| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| FGFR3 | 4K33A | P22607 | 459 | 755 | 806.0 | ACP:801 | ATPlike | Active | DFGin | 6.2519 | 13.787 | BLAminus | -133.88, -173.58 | 58.49, 82.81 | -96.43, 27.55 | 291.81, 80.95 | -59.32, -31.32 | in-in | in | 8.2114 | Saltbr-in | 2.895 | HRD-in | -87.09, -47.34 | 67.06, 1.63 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9905 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -55.89, 133.11 | APE9-dihe-in | -125.43, 130.21 | APE8-dihe-in | -78.76, 72.58 | APE8-rot-na | 29.71 | APE67-dihe-in | -71.45, -4.47 | -50.14, -48.75 | APE12-dist-na | 13.3098 | APE11-dist-na | 9.6016 | APE10-dist-na | 8.3051 | APE9-dist-in | 6.8731 | C482A,C582S,K650E | None | None | XRAY | 2.341 | 0.181 | 0.228 | A | 325.0 | 293.0 | 4 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 4k33 | TYR_FGFR3_HUMAN | TYR | 2.3e-104 | 354.2 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | AF-P22607-K1A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.5621 | 13.7198 | BLAminus | -135.6, -172.84 | 54.36, 70.3 | -87.69, 11.11 | 291.08, 95.72 | -59.35, -30.65 | in-in | in | 7.4386 | Saltbr-in | 2.6502 | HRD-in | -71.1, -43.09 | 66.59, -18.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8909 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.08, 128.6 | APE9-dihe-in | -136.51, 151.31 | APE8-dihe-in | -81.26, 77.84 | APE8-rot-na | 37.52 | APE67-dihe-in | -66.67, -14.17 | -46.27, -41.56 | APE12-dist-na | 14.3905 | APE11-dist-na | 9.9039 | APE10-dist-na | 9.996 | APE9-dist-in | 6.5212 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K1 | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | AF-P22607-K3A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.3619 | 13.7626 | BLAminus | -140.11, -178.74 | 60.69, 64.92 | -81.11, 10.08 | 291.09, 95.14 | -60.2, -27.32 | in-in | in | 7.6939 | Saltbr-in | 2.724 | HRD-in | -81.64, -44.23 | 60.23, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9077 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.46, 141.09 | APE9-dihe-in | -143.98, 144.08 | APE8-dihe-in | -81.78, 61.47 | APE8-rot-na | 36.97 | APE67-dihe-in | -68.61, -8.42 | -45.34, -43.48 | APE12-dist-na | 14.4543 | APE11-dist-na | 10.9342 | APE10-dist-na | 10.3642 | APE9-dist-in | 6.9461 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K3 | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 6LVMA | P22607 | 472 | 755 | 806.0 | EVR:60801 | Type1.5_Back | Active | DFGin | 6.5277 | 14.2505 | BLAminus | -141.75, -180.0 | 67.67, 74.35 | -89.33, 29.0 | 297.0, 117.38 | -56.22, -44.89 | in-in | in | 7.87 | Saltbr-in | 3.3042 | HRD-in | -81.99, -57.17 | 74.69, 3.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0228 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -86.44, 126.31 | APE9-dihe-in | -128.79, 145.49 | APE8-dihe-in | -85.23, 77.25 | APE8-rot-na | 30.53 | APE67-dihe-in | -75.5, -6.21 | -67.03, -34.23 | APE12-dist-na | 14.1311 | APE11-dist-na | 10.493 | APE10-dist-na | 10.6197 | APE9-dist-in | 6.8201 | None | PTR577,PTR647,PTR648 | PTR577,PTR647,PTR648 | XRAY | 2.53 | 0.211 | 0.279 | A | 313.0 | 276.0 | 8 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6lvm | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 7DHLA | P22607 | 472 | 755 | 806.0 | H6X:60801 | Type1.5_Back | Active | DFGin | 5.9046 | 13.8906 | BLAminus | -128.75, 172.71 | 75.89, 84.08 | -98.64, 30.77 | 301.65, 163.04 | -59.86, -43.17 | in-in | in | 7.8037 | Saltbr-in | 3.2049 | HRD-in | -74.83, -62.31 | 81.14, 3.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9371 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -89.21, 114.53 | APE9-dihe-in | -123.29, 143.17 | APE8-dihe-in | -76.55, 75.16 | APE8-rot-na | 29.19 | APE67-dihe-in | -80.84, -3.09 | -66.95, -32.19 | APE12-dist-na | 14.4146 | APE11-dist-na | 10.4878 | APE10-dist-na | 10.067 | APE9-dist-in | 6.8206 | None | PTR577,PTR647,PTR648 | PTR577,PTR647,PTR648 | XRAY | 2.57 | 0.197 | 0.254 | A | 313.0 | 277.0 | 7 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 7dhl | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDUB | P22607 | 459 | 755 | 806.0 | WIQ:61002 | Type1.5_Front | Active | DFGin | 6.4209 | 14.4148 | BLAminus | -138.69, 176.26 | 64.2, 86.01 | -100.28, 24.84 | 287.71, 79.66 | -57.6, -41.09 | in-in | in | 8.1853 | Saltbr-in | 2.9464 | HRD-in | -71.69, -47.92 | 71.62, 0.