -163.38 | 48.35, 84.73 | -99.0, 25.48 | 280.41, 70.13 | -63.69, -28.85 | in-in | in | 8.0989 | Saltbr-in | 2.7319 | HRD-in | -80.63, -44.7 | 74.93, -48.31 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.7771 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -141.78, 126.08 | APE9-dihe-in | -146.46, 155.19 | APE8-dihe-in | -90.31, 98.72 | APE8-rot-na | 9.96 | APE67-dihe-in | -78.0, -2.22 | -75.31, -23.81 | APE12-dist-na | 9.6188 | APE11-dist-na | 13.0285 | APE10-dist-na | 12.5423 | APE9-dist-out | 9.1313 | None | None | None | XRAY | 1.95 | 0.206 | 0.255 | B | 294.0 | 285.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apf | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7APGA | P52333 | 813 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0309 | 13.9524 | BLAminus | -145.19, -172.66 | 53.39, 85.17 | -97.7, 25.99 | 284.4, 73.93 | -62.87, -25.47 | in-in | in | 8.4915 | Saltbr-in | 3.0886 | HRD-in | -83.97, -50.23 | 79.99, -46.84 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9125 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -120.14, 50.45 | APE9-dihe-in | -76.86, 156.83 | APE8-dihe-in | -73.67, 136.77 | APE8-rot-na | 351.29 | APE67-dihe-in | -81.27, -2.59 | -94.73, -13.37 | APE12-dist-na | 10.6785 | APE11-dist-na | 10.8995 | APE10-dist-na | 13.6012 | APE9-dist-out | 8.9847 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | A | 294.0 | 279.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7APGB | P52333 | 814 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0387 | 14.0695 | BLAminus | -144.05, -171.58 | 55.33, 84.79 | -97.11, 25.47 | 284.03, 75.74 | -64.12, -25.92 | in-in | in | 8.44 | Saltbr-in | 3.0791 | HRD-in | -83.8, -49.69 | 80.24, -45.58 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9057 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -121.16, 48.46 | APE9-dihe-in | -74.89, 156.25 | APE8-dihe-in | -72.87, 137.28 | APE8-rot-na | 354.01 | APE67-dihe-in | -82.99, -1.84 | -93.81, -9.25 | APE12-dist-na | 10.8058 | APE11-dist-na | 10.8121 | APE10-dist-na | 13.4192 | APE9-dist-out | 8.9175 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | B | 294.0 | 278.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7APGC | P52333 | 812 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0574 | 14.0501 | BLAminus | -143.35, -172.89 | 56.23, 84.96 | -97.07, 24.64 | 284.44, 74.77 | -64.51, -25.55 | in-in | in | 8.468 | Saltbr-in | 3.0668 | HRD-in | -82.68, -50.65 | 80.68, -46.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9124 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -120.01, 55.65 | APE9-dihe-in | -74.89, 157.1 | APE8-dihe-in | -74.45, 136.81 | APE8-rot-na | 351.06 | APE67-dihe-in | -81.76, -1.91 | -93.74, -14.98 | APE12-dist-na | 10.5477 | APE11-dist-na | 11.1621 | APE10-dist-na | 13.9629 | APE9-dist-out | 8.9485 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | C | 294.0 | 287.0 | 5 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7APGD | P52333 | 815 | 1103 | 1124.0 | RQT:61201 | Type1 | Inactive | DFGin | 6.0092 | 14.041 | BLAminus | -143.73, -171.03 | 51.78, 85.49 | -96.62, 26.59 | 283.85, 72.76 | -64.13, -26.23 | in-in | in | 8.434 | Saltbr-in | 3.0873 | HRD-in | -83.66, -49.57 | 81.52, -47.38 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9154 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -120.66, 45.43 | APE9-dihe-in | -76.74, 156.2 | APE8-dihe-in | -73.01, 137.72 | APE8-rot-na | 354.08 | APE67-dihe-in | -79.85, -1.41 | -95.44, -12.08 | APE12-dist-na | 10.8366 | APE11-dist-na | 10.5366 | APE10-dist-na | 13.2359 | APE9-dist-out | 8.9582 | None | None | None | XRAY | 2.4 | 0.214 | 0.256 | D | 294.0 | 277.0 | 12 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 7apg | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5LWNA | P52333 | 814 | 1103 | 1124.0 | 79R:1208,79S:1209 | Type1,Type1 | Inactive | DFGin | 6.1459 | 14.132 | BLAminus | -129.49, -162.36 | 48.02, 73.73 | -88.01, 20.06 | 281.83, 72.86 | -61.77, -25.11 | in-in | in | 7.8172 | Saltbr-in | 2.7083 | HRD-in | -84.52, -44.16 | 75.64, -46.