AGC_GRK6 (G protein-coupled receptor kinase 6)

Total number of chains: 8
Active chains: 8
Uniprot: GRK6_HUMAN
Kinase Domain Residues: 186 - 448
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 8 100.0% AF-P43250-K1A

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GRK6 2ACXA P43250 14 532 576.0 ANP:577 ATPlike Active DFGin 6.2066 13.2835 BLAminus -133.82, 164.79 58.79, 76.03 -96.19, 24.41 281.42, 82.4 -59.68, -24.05 in-in in 9.3415 Saltbr-in 3.2194 HRD-in -78.26, -56.85 77.2, -1.95 in-in-in SNCiii in-in ActLoopNT-in 2.9714 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.49, 157.4 APE9-dihe-na 123.02, -168.26 APE8-dihe-in -95.03, 140.31 APE8-rot-in 303.17 APE67-dihe-in -86.56, -0.13 -45.11, -52.69 APE12-dist-in 10.4784 APE11-dist-in 11.834 APE10-dist-in 6.0832 APE9-dist-in 3.9058 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 A 576.0 495.0 0 27 27 0 [[186, 448]] 1.0 2acx AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 2ACXB P43250 14 535 576.0 ANP:577 ATPlike Active DFGin 6.0903 13.1455 BLAminus -128.37, 163.87 55.35, 87.14 -100.56, 21.26 285.61, 77.77 -55.4, -30.56 in-in in 9.2313 Saltbr-in 2.4394 HRD-in -77.3, -59.12 75.78, 1.97 in-in-in SNCiii in-in ActLoopNT-in 2.9766 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.83, 161.38 APE9-dihe-na 125.99, -167.44 APE8-dihe-in -95.89, 144.8 APE8-rot-in 307.19 APE67-dihe-in -70.72, -14.39 -48.06, -55.51 APE12-dist-in 10.4768 APE11-dist-in 11.8719 APE10-dist-in 6.1674 APE9-dist-in 3.7096 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 B 576.0 492.0 5 27 27 0 [[186, 448]] 1.0 2acx AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 3NYOA P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.4231 12.9864 BLAminus -150.32, 176.66 46.57, 93.99 -112.64, 27.92 269.12, 56.38 -53.19, -36.92 in-in in 8.4918 Saltbr-in 3.1334 HRD-in -67.42, -53.58 67.41, 17.23 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.58, 145.08 APE9-dihe-na 153.72, -154.4 APE8-dihe-in -119.63, 125.01 APE8-rot-in 309.24 APE67-dihe-inflip 99.19, -30.43 -48.0, 129.76 APE12-dist-in 10.102 APE11-dist-in 11.8813 APE10-dist-in 6.1522 APE9-dist-in 3.9847 None None None XRAY 2.92 0.222 0.253 A 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyo AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 3NYOB P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.4686 12.9206 BLAminus -147.57, -176.88 49.48, 66.09 -89.42, 43.68 283.74, 78.16 -61.9, -48.01 in-in in 8.4292 Saltbr-in 2.8589 HRD-in -67.89, -44.49 63.77, 4.77 in-in-in SNCiii in-in ActLoopNT-in 2.9592 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.44, 138.67 APE9-dihe-na 143.94, 179.93 APE8-dihe-in -100.37, 135.53 APE8-rot-in 311.67 APE67-dihe-inflip 96.9, -39.59 -38.27, 126.0 APE12-dist-in 10.1477 APE11-dist-in 11.7313 APE10-dist-in 5.9599 APE9-dist-in 3.734 None None None XRAY 2.92 0.222 0.253 B 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyo AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 