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9471 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.88, 155.75 | APE9-dihe-in | -122.51, 89.95 | APE8-dihe-in | -81.37, 70.05 | APE8-rot-na | 30.61 | APE67-dihe-in | -66.22, -12.9 | -45.0, -50.18 | APE12-dist-na | 999.0 | APE11-dist-na | 7.6606 | APE10-dist-na | 8.4893 | APE9-dist-in | 7.717 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | B | 297.0 | 276.0 | 9 | 30 | 29 | 1 | [[472, 750]] | 1.0 | 8udu | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 9KFUA | P22607 | 448 | 756 | 806.0 | A1L5T:801 | Type1 | Inactive | DFGin | 7.0189 | 14.4915 | BLAminus | -131.22, -178.97 | 62.43, 68.96 | -89.65, 16.94 | 287.35, 89.22 | -61.48, -27.48 | in-in | in | 7.689 | Saltbr-in | 2.7663 | HRD-in | -73.03, -51.34 | 76.73, -9.72 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.898 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -98.53, 13.75 | APE9-dihe-in | -98.46, 127.45 | APE8-dihe-in | -57.08, 120.6 | APE8-rot-na | 333.93 | APE67-dihe-in | -72.45, -11.1 | -67.2, -26.43 | APE12-dist-na | 9.9702 | APE11-dist-na | 10.7644 | APE10-dist-na | 7.0416 | APE9-dist-in | 4.7988 | None | None | None | XRAY | 1.4 | 0.229 | 0.251 | A | 309.0 | 288.0 | 21 | 30 | 24 | 6 | [[472, 750]] | 1.0 | 9kfu | TYR_FGFR3_HUMAN | TYR | 1.7e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 6PNXA | P22607 | 456 | 757 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1832 | 13.2568 | BLAplus | -117.43, 165.96 | 59.53, 36.21 | -90.35, -22.61 | 56.49, 88.29 | -100.71, 20.75 | in-out | in | 7.758 | Saltbr-out | 3.8922 | HRD-in | -72.74, -43.96 | 72.66, -12.59 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.6112 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 61.32, -168.18 | APE9-dihe-in | -95.45, 138.6 | APE8-dihe-in | -83.08, 62.92 | APE8-rot-na | 32.84 | APE67-dihe-in | -77.59, -4.01 | -63.19, -31.79 | APE12-dist-na | 17.76 | APE11-dist-na | 14.3869 | APE10-dist-na | 16.4747 | APE9-dist-in | 7.9796 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | A | 324.0 | 291.0 | 11 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 6PNXB | P22607 | 455 | 756 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1024 | 12.8796 | BLAplus | -116.22, 163.18 | 57.59, 45.48 | -96.33, -11.84 | 56.51, 88.18 | -107.89, 22.55 | in-in | in | 7.3718 | Saltbr-in | 2.3809 | HRD-in | -94.02, -38.66 | 69.29, -17.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 4.1485 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 54.33, 74.29 | APE9-dihe-in | -157.39, 146.53 | APE8-dihe-in | -79.85, 92.16 | APE8-rot-na | 29.38 | APE67-dihe-in | -64.97, -14.94 | -62.55, -40.44 | APE12-dist-na | 17.5294 | APE11-dist-na | 16.9582 | APE10-dist-na | 14.6317 | APE9-dist-in | 7.491 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | B | 324.0 | 294.0 | 8 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDTA | P22607 | 457 | 756 | 806.0 | MLT:61001,MLT:61002,WGF:61003 | Allosteric,Allosteric,Type1.5_Front | Inactive | DFGin | 5.4408 | 13.493 | BLAplus | -114.8, 158.79 | 55.69, 43.2 | -82.19, -34.37 | 42.84, 89.08 | -83.27, -4.41 | in-out | in | 8.3828 | Saltbr-out | 5.2872 | HRD-in | -68.34, -46.54 | 75.89, -9.4 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.9211 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 112.29 | APE8-dihe-out | -63.06, -32.23 | APE8-rot-na | 340.92 | APE67-dihe-in | -68.35, -26.42 | -62.13, -28.