OTHER_HASPIN (Serine/threonine-protein kinase haspin)

Total number of chains: 42
Active chains: 33
Family: OTHER
Uniprot: HASP_HUMAN
Kinase Domain Residues: 484 - 797
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 41 97.6% AF-Q8TF76-K1A
DFGin None 1 2.4% 9B2TK

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PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
3DLZA 470 798 798.0 AMP:902 ATPlike Active DFGin 5.254 12.469 BLAminus -120.14, 174.05 73.32, 91.07 -105.92, 29.14 315.79, 130.04 -57.27, -36.15 in-in in 9.264 Saltbr-in 2.695 HRD-na-N -71.0, -49.07 68.99, 3.03 in-in-na SNCiia in-na ActLoopNT-in 2.821 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -122.28, 17.39 APE9-dihe-na -67.57, 157.85 APE8-dihe-na -149.51, 177.99 APE8-rot-na 58.52 APE67-dihe-na -159.03, 144.74 95.06, -6.22 APE12-dist-na 9.493 APE11-dist-na 13.466 APE10-dist-na 17.05 APE9-dist-na 12.819 None None None XRAY 1.85 0.167 0.216 A 357 329 0 0 0 0 [[484, 797]] 1.0 3dlz OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
AF-Q8TF76-K1A 476 798 798.0 No_ligand No_ligand Active DFGin 4.997 12.374 BLAminus -138.62, 174.68 57.97, 91.28 -100.94, 21.93 314.77, 120.9 -55.94, -45.23 in-in in 9.18 Saltbr-in 2.711 HRD-na-N -75.36, -43.16 61.41, 5.31 in-in-na SNCiia in-na ActLoopNT-in 2.839 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -93.17, -12.71 APE9-dihe-na -54.03, 150.53 APE8-dihe-na -147.69, 169.0 APE8-rot-na 193.38 APE67-dihe-na -135.11, 149.27 98.64, -16.5 APE12-dist-na 9.305 APE11-dist-na 13.309 APE10-dist-na 16.98 APE9-dist-na 12.992 None None None AF2 -1.0 1.0 1.0 A 323 323 0 0 0 0 [[484, 797]] 1.0 AF-Q8TF76-K1 OTHER_HASPIN_HUMAN HASP 9.2e-227 757.1 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
AF-Q8TF76-K3A 476 798 798.0 No_ligand No_ligand Active DFGin 4.951 12.431 BLAminus -133.71, 176.01 54.85, 96.46 -104.75, 21.31 315.54, 124.63 -56.24, -41.59 in-in in 9.299 Saltbr-in 2.719 HRD-na-N -75.19, -42.52 61.0, 1.07 in-in-na SNCiia in-na ActLoopNT-in 2.885 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -93.31, -18.43 APE9-dihe-na -56.71, 155.17 APE8-dihe-na -141.59, -175.7 APE8-rot-na 73.98 APE67-dihe-na -125.54, 149.77 84.64, -25.13 APE12-dist-na 9.207 APE11-dist-na 13.228 APE10-dist-na 16.926 APE9-dist-na 13.133 None None None AF2 -1.0 1.0 1.0 A 323 323 0 0 0 0 [[484, 797]] 1.0 AF-Q8TF76-K3 OTHER_HASPIN_HUMAN HASP 9.2e-227 757.1 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
2WB8A 447 798 798.0 No_ligand No_ligand Active DFGin 5.22 12.191 BLAminus -120.69, 176.87 68.15, 91.75 -104.26, 25.9 315.71, 126.12 -56.01, -32.87 in-in in 9.095 Saltbr-in 2.281 HRD-na-N -69.54, -53.11 72.35, 6.09 in-in-na SNCiia in-na ActLoopNT-in 2.857 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -129.5, 34.17 APE9-dihe-na -83.79, 164.98 APE8-dihe-na -149.79, 174.65 APE8-rot-na 31.25 APE67-dihe-na -168.04, 143.08 80.64, 14.62 APE12-dist-na 9.206 APE11-dist-na 12.948 APE10-dist-na 16.727 APE9-dist-na 12.724 None None None XRAY 2.15 0.23 0.267 A 352 351 1 0 0 0 [[484, 797]] 1.0 2wb8 OTHER_HASPIN_HUMAN HASP 1.3e-226 756.7 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
5HTBA 471 798 798.0 No_ligand No_ligand Active DFGin 4.886 12.713 BLAminus -127.82, 172.38 75.8, 95.98 -111.9, 24.65 313.35, 119.25 -57.64, -36.0 in-in in 9.095 Saltbr-in 2.722 HRD-na-N -72.45, -46.3 70.77, -0.27 in-in-na SNCiia in-na ActLoopNT-in 2.859 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.52, 17.28 APE9-dihe-na -71.3, 162.17 APE8-dihe-na -148.2, 163.96 APE8-rot-na 208.0 APE67-dihe-na -159.11, 139.67 91.05, 1.41 APE12-dist-na 9.417 APE11-dist-na 13.298 APE10-dist-na 16.873 APE9-dist-na 12.933 None None None XRAY 1.7 0.163 0.181 A 357 328 0 0 0 0 [[484, 797]] 1.0 5htb OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
5HTCA 471 798 798.0 No_ligand No_ligand Active DFGin 5.008 12.77 BLAminus -124.68, 170.56 74.88, 95.44 -108.39, 22.99 316.66, 123.43 -55.96, -37.72 in-in in 9.222 Saltbr-in 2.671 HRD-na-N -71.81, -49.47 73.17, 0.66 in-in-na SNCiia in-na ActLoopNT-in 2.875 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.86, 18.07 APE9-dihe-na -74.58, 161.83 APE8-dihe-na -153.14, 168.43 APE8-rot-na 79.76 APE67-dihe-na -159.07, 137.97 97.79, -1.9 APE12-dist-na 9.518 APE11-dist-na 13.376 APE10-dist-na 16.983 APE9-dist-na 12.965 None None None XRAY 1.5 0.151 0.171 A 357 328 0 0 0 0 [[484, 797]] 1.0 5htc OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6G39A 471 798 798.0 5ID:802 Type1 Active DFGin 5.021 12.32 BLAminus -127.21, 173.16 74.1, 91.77 -104.6, 25.15 318.27, 124.04 -54.52, -37.44 in-in in 9.223 Saltbr-in 2.607 HRD-na-N -72.86, -48.93 72.97, 0.92 in-in-na SNCiia in-na ActLoopNT-in 2.865 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.61, 13.68 APE9-dihe-na -74.05, 162.55 APE8-dihe-na -147.53, 161.22 APE8-rot-na 206.35 APE67-dihe-na -163.09, 139.78 96.44, 2.71 APE12-dist-na 9.496 APE11-dist-na 13.491 APE10-dist-na 16.919 APE9-dist-na 13.026 F605Y None None XRAY 1.45 0.159 0.175 A 357 328 0 0 0 0 [[484, 797]] 1.0 6g39 OTHER_HASPIN_HUMAN HASP 3.9e-226 755.1 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
2VUWA 470 798 798.0 5ID:1800 Type1 Active DFGin 4.977 12.344 BLAminus -126.7, 172.42 73.13, 94.6 -106.22, 25.34 317.03, 123.17 -59.06, -30.58 in-in in 9.293 Saltbr-in 2.791 HRD-na-N -69.06, -49.8 71.93, -0.86 in-in-na SNCiia in-na ActLoopNT-in 2.886 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.41, 21.25 APE9-dihe-na -74.65, 162.69 APE8-dihe-na -150.22, 164.21 APE8-rot-na 197.92 APE67-dihe-na -163.26, 143.62 93.5, 5.23 APE12-dist-na 9.51 APE11-dist-na 13.492 APE10-dist-na 17.046 APE9-dist-na 12.946 None None MSE615,MSE706,MSE725,MSE752,MSE756,MSE767,MSE781 XRAY 1.8 0.148 0.169 A 336 329 0 0 0 0 [[484, 797]] 1.0 2vuw OTHER_HASPIN_HUMAN HASP 1.1e-226 756.9 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9FLTA 471 798 798.0 A1IDF:801 Type1 Active DFGin 5.178 12.218 BLAminus -141.02, 178.95 59.99, 70.73 -81.95, 27.03 316.78, 141.24 -69.29, -28.67 in-in in 8.759 Saltbr-in 2.463 HRD-na-N -66.6, -53.16 75.71, 6.9 in-in-na SNCiia in-na ActLoopNT-in 2.905 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -131.58, 41.34 APE9-dihe-na -102.69, 164.5 APE8-dihe-na -162.68, -171.46 APE8-rot-na 41.52 APE67-dihe-na -134.91, 146.64 100.36, -24.97 APE12-dist-na 9.64 APE11-dist-na 13.509 APE10-dist-na 17.247 APE9-dist-na 13.279 None None None XRAY 2.4 0.187 0.239 A 336 320 8 0 0 0 [[484, 797]] 1.0 9flt OTHER_HASPIN_HUMAN HASP 1.1e-226 756.9 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
3E7VA 471 798 798.0 DZO:1 Type1 Active DFGin 5.227 12.203 BLAminus -130.14, 169.21 72.6, 84.89 -101.25, 35.48 316.82, 123.9 -62.16, -34.97 in-in in 9.014 Saltbr-in 2.481 HRD-na-N -68.11, -48.56 71.09, -0.57 in-in-na SNCiia in-na ActLoopNT-in 2.917 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -113.43, 18.49 APE9-dihe-na -73.97, 165.86 APE8-dihe-na -158.09, 152.51 APE8-rot-na 206.55 APE67-dihe-na -159.89, 140.52 100.1, 0.81 APE12-dist-na 9.459 APE11-dist-na 13.36 APE10-dist-na 17.023 APE9-dist-na 12.905 None None None XRAY 2.0 0.17 0.225 A 357 328 0 0 0 0 [[484, 797]] 1.0 3e7v OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
