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| PDB | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AF-Q92630-K1A | 214 | 543 | 601.0 | No_ligand | No_ligand | Active | DFGin | 6.939 | 14.864 | BLAminus | -126.07, 177.15 | 62.42, 65.44 | -81.73, 10.25 | 284.63, 80.53 | -64.64, -17.85 | in-in | in | 8.728 | Saltbr-in | 2.723 | HRD-in | -66.96, -37.74 | 67.08, -16.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.848 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.84, 175.12 | APE9-dihe-na | 60.6, 144.79 | APE8-dihe-in | -65.13, 137.41 | APE8-rot-in | 294.19 | APE67-dihe-in | -65.52, -19.21 | -50.69, -46.33 | APE12-dist-in | 12.882 | APE11-dist-in | 11.334 | APE10-dist-in | 7.287 | APE9-dist-in | 3.021 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 330 | 330 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | AF-Q92630-K1 | CMGC_DYRK2_HUMAN | CMGC | 5.8e-99 | 337.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| AF-Q92630-K3A | 214 | 543 | 601.0 | No_ligand | No_ligand | Active | DFGin | 6.623 | 14.471 | BLAminus | -128.09, 177.13 | 63.4, 64.99 | -80.7, 10.08 | 289.17, 77.94 | -66.05, -16.49 | in-in | in | 8.839 | Saltbr-in | 2.734 | HRD-in | -72.99, -34.76 | 62.62, -5.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.882 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.48, 175.5 | APE9-dihe-na | 61.64, 142.59 | APE8-dihe-in | -63.51, 134.37 | APE8-rot-in | 293.35 | APE67-dihe-in | -63.69, -20.47 | -54.61, -45.06 | APE12-dist-in | 12.796 | APE11-dist-in | 11.341 | APE10-dist-in | 7.03 | APE9-dist-in | 3.09 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 330 | 330 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | AF-Q92630-K3 | CMGC_DYRK2_HUMAN | CMGC | 5.8e-99 | 337.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7EJVA | 151 | 537 | 601.0 | YK2:60501 | Type1 | Active | DFGin | 6.9 | 15.424 | BLAminus | -121.6, -175.71 | 52.95, 74.47 | -89.12, 21.12 | 283.92, 70.74 | -60.92, -24.61 | in-in | in | 8.982 | Saltbr-in | 3.13 | HRD-in | -72.41, -42.76 | 75.36, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.755 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.92, 162.27 | APE9-dihe-na | 76.47, 145.84 | APE8-dihe-in | -66.78, 142.47 | APE8-rot-in | 275.38 | APE67-dihe-in | -56.79, -30.59 | -58.46, -46.41 | APE12-dist-in | 12.918 | APE11-dist-in | 11.297 | APE10-dist-in | 6.969 | APE9-dist-in | 3.304 | None | PTR382 | PTR382 | XRAY | 2.5 | 0.202 | 0.246 | A | 387 | 385 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7ejv | CMGC_DYRK2_HUMAN | CMGC | 1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 8HLTA | 151 | 535 | 601.0 | XSE:60501 | Type1 | Active | DFGin | 7.153 | 15.661 | BLAminus | -128.03, -174.41 | 42.45, 74.99 | -83.08, 17.4 | 279.93, 74.95 | -62.5, -19.89 | in-in | in | 9.177 | Saltbr-in | 2.717 | HRD-in | -71.74, -44.48 | 73.83, 0.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.747 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.16, 170.0 | APE9-dihe-na | 71.16, 164.17 | APE8-dihe-in | -84.62, 135.53 | APE8-rot-in | 250.25 | APE67-dihe-in | -56.1, -31.76 | -49.25, -50.28 | APE12-dist-in | 13.315 | APE11-dist-in | 11.966 | APE10-dist-in | 7.57 | APE9-dist-in | 3.21 | None | PTR382 | PTR382 | XRAY | 2.8 | 0.213 | 0.267 | A | 393 | 385 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 8hlt | CMGC_DYRK2_HUMAN | CMGC | 1.1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7AKHA | 146 | 535 | 601.0 | RK8:60601 | Type1 | Active | DFGin | 6.926 | 15.074 | BLAminus | -121.6, -171.14 | 52.21, 81.66 | -96.01, 25.36 | 287.39, 72.64 | -67.66, -23.05 | in-in | in | 9.121 | Saltbr-in | 2.705 | HRD-in | -56.66, -58.54 | 81.07, -0.