AF-P43250-K1A P43250 178 456 576.0 No_ligand No_ligand Active DFGin 6.2157 12.749 BLAminus -123.11, -178.58 47.67, 74.06 -87.65, 23.59 291.93, 77.77 -58.68, -35.83 in-in in 8.7118 Saltbr-in 2.6653 HRD-in -82.84, -44.36 66.32, 2.28 in-in-in SNCiii in-in ActLoopNT-in 2.9261 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.32, 157.5 APE9-dihe-na 121.0, 172.74 APE8-dihe-in -78.3, 135.32 APE8-rot-in 301.62 APE67-dihe-inflip 93.32, -20.35 -55.72, 131.85 APE12-dist-in 10.366 APE11-dist-in 12.1373 APE10-dist-in 6.1395 APE9-dist-in 3.4895 None None None AF2 -1.0 1.0 1.0 A 279.0 279.0 0 27 27 0 [[186, 448]] 1.0 AF-P43250-K1 AGC_GRK6_HUMAN AGC 2.2e-86 295.0 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 AF-P43250-K3A P43250 178 456 576.0 No_ligand No_ligand Active DFGin 6.0455 12.2821 BLAminus -130.79, 178.36 51.08, 64.04 -74.31, 18.83 302.42, 178.07 -60.87, -31.76 in-in in 8.6239 Saltbr-in 2.6188 HRD-in -87.79, -47.34 67.55, 3.73 in-in-in SNCiii in-in ActLoopNT-in 2.9098 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.34, 159.69 APE9-dihe-na 109.39, -175.73 APE8-dihe-in -92.28, 133.79 APE8-rot-in 298.55 APE67-dihe-inflip 96.49, -17.7 -57.25, 129.59 APE12-dist-in 10.5252 APE11-dist-in 11.9519 APE10-dist-in 5.9894 APE9-dist-in 3.1921 None None None AF2 -1.0 1.0 1.0 A 279.0 279.0 0 27 27 0 [[186, 448]] 1.0 AF-P43250-K3 AGC_GRK6_HUMAN AGC 2.2e-86 295.0 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 3NYNA P43250 2 557 576.0 SGV:60577 Type1 Active DFGin 6.6451 12.6795 BLAminus -161.03, 177.65 50.76, 84.33 -106.7, 25.79 281.1, 79.92 -51.73, -45.29 in-in in 8.3118 Saltbr-in 2.7656 HRD-in -85.94, -51.42 62.16, 25.53 in-in-in SNCiii in-in ActLoopNT-in 3.0 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.0, 146.47 APE9-dihe-na 148.26, -154.46 APE8-dihe-in -112.6, 137.1 APE8-rot-in 298.15 APE67-dihe-inflip 129.81, -32.33 -65.27, 111.53 APE12-dist-in 9.9474 APE11-dist-in 11.8071 APE10-dist-in 6.0596 APE9-dist-in 3.6569 None None None XRAY 2.72 0.227 0.238 A 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyn AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 3NYNB P43250 2 557 576.0 SGV:60577 Type1 Active DFGin 6.7271 12.8243 BLAminus -165.39, 175.41 57.11, 63.92 -91.01, 39.72 289.62, 84.65 -64.54, -42.76 in-in in 8.3207 Saltbr-in 2.9278 HRD-in -79.96, -51.35 60.14, 27.4 in-in-in SNCiii in-in ActLoopNT-in 3.1932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.23, 144.63 APE9-dihe-na 148.65, -158.33 APE8-dihe-in -111.02, 128.64 APE8-rot-in 289.73 APE67-dihe-inflip 120.73, -19.06 -60.78, 111.9 APE12-dist-in 10.0864 APE11-dist-in 11.7778 APE10-dist-in 6.0299 APE9-dist-in 3.5907 None None None XRAY 2.72 0.227 0.238 B 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyn AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6

AGC_GRK6 (G protein-coupled receptor kinase 6)

Total number of chains: 8
Active chains: 8
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 8 100.0% AF-P43250-K1A