3F2NA 471 798 798.0 IZZ:800 Type1 Active DFGin 5.227 12.509 BLAminus -132.35, 169.14 74.56, 87.66 -98.09, 25.18 316.3, 125.75 -57.05, -34.51 in-in in 8.729 Saltbr-in 2.737 HRD-na-N -71.51, -49.79 70.28, -0.25 in-in-na SNCiia in-na ActLoopNT-in 2.913 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -120.07, 21.25 APE9-dihe-na -75.2, 162.89 APE8-dihe-na -156.01, 176.32 APE8-rot-na 74.11 APE67-dihe-na -157.24, 143.14 98.22, -8.69 APE12-dist-na 9.565 APE11-dist-na 13.531 APE10-dist-na 17.149 APE9-dist-na 12.969 None None None XRAY 1.8 0.162 0.186 A 357 328 0 0 0 0 [[484, 797]] 1.0 3f2n OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
3FMDA 470 798 798.0 IQB:1 Type1 Active DFGin 4.817 12.737 BLAminus -134.95, 173.12 69.12, 93.36 -108.33, 23.11 309.03, 122.86 -58.61, -32.84 in-in in 9.417 Saltbr-in 2.578 HRD-na-N -64.91, -44.59 67.0, -1.51 in-in-na SNCiia in-na ActLoopNT-in 2.86 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -126.4, 30.5 APE9-dihe-na -82.22, 168.97 APE8-dihe-na -156.73, 170.22 APE8-rot-na 87.7 APE67-dihe-na -158.09, 144.39 88.76, -6.79 APE12-dist-na 9.533 APE11-dist-na 13.423 APE10-dist-na 17.115 APE9-dist-na 13.017 None None None XRAY 2.0 0.226 0.283 A 357 329 0 0 0 0 [[484, 797]] 1.0 3fmd OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
3IQ7A 471 798 798.0 5ID:799 Type1 Active DFGin 5.002 12.525 BLAminus -130.14, 168.59 78.5, 93.8 -107.03, 26.88 317.14, 123.36 -63.63, -28.13 in-in in 9.288 Saltbr-in 2.716 HRD-na-N -69.08, -54.14 69.34, 3.59 in-in-na SNCiia in-na ActLoopNT-in 2.842 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -119.96, 19.66 APE9-dihe-na -73.26, 163.53 APE8-dihe-na -151.13, 165.69 APE8-rot-na 217.79 APE67-dihe-na -160.55, 141.37 91.74, 4.08 APE12-dist-na 9.31 APE11-dist-na 13.171 APE10-dist-na 16.954 APE9-dist-na 12.798 None None None XRAY 2.0 0.174 0.207 A 357 328 0 0 0 0 [[484, 797]] 1.0 3iq7 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
4OUCA 470 798 798.0 5ID:60808 Type1 Active DFGin 5.142 12.398 BLAminus -123.14, 171.36 70.83, 89.85 -103.14, 24.75 317.85, 126.13 -50.7, -43.23 in-in in 9.227 Saltbr-in 2.635 HRD-na-N -73.5, -49.82 73.73, 4.15 in-in-na SNCiia in-na ActLoopNT-in 2.897 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.93, 10.97 APE9-dihe-na -70.72, 155.25 APE8-dihe-na -144.93, 165.92 APE8-rot-na 81.62 APE67-dihe-na -154.34, 142.15 101.34, -0.24 APE12-dist-na 9.521 APE11-dist-na 13.627 APE10-dist-na 17.119 APE9-dist-na 12.997 None None None XRAY 1.9 0.166 0.211 A 357 329 0 0 0 0 [[484, 797]] 1.0 4ouc OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
4QTCA 469 798 798.0 38Z:804 Type1 Active DFGin 4.743 12.697 BLAminus -128.25, 174.11 72.8, 94.29 -100.86, 22.55 311.48, 126.56 -49.88, -46.32 in-in in 9.244 Saltbr-in 2.767 HRD-na-N -70.64, -49.71 73.49, 0.07 in-in-na SNCiia in-na ActLoopNT-in 2.862 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.14, 15.58 APE9-dihe-na -74.4, 166.34 APE8-dihe-na -155.61, 167.98 APE8-rot-na 54.8 APE67-dihe-na -159.6, 141.49 96.89, -1.32 APE12-dist-na 9.4 APE11-dist-na 13.293 APE10-dist-na 16.89 APE9-dist-na 13.142 None None None XRAY 1.4 0.15 0.164 A 357 330 0 0 0 0 [[484, 797]] 1.0 4qtc OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6G34A 472 798 798.0 5ID:60401 Type1 Active DFGin 4.991 12.367 BLAminus -127.35, 171.15 74.89, 93.11 -104.99, 26.96 316.16, 126.1 -57.37, -32.12 in-in in 9.292 Saltbr-in 2.721 HRD-na-N -71.53, -47.32 70.63, -2.3 in-in-na SNCiia in-na ActLoopNT-in 2.893 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.68, 18.32 APE9-dihe-na -70.1, 157.86 APE8-dihe-na -146.1, 158.98 APE8-rot-na 202.21 APE67-dihe-na -162.15, 141.91 96.58, 0.13 APE12-dist-na 9.436 APE11-dist-na 13.462 APE10-dist-na 16.952 APE9-dist-na 12.837 None None None XRAY 1.76 0.14 0.174 A 357 327 0 0 0 0 [[484, 797]] 1.0 6g34 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6G35A 465 798 798.0 EKK:60802 Type1 Active DFGin 5.005 12.39 BLAminus -126.0, 169.52 78.13, 90.25 -104.66, 24.26 315.74, 125.01 -60.88, -28.25 in-in in 9.306 Saltbr-in 2.713 HRD-na-N -70.57, -49.54 72.42, 1.39 in-in-na SNCiia in-na ActLoopNT-in 2.901 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.32, 17.8 APE9-dihe-na -73.2, 161.57 APE8-dihe-na -146.96, 162.71 APE8-rot-na 196.59 APE67-dihe-na -162.63, 137.82 97.88, 1.51 APE12-dist-na 9.478 APE11-dist-na 13.461 APE10-dist-na 17.008 APE9-dist-na 13.016 None None None XRAY 1.55 0.161 0.183 A 357 334 0 0 0 0 [[484, 797]] 1.0 6g35 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6G36A 465 798 798.0 EKH:60401 Type1 Active DFGin 4.952 12.328 BLAminus -126.44, 170.29 76.27, 92.19 -105.23, 26.61 316.28, 124.1 -57.25, -32.63 in-in in 9.282 Saltbr-in 2.744 HRD-na-N -71.83, -48.64 74.84, -0.58 in-in-na SNCiia in-na ActLoopNT-in 2.89 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.55, 15.17 APE9-dihe-na -70.08, 160.85 APE8-dihe-na -149.64, 167.11 APE8-rot-na 67.1 APE67-dihe-na -162.45, 137.7 92.15, 4.46 APE12-dist-na 9.491 APE11-dist-na 13.449 APE10-dist-na 17.015 APE9-dist-na 12.972 None None None XRAY 1.46 0.151 0.176 A 357 334 0 0 0 0 [[484, 797]] 1.0 6g36 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6G37A 472 798 798.0 FTU:801 Type1 Active DFGin 5.035 12.401 BLAminus -125.49, 171.67 75.49, 90.88 -104.56, 25.99 317.99, 122.48 -54.51, -35.12 in-in in 9.318 Saltbr-in 2.736 HRD-na-N -70.97, -50.1 72.78, 2.06 in-in-na SNCiia in-na ActLoopNT-in 2.889 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -114.17, 14.96 APE9-dihe-na -72.53, 161.37 APE8-dihe-na -147.52, 165.41 APE8-rot-na 216.83 APE67-dihe-na -159.62, 143.17 92.11, 0.24 APE12-dist-na 9.422 APE11-dist-na 13.433 APE10-dist-na 16.884 APE9-dist-na 12.914 None None None XRAY 1.48 0.149 0.167 A 357 327 0 0 0 0 [[484, 797]] 1.0 6g37 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6G38A 472 798 798.0 TBN:800 Type1 Active DFGin 5.155 12.468 BLAminus -124.6, 171.17 73.49, 90.96 -102.58, 23.98 318.22, 128.64 -60.91, -27.39 in-in in 9.286 Saltbr-in 2.681 HRD-na-N -70.12, -48.6 70.78, 0.07 in-in-na SNCiia in-na ActLoopNT-in 2.865 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.63, 17.26 APE9-dihe-na -74.94, 161.54 APE8-dihe-na -150.43, 171.99 APE8-rot-na 81.52 APE67-dihe-na -161.74, 140.31 94.52, 1.17 APE12-dist-na 9.54 APE11-dist-na 13.547 APE10-dist-na 17.024 APE9-dist-na 13.008 None None None XRAY 1.47 0.144 0.165 A 357 327 0 0 0 0 [[484, 797]] 1.0 6g38 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z57A 470 798 798.0 Q8W:801 Type1 Active DFGin 5.108 12.544 BLAminus -128.55, 170.14 70.49, 89.65 -99.72, 23.55 319.85, 122.5 -60.24, -32.24 in-in in 9.047 Saltbr-in 2.63 HRD-na-N -69.51, -48.64 73.21, 1.64 in-in-na SNCiia in-na ActLoopNT-in 2.906 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.13, 24.13 APE9-dihe-na -80.04, 165.59 APE8-dihe-na -154.67, 168.36 APE8-rot-na 59.7 APE67-dihe-na -158.19, 141.65 89.15, 3.9 APE12-dist-na 9.623 APE11-dist-na 13.634 APE10-dist-na 17.184 APE9-dist-na 13.001 None None None XRAY 1.5 0.164 0.188 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z57 