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.821 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.43, 168.94 | APE9-dihe-na | 72.6, 150.47 | APE8-dihe-in | -61.43, 140.56 | APE8-rot-in | 278.26 | APE67-dihe-in | -62.31, -24.44 | -52.56, -49.45 | APE12-dist-in | 12.815 | APE11-dist-in | 11.442 | APE10-dist-in | 6.914 | APE9-dist-in | 3.229 | None | SEP232,PTR382,SEP458 | SEP232,PTR382,SEP458 | XRAY | 2.85 | 0.188 | 0.245 | A | 429 | 390 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7akh | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 3K2LA | 146 | 543 | 601.0 | No_ligand | No_ligand | Inactive | DFGin | 7.095 | 15.241 | BLAminus | -127.38, 178.65 | 61.29, 89.71 | -107.22, 23.8 | 277.85, 81.5 | -75.9, -16.57 | in-in | in | 8.858 | Saltbr-in | 2.965 | HRD-in | -80.34, -48.51 | 75.91, -1.73 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.974 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.89, 168.99 | APE9-dihe-na | 66.37, 164.94 | APE8-dihe-in | -92.92, 137.86 | APE8-rot-out | 183.76 | APE67-dihe-in | -63.43, -18.18 | -49.75, -48.38 | APE12-dist-in | 12.59 | APE11-dist-in | 11.884 | APE10-dist-in | 7.261 | APE9-dist-in | 3.098 | None | SEP232,TPO381,PTR382,SEP442,SEP458 | SEP232,TPO381,PTR382,SEP442,SEP458 | XRAY | 2.36 | 0.228 | 0.288 | A | 429 | 397 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 3k2l | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DG4A | 215 | 538 | 601.0 | H5R:601 | Type1 | Inactive | DFGin | 7.076 | 15.315 | BLAminus | -112.18, -176.63 | 54.26, 82.32 | -95.55, 24.49 | 281.35, 68.71 | -70.68, -16.69 | in-in | in | 9.062 | Saltbr-in | 2.632 | HRD-in | -72.69, -45.13 | 72.43, 4.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.829 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -123.35, 168.65 | APE9-dihe-na | 72.59, 152.62 | APE8-dihe-in | -75.5, 133.34 | APE8-rot-out | 190.89 | APE67-dihe-in | -53.88, -27.24 | -50.74, -49.3 | APE12-dist-in | 13.02 | APE11-dist-in | 11.794 | APE10-dist-in | 7.365 | APE9-dist-in | 3.357 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.58 | 0.206 | 0.249 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dg4 | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DH9A | 215 | 538 | 601.0 | H7F:601 | Type1 | Inactive | DFGin | 6.955 | 15.393 | BLAminus | -118.25, -176.44 | 52.33, 72.66 | -86.4, 22.32 | 285.5, 71.17 | -68.46, -16.6 | in-in | in | 9.091 | Saltbr-in | 2.818 | HRD-in | -67.52, -48.86 | 77.78, -1.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.826 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.21, 165.64 | APE9-dihe-na | 77.26, 152.01 | APE8-dihe-in | -71.35, 136.19 | APE8-rot-out | 186.16 | APE67-dihe-in | -56.24, -27.47 | -53.15, -48.91 | APE12-dist-in | 13.085 | APE11-dist-in | 11.935 | APE10-dist-in | 7.588 | APE9-dist-in | 3.308 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.194 | 0.19 | 0.218 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dh9 | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DHCA | 215 | 538 | 601.0 | H99:601 | Type1 | Inactive | DFGin | 6.897 | 15.183 | BLAminus | -120.85, -173.65 | 54.47, 76.85 | -89.75, 13.16 | 285.05, 71.42 | -59.73, -14.3 | in-in | in | 9.165 | Saltbr-in | 2.836 | HRD-in | -67.26, -47.7 | 73.48, 5.