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
GRK6 GRK6_HUMAN 2ACXA P43250 14 532 576.0 ANP:577 ATPlike Active DFGin 6.2066 13.2835 BLAminus -133.82, 164.79 58.79, 76.03 -96.19, 24.41 281.42, 82.4 -59.68, -24.05 in-in in 9.3415 Saltbr-in 3.2194 HRD-in -78.26, -56.85 77.2, -1.95 in-in-in SNCiii in-in ActLoopNT-in 2.9714 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -139.49, 157.4 APE9-dihe-na 123.02, -168.26 APE8-dihe-in -95.03, 140.31 APE8-rot-in 303.17 APE67-dihe-in -86.56, -0.13 -45.11, -52.69 APE12-dist-in 10.4784 APE11-dist-in 11.834 APE10-dist-in 6.0832 APE9-dist-in 3.9058 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 A 576.0 495.0 0 27 27 0 [[186, 448]] 1.0 2acx Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 GRK6_HUMAN 2ACXB P43250 14 535 576.0 ANP:577 ATPlike Active DFGin 6.0903 13.1455 BLAminus -128.37, 163.87 55.35, 87.14 -100.56, 21.26 285.61, 77.77 -55.4, -30.56 in-in in 9.2313 Saltbr-in 2.4394 HRD-in -77.3, -59.12 75.78, 1.97 in-in-in SNCiii in-in ActLoopNT-in 2.9766 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -140.83, 161.38 APE9-dihe-na 125.99, -167.44 APE8-dihe-in -95.89, 144.8 APE8-rot-in 307.19 APE67-dihe-in -70.72, -14.39 -48.06, -55.51 APE12-dist-in 10.4768 APE11-dist-in 11.8719 APE10-dist-in 6.1674 APE9-dist-in 3.7096 C561S,C562S,C565S None None XRAY 2.6 0.204 0.243 B 576.0 492.0 5 27 27 0 [[186, 448]] 1.0 2acx Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 GRK6_HUMAN 3NYOA P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.4231 12.9864 BLAminus -150.32, 176.66 46.57, 93.99 -112.64, 27.92 269.12, 56.38 -53.19, -36.92 in-in in 8.4918 Saltbr-in 3.1334 HRD-in -67.42, -53.58 67.41, 17.23 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.58, 145.08 APE9-dihe-na 153.72, -154.4 APE8-dihe-in -119.63, 125.01 APE8-rot-in 309.24 APE67-dihe-inflip 99.19, -30.43 -48.0, 129.76 APE12-dist-in 10.102 APE11-dist-in 11.8813 APE10-dist-in 6.1522 APE9-dist-in 3.9847 None None None XRAY 2.92 0.222 0.253 A 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyo Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 GRK6_HUMAN 3NYOB P43250 2 557 576.0 AMP:60577 ATPlike Active DFGin 6.4686 12.9206 BLAminus -147.57, -176.88 49.48, 66.09 -89.42, 43.68 283.74, 78.16 -61.9, -48.01 in-in in 8.4292 Saltbr-in 2.8589 HRD-in -67.89, -44.49 63.77, 4.77 in-in-in SNCiii in-in ActLoopNT-in 2.9592 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -138.44, 138.67 APE9-dihe-na 143.94, 179.93 APE8-dihe-in -100.37, 135.53 APE8-rot-in 311.67 APE67-dihe-inflip 96.9, -39.59 -38.27, 126.0 APE12-dist-in 10.1477 APE11-dist-in 11.7313 APE10-dist-in 5.9599 APE9-dist-in 3.734 None None None XRAY 2.92 0.222 0.253 B 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyo Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 GRK6_HUMAN AF-P43250-K1A P43250 178 456 576.0 No_ligand No_ligand Active DFGin 6.2157 12.749 BLAminus -123.11, -178.58 47.67, 74.06 -87.65, 23.59 291.93, 77.77 -58.68, -35.83 in-in in 8.7118 Saltbr-in 2.6653 HRD-in -82.84, -44.36 66.32, 2.28 in-in-in SNCiii in-in ActLoopNT-in 2.9261 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.32, 157.5 APE9-dihe-na 121.0, 172.74 APE8-dihe-in -78.3, 135.32 APE8-rot-in 301.62 APE67-dihe-inflip 93.32, -20.35 -55.72, 131.85 APE12-dist-in 10.366 APE11-dist-in 12.1373 APE10-dist-in 6.1395 APE9-dist-in 3.4895 None None None AF2 -1.0 1.0 1.0 A 279.0 279.0 0 27 27 0 [[186, 448]] 1.0 AF-P43250-K1 Homo sapiens AGC_GRK6_HUMAN AGC 2.2e-86 295.0 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 GRK6_HUMAN AF-P43250-K3A P43250 178 456 576.0 No_ligand No_ligand Active DFGin 6.0455 12.2821 BLAminus -130.79, 178.36 51.08, 64.04 -74.31, 18.83 302.42, 178.07 -60.87, -31.76 in-in in 8.6239 Saltbr-in 2.6188 HRD-in -87.79, -47.34 67.55, 3.73 in-in-in SNCiii in-in ActLoopNT-in 2.9098 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.34, 159.69 APE9-dihe-na 109.39, -175.73 APE8-dihe-in -92.28, 133.79 APE8-rot-in 298.55 APE67-dihe-inflip 96.49, -17.7 -57.25, 129.59 APE12-dist-in 10.5252 APE11-dist-in 11.9519 APE10-dist-in 5.9894 APE9-dist-in 3.1921 None None None AF2 -1.0 1.0 1.0 A 279.0 279.0 0 27 27 0 [[186, 448]] 1.0 AF-P43250-K3 Homo sapiens AGC_GRK6_HUMAN AGC 2.2e-86 295.0 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 GRK6_HUMAN 3NYNA P43250 2 557 576.0 SGV:60577 Type1 Active DFGin 6.6451 12.6795 BLAminus -161.03, 177.65 50.76, 84.33 -106.7, 25.79 281.1, 79.92 -51.73, -45.29 in-in in 8.3118 Saltbr-in 2.7656 HRD-in -85.94, -51.42 62.16, 25.53 in-in-in SNCiii in-in ActLoopNT-in 3.0 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.0, 146.47 APE9-dihe-na 148.26, -154.46 APE8-dihe-in -112.6, 137.1 APE8-rot-in 298.15 APE67-dihe-inflip 129.81, -32.33 -65.27, 111.53 APE12-dist-in 9.9474 APE11-dist-in 11.8071 APE10-dist-in 6.0596 APE9-dist-in 3.6569 None None None XRAY 2.72 0.227 0.238 A 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyn Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6
GRK6 GRK6_HUMAN 3NYNB P43250 2 557 576.0 SGV:60577 Type1 Active DFGin 6.7271 12.8243 BLAminus -165.39, 175.41 57.11, 63.92 -91.01, 39.72 289.62, 84.65 -64.54, -42.76 in-in in 8.3207 Saltbr-in 2.9278 HRD-in -79.96, -51.35 60.14, 27.4 in-in-in SNCiii in-in ActLoopNT-in 3.1932 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.23, 144.63 APE9-dihe-na 148.65, -158.33 APE8-dihe-in -111.02, 128.64 APE8-rot-in 289.73 APE67-dihe-inflip 120.73, -19.06 -60.78, 111.9 APE12-dist-in 10.0864 APE11-dist-in 11.7778 APE10-dist-in 6.0299 APE9-dist-in 3.5907 None None None XRAY 2.72 0.227 0.238 B 576.0 553.0 3 27 27 0 [[186, 448]] 1.0 3nyn Homo sapiens AGC_GRK6_HUMAN AGC 2e-85 292.1 1.0 260.0 260.0 328 329 330 332 334 215 234 238 308 310 309 311.0 367 355 350 349 348 347 346 345 344 264 G protein-coupled receptor kinase 6

AGC_GRK6 (G protein-coupled receptor kinase 6)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name