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z58A 470 798 798.0 Q9B:801 Type1 Active DFGin 5.29 11.882 BLAminus -131.62, 178.98 63.69, 89.83 -101.06, 25.15 318.41, 128.59 -53.25, -41.36 in-in in 8.999 Saltbr-in 2.668 HRD-na-N -74.24, -49.55 73.51, 2.01 in-in-na SNCiia in-na ActLoopNT-in 2.86 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.26, 20.54 APE9-dihe-na -78.55, 163.28 APE8-dihe-na -149.94, 172.24 APE8-rot-na 51.88 APE67-dihe-na -158.7, 145.23 97.38, -8.51 APE12-dist-na 9.654 APE11-dist-na 13.592 APE10-dist-na 17.186 APE9-dist-na 13.103 None None None XRAY 1.8 0.164 0.19 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z58 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z59A 471 798 798.0 Q98:801 Type1 Active DFGin 5.136 12.054 BLAminus -130.43, 175.42 66.1, 93.37 -104.47, 26.06 315.68, 130.09 -58.56, -40.67 in-in in 9.082 Saltbr-in 2.794 HRD-na-N -73.99, -49.28 75.88, 2.33 in-in-na SNCiia in-na ActLoopNT-in 2.831 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.38, 14.19 APE9-dihe-na -67.33, 158.61 APE8-dihe-na -154.66, -177.03 APE8-rot-na 74.44 APE67-dihe-na -159.78, 146.47 89.13, -0.56 APE12-dist-na 9.712 APE11-dist-na 13.618 APE10-dist-na 17.166 APE9-dist-na 12.987 None None None XRAY 2.0 0.201 0.24 A 357 328 0 0 0 0 [[484, 797]] 1.0 6z59 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z5DA 470 798 798.0 Q8Q:805 Type1 Active DFGin 5.053 12.308 BLAminus -128.1, 170.45 73.65, 93.08 -105.2, 21.18 315.55, 125.26 -62.8, -29.15 in-in in 9.073 Saltbr-in 2.688 HRD-na-N -71.9, -46.78 72.06, -1.5 in-in-na SNCiia in-na ActLoopNT-in 2.861 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.04, 23.91 APE9-dihe-na -77.44, 160.96 APE8-dihe-na -149.27, 168.07 APE8-rot-na 78.22 APE67-dihe-na -158.56, 145.68 94.91, -2.03 APE12-dist-na 9.558 APE11-dist-na 13.567 APE10-dist-na 17.139 APE9-dist-na 13.019 None None None XRAY 1.75 0.154 0.178 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z5d OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z5EA 471 798 798.0 Q8K:806 Type1 Active DFGin 5.08 12.459 BLAminus -128.44, 172.31 71.81, 90.69 -103.13, 26.31 316.73, 125.57 -64.15, -28.51 in-in in 9.143 Saltbr-in 2.729 HRD-na-N -68.18, -49.54 73.75, 2.15 in-in-na SNCiia in-na ActLoopNT-in 2.888 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.8, 21.0 APE9-dihe-na -73.94, 160.68 APE8-dihe-na -150.44, 166.42 APE8-rot-na 75.48 APE67-dihe-na -157.25, 143.6 92.62, -2.15 APE12-dist-na 9.572 APE11-dist-na 13.485 APE10-dist-na 17.146 APE9-dist-na 12.936 None None None XRAY 1.5 0.159 0.183 A 357 328 0 0 0 0 [[484, 797]] 1.0 6z5e OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
7AVQA 471 798 798.0 S1Z:801 Type1 Active DFGin 5.149 12.146 BLAminus -126.06, 173.12 69.03, 91.95 -102.42, 24.12 320.3, 125.97 -52.79, -41.95 in-in in 8.998 Saltbr-in 2.659 HRD-na-N -75.14, -46.38 71.99, 2.8 in-in-na SNCiia in-na ActLoopNT-in 2.891 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.18, 22.84 APE9-dihe-na -73.32, 160.09 APE8-dihe-na -148.12, 160.7 APE8-rot-na 195.64 APE67-dihe-na -157.46, 142.25 95.7, -0.72 APE12-dist-na 9.574 APE11-dist-na 13.487 APE10-dist-na 17.118 APE9-dist-na 12.952 None None None XRAY 1.65 0.16 0.179 A 357 328 0 0 0 0 [[484, 797]] 1.0 7avq OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
7OPSA 471 798 798.0 07C:801 Type1 Active DFGin 4.955 12.409 BLAminus -120.84, 168.72 74.52, 94.25 -110.46, 32.79 314.75, 129.03 -72.39, -27.54 in-in in 9.209 Saltbr-in 2.891 HRD-na-N -67.82, -53.79 76.87, 1.09 in-in-na SNCiia in-na ActLoopNT-in 2.935 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.38, 10.26 APE9-dihe-na -73.55, 156.67 APE8-dihe-na -147.73, 179.58 APE8-rot-na 67.78 APE67-dihe-na -167.67, 141.52 97.91, 1.48 APE12-dist-na 9.463 APE11-dist-na 13.499 APE10-dist-na 16.964 APE9-dist-na 13.035 None None None XRAY 2.38 0.179 0.229 A 357 328 0 0 0 0 [[484, 797]] 1.0 7ops OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
8RDKA 471 798 798.0 YQT:803 Type1 Active DFGin 5.304 12.291 BLAminus -126.79, 170.58 68.55, 97.1 -105.65, 24.46 315.14, 130.76 -63.91, -28.61 in-in in 8.949 Saltbr-in 2.684 HRD-na-N -70.8, -52.97 75.33, 1.85 in-in-na SNCiia in-na ActLoopNT-in 2.843 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.88, 25.66 APE9-dihe-na -78.67, 156.59 APE8-dihe-na -150.7, 178.52 APE8-rot-na 74.04 APE67-dihe-na -162.89, 139.09 96.18, -5.83 APE12-dist-na 9.438 APE11-dist-na 13.401 APE10-dist-na 17.106 APE9-dist-na 12.963 None None None XRAY 2.0 0.199 0.233 A 357 328 0 0 0 0 [[484, 797]] 1.0 8rdk OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9FLBA 471 798 798.0 A1IDB:802 Type1 Active DFGin 5.017 12.499 BLAminus -122.75, 164.93 78.09, 95.44 -111.48, 32.7 311.33, 133.52 -69.25, -37.29 in-in in 8.846 Saltbr-in 2.663 HRD-na-N -65.06, -57.81 86.13, 3.33 in-in-na SNCiia in-na ActLoopNT-in 2.883 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -97.12, -24.47 APE9-dihe-na -48.97, 165.86 APE8-dihe-na -171.41, -171.26 APE8-rot-na 65.27 APE67-dihe-na -131.18, 150.53 102.5, -31.2 APE12-dist-na 9.656 APE11-dist-na 13.445 APE10-dist-na 16.901 APE9-dist-na 13.075 None None None XRAY 2.5 0.195 0.245 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flb OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9FLQA 471 798 798.0 A1IDD:806 Type1 Active DFGin 5.277 11.995 BLAminus -131.52, 170.51 72.45, 91.56 -104.74, 27.71 313.77, 132.43 -58.36, -40.16 in-in in 9.194 Saltbr-in 2.385 HRD-na-N -72.62, -50.16 74.03, 2.04 in-in-na SNCiia in-na ActLoopNT-in 2.89 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -123.97, 17.68 APE9-dihe-na -77.54, 163.56 APE8-dihe-na -154.04, 168.58 APE8-rot-na 56.93 APE67-dihe-na -156.8, 141.47 98.45, -3.96 APE12-dist-na 9.579 APE11-dist-na 13.504 APE10-dist-na 17.048 APE9-dist-na 13.042 None None None XRAY 1.85 0.176 0.202 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flq OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9FLRA 471 798 798.0 A1IDE:803 Type1 Active DFGin 5.257 11.905 BLAminus -132.45, 173.37 67.71, 90.56 -101.27, 25.05 315.0, 128.67 -53.75, -42.86 in-in in 9.406 Saltbr-in 2.535 HRD-na-N -70.9, -52.21 71.26, 4.74 in-in-na SNCiia in-na ActLoopNT-in 2.852 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.29, 14.34 APE9-dihe-na -78.07, 164.28 APE8-dihe-na -157.67, 170.99 APE8-rot-na 58.59 APE67-dihe-na -164.88, 135.66 97.12, 4.81 APE12-dist-na 9.597 APE11-dist-na 13.566 APE10-dist-na 17.045 APE9-dist-na 13.109 None None None XRAY 1.91 0.173 0.209 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flr OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