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.79 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -124.28, 171.52 | APE9-dihe-na | 72.07, 147.78 | APE8-dihe-in | -70.3, 140.28 | APE8-rot-out | 189.19 | APE67-dihe-in | -57.12, -25.22 | -59.04, -44.86 | APE12-dist-in | 13.016 | APE11-dist-in | 11.9 | APE10-dist-in | 7.482 | APE9-dist-in | 3.275 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.592 | 0.17 | 0.217 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhc | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DHHA | 215 | 538 | 601.0 | H7L:601 | Type1 | Inactive | DFGin | 7.002 | 15.315 | BLAminus | -121.49, -175.98 | 53.38, 75.83 | -90.0, 17.27 | 285.73, 67.63 | -60.12, -17.2 | in-in | in | 9.069 | Saltbr-in | 2.831 | HRD-in | -72.48, -43.45 | 72.8, 3.03 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.934 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -112.98, 162.3 | APE9-dihe-na | 71.38, 148.19 | APE8-dihe-in | -71.4, 141.57 | APE8-rot-out | 161.34 | APE67-dihe-in | -65.17, -19.89 | -55.14, -43.22 | APE12-dist-in | 12.9 | APE11-dist-in | 11.849 | APE10-dist-in | 7.619 | APE9-dist-in | 3.387 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.486 | 0.195 | 0.245 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhh | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DHKA | 215 | 538 | 601.0 | H7O:601 | Type1 | Inactive | DFGin | 7.052 | 15.35 | BLAminus | -117.35, 177.72 | 56.81, 75.07 | -85.18, 19.92 | 283.41, 63.05 | -63.85, -33.36 | in-in | in | 9.196 | Saltbr-in | 2.644 | HRD-in | -71.37, -46.63 | 75.15, -1.94 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.906 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -118.3, 166.48 | APE9-dihe-na | 68.65, 147.66 | APE8-dihe-in | -62.61, 137.42 | APE8-rot-out | 200.1 | APE67-dihe-in | -57.5, -27.74 | -53.83, -48.57 | APE12-dist-in | 12.955 | APE11-dist-in | 11.738 | APE10-dist-in | 7.593 | APE9-dist-in | 3.202 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.341 | 0.199 | 0.257 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhk | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DHNA | 215 | 538 | 601.0 | H7R:601 | Type1 | Inactive | DFGin | 6.943 | 15.204 | BLAminus | -121.26, -177.62 | 55.21, 78.31 | -90.06, 20.47 | 287.34, 73.71 | -59.07, -25.63 | in-out | in | 9.064 | Saltbr-out | 3.683 | HRD-in | -71.04, -47.07 | 70.57, 6.17 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.681 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.33, 167.28 | APE9-dihe-na | 70.26, 153.99 | APE8-dihe-in | -74.79, 138.71 | APE8-rot-out | 162.7 | APE67-dihe-in | -57.15, -24.62 | -55.14, -47.5 | APE12-dist-in | 13.035 | APE11-dist-in | 11.859 | APE10-dist-in | 7.473 | APE9-dist-in | 3.339 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.38 | 0.187 | 0.223 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhn | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DHOA | 215 | 538 | 601.0 | H7U:601 | Type1 | Inactive | DFGin | 7.024 | 15.384 | BLAminus | -119.43, -172.42 | 42.56, 78.27 | -84.62, 15.62 | 281.95, 67.94 | -55.62, -33.56 | in-in | in | 9.274 | Saltbr-in | 2.624 | HRD-in | -82.16, -38.69 | 68.11, 7.67 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.83 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -109.77, 178.86 | APE9-dihe-na | 69.78, 147.69 | APE8-dihe-in | -69.75, 134.88 | APE8-rot-out | 211.6 | APE67-dihe-in | -60.55, -23.47 | -49.02, -52.25 | APE12-dist-in | 12.813 | APE11-dist-in | 11.959 | APE10-dist-in | 7.417 | APE9-dist-in | 3.473 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 3.29 | 0.188 | 0.259 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dho | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DJOA | 215 | 538 | 601.0 | H80:601 | Type1 | Inactive | DFGin | 6.825 | 15.46 | BLAminus | -127.28, -171.08 | 53.55, 75.01 | -93.19, 14.88 | 276.88, 71.94 | -62.8, -14.89 | in-in | in | 9.123 | Saltbr-in | 2.61 | HRD-in | -68.11, -47.05 | 70.53, 3.02 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.794 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -112.85, 165.38 | APE9-dihe-na | 72.88, 157.2 | APE8-dihe-in | -82.18, 142.51 | APE8-rot-out | 184.87 | APE67-dihe-in | -72.03, -23.08 | -61.29, -39.89 | APE12-dist-in | 12.99 | APE11-dist-in | 11.881 | APE10-dist-in | 7.591 | APE9-dist-in | 3.376 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.499 | 0.184 | 0.234 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7djo | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DL6A | 215 | 538 | 601.0 | H96:601 | Type1 | Inactive | DFGin | 7.152 | 15.218 | BLAminus | -117.62, -177.39 | 53.85, 78.98 | -93.5, 18.12 | 285.84, 68.07 | -63.99, -13.06 | in-in | in | 9.043 | Saltbr-in | 2.543 | HRD-in | -67.53, -45.24 | 75.47, 0.91 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.92 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -125.16, 165.64 | APE9-dihe-na | 68.7, 158.66 | APE8-dihe-in | -84.48, 139.38 | APE8-rot-out | 172.15 | APE67-dihe-in | -59.22, -22.44 | -52.23, -48.32 | APE12-dist-in | 13.001 | APE11-dist-in | 11.777 | APE10-dist-in | 7.505 | APE9-dist-in | 3.173 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.648 | 0.177 | 0.232 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dl6 | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DH3A | 213 | 538 | 601.0 | H7C:601 | Type1 | Inactive | DFGin | 7.045 | 15.26 | BLAminus | -119.08, -179.53 | 58.29, 74.58 | -88.67, 21.96 | 286.19, 71.25 | -64.16, -21.81 | in-in | in | 8.924 | Saltbr-in | 3.399 | HRD-in | -71.55, -47.36 | 71.56, 3.54 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.739 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -134.02, 171.08 | APE9-dihe-na | 72.29, 151.84 | APE8-dihe-in | -71.94, 135.94 | APE8-rot-out | 194.0 | APE67-dihe-in | -56.42, -28.28 | -53.31, -46.8 | APE12-dist-in | 13.015 | APE11-dist-in | 11.909 | APE10-dist-in | 7.475 | APE9-dist-in | 3.347 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.33 | 0.195 | 0.217 | A | 326 | 326 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dh3 | CMGC_DYRK2_HUMAN | CMGC | 5.5e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7DHVA | 212 | 538 | 601.0 | H7X:601 | Type1 | Inactive | DFGin | 7.004 | 15.218 | BLAminus | -128.46, -170.28 | 43.26, 83.31 | -95.73, 25.21 | 286.23, 69.56 | -68.03, -32.6 | in-in | in | 8.932 | Saltbr-in | 2.635 | HRD-in | -77.4, -41.95 | 73.79, 2.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.712 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -125.51, 169.17 | APE9-dihe-na | 70.62, 163.65 | APE8-dihe-in | -91.1, 137.8 | APE8-rot-out | 165.09 | APE67-dihe-in | -63.71, -20.64 | -53.82, -42.56 | APE12-dist-in | 12.705 | APE11-dist-in | 11.639 | APE10-dist-in | 7.382 | APE9-dist-in | 3.329 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.679 | 0.193 | 0.249 | A | 327 | 327 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhv | CMGC_DYRK2_HUMAN | CMGC | 5.6e-99 | 337.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 4AZFA | 146 | 536 | 601.0 | 3RA:60600 | Type1 | Inactive | DFGin | 6.995 | 15.39 | BLAminus | -118.77, 179.61 | 61.33, 77.52 | -93.54, 30.44 | 283.47, 77.53 | -76.64, -12.42 | in-in | in | 9.082 | Saltbr-in | 2.733 | HRD-in | -73.11, -47.79 | 80.4, -7.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.921 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -141.82, 174.61 | APE9-dihe-na | 70.03, 158.03 | APE8-dihe-in | -81.89, 134.84 | APE8-rot-out | 174.41 | APE67-dihe-in | -64.03, -20.73 | -38.64, -55.03 | APE12-dist-in | 10.247 | APE11-dist-in | 11.617 | APE10-dist-in | 7.116 | APE9-dist-in | 3.212 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.55 | 0.2 | 0.255 | A | 417 | 389 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 4azf | CMGC_DYRK2_HUMAN | CMGC | 1.3e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7EJVB | 153 | 543 | 601.0 | YK2:60501 | Type1 | Inactive | DFGin | 7.155 | 15.775 | BLAminus | -119.43, -178.81 | 52.81, 76.66 | -89.1, 19.14 | 283.4, 73.64 | -64.56, -23.63 | in-out | in | 8.918 | Saltbr-out | 3.623 | HRD-in | -70.75, -42.53 | 75.19, 1.74 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.874 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.05, 163.39 | APE9-dihe-na | 74.33, 145.19 | APE8-dihe-in | -65.87, 144.25 | APE8-rot-in | 282.1 | APE67-dihe-in | -56.42, -28.58 | -55.11, -50.7 | APE12-dist-in | 13.028 | APE11-dist-in | 11.768 | APE10-dist-in | 7.569 | APE9-dist-in | 3.367 | None | PTR382 | PTR382 | XRAY | 2.5 | 0.202 | 0.246 | B | 391 | 391 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7ejv | CMGC_DYRK2_HUMAN | CMGC | 1.1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 3KVWA | 146 | 536 | 601.0 | IRB:60001 | Type1 | Inactive | DFGin | 6.948 | 15.117 | BLAminus | -111.07, -179.04 | 64.3, 75.68 | -93.62, 22.45 | 282.14, 79.62 | -72.21, -11.84 | in-in | in | 9.088 | Saltbr-in | 2.684 | HRD-in | -73.11, -47.89 | 78.54, -3.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.901 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -142.44, 168.47 | APE9-dihe-na | 69.36, 159.88 | APE8-dihe-in | -78.87, 139.14 | APE8-rot-out | 177.13 | APE67-dihe-in | -55.72, -26.97 | -53.0, -51.24 | APE12-dist-in | 13.447 | APE11-dist-in | 11.708 | APE10-dist-in | 7.236 | APE9-dist-in | 3.158 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.28 | 0.211 | 0.26 | A | 429 | 389 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 3kvw | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 5ZTNA | 146 | 536 | 601.0 | CUR:60501 | Type1 | Inactive | DFGin | 7.044 | 14.917 | BLAminus | -121.02, -170.84 | 55.37, 74.14 | -90.27, 24.89 | 284.91, 71.59 | -68.02, -21.72 | in-in | in | 9.038 | Saltbr-in | 3.201 | HRD-in | -75.34, -43.05 | 70.76, 4.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.991 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.75, -1.92 | APE9-dihe-na | -118.6, 178.64 | APE8-dihe-in | -75.97, 135.26 | APE8-rot-out | 181.93 | APE67-dihe-in | -60.16, -23.88 | -54.39, -47.99 | APE12-dist-in | 13.019 | APE11-dist-in | 11.6 | APE10-dist-in | 7.156 | APE9-dist-in | 3.639 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.496 | 0.2 | 0.244 | A | 429 | 384 | 7 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5ztn | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 5ZTNB | 146 | 536 | 601.0 | CUR:60501 | Type1 | Inactive | DFGin | 6.985 | 14.938 | BLAminus | -121.23, -170.26 | 54.62, 73.44 | -89.58, 24.17 | 284.13, 70.16 | -67.88, -20.27 | in-in | in | 9.125 | Saltbr-in | 3.318 | HRD-in | -75.96, -42.97 | 70.51, 4.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.915 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.98, -2.03 | APE9-dihe-na | -118.4, 178.1 | APE8-dihe-in | -73.54, 134.92 | APE8-rot-out | 181.22 | APE67-dihe-in | -60.19, -23.13 | -53.91, -47.68 | APE12-dist-in | 13.056 | APE11-dist-in | 11.551 | APE10-dist-in | 7.147 | APE9-dist-in | 3.663 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.496 | 0.2 | 0.244 | B | 429 | 384 | 7 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5ztn | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 6HDPA | 146 | 542 | 601.0 | FZ5:60501 | Type1 | Inactive | DFGin | 6.931 | 15.235 | BLAminus | -114.28, 179.49 | 62.03, 77.41 | -96.04, 25.56 | 278.7, 72.31 | -76.29, -11.59 | in-in | in | 9.224 | Saltbr-in | 3.383 | HRD-in | -70.91, -50.83 | 77.22, 0.35 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.763 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -141.94, 167.37 | APE9-dihe-na | 71.47, 153.79 | APE8-dihe-in | -72.94, 137.06 | APE8-rot-out | 179.54 | APE67-dihe-in | -60.52, -24.48 | -51.62, -50.78 | APE12-dist-in | 13.278 | APE11-dist-in | 11.659 | APE10-dist-in | 7.064 | APE9-dist-in | 3.22 