| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK6 | 2ACXA | P43250 | 14 | 532 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.2066 | 13.2835 | BLAminus | -133.82, 164.79 | 58.79, 76.03 | -96.19, 24.41 | 281.42, 82.4 | -59.68, -24.05 | in-in | in | 9.3415 | Saltbr-in | 3.2194 | HRD-in | -78.26, -56.85 | 77.2, -1.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9714 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.49, 157.4 | APE9-dihe-na | 123.02, -168.26 | APE8-dihe-in | -95.03, 140.31 | APE8-rot-in | 303.17 | APE67-dihe-in | -86.56, -0.13 | -45.11, -52.69 | APE12-dist-in | 10.4784 | APE11-dist-in | 11.834 | APE10-dist-in | 6.0832 | APE9-dist-in | 3.9058 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | A | 576.0 | 495.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | 2ACXB | P43250 | 14 | 535 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.0903 | 13.1455 | BLAminus | -128.37, 163.87 | 55.35, 87.14 | -100.56, 21.26 | 285.61, 77.77 | -55.4, -30.56 | in-in | in | 9.2313 | Saltbr-in | 2.4394 | HRD-in | -77.3, -59.12 | 75.78, 1.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.83, 161.38 | APE9-dihe-na | 125.99, -167.44 | APE8-dihe-in | -95.89, 144.8 | APE8-rot-in | 307.19 | APE67-dihe-in | -70.72, -14.39 | -48.06, -55.51 | APE12-dist-in | 10.4768 | APE11-dist-in | 11.8719 | APE10-dist-in | 6.1674 | APE9-dist-in | 3.7096 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | B | 576.0 | 492.0 | 5 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | 3NYOA | P43250 | 2 | 557 | 576.0 | AMP:60577 | ATPlike | Active | DFGin | 6.4231 | 12.9864 | BLAminus | -150.32, 176.66 | 46.57, 93.99 | -112.64, 27.92 | 269.12, 56.38 | -53.19, -36.92 | in-in | in | 8.4918 | Saltbr-in | 3.1334 | HRD-in | -67.42, -53.58 | 67.41, 17.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.875 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.58, 145.08 | APE9-dihe-na | 153.72, -154.4 | APE8-dihe-in | -119.63, 125.01 | APE8-rot-in | 309.24 | APE67-dihe-inflip | 99.19, -30.43 | -48.0, 129.76 | APE12-dist-in | 10.102 | APE11-dist-in | 11.8813 | APE10-dist-in | 6.1522 | APE9-dist-in | 3.9847 | None | None | None | XRAY | 2.92 | 0.222 | 0.253 | A | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyo | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | 3NYOB | P43250 | 2 | 557 | 576.0 | AMP:60577 | ATPlike | Active | DFGin | 6.4686 | 12.9206 | BLAminus | -147.57, -176.88 | 49.48, 66.09 | -89.42, 43.68 | 283.74, 78.16 | -61.9, -48.01 | in-in | in | 8.4292 | Saltbr-in | 2.8589 | HRD-in | -67.89, -44.49 | 63.77, 4.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9592 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.44, 138.67 | APE9-dihe-na | 143.94, 179.93 | APE8-dihe-in | -100.37, 135.53 | APE8-rot-in | 311.67 | APE67-dihe-inflip | 96.9, -39.59 | -38.27, 126.0 | APE12-dist-in | 10.1477 | APE11-dist-in | 11.7313 | APE10-dist-in | 5.9599 | APE9-dist-in | 3.734 | None | None | None | XRAY | 2.92 | 0.222 | 0.253 | B | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyo | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | AF-P43250-K1A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.2157 | 12.749 | BLAminus | -123.11, -178.58 | 47.67, 74.06 | -87.65, 23.59 | 291.93, 77.77 | -58.68, -35.83 | in-in | in | 8.7118 | Saltbr-in | 2.6653 | HRD-in | -82.84, -44.36 | 66.32, 2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9261 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.32, 157.5 | APE9-dihe-na | 121.0, 172.74 | APE8-dihe-in | -78.3, 135.32 | APE8-rot-in | 301.62 | APE67-dihe-inflip | 93.32, -20.35 | -55.72, 131.85 | APE12-dist-in | 10.366 | APE11-dist-in | 12.1373 | APE10-dist-in | 6.1395 | APE9-dist-in | 3.4895 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K1 | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | AF-P43250-K3A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.0455 | 12.2821 | BLAminus | -130.79, 178.36 | 51.08, 64.04 | -74.31, 18.83 | 302.42, 178.07 | -60.87, -31.76 | in-in | in | 8.6239 | Saltbr-in | 2.6188 | HRD-in | -87.79, -47.34 | 67.55, 3.