7SQMA 453 798 798.0 A5G:801 Type1 Active DFGin 5.294 12.385 BLAminus -126.59, 168.89 78.77, 90.66 -103.22, 31.48 318.95, 126.98 -62.97, -29.65 in-in in 9.033 Saltbr-in 2.862 HRD-na-N -74.3, -49.72 73.45, 2.57 in-in-na SNCiia in-na ActLoopNT-in 2.956 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.03, 13.48 APE9-dihe-na -73.56, 163.48 APE8-dihe-na -150.66, 160.36 APE8-rot-na 211.61 APE67-dihe-na -164.54, 145.89 99.66, 4.4 APE12-dist-na 9.225 APE11-dist-na 13.189 APE10-dist-na 16.762 APE9-dist-na 12.944 None None None XRAY 1.78 0.175 0.205 A 357 346 0 0 0 0 [[484, 797]] 1.0 7sqm OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9FLCA 471 798 798.0 A1IDA:801 Type1.5_Back Active DFGin 4.715 12.46 BLAminus -134.34, 171.12 67.31, 104.11 -111.35, 24.44 309.33, 129.38 -43.69, -56.59 in-in in 9.127 Saltbr-in 2.572 HRD-na-N -70.37, -50.71 74.43, 4.41 in-in-na SNCiia in-na ActLoopNT-in 2.846 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -124.8, 13.59 APE9-dihe-na -68.86, 164.74 APE8-dihe-na -159.81, 175.83 APE8-rot-na 49.95 APE67-dihe-na -162.39, 140.7 102.66, -4.36 APE12-dist-na 9.337 APE11-dist-na 13.24 APE10-dist-na 16.865 APE9-dist-na 12.997 None None None XRAY 2.18 0.166 0.197 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flc OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9B2SK 470 798 798.0 No_ligand No_ligand Inactive DFGin 6.064 12.671 BLAminus -142.15, 178.43 60.64, 69.74 -94.32, 35.13 330.57, 110.31 -71.54, -20.41 out-out out 10.509 Saltbr-out 8.91 HRD-na-N -103.48, -39.3 72.01, 16.12 out-in-na SNCoia in-na ActLoopNT-in 2.662 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -93.15, 4.32 APE9-dihe-na -71.11, 161.22 APE8-dihe-na -159.47, 164.4 APE8-rot-na 76.0 APE67-dihe-na -157.32, 146.25 103.48, -10.17 APE12-dist-na 10.384 APE11-dist-na 14.356 APE10-dist-na 17.698 APE9-dist-na 13.728 None None None EM 3.01 999.0 999.0 K 357 329 0 0 0 0 [[484, 797]] 1.0 9b2s OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9B2UK 470 798 798.0 No_ligand No_ligand Inactive DFGin 5.926 12.627 BLAminus -136.69, -178.38 59.48, 67.33 -92.11, 31.61 333.66, 107.16 -67.05, -16.22 out-out out 10.457 Saltbr-out 8.398 HRD-na-N -100.22, -40.69 78.07, 2.57 out-in-na SNCoia in-na ActLoopNT-in 2.756 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -100.28, 9.24 APE9-dihe-na -71.6, 162.97 APE8-dihe-na -157.23, 160.72 APE8-rot-na 81.21 APE67-dihe-na -151.55, 148.6 98.32, -9.69 APE12-dist-na 10.577 APE11-dist-na 14.628 APE10-dist-na 17.968 APE9-dist-na 13.833 None None None EM 3.64 999.0 999.0 K 357 329 0 0 0 0 [[484, 797]] 1.0 9b2u OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z5CA 470 798 798.0 PQ5:805 Type1 Inactive DFGin 4.731 13.108 BLAminus -133.84, 170.31 75.72, 94.52 -110.21, 19.19 311.37, 116.86 -61.87, -31.19 out-out out 10.462 Saltbr-out 3.7 HRD-na-N -70.06, -50.84 74.01, -0.31 out-in-na SNCoia in-na ActLoopNT-in 2.931 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.88, 20.45 APE9-dihe-na -80.43, 159.13 APE8-dihe-na -144.39, 165.92 APE8-rot-na 214.89 APE67-dihe-na -162.19, 147.1 97.48, -3.07 APE12-dist-na 9.488 APE11-dist-na 13.52 APE10-dist-na 17.05 APE9-dist-na 13.1 None None None XRAY 1.75 0.16 0.188 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z5c OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9FLOA 466 797 798.0 A1IDC:802 Type1 Inactive DFGin 5.355 12.318 BLAminus -140.34, 174.89 75.76, 76.52 -89.13, 31.66 305.79, 159.49 -77.78, -25.85 in-out in 9.084 Saltbr-out 3.76 HRD-na-N -85.47, -46.33 68.95, 25.87 out-in-na SNCoia in-na ActLoopNT-in 2.616 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.51, 102.44 APE9-dihe-na 136.93, 133.28 APE8-dihe-na -151.7, -143.81 APE8-rot-na 72.42 APE67-dihe-na -90.21, 160.33 109.28, -71.54 APE12-dist-na 9.638 APE11-dist-na 13.586 APE10-dist-na 17.18 APE9-dist-na 14.433 None None None XRAY 2.9 0.214 0.247 A 357 332 0 0 0 0 [[484, 797]] 1.0 9flo OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6G3AA 471 798 798.0 5ID:805 Type1 Inactive DFGin 4.953 12.443 BLAminus -127.41, 171.94 74.51, 93.23 -106.28, 26.81 312.44, 123.45 -60.95, -29.67 in-out in 9.904 Saltbr-out 4.42 HRD-na-N -72.27, -48.82 73.62, 1.17 out-in-na SNCoia in-na ActLoopNT-in 2.883 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.57, 14.66 APE9-dihe-na -70.85, 159.17 APE8-dihe-na -152.35, 172.74 APE8-rot-na 72.92 APE67-dihe-na -156.95, 142.2 92.44, -2.34 APE12-dist-na 9.454 APE11-dist-na 13.382 APE10-dist-na 16.931 APE9-dist-na 12.993 F605T None None XRAY 1.43 0.151 0.175 A 357 328 0 0 0 0 [[484, 797]] 1.0 6g3a OTHER_HASPIN_HUMAN HASP 1.8e-225 752.9 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z56A 470 798 798.0 Q7Q:801 Type1.5_Back Inactive DFGin 4.602 12.569 BLAminus -129.58, 171.28 69.16, 102.48 -109.85, 26.06 309.6, 123.99 -45.33, -46.61 out-out out 10.104 Saltbr-out 4.52 HRD-na-N -69.89, -50.01 74.0, -0.03 out-in-na SNCoia in-na ActLoopNT-in 2.821 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -120.86, 18.07 APE9-dihe-na -73.34, 162.1 APE8-dihe-na -143.73, 169.15 APE8-rot-na 201.43 APE67-dihe-na -162.09, 141.44 91.95, 4.24 APE12-dist-na 9.424 APE11-dist-na 13.25 APE10-dist-na 17.008 APE9-dist-na 13.071 None None None XRAY 1.9 0.178 0.221 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z56 OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z5BA 469 798 798.0 Q7Z:803 Type1.5_Back Inactive DFGin 4.548 12.709 BLAminus -135.9, 170.26 70.64, 101.28 -110.64, 25.44 308.83, 121.13 -45.93, -45.39 out-out out 10.049 Saltbr-out 4.556 HRD-na-N -70.65, -51.98 77.17, -0.49 out-in-na SNCoia in-na ActLoopNT-in 2.906 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -114.59, 17.24 APE9-dihe-na -73.9, 162.49 APE8-dihe-na -150.9, 168.36 APE8-rot-na 77.43 APE67-dihe-na -163.72, 140.01 97.4, -1.55 APE12-dist-na 9.36 APE11-dist-na 13.278 APE10-dist-na 16.905 APE9-dist-na 12.945 None None None XRAY 1.9 0.157 0.198 A 357 330 0 0 0 0 [[484, 797]] 1.0 6z5b OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
6Z5AA 465 798 798.0 Q8B:60807 Type1.5_Front Inactive DFGin 4.746 13.158 BLAminus -130.52, 170.23 77.78, 97.19 -110.55, 22.86 309.49, 126.33 -50.19, -42.61 out-out out 10.928 Saltbr-out 6.049 HRD-na-N -69.87, -51.48 73.76, 2.92 out-in-na SNCoia in-na ActLoopNT-in 2.957 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -114.05, 16.57 APE9-dihe-na -70.55, 162.23 APE8-dihe-na -152.03, 159.2 APE8-rot-na 218.93 APE67-dihe-na -157.88, 144.9 96.43, 3.83 APE12-dist-na 9.408 APE11-dist-na 13.313 APE10-dist-na 16.953 APE9-dist-na 12.968 None None None XRAY 1.55 0.157 0.182 A 357 334 0 0 0 0 [[484, 797]] 1.0 6z5a OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
9B2TK 470 798 798.0 No_ligand No_ligand Inactive DFGin 10.473 16.998 None -74.01, 167.84 -68.22, 151.89 -112.4, 131.65 323.3, 85.18 -72.17, -31.47 out-out out 10.371 Saltbr-out 8.739 HRD-na-N -90.05, -46.55 60.89, 17.99 out-in-na SNCoia in-na ActLoopNT-in 2.509 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -99.75, 7.12 APE9-dihe-na -76.13, 178.32 APE8-dihe-na -157.85, 172.7 APE8-rot-na 78.9 APE67-dihe-na -161.94, 175.92 118.79, -26.14 APE12-dist-na 11.19 APE11-dist-na 13.535 APE10-dist-na 18.064 APE9-dist-na 14.027 None None None EM 2.99 999.0 999.0 K 357 329 0 0 0 0 [[484, 797]] 1.0 9b2t OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin

OTHER_HASPIN (Serine/threonine-protein kinase haspin)

Total number of chains: 42
Active chains: 33
Family: OTHER
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 41 97.6% AF-Q8TF76-K1A
DFGin None 1 2.4% 9B2TK

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