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.1982 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | A | 297.0 | 284.0 | 4 | 30 | 26 | 4 | [[472, 750]] | 1.0 | 8udt | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 9D1XA | P22607 | 461 | 754 | 806.0 | A1A6M:2001 | Type1 | Inactive | DFGin | 5.1196 | 12.6323 | BLAplus | -108.03, 159.86 | 61.02, 36.65 | -81.76, -20.43 | 56.47, 81.47 | -95.6, 7.99 | in-in | in | 7.8726 | Saltbr-in | 3.0881 | HRD-in | -69.72, -49.85 | 77.77, -9.05 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.4139 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -149.56, 157.12 | APE9-dihe-in | -112.69, 98.2 | APE8-dihe-out | -58.57, -23.42 | APE8-rot-na | 337.44 | APE67-dihe-in | -70.39, -9.82 | -57.35, -25.35 | APE12-dist-na | 16.0046 | APE11-dist-na | 20.0862 | APE10-dist-na | 17.5026 | APE9-dist-out | 11.3051 | P572S,P573G | None | None | XRAY | 1.6 | 0.18 | 0.19 | A | 297.0 | 282.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 9d1x | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 9CD7A | P22607 | 451 | 755 | 806.0 | A1AV2:801 | Type1 | Inactive | DFGin | 5.0186 | 12.7277 | BLAplus | -114.49, 161.16 | 51.06, 50.03 | -90.62, -20.91 | 50.11, 84.08 | -82.82, 141.47 | in-in | in | 7.0948 | Saltbr-in | 2.5832 | HRD-in | -75.51, -51.62 | 85.64, -15.78 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 85.15 | APE8-dihe-out | -64.87, -3.22 | APE8-rot-na | 28.88 | APE67-dihe-in | -77.21, -9.06 | -69.64, -25.05 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3457 | C482A,C582S,K650E | None | None | XRAY | 2.53 | 0.23 | 0.267 | A | 312.0 | 276.0 | 29 | 30 | 13 | 17 | [[472, 750]] | 1.0 | 9cd7 | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 9CD7B | P22607 | 458 | 755 | 806.0 | A1AV2:801 | Type1 | Inactive | DFGin | 5.0653 | 12.8593 | BLAplus | -114.57, 159.12 | 51.43, 51.5 | -92.22, -19.36 | 49.89, 84.09 | -76.73, -39.85 | in-in | in | 7.4133 | Saltbr-in | 2.5967 | HRD-in | -74.94, -51.38 | 85.94, -16.13 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.5988 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 48.12 | APE8-dihe-out | -65.12, -2.8 | APE8-rot-na | 29.36 | APE67-dihe-in | -77.72, -8.63 | -66.93, -28.5 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2175 | C482A,C582S,K650E | None | None | XRAY | 2.53 | 0.23 | 0.267 | B | 312.0 | 278.0 | 20 | 30 | 24 | 6 | [[472, 750]] | 1.0 | 9cd7 | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 9CD7C | P22607 | 458 | 755 | 806.0 | A1AV2:801 | Type1 | Inactive | DFGin | 5.0552 | 12.9174 | BLAplus | -113.11, 157.29 | 52.27, 52.26 | -91.9, -19.06 | 50.44, 84.08 | -76.91, -39.15 | in-in | in | 7.4207 | Saltbr-in | 2.6017 | HRD-in | -75.28, -51.41 | 85.96, -15.25 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.7116 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 98.75 | APE8-dihe-out | -72.0, 23.1 | APE8-rot-na | 34.26 | APE67-dihe-in | -76.94, -9.16 | -66.89, -26.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.796 | C482A,C582S,K650E | None | None | XRAY | 2.53 | 0.23 | 0.267 | C | 312.0 | 278.0 | 20 | 30 | 24 | 6 | [[472, 750]] | 1.0 | 9cd7 | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDVA | P22607 | 458 | 755 | 806.0 | WIQ:1003 | Type1.5_Back | Inactive | DFGin | 6.0012 | 13.4764 | BLAplus | -124.26, 161.29 | 66.5, 36.68 | -91.33, -43.75 | 46.96, 90.73 | -84.73, 13.25 | in-in | in | 7.6609 | Saltbr-in | 2.9402 | HRD-in | -66.26, -46.33 | 75.0, -11.55 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.16 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -144.63, 151.27 | APE9-dihe-in | -107.88, 92.32 | APE8-dihe-out | -54.6, -21.22 | APE8-rot-na | 338.66 | APE67-dihe-in | -68.84, -8.83 | -57.22, -29.15 | APE12-dist-na | 15.9556 | APE11-dist-na | 19.9983 | APE10-dist-na | 17.2851 | APE9-dist-out | 11.6116 | V555M | None | None | XRAY | 2.348 | 0.237 | 0.261 | A | 297.0 | 279.0 | 7 | 30 | 23 | 7 | [[472, 750]] | 1.0 | 8udv | TYR_FGFR3_HUMAN | TYR | 4.5e-105 | 356.6 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDVB | P22607 | 455 | 755 | 806.0 | WIQ:803 | Type1.5_Back | Inactive | DFGin | 5.4813 | 13.2542 | BLAplus | -124.6, 164.38 | 63.05, 27.71 | -82.13, -38.21 | 55.85, 89.15 | -91.32, 13.57 | in-in | in | 7.68 | Saltbr-in | 2.9036 | HRD-in | -63.59, -46.44 | 79.4, -13.95 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.9067 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -136.87, 152.88 | APE9-dihe-in | -110.79, 96.93 | APE8-dihe-out | -58.89, -20.81 | APE8-rot-na | 338.74 | APE67-dihe-in | -70.46, -8.74 | -52.69, -32.19 | APE12-dist-na | 15.4794 | APE11-dist-na | 19.3858 | APE10-dist-na | 16.7032 | APE9-dist-out | 11.4241 | V555M | None | None | XRAY | 2.348 | 0.237 | 0.261 | B | 297.0 | 281.0 | 8 | 30 | 22 | 8 | [[472, 750]] | 1.0 | 8udv | TYR_FGFR3_HUMAN | TYR | 4.5e-105 | 356.6 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDVC | P22607 | 458 | 755 | 806.0 | WIQ:1004 | Type1.5_Back | Inactive | DFGin | 6.071 | 13.4313 | BLAplus | -124.65, 164.21 | 70.39, 38.16 | -109.8, -21.91 | 57.41, 87.59 | -78.9, -34.05 | in-in | in | 7.6549 | Saltbr-in | 2.8879 | HRD-in | -64.72, -49.48 | 77.07, -10.54 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 91.25 | APE8-dihe-out | -54.32, -20.59 | APE8-rot-na | 338.75 | APE67-dihe-in | -71.87, -8.91 | -59.36, -26.12 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.6264 | V555M | None | None | XRAY | 2.348 | 0.237 | 0.261 | C | 297.0 | 269.0 | 17 | 30 | 14 | 16 | [[472, 750]] | 1.0 | 8udv | TYR_FGFR3_HUMAN | TYR | 4.5e-105 | 356.6 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDTB | P22607 | 457 | 754 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.2581 | 13.7103 | BLAplus | -108.64, 157.87 | 56.15, 40.62 | -79.39, -35.54 | 45.72, 88.06 | -80.67, 0.1 | in-out | in | 8.4451 | Saltbr-out | 5.3977 | HRD-in | -67.98, -43.8 | 74.91, -8.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.8672 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -64.67 | APE9-dihe-out | -68.82, -39.67 | APE8-dihe-out | -56.45, -17.85 | APE8-rot-na | 337.42 | APE67-dihe-in | -61.76, -27.35 | -59.02, -40.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.6665 | APE9-dist-out | 10.854 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | B | 297.0 | 283.0 | 3 | 30 | 27 | 3 | [[472, 750]] | 1.0 | 8udt | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDTC | P22607 | 457 | 756 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.2583 | 13.8238 | BLAplus | -109.74, 157.08 | 55.91, 40.67 | -78.94, -35.79 | 45.97, 87.77 | -81.04, -4.46 | in-out | in | 8.545 | Saltbr-out | 4.1026 | HRD-in | -68.09, -46.3 | 75.11, -4.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.8702 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -150.08 | APE9-dihe-out | -67.3, -42.56 | APE8-dihe-out | -46.98, -31.66 | APE8-rot-na | 333.46 | APE67-dihe-in | -60.08, -29.46 | -58.03, -43.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.4047 | APE9-dist-out | 11.049 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | C | 297.0 | 284.0 | 4 | 30 | 26 | 4 | [[472, 750]] | 1.0 | 8udt | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | 8UDUA | P22607 | 460 | 756 | 806.0 | WIQ:61002 | Type1.5_Back | Inactive | DFGin | 5.7614 | 13.5292 | BLBplus | -121.3, 171.32 | 71.72, 21.7 | -99.77, 166.76 | 66.11, 93.34 | 95.58, -59.45 | in-in | in | 7.9172 | Saltbr-in | 2.7343 | HRD-in | -77.2, -48.45 | 77.61, -12.83 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -71.65, 162.44 | APE9-dihe-in | -54.1, 129.25 | APE8-dihe-in | -83.64, 61.19 | APE8-rot-na | 34.62 | APE67-dihe-in | -73.43, -8.03 | -52.16, -35.97 | APE12-dist-na | 999.0 | APE11-dist-na | 14.2323 | APE10-dist-na | 17.7469 | APE9-dist-out | 8.253 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | A | 297.0 | 277.0 | 8 | 30 | 22 | 8 | [[472, 750]] | 1.0 | 8udu | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| FGFR3 | FGFR3_HUMAN | 4K33A | P22607 | 459 | 755 | 806.0 | ACP:801 | ATPlike | Active | DFGin | 6.2519 | 13.787 | BLAminus | -133.88, -173.58 | 58.49, 82.81 | -96.43, 27.55 | 291.81, 80.95 | -59.32, -31.32 | in-in | in | 8.2114 | Saltbr-in | 2.895 | HRD-in | -87.09, -47.34 | 67.06, 1.63 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9905 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -55.89, 133.11 | APE9-dihe-in | -125.43, 130.21 | APE8-dihe-in | -78.76, 72.58 | APE8-rot-na | 29.71 | APE67-dihe-in | -71.45, -4.47 | -50.14, -48.75 | APE12-dist-na | 13.3098 | APE11-dist-na | 9.6016 | APE10-dist-na | 8.3051 | APE9-dist-in | 6.8731 | C482A,C582S,K650E | None | None | XRAY | 2.341 | 0.181 | 0.228 | A | 325.0 | 293.0 | 4 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 4k33 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2.3e-104 | 354.2 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | AF-P22607-K1A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.5621 | 13.7198 | BLAminus | -135.6, -172.84 | 54.36, 70.3 | -87.69, 11.11 | 291.08, 95.72 | -59.35, -30.65 | in-in | in | 7.4386 | Saltbr-in | 2.6502 | HRD-in | -71.1, -43.09 | 66.59, -18.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8909 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.08, 128.6 | APE9-dihe-in | -136.51, 151.31 | APE8-dihe-in | -81.26, 77.84 | APE8-rot-na | 37.52 | APE67-dihe-in | -66.67, -14.17 | -46.27, -41.56 | APE12-dist-na | 14.3905 | APE11-dist-na | 9.9039 | APE10-dist-na | 9.996 | APE9-dist-in | 6.5212 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K1 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | AF-P22607-K3A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.3619 | 13.7626 | BLAminus | -140.11, -178.74 | 60.69, 64.92 | -81.11, 10.08 | 291.09, 95.14 | -60.2, -27.32 | in-in | in | 7.6939 | Saltbr-in | 2.724 | HRD-in | -81.64, -44.23 | 60.23, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9077 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.46, 141.09 | APE9-dihe-in | -143.98, 144.08 | APE8-dihe-in | -81.78, 61.47 | APE8-rot-na | 36.97 | APE67-dihe-in | -68.61, -8.42 | -45.34, -43.48 | APE12-dist-na | 14.4543 | APE11-dist-na | 10.9342 | APE10-dist-na | 10.3642 | APE9-dist-in | 6.9461 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K3 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 6LVMA | P22607 | 472 | 755 | 806.0 | EVR:60801 | Type1.5_Back | Active | DFGin | 6.5277 | 14.2505 | BLAminus | -141.75, -180.0 | 67.67, 74.35 | -89.33, 29.0 | 297.0, 117.38 | -56.22, -44.89 | in-in | in | 7.87 | Saltbr-in | 3.3042 | HRD-in | -81.99, -57.17 | 74.69, 3.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0228 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -86.44, 126.31 | APE9-dihe-in | -128.79, 145.49 | APE8-dihe-in | -85.23, 77.25 | APE8-rot-na | 30.53 | APE67-dihe-in | -75.5, -6.21 | -67.03, -34.23 | APE12-dist-na | 14.1311 | APE11-dist-na | 10.493 | APE10-dist-na | 10.6197 | APE9-dist-in | 6.8201 | None | PTR577,PTR647,PTR648 | PTR577,PTR647,PTR648 | XRAY | 2.53 | 0.211 | 0.279 | A | 313.0 | 276.0 | 8 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6lvm | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 7DHLA | P22607 | 472 | 755 | 806.0 | H6X:60801 | Type1.5_Back | Active | DFGin | 5.9046 | 13.8906 | BLAminus | -128.75, 172.71 | 75.89, 84.08 | -98.64, 30.77 | 301.65, 163.04 | -59.86, -43.17 | in-in | in | 7.8037 | Saltbr-in | 3.2049 | HRD-in | -74.83, -62.31 | 81.14, 3.67 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9371 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -89.21, 114.53 | APE9-dihe-in | -123.29, 143.17 | APE8-dihe-in | -76.55, 75.16 | APE8-rot-na | 29.19 | APE67-dihe-in | -80.84, -3.09 | -66.95, -32.19 | APE12-dist-na | 14.4146 | APE11-dist-na | 10.4878 | APE10-dist-na | 10.067 | APE9-dist-in | 6.8206 | None | PTR577,PTR647,PTR648 | PTR577,PTR647,PTR648 | XRAY | 2.57 | 0.197 | 0.254 | A | 313.0 | 277.0 | 7 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 7dhl | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDUB | P22607 | 459 | 755 | 806.0 | WIQ:61002 | Type1.5_Front | Active | DFGin | 6.4209 | 14.4148 | BLAminus | -138.69, 176.26 | 64.2, 86.01 | -100.28, 24.84 | 287.71, 79.66 | -57.6, -41.09 | in-in | in | 8.1853 | Saltbr-in | 2.9464 | HRD-in | -71.69, -47.92 | 71.62, 0.