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9098 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.34, 159.69 | APE9-dihe-na | 109.39, -175.73 | APE8-dihe-in | -92.28, 133.79 | APE8-rot-in | 298.55 | APE67-dihe-inflip | 96.49, -17.7 | -57.25, 129.59 | APE12-dist-in | 10.5252 | APE11-dist-in | 11.9519 | APE10-dist-in | 5.9894 | APE9-dist-in | 3.1921 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K3 | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | 3NYNA | P43250 | 2 | 557 | 576.0 | SGV:60577 | Type1 | Active | DFGin | 6.6451 | 12.6795 | BLAminus | -161.03, 177.65 | 50.76, 84.33 | -106.7, 25.79 | 281.1, 79.92 | -51.73, -45.29 | in-in | in | 8.3118 | Saltbr-in | 2.7656 | HRD-in | -85.94, -51.42 | 62.16, 25.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.0, 146.47 | APE9-dihe-na | 148.26, -154.46 | APE8-dihe-in | -112.6, 137.1 | APE8-rot-in | 298.15 | APE67-dihe-inflip | 129.81, -32.33 | -65.27, 111.53 | APE12-dist-in | 9.9474 | APE11-dist-in | 11.8071 | APE10-dist-in | 6.0596 | APE9-dist-in | 3.6569 | None | None | None | XRAY | 2.72 | 0.227 | 0.238 | A | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyn | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | 3NYNB | P43250 | 2 | 557 | 576.0 | SGV:60577 | Type1 | Active | DFGin | 6.7271 | 12.8243 | BLAminus | -165.39, 175.41 | 57.11, 63.92 | -91.01, 39.72 | 289.62, 84.65 | -64.54, -42.76 | in-in | in | 8.3207 | Saltbr-in | 2.9278 | HRD-in | -79.96, -51.35 | 60.14, 27.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1932 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.23, 144.63 | APE9-dihe-na | 148.65, -158.33 | APE8-dihe-in | -111.02, 128.64 | APE8-rot-in | 289.73 | APE67-dihe-inflip | 120.73, -19.06 | -60.78, 111.9 | APE12-dist-in | 10.0864 | APE11-dist-in | 11.7778 | APE10-dist-in | 6.0299 | APE9-dist-in | 3.5907 | None | None | None | XRAY | 2.72 | 0.227 | 0.238 | B | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyn | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GRK6 | GRK6_HUMAN | 2ACXA | P43250 | 14 | 532 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.2066 | 13.2835 | BLAminus | -133.82, 164.79 | 58.79, 76.03 | -96.19, 24.41 | 281.42, 82.4 | -59.68, -24.05 | in-in | in | 9.3415 | Saltbr-in | 3.2194 | HRD-in | -78.26, -56.85 | 77.2, -1.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9714 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -139.49, 157.4 | APE9-dihe-na | 123.02, -168.26 | APE8-dihe-in | -95.03, 140.31 | APE8-rot-in | 303.17 | APE67-dihe-in | -86.56, -0.13 | -45.11, -52.69 | APE12-dist-in | 10.4784 | APE11-dist-in | 11.834 | APE10-dist-in | 6.0832 | APE9-dist-in | 3.9058 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | A | 576.0 | 495.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | GRK6_HUMAN | 2ACXB | P43250 | 14 | 535 | 576.0 | ANP:577 | ATPlike | Active | DFGin | 6.0903 | 13.1455 | BLAminus | -128.37, 163.87 | 55.35, 87.14 | -100.56, 21.26 | 285.61, 77.77 | -55.4, -30.56 | in-in | in | 9.2313 | Saltbr-in | 2.4394 | HRD-in | -77.3, -59.12 | 75.78, 1.97 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9766 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.83, 161.38 | APE9-dihe-na | 125.99, -167.44 | APE8-dihe-in | -95.89, 144.8 | APE8-rot-in | 307.19 | APE67-dihe-in | -70.72, -14.39 | -48.06, -55.51 | APE12-dist-in | 10.4768 | APE11-dist-in | 11.8719 | APE10-dist-in | 6.1674 | APE9-dist-in | 3.7096 | C561S,C562S,C565S | None | None | XRAY | 2.6 | 0.204 | 0.243 | B | 576.0 | 492.0 | 5 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 2acx | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | GRK6_HUMAN | 3NYOA | P43250 | 2 | 557 | 576.0 | AMP:60577 | ATPlike | Active | DFGin | 6.4231 | 12.9864 | BLAminus | -150.32, 176.66 | 46.57, 93.99 | -112.64, 27.92 | 269.12, 56.38 | -53.19, -36.92 | in-in | in | 8.4918 | Saltbr-in | 3.1334 | HRD-in | -67.42, -53.58 | 67.41, 17.