HASP_HUMAN 3DLZA Q8TF76 470 798 798.0 AMP:902 ATPlike Active DFGin 5.254 12.469 BLAminus -120.14, 174.05 73.32, 91.07 -105.92, 29.14 315.79, 130.04 -57.27, -36.15 in-in in 9.264 Saltbr-in 2.695 HRD-na-N -71.0, -49.07 68.99, 3.03 in-in-na SNCiia in-na ActLoopNT-in 2.821 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -122.28, 17.39 APE9-dihe-na -67.57, 157.85 APE8-dihe-na -149.51, 177.99 APE8-rot-na 58.52 APE67-dihe-na -159.03, 144.74 95.06, -6.22 APE12-dist-na 9.493 APE11-dist-na 13.466 APE10-dist-na 17.05 APE9-dist-na 12.819 None None None XRAY 1.85 0.167 0.216 A 357 329 0 0 0 0 [[484, 797]] 1.0 3dlz Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN AF-Q8TF76-K1A Q8TF76 476 798 798.0 No_ligand No_ligand Active DFGin 4.997 12.374 BLAminus -138.62, 174.68 57.97, 91.28 -100.94, 21.93 314.77, 120.9 -55.94, -45.23 in-in in 9.18 Saltbr-in 2.711 HRD-na-N -75.36, -43.16 61.41, 5.31 in-in-na SNCiia in-na ActLoopNT-in 2.839 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -93.17, -12.71 APE9-dihe-na -54.03, 150.53 APE8-dihe-na -147.69, 169.0 APE8-rot-na 193.38 APE67-dihe-na -135.11, 149.27 98.64, -16.5 APE12-dist-na 9.305 APE11-dist-na 13.309 APE10-dist-na 16.98 APE9-dist-na 12.992 None None None AF2 -1.0 1.0 1.0 A 323 323 0 0 0 0 [[484, 797]] 1.0 AF-Q8TF76-K1 Homo sapiens OTHER_HASPIN_HUMAN HASP 9.2e-227 757.1 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN AF-Q8TF76-K3A Q8TF76 476 798 798.0 No_ligand No_ligand Active DFGin 4.951 12.431 BLAminus -133.71, 176.01 54.85, 96.46 -104.75, 21.31 315.54, 124.63 -56.24, -41.59 in-in in 9.299 Saltbr-in 2.719 HRD-na-N -75.19, -42.52 61.0, 1.07 in-in-na SNCiia in-na ActLoopNT-in 2.885 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -93.31, -18.43 APE9-dihe-na -56.71, 155.17 APE8-dihe-na -141.59, -175.7 APE8-rot-na 73.98 APE67-dihe-na -125.54, 149.77 84.64, -25.13 APE12-dist-na 9.207 APE11-dist-na 13.228 APE10-dist-na 16.926 APE9-dist-na 13.133 None None None AF2 -1.0 1.0 1.0 A 323 323 0 0 0 0 [[484, 797]] 1.0 AF-Q8TF76-K3 Homo sapiens OTHER_HASPIN_HUMAN HASP 9.2e-227 757.1 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 2WB8A Q8TF76 447 798 798.0 No_ligand No_ligand Active DFGin 5.22 12.191 BLAminus -120.69, 176.87 68.15, 91.75 -104.26, 25.9 315.71, 126.12 -56.01, -32.87 in-in in 9.095 Saltbr-in 2.281 HRD-na-N -69.54, -53.11 72.35, 6.09 in-in-na SNCiia in-na ActLoopNT-in 2.857 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -129.5, 34.17 APE9-dihe-na -83.79, 164.98 APE8-dihe-na -149.79, 174.65 APE8-rot-na 31.25 APE67-dihe-na -168.04, 143.08 80.64, 14.62 APE12-dist-na 9.206 APE11-dist-na 12.948 APE10-dist-na 16.727 APE9-dist-na 12.724 None None None XRAY 2.15 0.23 0.267 A 352 351 1 0 0 0 [[484, 797]] 1.0 2wb8 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.3e-226 756.7 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 5HTBA Q8TF76 471 798 798.0 No_ligand No_ligand Active DFGin 4.886 12.713 BLAminus -127.82, 172.38 75.8, 95.98 -111.9, 24.65 313.35, 119.25 -57.64, -36.0 in-in in 9.095 Saltbr-in 2.722 HRD-na-N -72.45, -46.3 70.77, -0.27 in-in-na SNCiia in-na ActLoopNT-in 2.859 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.52, 17.28 APE9-dihe-na -71.3, 162.17 APE8-dihe-na -148.2, 163.96 APE8-rot-na 208.0 APE67-dihe-na -159.11, 139.67 91.05, 1.41 APE12-dist-na 9.417 APE11-dist-na 13.298 APE10-dist-na 16.873 APE9-dist-na 12.933 None None None XRAY 1.7 0.163 0.181 A 357 328 0 0 0 0 [[484, 797]] 1.0 5htb Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 5HTCA Q8TF76 471 798 798.0 No_ligand No_ligand Active DFGin 5.008 12.77 BLAminus -124.68, 170.56 74.88, 95.44 -108.39, 22.99 316.66, 123.43 -55.96, -37.72 in-in in 9.222 Saltbr-in 2.671 HRD-na-N -71.81, -49.47 73.17, 0.66 in-in-na SNCiia in-na ActLoopNT-in 2.875 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.86, 18.07 APE9-dihe-na -74.58, 161.83 APE8-dihe-na -153.14, 168.43 APE8-rot-na 79.76 APE67-dihe-na -159.07, 137.97 97.79, -1.9 APE12-dist-na 9.518 APE11-dist-na 13.376 APE10-dist-na 16.983 APE9-dist-na 12.965 None None None XRAY 1.5 0.151 0.171 A 357 328 0 0 0 0 [[484, 797]] 1.0 5htc Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6G39A Q8TF76 471 798 798.0 5ID:802 Type1 Active DFGin 5.021 12.32 BLAminus -127.21, 173.16 74.1, 91.77 -104.6, 25.15 318.27, 124.04 -54.52, -37.44 in-in in 9.223 Saltbr-in 2.607 HRD-na-N -72.86, -48.93 72.97, 0.92 in-in-na SNCiia in-na ActLoopNT-in 2.865 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.61, 13.68 APE9-dihe-na -74.05, 162.55 APE8-dihe-na -147.53, 161.22 APE8-rot-na 206.35 APE67-dihe-na -163.09, 139.78 96.44, 2.71 APE12-dist-na 9.496 APE11-dist-na 13.491 APE10-dist-na 16.919 APE9-dist-na 13.026 F605Y None None XRAY 1.45 0.159 0.175 A 357 328 0 0 0 0 [[484, 797]] 1.0 6g39 Homo sapiens OTHER_HASPIN_HUMAN HASP 3.9e-226 755.1 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 2VUWA Q8TF76 470 798 798.0 5ID:1800 Type1 Active DFGin 4.977 12.344 BLAminus -126.7, 172.42 73.13, 94.6 -106.22, 25.34 317.03, 123.17 -59.06, -30.58 in-in in 9.293 Saltbr-in 2.791 HRD-na-N -69.06, -49.8 71.93, -0.86 in-in-na SNCiia in-na ActLoopNT-in 2.886 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.41, 21.25 APE9-dihe-na -74.65, 162.69 APE8-dihe-na -150.22, 164.21 APE8-rot-na 197.92 APE67-dihe-na -163.26, 143.62 93.5, 5.23 APE12-dist-na 9.51 APE11-dist-na 13.492 APE10-dist-na 17.046 APE9-dist-na 12.946 None None MSE615,MSE706,MSE725,MSE752,MSE756,MSE767,MSE781 XRAY 1.8 0.148 0.169 A 336 329 0 0 0 0 [[484, 797]] 1.0 2vuw Homo sapiens OTHER_HASPIN_HUMAN HASP 1.1e-226 756.9 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9FLTA Q8TF76 471 798 798.0 A1IDF:801 Type1 Active DFGin 5.178 12.218 BLAminus -141.02, 178.95 59.99, 70.73 -81.95, 27.03 316.78, 141.24 -69.29, -28.67 in-in in 8.759 Saltbr-in 2.463 HRD-na-N -66.6, -53.16 75.71, 6.9 in-in-na SNCiia in-na ActLoopNT-in 2.905 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -131.58, 41.34 APE9-dihe-na -102.69, 164.5 APE8-dihe-na -162.68, -171.46 APE8-rot-na 41.52 APE67-dihe-na -134.91, 146.64 100.36, -24.97 APE12-dist-na 9.64 APE11-dist-na 13.509 APE10-dist-na 17.247 APE9-dist-na 13.279 None None None XRAY 2.4 0.187 0.239 A 336 320 8 0 0 0 [[484, 797]] 1.0 9flt Homo sapiens OTHER_HASPIN_HUMAN HASP 1.1e-226 756.9 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 3E7VA Q8TF76 471 798 798.0 DZO:1 Type1 Active DFGin 5.227 12.203 BLAminus -130.14, 169.21 72.6, 84.89 -101.25, 35.48 316.82, 123.9 -62.16, -34.97 in-in in 9.014 Saltbr-in 2.481 HRD-na-N -68.11, -48.56 71.09, -0.57 in-in-na SNCiia in-na ActLoopNT-in 2.917 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -113.43, 18.49 APE9-dihe-na -73.97, 165.86 APE8-dihe-na -158.09, 152.51 APE8-rot-na 206.55 APE67-dihe-na -159.89, 140.52 100.1, 0.81 APE12-dist-na 9.459 APE11-dist-na 13.36 APE10-dist-na 17.023 APE9-dist-na 12.905 None None None XRAY 2.0 0.17 0.225 A 357 328 0 0 0 0 [[484, 797]] 1.0 3e7v Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 3F2NA Q8TF76 471 798 798.0 IZZ:800 Type1 Active DFGin 5.227 12.509 BLAminus -132.35, 169.14 74.56, 87.66 -98.09, 25.18 316.3, 125.75 -57.05, -34.51 in-in in 8.729 Saltbr-in 2.737 HRD-na-N -71.51, -49.79 70.28, -0.25 in-in-na SNCiia in-na ActLoopNT-in 2.913 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -120.07, 21.25 APE9-dihe-na -75.2, 162.89 APE8-dihe-na -156.01, 176.32 APE8-rot-na 74.11 APE67-dihe-na -157.24, 143.14 98.22, -8.69 APE12-dist-na 9.565 APE11-dist-na 13.531 APE10-dist-na 17.149 APE9-dist-na 12.969 None None None XRAY 1.8 0.162 0.186 A 357 328 0 0 0 0 [[484, 797]] 1.0 3f2n Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 3FMDA Q8TF76 470 798 798.0 IQB:1 Type1 Active DFGin 4.817 12.737 BLAminus -134.95, 173.12 69.12, 93.36 -108.33, 23.11 309.03, 122.86 -58.61, -32.84 in-in in 9.417 Saltbr-in 2.578 HRD-na-N -64.91, -44.59 67.0, -1.51 in-in-na SNCiia in-na ActLoopNT-in 2.86 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -126.4, 30.5 APE9-dihe-na -82.22, 168.97 APE8-dihe-na -156.73, 170.22 APE8-rot-na 87.7 APE67-dihe-na -158.09, 144.39 88.76, -6.79 APE12-dist-na 9.533 APE11-dist-na 13.423 APE10-dist-na 17.115 APE9-dist-na 13.017 None None None XRAY 2.0 0.226 0.283 A 357 329 0 0 0 0 [[484, 797]] 1.0 3fmd Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 3IQ7A Q8TF76 471 798 798.0 5ID:799 Type1 Active DFGin 5.002 12.525 BLAminus -130.14, 168.59 78.5, 93.8 -107.03, 26.88 317.14, 123.36 -63.63, -28.13 in-in in 9.288 Saltbr-in 2.716 HRD-na-N -69.08, -54.14 69.34, 3.59 in-in-na SNCiia in-na ActLoopNT-in 2.842 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -119.96, 19.66 APE9-dihe-na -73.26, 163.53 APE8-dihe-na -151.13, 165.69 APE8-rot-na 217.79 APE67-dihe-na -160.55, 141.37 91.74, 4.08 APE12-dist-na 9.31 APE11-dist-na 13.171 APE10-dist-na 16.954 APE9-dist-na 12.798 None None None XRAY 2.0 0.174 0.207 A 357 328 0 0 0 0 [[484, 797]] 1.0 3iq7 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 4OUCA Q8TF76 470 798 798.0 5ID:60808 Type1 Active DFGin 5.142 12.398 BLAminus -123.14, 171.36 70.83, 89.85 -103.14, 24.75 317.85, 126.13 -50.7, -43.23 in-in in 9.227 Saltbr-in 2.635 HRD-na-N -73.5, -49.82 73.73, 4.15 in-in-na SNCiia in-na ActLoopNT-in 2.897 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.93, 10.97 APE9-dihe-na -70.72, 155.25 APE8-dihe-na -144.93, 165.92 APE8-rot-na 81.62 APE67-dihe-na -154.34, 142.15 101.34, -0.24 APE12-dist-na 9.521 APE11-dist-na 13.627 APE10-dist-na 17.119 APE9-dist-na 12.997 None None None XRAY 1.9 0.166 0.211 A 357 329 0 0 0 0 [[484, 797]] 1.0 4ouc Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 4QTCA Q8TF76 469 798 798.0 38Z:804 Type1 Active DFGin 4.743 12.697 BLAminus -128.25, 174.11 72.8, 94.29 -100.86, 22.55 311.48, 126.56 -49.88, -46.32 in-in in 9.244 Saltbr-in 2.767 HRD-na-N -70.64, -49.71 73.49, 0.07 in-in-na SNCiia in-na ActLoopNT-in 2.862 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.14, 15.58 APE9-dihe-na -74.4, 166.34 APE8-dihe-na -155.61, 167.98 APE8-rot-na 54.8 APE67-dihe-na -159.6, 141.49 96.89, -1.32 APE12-dist-na 9.4 APE11-dist-na 13.293 APE10-dist-na 16.89 APE9-dist-na 13.142 None None None XRAY 1.4 0.15 0.164 A 357 330 0 0 0 0 [[484, 797]] 1.0 4qtc Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6G34A Q8TF76 472 798 798.0 5ID:60401 Type1 Active DFGin 4.991 12.367 BLAminus -127.35, 171.15 74.89, 93.11 -104.99, 26.96 316.16, 126.1 -57.37, -32.12 in-in in 9.292 Saltbr-in 2.721 HRD-na-N -71.53, -47.32 70.63, -2.3 in-in-na SNCiia in-na ActLoopNT-in 2.893 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.68, 18.32 APE9-dihe-na -70.1, 157.86 APE8-dihe-na -146.1, 158.98 APE8-rot-na 202.21 APE67-dihe-na -162.15, 141.91 96.58, 0.13 APE12-dist-na 9.436 APE11-dist-na 13.462 APE10-dist-na 16.952 APE9-dist-na 12.837 None None None XRAY 1.76 0.14 0.174 A 357 327 0 0 0 0 [[484, 797]] 1.0 6g34 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6G35A Q8TF76 465 798 798.0 EKK:60802 Type1 Active DFGin 5.005 12.39 BLAminus -126.0, 169.52 78.13, 90.25 -104.66, 24.26 315.74, 125.01 -60.88, -28.25 in-in in 9.306 Saltbr-in 2.713 HRD-na-N -70.57, -49.54 72.42, 1.39 in-in-na SNCiia in-na ActLoopNT-in 2.901 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.32, 17.8 APE9-dihe-na -73.2, 161.57 APE8-dihe-na -146.96, 162.71 APE8-rot-na 196.59 APE67-dihe-na -162.63, 137.82 97.88, 1.51 APE12-dist-na 9.478 APE11-dist-na 13.461 APE10-dist-na 17.008 APE9-dist-na 13.016 None None None XRAY 1.55 0.161 0.183 A 357 334 0 0 0 0 [[484, 797]] 1.0 6g35 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6G36A Q8TF76 465 798 798.0 EKH:60401 Type1 Active DFGin 4.952 12.328 BLAminus -126.44, 170.29 76.27, 92.19 -105.23, 26.61 316.28, 124.1 -57.25, -32.63 in-in in 9.282 Saltbr-in 2.744 HRD-na-N -71.83, -48.64 74.84, -0.58 in-in-na SNCiia in-na ActLoopNT-in 2.89 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.55, 15.17 APE9-dihe-na -70.08, 160.85 APE8-dihe-na -149.64, 167.11 APE8-rot-na 67.1 APE67-dihe-na -162.45, 137.7 92.15, 4.46 APE12-dist-na 9.491 APE11-dist-na 13.449 APE10-dist-na 17.015 APE9-dist-na 12.972 None None None XRAY 1.46 0.151 0.176 A 357 334 0 0 0 0 [[484, 797]] 1.0 6g36 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6G37A Q8TF76 472 798 798.0 FTU:801 Type1 Active DFGin 5.035 12.401 BLAminus -125.49, 171.67 75.49, 90.88 -104.56, 25.99 317.99, 122.48 -54.51, -35.12 in-in in 9.318 Saltbr-in 2.736 HRD-na-N -70.97, -50.1 72.78, 2.06 in-in-na SNCiia in-na ActLoopNT-in 2.889 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -114.17, 14.96 APE9-dihe-na -72.53, 161.37 APE8-dihe-na -147.52, 165.41 APE8-rot-na 216.83 APE67-dihe-na -159.62, 143.17 92.11, 0.24 APE12-dist-na 9.422 APE11-dist-na 13.433 APE10-dist-na 16.884 APE9-dist-na 12.914 None None None XRAY 1.48 0.149 0.167 A 357 327 0 0 0 0 [[484, 797]] 1.0 6g37 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6G38A Q8TF76 472 798 798.0 TBN:800 Type1 Active DFGin 5.155 12.468 BLAminus -124.6, 171.17 73.49, 90.96 -102.58, 23.98 318.22, 128.64 -60.91, -27.39 in-in in 9.286 Saltbr-in 2.681 HRD-na-N -70.12, -48.6 70.78, 0.07 in-in-na SNCiia in-na ActLoopNT-in 2.865 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.63, 17.26 APE9-dihe-na -74.94, 161.54 APE8-dihe-na -150.43, 171.99 APE8-rot-na 81.52 APE67-dihe-na -161.74, 140.31 94.52, 1.17 APE12-dist-na 9.54 APE11-dist-na 13.547 APE10-dist-na 17.024 APE9-dist-na 13.008 None None None XRAY 1.47 0.144 0.165 A 357 327 0 0 0 0 [[484, 797]] 1.0 6g38 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z57A Q8TF76 470 798 798.0 Q8W:801 Type1 Active DFGin 5.108 12.544 BLAminus -128.55, 170.14 70.49, 89.65 -99.72, 23.55 319.85, 122.5 -60.24, -32.24 in-in in 9.047 Saltbr-in 2.63 HRD-na-N -69.51, -48.64 73.21, 1.64 in-in-na SNCiia in-na ActLoopNT-in 2.906 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.13, 24.13 APE9-dihe-na -80.04, 165.59 APE8-dihe-na -154.67, 168.36 APE8-rot-na 59.7 APE67-dihe-na -158.19, 141.65 89.15, 3.9 APE12-dist-na 9.623 APE11-dist-na 13.634 APE10-dist-na 17.184 APE9-dist-na 13.001 None None None XRAY 1.5 0.164 0.188 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z57 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z58A Q8TF76 470 798 798.0 Q9B:801 Type1 Active DFGin 5.29 11.882 BLAminus -131.62, 178.98 63.69, 89.83 -101.06, 25.15 318.41, 128.59 -53.25, -41.36 in-in in 8.999 Saltbr-in 2.668 HRD-na-N -74.24, -49.55 73.51, 2.01 in-in-na SNCiia in-na ActLoopNT-in 2.86 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.26, 20.54 APE9-dihe-na -78.55, 163.28 APE8-dihe-na -149.94, 172.24 APE8-rot-na 51.88 APE67-dihe-na -158.7, 145.23 97.38, -8.51 APE12-dist-na 9.654 APE11-dist-na 13.592 APE10-dist-na 17.186 APE9-dist-na 13.103 None None None XRAY 1.8 0.164 0.19 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z58 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z59A Q8TF76 471 798 798.0 Q98:801 Type1 Active DFGin 5.136 12.054 BLAminus -130.43, 175.42 66.1, 93.37 -104.47, 26.06 315.68, 130.09 -58.56, -40.67 in-in in 9.082 Saltbr-in 2.794 HRD-na-N -73.99, -49.28 75.88, 2.33 in-in-na SNCiia in-na ActLoopNT-in 2.831 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.38, 14.19 APE9-dihe-na -67.33, 158.61 APE8-dihe-na -154.66, -177.03 APE8-rot-na 74.44 APE67-dihe-na -159.78, 146.47 89.13, -0.56 APE12-dist-na 9.712 APE11-dist-na 13.618 APE10-dist-na 17.166 APE9-dist-na 12.987 None None None XRAY 2.0 0.201 0.24 A 357 328 0 0 0 0 [[484, 797]] 1.0 6z59 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z5DA Q8TF76 470 798 798.0 Q8Q:805 Type1 Active DFGin 5.053 12.308 BLAminus -128.1, 170.45 73.65, 93.08 -105.2, 21.18 315.55, 125.26 -62.8, -29.15 in-in in 9.073 Saltbr-in 2.688 HRD-na-N -71.9, -46.78 72.06, -1.5 in-in-na SNCiia in-na ActLoopNT-in 2.861 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.04, 23.91 APE9-dihe-na -77.44, 160.96 APE8-dihe-na -149.27, 168.07 APE8-rot-na 78.22 APE67-dihe-na -158.56, 145.68 94.91, -2.03 APE12-dist-na 9.558 APE11-dist-na 13.567 APE10-dist-na 17.139 APE9-dist-na 13.019 None None None XRAY 1.75 0.154 0.178 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z5d Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z5EA Q8TF76 471 798 798.0 Q8K:806 Type1 Active DFGin 5.08 12.459 BLAminus -128.44, 172.31 71.81, 90.69 -103.13, 26.31 316.73, 125.57 -64.15, -28.51 in-in in 9.143 Saltbr-in 2.729 HRD-na-N -68.18, -49.54 73.75, 2.15 in-in-na SNCiia in-na ActLoopNT-in 2.888 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.8, 21.0 APE9-dihe-na -73.94, 160.68 APE8-dihe-na -150.44, 166.42 APE8-rot-na 75.48 APE67-dihe-na -157.25, 143.6 92.62, -2.15 APE12-dist-na 9.572 APE11-dist-na 13.485 APE10-dist-na 17.146 APE9-dist-na 12.936 None None None XRAY 1.5 0.159 0.183 A 357 328 0 0 0 0 [[484, 797]] 1.0 6z5e Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 7AVQA Q8TF76 471 798 798.0 S1Z:801 Type1 Active DFGin 5.149 12.146 BLAminus -126.06, 173.12 69.03, 91.95 -102.42, 24.12 320.3, 125.97 -52.79, -41.95 in-in in 8.998 Saltbr-in 2.659 HRD-na-N -75.14, -46.38 71.99, 2.8 in-in-na SNCiia in-na ActLoopNT-in 2.891 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.18, 22.84 APE9-dihe-na -73.32, 160.09 APE8-dihe-na -148.12, 160.7 APE8-rot-na 195.64 APE67-dihe-na -157.46, 142.25 95.7, -0.72 APE12-dist-na 9.574 APE11-dist-na 13.487 APE10-dist-na 17.118 APE9-dist-na 12.952 None None None XRAY 1.65 0.16 0.179 A 357 328 0 0 0 0 [[484, 797]] 1.0 7avq Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 7OPSA Q8TF76 471 798 798.0 07C:801 Type1 Active DFGin 4.955 12.409 BLAminus -120.84, 168.72 74.52, 94.25 -110.46, 32.79 314.75, 129.03 -72.39, -27.54 in-in in 9.209 Saltbr-in 2.891 HRD-na-N -67.82, -53.79 76.87, 1.09 in-in-na SNCiia in-na ActLoopNT-in 2.935 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.38, 10.26 APE9-dihe-na -73.55, 156.67 APE8-dihe-na -147.73, 179.58 APE8-rot-na 67.78 APE67-dihe-na -167.67, 141.52 97.91, 1.48 APE12-dist-na 9.463 APE11-dist-na 13.499 APE10-dist-na 16.964 APE9-dist-na 13.035 None None None XRAY 2.38 0.179 0.229 A 357 328 0 0 0 0 [[484, 797]] 1.0 7ops Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 8RDKA Q8TF76 471 798 798.0 YQT:803 Type1 Active DFGin 5.304 12.291 BLAminus -126.79, 170.58 68.55, 97.1 -105.65, 24.46 315.14, 130.76 -63.91, -28.61 in-in in 8.949 Saltbr-in 2.684 HRD-na-N -70.8, -52.97 75.33, 1.85 in-in-na SNCiia in-na ActLoopNT-in 2.843 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -121.88, 25.66 APE9-dihe-na -78.67, 156.59 APE8-dihe-na -150.7, 178.52 APE8-rot-na 74.04 APE67-dihe-na -162.89, 139.09 96.18, -5.83 APE12-dist-na 9.438 APE11-dist-na 13.401 APE10-dist-na 17.106 APE9-dist-na 12.963 None None None XRAY 2.0 0.199 0.233 A 357 328 0 0 0 0 [[484, 797]] 1.0 8rdk Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9FLBA Q8TF76 471 798 798.0 A1IDB:802 Type1 Active DFGin 5.017 12.499 BLAminus -122.75, 164.93 78.09, 95.44 -111.48, 32.7 311.33, 133.52 -69.25, -37.29 in-in in 8.846 Saltbr-in 2.663 HRD-na-N -65.06, -57.81 86.13, 3.33 in-in-na SNCiia in-na ActLoopNT-in 2.883 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -97.12, -24.47 APE9-dihe-na -48.97, 165.86 APE8-dihe-na -171.41, -171.26 APE8-rot-na 65.27 APE67-dihe-na -131.18, 150.53 102.5, -31.2 APE12-dist-na 9.656 APE11-dist-na 13.445 APE10-dist-na 16.901 APE9-dist-na 13.075 None None None XRAY 2.5 0.195 0.245 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flb Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9FLQA Q8TF76 471 798 798.0 A1IDD:806 Type1 Active DFGin 5.277 11.995 BLAminus -131.52, 170.51 72.45, 91.56 -104.74, 27.71 313.77, 132.43 -58.36, -40.16 in-in in 9.194 Saltbr-in 2.385 HRD-na-N -72.62, -50.16 74.03, 2.04 in-in-na SNCiia in-na ActLoopNT-in 2.89 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -123.97, 17.68 APE9-dihe-na -77.54, 163.56 APE8-dihe-na -154.04, 168.58 APE8-rot-na 56.93 APE67-dihe-na -156.8, 141.47 98.45, -3.96 APE12-dist-na 9.579 APE11-dist-na 13.504 APE10-dist-na 17.048 APE9-dist-na 13.042 None None None XRAY 1.85 0.176 0.202 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flq Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9FLRA Q8TF76 471 798 798.0 A1IDE:803 Type1 Active DFGin 5.257 11.905 BLAminus -132.45, 173.37 67.71, 90.56 -101.27, 25.05 315.0, 128.67 -53.75, -42.86 in-in in 9.406 Saltbr-in 2.535 HRD-na-N -70.9, -52.21 71.26, 4.74 in-in-na SNCiia in-na ActLoopNT-in 2.852 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.29, 14.34 APE9-dihe-na -78.07, 164.28 APE8-dihe-na -157.67, 170.99 APE8-rot-na 58.59 APE67-dihe-na -164.88, 135.66 97.12, 4.81 APE12-dist-na 9.597 APE11-dist-na 13.566 APE10-dist-na 17.045 APE9-dist-na 13.109 None None None XRAY 1.91 0.173 0.209 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flr Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 7SQMA Q8TF76 453 798 798.0 A5G:801 Type1 Active DFGin 5.294 12.385 BLAminus -126.59, 168.89 78.77, 90.66 -103.22, 31.48 318.95, 126.98 -62.97, -29.65 in-in in 9.033 Saltbr-in 2.862 HRD-na-N -74.3, -49.72 73.45, 2.57 in-in-na SNCiia in-na ActLoopNT-in 2.956 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -117.03, 13.48 APE9-dihe-na -73.56, 163.48 APE8-dihe-na -150.66, 160.36 APE8-rot-na 211.61 APE67-dihe-na -164.54, 145.89 99.66, 4.4 APE12-dist-na 9.225 APE11-dist-na 13.189 APE10-dist-na 16.762 APE9-dist-na 12.944 None None None XRAY 1.78 0.175 0.205 A 357 346 0 0 0 0 [[484, 797]] 1.0 7sqm Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9FLCA