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9471 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.88, 155.75 | APE9-dihe-in | -122.51, 89.95 | APE8-dihe-in | -81.37, 70.05 | APE8-rot-na | 30.61 | APE67-dihe-in | -66.22, -12.9 | -45.0, -50.18 | APE12-dist-na | 999.0 | APE11-dist-na | 7.6606 | APE10-dist-na | 8.4893 | APE9-dist-in | 7.717 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | B | 297.0 | 276.0 | 9 | 30 | 29 | 1 | [[472, 750]] | 1.0 | 8udu | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 9KFUA | P22607 | 448 | 756 | 806.0 | A1L5T:801 | Type1 | Inactive | DFGin | 7.0189 | 14.4915 | BLAminus | -131.22, -178.97 | 62.43, 68.96 | -89.65, 16.94 | 287.35, 89.22 | -61.48, -27.48 | in-in | in | 7.689 | Saltbr-in | 2.7663 | HRD-in | -73.03, -51.34 | 76.73, -9.72 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.898 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -98.53, 13.75 | APE9-dihe-in | -98.46, 127.45 | APE8-dihe-in | -57.08, 120.6 | APE8-rot-na | 333.93 | APE67-dihe-in | -72.45, -11.1 | -67.2, -26.43 | APE12-dist-na | 9.9702 | APE11-dist-na | 10.7644 | APE10-dist-na | 7.0416 | APE9-dist-in | 4.7988 | None | None | None | XRAY | 1.4 | 0.229 | 0.251 | A | 309.0 | 288.0 | 21 | 30 | 24 | 6 | [[472, 750]] | 1.0 | 9kfu | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 1.7e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 6PNXA | P22607 | 456 | 757 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1832 | 13.2568 | BLAplus | -117.43, 165.96 | 59.53, 36.21 | -90.35, -22.61 | 56.49, 88.29 | -100.71, 20.75 | in-out | in | 7.758 | Saltbr-out | 3.8922 | HRD-in | -72.74, -43.96 | 72.66, -12.59 | out-out-out | SNCooo | out-out | ActLoopNT-out | 8.6112 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 61.32, -168.18 | APE9-dihe-in | -95.45, 138.6 | APE8-dihe-in | -83.08, 62.92 | APE8-rot-na | 32.84 | APE67-dihe-in | -77.59, -4.01 | -63.19, -31.79 | APE12-dist-na | 17.76 | APE11-dist-na | 14.3869 | APE10-dist-na | 16.4747 | APE9-dist-in | 7.9796 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | A | 324.0 | 291.0 | 11 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 6PNXB | P22607 | 455 | 756 | 806.0 | ACP:801 | ATPlike | Inactive | DFGin | 5.1024 | 12.8796 | BLAplus | -116.22, 163.18 | 57.59, 45.48 | -96.33, -11.84 | 56.51, 88.18 | -107.89, 22.55 | in-in | in | 7.3718 | Saltbr-in | 2.3809 | HRD-in | -94.02, -38.66 | 69.29, -17.12 | in-out-out | SNCioo | out-out | ActLoopNT-out | 4.1485 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 54.33, 74.29 | APE9-dihe-in | -157.39, 146.53 | APE8-dihe-in | -79.85, 92.16 | APE8-rot-na | 29.38 | APE67-dihe-in | -64.97, -14.94 | -62.55, -40.44 | APE12-dist-na | 17.5294 | APE11-dist-na | 16.9582 | APE10-dist-na | 14.6317 | APE9-dist-in | 7.491 | C482A,C582S,R669E | None | None | XRAY | 2.199 | 0.195 | 0.23 | B | 324.0 | 294.0 | 8 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 6pnx | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDTA | P22607 | 457 | 756 | 806.0 | MLT:61001,MLT:61002,WGF:61003 | Allosteric,Allosteric,Type1.5_Front | Inactive | DFGin | 5.4408 | 13.493 | BLAplus | -114.8, 158.79 | 55.69, 43.2 | -82.19, -34.37 | 42.84, 89.08 | -83.27, -4.41 | in-out | in | 8.3828 | Saltbr-out | 5.2872 | HRD-in | -68.34, -46.54 | 75.89, -9.4 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.9211 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 112.29 | APE8-dihe-out | -63.06, -32.23 | APE8-rot-na | 340.92 | APE67-dihe-in | -68.35, -26.42 | -62.13, -28.18 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.1982 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | A | 297.0 | 284.0 | 4 | 30 | 26 | 4 | [[472, 750]] | 1.0 | 8udt | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 9D1XA | P22607 | 461 | 754 | 806.0 | A1A6M:2001 | Type1 | Inactive | DFGin | 5.1196 | 12.6323 | BLAplus | -108.03, 159.86 | 61.02, 36.65 | -81.76, -20.43 | 56.47, 81.47 | -95.6, 7.99 | in-in | in | 7.8726 | Saltbr-in | 3.0881 | HRD-in | -69.72, -49.85 | 77.77, -9.05 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.4139 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -149.56, 157.12 | APE9-dihe-in | -112.69, 98.2 | APE8-dihe-out | -58.57, -23.42 | APE8-rot-na | 337.44 | APE67-dihe-in | -70.39, -9.82 | -57.35, -25.35 | APE12-dist-na | 16.0046 | APE11-dist-na | 20.0862 | APE10-dist-na | 17.5026 | APE9-dist-out | 11.3051 | P572S,P573G | None | None | XRAY | 1.6 | 0.18 | 0.19 | A | 297.0 | 282.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | 9d1x | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 9CD7A | P22607 | 451 | 755 | 806.0 | A1AV2:801 | Type1 | Inactive | DFGin | 5.0186 | 12.7277 | BLAplus | -114.49, 161.16 | 51.06, 50.03 | -90.62, -20.91 | 50.11, 84.08 | -82.82, 141.47 | in-in | in | 7.0948 | Saltbr-in | 2.5832 | HRD-in | -75.51, -51.62 | 85.64, -15.78 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 85.15 | APE8-dihe-out | -64.87, -3.22 | APE8-rot-na | 28.88 | APE67-dihe-in | -77.21, -9.06 | -69.64, -25.05 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.3457 | C482A,C582S,K650E | None | None | XRAY | 2.53 | 0.23 | 0.267 | A | 312.0 | 276.0 | 29 | 30 | 13 | 17 | [[472, 750]] | 1.0 | 9cd7 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 9CD7B | P22607 | 458 | 755 | 806.0 | A1AV2:801 | Type1 | Inactive | DFGin | 5.0653 | 12.8593 | BLAplus | -114.57, 159.12 | 51.43, 51.5 | -92.22, -19.36 | 49.89, 84.09 | -76.73, -39.85 | in-in | in | 7.4133 | Saltbr-in | 2.5967 | HRD-in | -74.94, -51.38 | 85.94, -16.13 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.5988 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 48.12 | APE8-dihe-out | -65.12, -2.8 | APE8-rot-na | 29.36 | APE67-dihe-in | -77.72, -8.63 | -66.93, -28.5 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2175 | C482A,C582S,K650E | None | None | XRAY | 2.53 | 0.23 | 0.267 | B | 312.0 | 278.0 | 20 | 30 | 24 | 6 | [[472, 750]] | 1.0 | 9cd7 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 9CD7C | P22607 | 458 | 755 | 806.0 | A1AV2:801 | Type1 | Inactive | DFGin | 5.0552 | 12.9174 | BLAplus | -113.11, 157.29 | 52.27, 52.26 | -91.9, -19.06 | 50.44, 84.08 | -76.91, -39.15 | in-in | in | 7.4207 | Saltbr-in | 2.6017 | HRD-in | -75.28, -51.41 | 85.96, -15.25 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.7116 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 98.75 | APE8-dihe-out | -72.0, 23.1 | APE8-rot-na | 34.26 | APE67-dihe-in | -76.94, -9.16 | -66.89, -26.41 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 10.796 | C482A,C582S,K650E | None | None | XRAY | 2.53 | 0.23 | 0.267 | C | 312.0 | 278.0 | 20 | 30 | 24 | 6 | [[472, 750]] | 1.0 | 9cd7 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 2e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDVA | P22607 | 458 | 755 | 806.0 | WIQ:1003 | Type1.5_Back | Inactive | DFGin | 6.0012 | 13.4764 | BLAplus | -124.26, 161.29 | 66.5, 36.68 | -91.33, -43.75 | 46.96, 90.73 | -84.73, 13.25 | in-in | in | 7.6609 | Saltbr-in | 2.9402 | HRD-in | -66.26, -46.33 | 75.0, -11.55 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.16 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -144.63, 151.27 | APE9-dihe-in | -107.88, 92.32 | APE8-dihe-out | -54.6, -21.22 | APE8-rot-na | 338.66 | APE67-dihe-in | -68.84, -8.83 | -57.22, -29.15 | APE12-dist-na | 15.9556 | APE11-dist-na | 19.9983 | APE10-dist-na | 17.2851 | APE9-dist-out | 11.6116 | V555M | None | None | XRAY | 2.348 | 0.237 | 0.261 | A | 297.0 | 279.0 | 7 | 30 | 23 | 7 | [[472, 750]] | 1.0 | 8udv | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 4.5e-105 | 356.6 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDVB | P22607 | 455 | 755 | 806.0 | WIQ:803 | Type1.5_Back | Inactive | DFGin | 5.4813 | 13.2542 | BLAplus | -124.6, 164.38 | 63.05, 27.71 | -82.13, -38.21 | 55.85, 89.15 | -91.32, 13.57 | in-in | in | 7.68 | Saltbr-in | 2.9036 | HRD-in | -63.59, -46.44 | 79.4, -13.95 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.9067 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -136.87, 152.88 | APE9-dihe-in | -110.79, 96.93 | APE8-dihe-out | -58.89, -20.81 | APE8-rot-na | 338.74 | APE67-dihe-in | -70.46, -8.74 | -52.69, -32.19 | APE12-dist-na | 15.4794 | APE11-dist-na | 19.3858 | APE10-dist-na | 16.7032 | APE9-dist-out | 11.4241 | V555M | None | None | XRAY | 2.348 | 0.237 | 0.261 | B | 297.0 | 281.0 | 8 | 30 | 22 | 8 | [[472, 750]] | 1.0 | 8udv | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 4.5e-105 | 356.6 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDVC | P22607 | 458 | 755 | 806.0 | WIQ:1004 | Type1.5_Back | Inactive | DFGin | 6.071 | 13.4313 | BLAplus | -124.65, 164.21 | 70.39, 38.16 | -109.8, -21.91 | 57.41, 87.59 | -78.9, -34.05 | in-in | in | 7.6549 | Saltbr-in | 2.8879 | HRD-in | -64.72, -49.48 | 77.07, -10.54 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 91.25 | APE8-dihe-out | -54.32, -20.59 | APE8-rot-na | 338.75 | APE67-dihe-in | -71.87, -8.91 | -59.36, -26.12 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.6264 | V555M | None | None | XRAY | 2.348 | 0.237 | 0.261 | C | 297.0 | 269.0 | 17 | 30 | 14 | 16 | [[472, 750]] | 1.0 | 8udv | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 4.5e-105 | 356.6 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDTB | P22607 | 457 | 754 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.2581 | 13.7103 | BLAplus | -108.64, 157.87 | 56.15, 40.62 | -79.39, -35.54 | 45.72, 88.06 | -80.67, 0.1 | in-out | in | 8.4451 | Saltbr-out | 5.3977 | HRD-in | -67.98, -43.8 | 74.91, -8.8 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.8672 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -64.67 | APE9-dihe-out | -68.82, -39.67 | APE8-dihe-out | -56.45, -17.85 | APE8-rot-na | 337.42 | APE67-dihe-in | -61.76, -27.35 | -59.02, -40.48 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.6665 | APE9-dist-out | 10.854 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | B | 297.0 | 283.0 | 3 | 30 | 27 | 3 | [[472, 750]] | 1.0 | 8udt | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDTC | P22607 | 457 | 756 | 806.0 | WGF:62001 | Type1.5_Front | Inactive | DFGin | 5.2583 | 13.8238 | BLAplus | -109.74, 157.08 | 55.91, 40.67 | -78.94, -35.79 | 45.97, 87.77 | -81.04, -4.46 | in-out | in | 8.545 | Saltbr-out | 4.1026 | HRD-in | -68.09, -46.3 | 75.11, -4.3 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.8702 | ActLoopCT-out | TYR | APEdihe_nooai | APEdist_aaao | APE10-dihe-none | 999.0, -150.08 | APE9-dihe-out | -67.3, -42.56 | APE8-dihe-out | -46.98, -31.66 | APE8-rot-na | 333.46 | APE67-dihe-in | -60.08, -29.46 | -58.03, -43.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 18.4047 | APE9-dist-out | 11.049 | P572S,P573G | None | None | XRAY | 2.829 | 0.263 | 0.274 | C | 297.0 | 284.0 | 4 | 30 | 26 | 4 | [[472, 750]] | 1.0 | 8udt | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| FGFR3 | FGFR3_HUMAN | 8UDUA | P22607 | 460 | 756 | 806.0 | WIQ:61002 | Type1.5_Back | Inactive | DFGin | 5.7614 | 13.5292 | BLBplus | -121.3, 171.32 | 71.72, 21.7 | -99.77, 166.76 | 66.11, 93.34 | 95.58, -59.45 | in-in | in | 7.9172 | Saltbr-in | 2.7343 | HRD-in | -77.2, -48.45 | 77.61, -12.83 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iiiai | APEdist_aaao | APE10-dihe-in | -71.65, 162.44 | APE9-dihe-in | -54.1, 129.25 | APE8-dihe-in | -83.64, 61.19 | APE8-rot-na | 34.62 | APE67-dihe-in | -73.43, -8.03 | -52.16, -35.97 | APE12-dist-na | 999.0 | APE11-dist-na | 14.2323 | APE10-dist-na | 17.7469 | APE9-dist-out | 8.253 | P572S,P573G | None | None | XRAY | 1.737 | 0.231 | 0.256 | A | 297.0 | 277.0 | 8 | 30 | 22 | 8 | [[472, 750]] | 1.0 | 8udu | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|