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.875 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -146.58, 145.08 | APE9-dihe-na | 153.72, -154.4 | APE8-dihe-in | -119.63, 125.01 | APE8-rot-in | 309.24 | APE67-dihe-inflip | 99.19, -30.43 | -48.0, 129.76 | APE12-dist-in | 10.102 | APE11-dist-in | 11.8813 | APE10-dist-in | 6.1522 | APE9-dist-in | 3.9847 | None | None | None | XRAY | 2.92 | 0.222 | 0.253 | A | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyo | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | GRK6_HUMAN | 3NYOB | P43250 | 2 | 557 | 576.0 | AMP:60577 | ATPlike | Active | DFGin | 6.4686 | 12.9206 | BLAminus | -147.57, -176.88 | 49.48, 66.09 | -89.42, 43.68 | 283.74, 78.16 | -61.9, -48.01 | in-in | in | 8.4292 | Saltbr-in | 2.8589 | HRD-in | -67.89, -44.49 | 63.77, 4.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9592 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.44, 138.67 | APE9-dihe-na | 143.94, 179.93 | APE8-dihe-in | -100.37, 135.53 | APE8-rot-in | 311.67 | APE67-dihe-inflip | 96.9, -39.59 | -38.27, 126.0 | APE12-dist-in | 10.1477 | APE11-dist-in | 11.7313 | APE10-dist-in | 5.9599 | APE9-dist-in | 3.734 | None | None | None | XRAY | 2.92 | 0.222 | 0.253 | B | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyo | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | GRK6_HUMAN | AF-P43250-K1A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.2157 | 12.749 | BLAminus | -123.11, -178.58 | 47.67, 74.06 | -87.65, 23.59 | 291.93, 77.77 | -58.68, -35.83 | in-in | in | 8.7118 | Saltbr-in | 2.6653 | HRD-in | -82.84, -44.36 | 66.32, 2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9261 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.32, 157.5 | APE9-dihe-na | 121.0, 172.74 | APE8-dihe-in | -78.3, 135.32 | APE8-rot-in | 301.62 | APE67-dihe-inflip | 93.32, -20.35 | -55.72, 131.85 | APE12-dist-in | 10.366 | APE11-dist-in | 12.1373 | APE10-dist-in | 6.1395 | APE9-dist-in | 3.4895 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K1 | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | GRK6_HUMAN | AF-P43250-K3A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.0455 | 12.2821 | BLAminus | -130.79, 178.36 | 51.08, 64.04 | -74.31, 18.83 | 302.42, 178.07 | -60.87, -31.76 | in-in | in | 8.6239 | Saltbr-in | 2.6188 | HRD-in | -87.79, -47.34 | 67.55, 3.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9098 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.34, 159.69 | APE9-dihe-na | 109.39, -175.73 | APE8-dihe-in | -92.28, 133.79 | APE8-rot-in | 298.55 | APE67-dihe-inflip | 96.49, -17.7 | -57.25, 129.59 | APE12-dist-in | 10.5252 | APE11-dist-in | 11.9519 | APE10-dist-in | 5.9894 | APE9-dist-in | 3.1921 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K3 | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | GRK6_HUMAN | 3NYNA | P43250 | 2 | 557 | 576.0 | SGV:60577 | Type1 | Active | DFGin | 6.6451 | 12.6795 | BLAminus | -161.03, 177.65 | 50.76, 84.33 | -106.7, 25.79 | 281.1, 79.92 | -51.73, -45.29 | in-in | in | 8.3118 | Saltbr-in | 2.7656 | HRD-in | -85.94, -51.42 | 62.16, 25.53 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -145.0, 146.47 | APE9-dihe-na | 148.26, -154.46 | APE8-dihe-in | -112.6, 137.1 | APE8-rot-in | 298.15 | APE67-dihe-inflip | 129.81, -32.33 | -65.27, 111.53 | APE12-dist-in | 9.9474 | APE11-dist-in | 11.8071 | APE10-dist-in | 6.0596 | APE9-dist-in | 3.6569 | None | None | None | XRAY | 2.72 | 0.227 | 0.238 | A | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyn | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| GRK6 | GRK6_HUMAN | 3NYNB | P43250 | 2 | 557 | 576.0 | SGV:60577 | Type1 | Active | DFGin | 6.7271 | 12.8243 | BLAminus | -165.39, 175.41 | 57.11, 63.92 | -91.01, 39.72 | 289.62, 84.65 | -64.54, -42.76 | in-in | in | 8.3207 | Saltbr-in | 2.9278 | HRD-in | -79.96, -51.35 | 60.14, 27.4 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.1932 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -144.23, 144.63 | APE9-dihe-na | 148.65, -158.33 | APE8-dihe-in | -111.02, 128.64 | APE8-rot-in | 289.73 | APE67-dihe-inflip | 120.73, -19.06 | -60.78, 111.9 | APE12-dist-in | 10.0864 | APE11-dist-in | 11.7778 | APE10-dist-in | 6.0299 | APE9-dist-in | 3.5907 | None | None | None | XRAY | 2.72 | 0.227 | 0.238 | B | 576.0 | 553.0 | 3 | 27 | 27 | 0 | [[186, 448]] | 1.0 | 3nyn | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2e-85 | 292.1 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|