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.3 | 0.186 | 0.238 | A | 429 | 397 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 6hdp | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 6HDRA | 146 | 536 | 601.0 | CC9:60501 | Type1 | Inactive | DFGin | 6.939 | 14.832 | BLAminus | -116.98, -175.8 | 60.97, 77.21 | -96.77, 23.88 | 280.67, 81.52 | -78.88, -6.9 | in-in | in | 9.328 | Saltbr-in | 3.505 | HRD-in | -71.46, -52.99 | 79.25, 3.29 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.804 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.88, 167.44 | APE9-dihe-na | 70.73, 153.88 | APE8-dihe-in | -70.98, 134.66 | APE8-rot-out | 177.54 | APE67-dihe-in | -61.24, -20.91 | -50.8, -48.3 | APE12-dist-in | 12.885 | APE11-dist-in | 11.357 | APE10-dist-in | 6.899 | APE9-dist-in | 3.222 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.2 | 0.192 | 0.243 | A | 429 | 389 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 6hdr | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 7AKFA | 146 | 535 | 601.0 | RK5:60601 | Type1 | Inactive | DFGin | 6.785 | 14.751 | BLAminus | -116.54, -178.37 | 61.83, 93.06 | -112.09, 28.57 | 283.6, 77.78 | -86.48, 0.57 | in-in | in | 8.763 | Saltbr-in | 2.658 | HRD-in | -67.66, -54.85 | 75.7, 9.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.989 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -135.94, 166.25 | APE9-dihe-na | 63.8, 156.1 | APE8-dihe-in | -67.55, 128.45 | APE8-rot-out | 225.46 | APE67-dihe-in | -65.91, -25.18 | -38.34, -48.5 | APE12-dist-in | 12.873 | APE11-dist-in | 11.166 | APE10-dist-in | 6.714 | APE9-dist-in | 3.342 | None | SEP232,PTR382,SEP458 | SEP232,PTR382,SEP458 | XRAY | 2.6 | 0.192 | 0.259 | A | 429 | 390 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7akf | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 5LXCA | 153 | 536 | 601.0 | 7AA:60501 | Type1 | Inactive | DFGin | 7.077 | 15.396 | BLAminus | -127.7, 168.29 | 65.71, 89.28 | -103.99, 15.3 | 281.54, 81.72 | -66.81, -20.15 | in-in | in | 8.692 | Saltbr-in | 2.893 | HRD-in | -69.9, -43.78 | 75.48, 2.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.899 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.55, 166.23 | APE9-dihe-na | 72.78, 145.6 | APE8-dihe-in | -76.68, 135.17 | APE8-rot-out | 177.09 | APE67-dihe-in | -59.77, -30.24 | -44.95, -46.79 | APE12-dist-in | 13.342 | APE11-dist-in | 11.748 | APE10-dist-in | 7.517 | APE9-dist-in | 3.286 | None | PTR382 | PTR382 | XRAY | 2.15 | 0.208 | 0.254 | A | 408 | 384 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxc | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 5LXCB | 153 | 538 | 601.0 | 7AA:60501 | Type1 | Inactive | DFGin | 7.058 | 15.351 | BLAminus | -125.13, 171.0 | 62.64, 89.27 | -105.23, 19.5 | 281.52, 82.75 | -66.91, -27.57 | in-in | in | 8.807 | Saltbr-in | 2.978 | HRD-in | -70.76, -50.91 | 83.26, -7.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.943 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -139.21, 164.87 | APE9-dihe-na | 72.46, 149.37 | APE8-dihe-in | -74.96, 138.82 | APE8-rot-out | 175.15 | APE67-dihe-in | -59.45, -29.64 | -49.5, -49.1 | APE12-dist-in | 13.348 | APE11-dist-in | 11.697 | APE10-dist-in | 7.461 | APE9-dist-in | 3.137 | None | PTR382 | PTR382 | XRAY | 2.15 | 0.208 | 0.254 | B | 408 | 386 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxc | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 5LXDA | 153 | 538 | 601.0 | 7A7:60501 | Type1 | Inactive | DFGin | 7.044 | 15.038 | BLAminus | -123.98, 173.69 | 67.75, 85.87 | -103.32, 20.02 | 290.69, 80.27 | -60.79, -26.58 | in-in | in | 8.985 | Saltbr-in | 2.718 | HRD-in | -78.02, -45.82 | 73.2, 0.