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8251 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -141.38, 98.08 | APE9-dihe-in | -113.86, 140.78 | APE8-dihe-in | -73.27, 87.08 | APE8-rot-na | 29.33 | APE67-dihe-in | -77.95, -2.97 | -61.74, -27.63 | APE12-dist-na | 10.0824 | APE11-dist-na | 13.4052 | APE10-dist-na | 12.4459 | APE9-dist-out | 8.904 | None | None | None | XRAY | 1.6 | 0.169 | 0.209 | A | 294.0 | 290.0 | 0 | 31 | 31 | 0 | [[521, 779], [822, 1097]] | 2.0 | 5lwn | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6HZVA | P52333 | 815 | 1098 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.4293 | 14.257 | BLAminus | -133.87, 178.6 | 61.51, 90.4 | -109.85, 28.17 | 289.99, 77.52 | -67.6, -31.52 | in-in | in | 8.3241 | Saltbr-in | 2.9312 | HRD-in | -62.66, -43.13 | 71.32, -8.68 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7324 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 119.68 | APE8-rot-na | 14.07 | APE67-dihe-in | -79.55, -1.3 | -80.03, -13.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | A | 285.0 | 266.0 | 18 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6HZVB | P52333 | 815 | 1099 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.1943 | 14.2143 | BLAminus | -135.38, 176.48 | 64.47, 86.88 | -105.43, 20.89 | 286.69, 85.17 | -66.35, -29.51 | in-in | in | 8.1494 | Saltbr-in | 2.8265 | HRD-in | -61.18, -44.44 | 71.7, 4.93 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.6907 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 129.11 | APE8-rot-na | 330.57 | APE67-dihe-in | -79.98, -2.63 | -77.74, -18.2 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | B | 285.0 | 269.0 | 16 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6HZVC | P52333 | 815 | 1098 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.477 | 14.2719 | BLAminus | -130.86, 179.06 | 58.44, 90.28 | -109.09, 23.07 | 290.05, 84.12 | -62.59, -33.96 | in-in | in | 8.0905 | Saltbr-in | 2.8088 | HRD-in | -69.82, -48.24 | 78.15, -8.29 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.6892 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -41.25 | APE8-dihe-in | -66.72, 131.5 | APE8-rot-na | 341.69 | APE67-dihe-in | -75.5, -7.29 | -73.63, -18.87 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.346 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | C | 285.0 | 265.0 | 19 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6HZVD | P52333 | 815 | 1098 | 1124.0 | GYW:1101 | Type1 | None | DFGin | 6.418 | 14.1518 | BLAminus | -133.07, -178.12 | 58.66, 85.08 | -104.02, 25.84 | 292.67, 81.24 | -61.98, -32.78 | in-in | in | 8.1402 | Saltbr-in | 2.7701 | HRD-in | -71.74, -43.92 | 75.22, -14.51 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7079 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -35.5 | APE8-dihe-in | -66.27, 131.93 | APE8-rot-na | 340.52 | APE67-dihe-in | -79.97, 1.1 | -77.2, -17.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.6337 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.46 | 0.224 | 0.275 | D | 285.0 | 259.0 | 25 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6hzv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5W86B | P52333 | 816 | 1098 | 1124.0 | 9YV:4000 | Type1 | None | DFGin | 6.5719 | 14.1258 | BLAminus | -130.89, -177.7 | 55.33, 86.59 | -98.74, 23.53 | 285.65, 80.73 | -58.36, -36.34 | in-in | in | 8.1755 | Saltbr-in | 2.7815 | HRD-in | -61.09, -43.56 | 75.39, -22.05 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8266 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-in | -98.06, 144.28 | APE8-rot-na | 28.22 | APE67-dihe-in | -84.46, -5.87 | -122.29, -17.