Q8TF76 471 798 798.0 A1IDA:801 Type1.5_Back Active DFGin 4.715 12.46 BLAminus -134.34, 171.12 67.31, 104.11 -111.35, 24.44 309.33, 129.38 -43.69, -56.59 in-in in 9.127 Saltbr-in 2.572 HRD-na-N -70.37, -50.71 74.43, 4.41 in-in-na SNCiia in-na ActLoopNT-in 2.846 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -124.8, 13.59 APE9-dihe-na -68.86, 164.74 APE8-dihe-na -159.81, 175.83 APE8-rot-na 49.95 APE67-dihe-na -162.39, 140.7 102.66, -4.36 APE12-dist-na 9.337 APE11-dist-na 13.24 APE10-dist-na 16.865 APE9-dist-na 12.997 None None None XRAY 2.18 0.166 0.197 A 357 328 0 0 0 0 [[484, 797]] 1.0 9flc Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9B2SK Q8TF76 470 798 798.0 No_ligand No_ligand Inactive DFGin 6.064 12.671 BLAminus -142.15, 178.43 60.64, 69.74 -94.32, 35.13 330.57, 110.31 -71.54, -20.41 out-out out 10.509 Saltbr-out 8.91 HRD-na-N -103.48, -39.3 72.01, 16.12 out-in-na SNCoia in-na ActLoopNT-in 2.662 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -93.15, 4.32 APE9-dihe-na -71.11, 161.22 APE8-dihe-na -159.47, 164.4 APE8-rot-na 76.0 APE67-dihe-na -157.32, 146.25 103.48, -10.17 APE12-dist-na 10.384 APE11-dist-na 14.356 APE10-dist-na 17.698 APE9-dist-na 13.728 None None None EM 3.01 999.0 999.0 K 357 329 0 0 0 0 [[484, 797]] 1.0 9b2s Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9B2UK Q8TF76 470 798 798.0 No_ligand No_ligand Inactive DFGin 5.926 12.627 BLAminus -136.69, -178.38 59.48, 67.33 -92.11, 31.61 333.66, 107.16 -67.05, -16.22 out-out out 10.457 Saltbr-out 8.398 HRD-na-N -100.22, -40.69 78.07, 2.57 out-in-na SNCoia in-na ActLoopNT-in 2.756 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -100.28, 9.24 APE9-dihe-na -71.6, 162.97 APE8-dihe-na -157.23, 160.72 APE8-rot-na 81.21 APE67-dihe-na -151.55, 148.6 98.32, -9.69 APE12-dist-na 10.577 APE11-dist-na 14.628 APE10-dist-na 17.968 APE9-dist-na 13.833 None None None EM 3.64 999.0 999.0 K 357 329 0 0 0 0 [[484, 797]] 1.0 9b2u Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z5CA Q8TF76 470 798 798.0 PQ5:805 Type1 Inactive DFGin 4.731 13.108 BLAminus -133.84, 170.31 75.72, 94.52 -110.21, 19.19 311.37, 116.86 -61.87, -31.19 out-out out 10.462 Saltbr-out 3.7 HRD-na-N -70.06, -50.84 74.01, -0.31 out-in-na SNCoia in-na ActLoopNT-in 2.931 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.88, 20.45 APE9-dihe-na -80.43, 159.13 APE8-dihe-na -144.39, 165.92 APE8-rot-na 214.89 APE67-dihe-na -162.19, 147.1 97.48, -3.07 APE12-dist-na 9.488 APE11-dist-na 13.52 APE10-dist-na 17.05 APE9-dist-na 13.1 None None None XRAY 1.75 0.16 0.188 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z5c Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9FLOA Q8TF76 466 797 798.0 A1IDC:802 Type1 Inactive DFGin 5.355 12.318 BLAminus -140.34, 174.89 75.76, 76.52 -89.13, 31.66 305.79, 159.49 -77.78, -25.85 in-out in 9.084 Saltbr-out 3.76 HRD-na-N -85.47, -46.33 68.95, 25.87 out-in-na SNCoia in-na ActLoopNT-in 2.616 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -118.51, 102.44 APE9-dihe-na 136.93, 133.28 APE8-dihe-na -151.7, -143.81 APE8-rot-na 72.42 APE67-dihe-na -90.21, 160.33 109.28, -71.54 APE12-dist-na 9.638 APE11-dist-na 13.586 APE10-dist-na 17.18 APE9-dist-na 14.433 None None None XRAY 2.9 0.214 0.247 A 357 332 0 0 0 0 [[484, 797]] 1.0 9flo Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6G3AA Q8TF76 471 798 798.0 5ID:805 Type1 Inactive DFGin 4.953 12.443 BLAminus -127.41, 171.94 74.51, 93.23 -106.28, 26.81 312.44, 123.45 -60.95, -29.67 in-out in 9.904 Saltbr-out 4.42 HRD-na-N -72.27, -48.82 73.62, 1.17 out-in-na SNCoia in-na ActLoopNT-in 2.883 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -116.57, 14.66 APE9-dihe-na -70.85, 159.17 APE8-dihe-na -152.35, 172.74 APE8-rot-na 72.92 APE67-dihe-na -156.95, 142.2 92.44, -2.34 APE12-dist-na 9.454 APE11-dist-na 13.382 APE10-dist-na 16.931 APE9-dist-na 12.993 F605T None None XRAY 1.43 0.151 0.175 A 357 328 0 0 0 0 [[484, 797]] 1.0 6g3a Homo sapiens OTHER_HASPIN_HUMAN HASP 1.8e-225 752.9 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z56A Q8TF76 470 798 798.0 Q7Q:801 Type1.5_Back Inactive DFGin 4.602 12.569 BLAminus -129.58, 171.28 69.16, 102.48 -109.85, 26.06 309.6, 123.99 -45.33, -46.61 out-out out 10.104 Saltbr-out 4.52 HRD-na-N -69.89, -50.01 74.0, -0.03 out-in-na SNCoia in-na ActLoopNT-in 2.821 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -120.86, 18.07 APE9-dihe-na -73.34, 162.1 APE8-dihe-na -143.73, 169.15 APE8-rot-na 201.43 APE67-dihe-na -162.09, 141.44 91.95, 4.24 APE12-dist-na 9.424 APE11-dist-na 13.25 APE10-dist-na 17.008 APE9-dist-na 13.071 None None None XRAY 1.9 0.178 0.221 A 357 329 0 0 0 0 [[484, 797]] 1.0 6z56 Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z5BA Q8TF76 469 798 798.0 Q7Z:803 Type1.5_Back Inactive DFGin 4.548 12.709 BLAminus -135.9, 170.26 70.64, 101.28 -110.64, 25.44 308.83, 121.13 -45.93, -45.39 out-out out 10.049 Saltbr-out 4.556 HRD-na-N -70.65, -51.98 77.17, -0.49 out-in-na SNCoia in-na ActLoopNT-in 2.906 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -114.59, 17.24 APE9-dihe-na -73.9, 162.49 APE8-dihe-na -150.9, 168.36 APE8-rot-na 77.43 APE67-dihe-na -163.72, 140.01 97.4, -1.55 APE12-dist-na 9.36 APE11-dist-na 13.278 APE10-dist-na 16.905 APE9-dist-na 12.945 None None None XRAY 1.9 0.157 0.198 A 357 330 0 0 0 0 [[484, 797]] 1.0 6z5b Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 6Z5AA Q8TF76 465 798 798.0 Q8B:60807 Type1.5_Front Inactive DFGin 4.746 13.158 BLAminus -130.52, 170.23 77.78, 97.19 -110.55, 22.86 309.49, 126.33 -50.19, -42.61 out-out out 10.928 Saltbr-out 6.049 HRD-na-N -69.87, -51.48 73.76, 2.92 out-in-na SNCoia in-na ActLoopNT-in 2.957 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -114.05, 16.57 APE9-dihe-na -70.55, 162.23 APE8-dihe-na -152.03, 159.2 APE8-rot-na 218.93 APE67-dihe-na -157.88, 144.9 96.43, 3.83 APE12-dist-na 9.408 APE11-dist-na 13.313 APE10-dist-na 16.953 APE9-dist-na 12.968 None None None XRAY 1.55 0.157 0.182 A 357 334 0 0 0 0 [[484, 797]] 1.0 6z5a Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin
HASP_HUMAN 9B2TK Q8TF76 470 798 798.0 No_ligand No_ligand Inactive DFGin 10.473 16.998 None -74.01, 167.84 -68.22, 151.89 -112.4, 131.65 323.3, 85.18 -72.17, -31.47 out-out out 10.371 Saltbr-out 8.739 HRD-na-N -90.05, -46.55 60.89, 17.99 out-in-na SNCoia in-na ActLoopNT-in 2.509 ActLoopCT-na noAPE APEdihe_aaaaa APEdist_aaaa APE10-dihe-na -99.75, 7.12 APE9-dihe-na -76.13, 178.32 APE8-dihe-na -157.85, 172.7 APE8-rot-na 78.9 APE67-dihe-na -161.94, 175.92 118.79, -26.14 APE12-dist-na 11.19 APE11-dist-na 13.535 APE10-dist-na 18.064 APE9-dist-na 14.027 None None None EM 2.99 999.0 999.0 K 357 329 0 0 0 0 [[484, 797]] 1.0 9b2t Homo sapiens OTHER_HASPIN_HUMAN HASP 1.4e-226 756.6 1 314 314 686 687 688 690 692 511 535 539 646 648 647 649 741 721 716 715 714 713 712 711 710 604 Serine/threonine-protein kinase haspin

OTHER_HASPIN (Serine/threonine-protein kinase haspin)

Total number of chains: 0
Active chains: 0
Family: OTHER
Spatial label Dihedral label Number of Chains Percent Representative

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name