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.7561 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | B | 287.0 | 269.0 | 14 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5W86C | P52333 | 814 | 1099 | 1124.0 | 9YV:4000 | Type1 | None | DFGin | 6.5069 | 14.1113 | BLAminus | -131.5, -178.51 | 55.57, 86.1 | -97.59, 23.31 | 285.7, 80.13 | -57.67, -36.43 | in-in | in | 8.1655 | Saltbr-in | 2.9403 | HRD-in | -62.63, -48.44 | 77.31, -20.33 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8223 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -67.29 | APE8-rot-na | 15.79 | APE67-dihe-in | -70.13, -18.29 | -58.03, -20.5 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.61 | 0.211 | 0.264 | C | 287.0 | 275.0 | 11 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 5w86 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6AAKD | P52333 | 814 | 1098 | 1124.0 | 9T6:1201 | Type1 | None | DFGin | 6.3309 | 14.1383 | BLAminus | -145.03, 168.99 | 56.55, 97.11 | -103.75, 32.24 | 293.47, 81.71 | -62.01, -33.71 | in-in | in | 8.0179 | Saltbr-in | 2.8556 | HRD-in | -76.49, -42.81 | 76.74, -36.27 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7662 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 72.65 | APE8-dihe-in | -50.29, 134.06 | APE8-rot-na | 332.19 | APE67-dihe-in | -63.85, -16.03 | -70.13, -20.9 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.3842 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.67 | 0.269 | 0.326 | D | 287.0 | 268.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 6aak | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 1.9e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZC6B | P52333 | 813 | 1100 | 1124.0 | VFC:2103 | Type1 | None | DFGin | 6.2181 | 14.0462 | BLAminus | -128.88, -176.96 | 59.69, 81.97 | -99.61, 22.0 | 289.18, 82.46 | -63.53, -20.72 | in-in | in | 8.2087 | Saltbr-in | 2.7991 | HRD-in | -71.31, -49.71 | 79.31, 3.34 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7475 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 25.15 | APE9-dihe-in | -99.95, 171.81 | APE8-dihe-in | -50.02, 112.29 | APE8-rot-na | 325.04 | APE67-dihe-in | -73.29, -4.3 | -58.87, -25.22 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.4818 | APE9-dist-in | 6.8402 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | B | 288.0 | 278.0 | 10 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZC6D | P52333 | 814 | 1100 | 1124.0 | VFC:2103 | Type1 | None | DFGin | 6.3147 | 14.132 | BLAminus | -134.59, -176.68 | 59.2, 81.95 | -97.58, 24.75 | 285.45, 76.49 | -66.73, -25.04 | in-in | in | 8.057 | Saltbr-in | 2.7416 | HRD-in | -74.86, -52.02 | 77.99, -12.75 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7303 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 79.2 | APE8-rot-na | 32.25 | APE67-dihe-in | -80.63, -5.09 | -78.85, -21.32 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.42 | 0.193 | 0.254 | D | 288.0 | 269.0 | 18 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 3zc6 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZEPB | P52333 | 814 | 1100 | 1124.0 | 1NX:2101 | Type1 | None | DFGin | 6.3528 | 14.2219 | BLAminus | -142.2, 177.46 | 62.39, 84.45 | -101.38, 32.38 | 292.96, 77.07 | -73.1, -37.75 | in-in | in | 8.2407 | Saltbr-in | 2.735 | HRD-in | -71.3, -45.86 | 73.98, -5.89 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7688 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 174.81 | APE8-dihe-in | -59.17, 141.04 | APE8-rot-na | 332.8 | APE67-dihe-in | -80.76, -5.98 | -67.68, -15.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.4769 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | B | 288.0 | 270.0 | 17 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 3zep | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZEPC | P52333 | 814 | 1100 | 1124.0 | 1NX:2101 | Type1 | None | DFGin | 6.2667 | 14.2845 | BLAminus | -143.3, 179.56 | 63.59, 86.35 | -106.32, 31.56 | 290.45, 75.82 | -68.82, -32.0 | in-in | in | 8.1744 | Saltbr-in | 2.7545 | HRD-in | -76.43, -48.0 | 76.34, -21.16 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7144 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 45.01 | APE9-dihe-in | -93.38, 161.79 | APE8-dihe-in | -56.5, 116.98 | APE8-rot-na | 326.42 | APE67-dihe-in | -74.98, -4.7 | -72.25, -13.12 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.7287 | APE9-dist-in | 6.8497 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | C | 288.0 | 278.0 | 9 | 31 | 29 | 2 | [[521, 779], [822, 1097]] | 2.0 | 3zep | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 3ZEPD | P52333 | 814 | 1099 | 1124.0 | 1NX:2100 | Type1 | None | DFGin | 6.5755 | 14.572 | BLAminus | -134.12, 176.57 | 59.25, 80.73 | -100.38, 28.57 | 291.24, 76.13 | -63.83, -42.01 | in-in | in | 8.3615 | Saltbr-in | 2.6719 | HRD-in | -72.39, -47.07 | 79.2, -13.88 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7779 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 161.47 | APE8-dihe-in | -52.69, 138.76 | APE8-rot-na | 329.47 | APE67-dihe-in | -77.9, -7.22 | -77.25, -13.54 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.5559 | C1040S,C1048S | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.35 | 0.226 | 0.265 | D | 288.0 | 274.0 | 12 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 3zep | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.1 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 7UYVD | P52333 | 814 | 1100 | 1124.0 | OV5:1201 | Type1 | None | DFGin | 6.4207 | 14.2582 | BLAminus | -133.29, -179.06 | 58.4, 83.86 | -99.71, 22.65 | 285.23, 81.71 | -62.49, -28.09 | in-in | in | 8.2976 | Saltbr-in | 2.6722 | HRD-in | -64.99, -48.29 | 76.96, -0.25 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7457 | ActLoopCT-none | TYR | APEdihe_nniai | APEdist_aaai | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 163.98 | APE8-dihe-in | -58.27, 129.89 | APE8-rot-na | 335.93 | APE67-dihe-in | -80.69, -3.3 | -71.81, -12.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 7.4681 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.15 | 0.222 | 0.263 | D | 291.0 | 272.0 | 15 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 7uyv | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 5VO6A | P52333 | 815 | 1099 | 1124.0 | 9J4:4000 | Type1 | None | DFGin | 6.5587 | 13.7482 | BLAminus | -128.78, -173.97 | 61.05, 89.09 | -107.4, 19.66 | 285.17, 86.8 | -68.24, -28.8 | in-in | in | 7.5123 | Saltbr-in | 2.9107 | HRD-in | -75.3, -50.06 | 76.72, -16.95 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.9825 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 135.66 | APE8-rot-na | 332.57 | APE67-dihe-in | -81.44, -5.82 | -70.82, -9.6 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | C1040S,C1048S | None | None | XRAY | 2.65 | 0.215 | 0.284 | A | 293.0 | 271.0 | 14 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 5vo6 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6NY4A | P52333 | 815 | 1099 | 1124.0 | Z3A:4000 | Type1 | None | DFGin | 6.4319 | 13.7522 | BLAminus | -130.0, -166.41 | 50.15, 85.44 | -100.28, 21.12 | 284.91, 84.56 | -64.41, -23.36 | in-in | in | 7.6903 | Saltbr-in | 2.7769 | HRD-in | -74.4, -47.07 | 70.71, -6.14 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8428 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -0.08 | APE9-dihe-in | -95.23, 160.07 | APE8-dihe-in | -49.81, 129.43 | APE8-rot-na | 333.86 | APE67-dihe-in | -73.45, 2.08 | -64.08, -16.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 9.7064 | APE9-dist-in | 7.0951 | C811S,C1040S,C1048S | None | None | XRAY | 2.33 | 0.216 | 0.241 | A | 293.0 | 277.0 | 8 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 6ny4 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.1e-81 | 279.0 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4V0GB | P52333 | 816 | 1098 | 1124.0 | G9B:2099 | Type1 | None | DFGin | 6.202 | 14.6329 | BLAminus | -137.8, -174.69 | 52.03, 76.68 | -96.09, 37.57 | 296.46, 78.81 | -70.34, -40.16 | in-in | in | 8.7004 | Saltbr-in | 2.629 | HRD-in | -75.76, -37.0 | 67.95, -17.09 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8243 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -54.69 | APE8-rot-na | 331.57 | APE67-dihe-in | -77.98, -0.68 | -62.56, -42.14 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 3.0 | 0.254 | 0.295 | B | 283.0 | 274.0 | 9 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4v0g | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.3e-81 | 278.9 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4V0GA | P52333 | 817 | 1098 | 1124.0 | G9B:2099 | Type1 | None | DFGin | 6.198 | 14.7166 | BLAminus | -144.75, -176.45 | 39.25, 85.88 | -90.52, 22.25 | 286.27, 74.42 | -61.38, -18.98 | in-in | in | 8.3521 | Saltbr-in | 2.7066 | HRD-in | -65.46, -44.14 | 69.1, 4.41 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8503 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -33.75 | APE8-rot-na | 330.77 | APE67-dihe-in | -73.45, -1.83 | -68.02, -39.07 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 3.0 | 0.254 | 0.295 | A | 283.0 | 269.0 | 13 | 31 | 27 | 4 | [[521, 779], [822, 1097]] | 2.0 | 4v0g | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 2.3e-81 | 278.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4Z16A | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | None | DFGin | 6.693 | 14.5354 | BLAminus | -125.11, -170.67 | 46.31, 83.09 | -100.98, 26.25 | 290.17, 83.28 | -67.99, -29.42 | in-in | in | 8.3468 | Saltbr-in | 2.8339 | HRD-in | -67.29, -45.59 | 73.41, -19.17 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8291 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 77.57 | APE8-rot-na | 328.09 | APE67-dihe-in | -74.64, -13.67 | -80.93, -12.04 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | A | 316.0 | 273.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4Z16C | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | None | DFGin | 6.724 | 14.5409 | BLAminus | -124.89, -171.04 | 46.95, 83.36 | -101.0, 25.74 | 290.21, 83.17 | -68.15, -28.94 | in-in | in | 8.3723 | Saltbr-in | 2.8403 | HRD-in | -67.03, -45.78 | 73.53, -19.66 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7882 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 38.92 | APE8-rot-na | 335.43 | APE67-dihe-in | -76.63, -13.6 | -68.45, -18.81 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | C | 316.0 | 273.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4Z16D | P52333 | 814 | 1103 | 1124.0 | 4LH:2000 | Type1 | None | DFGin | 6.6883 | 14.5667 | BLAminus | -124.04, -170.5 | 45.94, 82.68 | -99.35, 24.89 | 290.17, 82.54 | -66.47, -27.42 | in-in | in | 8.3931 | Saltbr-in | 2.8748 | HRD-in | -67.23, -45.45 | 73.09, -20.62 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7942 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 52.48 | APE8-rot-na | 345.61 | APE67-dihe-in | -77.91, -13.97 | -72.79, -6.5 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.9 | 0.204 | 0.24 | D | 316.0 | 273.0 | 17 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 4z16 | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 7.5e-81 | 277.2 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 4QPSA | P52333 | 814 | 1100 | 1124.0 | 37Q:1201 | Type1 | None | DFGin | 6.8957 | 14.0909 | BLAminus | -130.94, -174.49 | 64.52, 86.82 | -104.86, 15.71 | 281.27, 81.21 | -57.28, -32.23 | in-in | in | 8.5879 | Saltbr-in | 2.8637 | HRD-in | -78.56, -46.33 | 74.55, -53.21 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.801 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 149.07 | APE8-rot-na | 18.94 | APE67-dihe-in | -69.31, -9.6 | -100.11, -5.26 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | D949A,C1040S,C1048S | None | None | XRAY | 1.8 | 0.21 | 0.251 | A | 293.0 | 270.0 | 17 | 31 | 25 | 6 | [[521, 779], [822, 1097]] | 2.0 | 4qps | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 3.9e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6GLAA | P52333 | 813 | 1103 | 1124.0 | F4B:1201 | Type1 | None | DFGin | 6.1255 | 14.0661 | BLAminus | -126.69, -163.69 | 45.61, 84.37 | -97.16, 18.74 | 276.14, 73.33 | -60.39, -30.05 | in-in | in | 7.8334 | Saltbr-in | 2.6744 | HRD-in | -80.36, -50.35 | 74.06, -4.7 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7495 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 115.39 | APE9-dihe-in | -100.65, 143.31 | APE8-dihe-in | -75.22, 92.35 | APE8-rot-na | 30.49 | APE67-dihe-in | -81.25, -0.82 | -60.88, -31.57 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.6793 | APE9-dist-in | 7.0014 | None | None | None | XRAY | 1.92 | 0.228 | 0.273 | A | 294.0 | 288.0 | 3 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6gla | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6GLAB | P52333 | 813 | 1103 | 1124.0 | F4B:1201 | Type1 | None | DFGin | 6.1346 | 14.0372 | BLAminus | -126.98, -166.17 | 47.87, 84.06 | -100.26, 19.16 | 275.64, 73.52 | -60.46, -30.51 | in-in | in | 7.8307 | Saltbr-in | 2.6702 | HRD-in | -83.39, -49.56 | 74.28, -3.93 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7748 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 114.52 | APE9-dihe-in | -101.31, 145.02 | APE8-dihe-in | -77.95, 91.55 | APE8-rot-na | 29.11 | APE67-dihe-in | -79.72, -1.04 | -62.76, -29.93 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.7449 | APE9-dist-in | 6.9663 | None | None | None | XRAY | 1.92 | 0.228 | 0.273 | B | 294.0 | 286.0 | 5 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6gla | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6GLBA | P52333 | 813 | 1103 | 1124.0 | F48:1201 | Type1 | None | DFGin | 6.0868 | 14.0047 | BLAminus | -127.29, -165.11 | 42.2, 80.94 | -98.99, 18.18 | 281.6, 72.22 | -46.91, -40.63 | in-in | in | 7.5761 | Saltbr-in | 2.7125 | HRD-in | -78.7, -52.76 | 77.75, 9.6 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7344 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 129.22 | APE9-dihe-in | -106.96, 151.72 | APE8-dihe-in | -79.63, 91.52 | APE8-rot-na | 32.17 | APE67-dihe-in | -74.91, -5.23 | -62.01, -34.09 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.734 | APE9-dist-in | 6.7274 | None | None | None | XRAY | 2.0 | 0.236 | 0.29 | A | 294.0 | 288.0 | 3 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6glb | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 6GLBB | P52333 | 813 | 1103 | 1124.0 | F48:1201 | Type1 | None | DFGin | 6.117 | 14.0249 | BLAminus | -125.81, -165.95 | 42.86, 80.87 | -97.87, 18.6 | 282.22, 74.99 | -51.1, -37.8 | in-in | in | 7.5451 | Saltbr-in | 2.7085 | HRD-in | -76.97, -51.62 | 77.21, 8.56 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.7568 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 130.97 | APE9-dihe-in | -105.16, 150.45 | APE8-dihe-in | -79.13, 89.35 | APE8-rot-na | 33.14 | APE67-dihe-in | -76.14, -3.82 | -57.76, -35.85 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.6293 | APE9-dist-in | 6.7039 | None | None | None | XRAY | 2.0 | 0.236 | 0.29 | B | 294.0 | 288.0 | 3 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 6glb | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 9R5ZA | P52333 | 822 | 1101 | 1124.0 | A1JJU:60301 | Type1 | None | DFGin | 6.1324 | 14.0012 | BLAminus | -127.52, -161.85 | 48.17, 81.61 | -92.0, 24.85 | 277.91, 73.75 | -73.44, -23.7 | in-in | in | 7.6679 | Saltbr-in | 2.7676 | HRD-in | -79.16, -47.46 | 79.61, -35.13 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8804 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 92.63 | APE8-rot-na | 20.77 | APE67-dihe-in | -76.47, -3.83 | -62.4, -34.74 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.8 | 0.239 | 0.289 | A | 294.0 | 258.0 | 22 | 31 | 26 | 5 | [[521, 779], [822, 1097]] | 2.0 | 9r5z | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| JAK3-2 | JAK3_HUMAN | 9R5ZB | P52333 | 816 | 1101 | 1124.0 | A1JJU:60301 | Type1 | None | DFGin | 6.2264 | 14.1304 | BLAminus | -127.35, -164.41 | 49.32, 77.12 | -91.09, 23.07 | 281.2, 72.28 | -62.52, -23.26 | in-in | in | 7.8816 | Saltbr-in | 2.8186 | HRD-in | -86.18, -46.89 | 79.27, -42.6 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.8747 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 79.25 | APE8-rot-na | 31.77 | APE67-dihe-in | -82.31, -0.99 | -65.94, -24.16 | APE12-dist-na | 11.0451 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.8 | 0.239 | 0.289 | B | 294.0 | 275.0 | 11 | 31 | 28 | 3 | [[521, 779], [822, 1097]] | 2.0 | 9r5z | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 4e-80 | 274.8 | 1.0 | 260.0 | 260.0 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949.0 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|