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.933 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.87, 166.87 | APE9-dihe-na | 75.57, 144.69 | APE8-dihe-in | -63.57, 135.03 | APE8-rot-out | 186.77 | APE67-dihe-in | -56.98, -18.46 | -55.94, -51.68 | APE12-dist-in | 13.257 | APE11-dist-in | 12.121 | APE10-dist-in | 7.648 | APE9-dist-in | 3.33 | None | PTR382 | PTR382 | XRAY | 2.58 | 0.2 | 0.253 | A | 408 | 386 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxd | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 5LXDB | 153 | 538 | 601.0 | 7A7:60501 | Type1 | Inactive | DFGin | 7.017 | 15.002 | BLAminus | -125.15, 174.13 | 66.86, 85.87 | -102.41, 18.55 | 290.97, 80.01 | -60.53, -24.71 | in-in | in | 8.991 | Saltbr-in | 2.786 | HRD-in | -79.02, -46.62 | 74.88, 2.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.867 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.84, 168.16 | APE9-dihe-na | 73.17, 145.14 | APE8-dihe-in | -63.72, 133.94 | APE8-rot-out | 182.75 | APE67-dihe-in | -55.28, -20.15 | -52.56, -53.24 | APE12-dist-in | 13.282 | APE11-dist-in | 12.127 | APE10-dist-in | 7.665 | APE9-dist-in | 3.299 | None | PTR382 | PTR382 | XRAY | 2.58 | 0.2 | 0.253 | B | 408 | 386 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxd | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 6K0JA | 212 | 536 | 601.0 | CQO:60601 | Type1 | Inactive | DFGin | 7.065 | 15.359 | BLAminus | -116.77, 179.78 | 59.52, 75.88 | -89.73, 24.44 | 286.49, 66.6 | -65.24, -18.56 | in-in | in | 9.258 | Saltbr-in | 2.849 | HRD-in | -66.29, -47.14 | 70.83, 1.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.859 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.01, 167.62 | APE9-dihe-na | 74.56, 150.55 | APE8-dihe-in | -69.83, 137.05 | APE8-rot-out | 181.49 | APE67-dihe-in | -55.27, -26.64 | -53.33, -50.0 | APE12-dist-in | 13.006 | APE11-dist-in | 11.846 | APE10-dist-in | 7.514 | APE9-dist-in | 3.362 | E256N,L349A | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.352 | 0.175 | 0.209 | A | 327 | 325 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 6k0j | CMGC_DYRK2_HUMAN | CMGC | 5.6e-98 | 333.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 9KQYA | 151 | 537 | 601.0 | No_ligand | No_ligand | Inactive | DFGin | 6.559 | 15.306 | None | -118.46, -58.2 | -76.39, 93.69 | -100.84, 14.42 | 280.8, 85.79 | -66.94, -30.92 | in-in | in | 8.842 | Saltbr-in | 2.954 | HRD-in | -69.15, -42.93 | 69.8, -4.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.747 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.16, 173.73 | APE9-dihe-na | 69.18, 145.61 | APE8-dihe-in | -65.57, 148.39 | APE8-rot-in | 308.71 | APE67-dihe-in | -62.63, -39.04 | -60.44, -42.14 | APE12-dist-in | 13.024 | APE11-dist-in | 11.654 | APE10-dist-in | 7.133 | APE9-dist-in | 3.15 | None | PTR382 | PTR382 | XRAY | 3.2 | 0.233 | 0.276 | A | 407 | 387 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 9kqy | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 8HLTB | 151 | 537 | 601.0 | XSE:60501 | Type1 | Inactive | DFGin | 6.677 | 15.172 | None | -123.1, -45.42 | -92.76, 76.97 | -82.13, 19.07 | 287.19, 77.16 | -64.05, -27.16 | in-in | in | 8.966 | Saltbr-in | 2.975 | HRD-in | -75.54, -44.65 | 72.51, -4.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.784 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.69, 168.46 | APE9-dihe-na | 73.66, 156.43 | APE8-dihe-in | -77.8, 146.18 | APE8-rot-in | 309.51 | APE67-dihe-in | -59.07, -35.58 | -50.16, -47.35 | APE12-dist-in | 12.987 | APE11-dist-in | 11.623 | APE10-dist-in | 7.106 | APE9-dist-in | 3.124 | None | PTR382 | PTR382 | XRAY | 2.8 | 0.213 | 0.267 | B | 393 | 387 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 8hlt | CMGC_DYRK2_HUMAN | CMGC | 1.1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| 9KQYB | 151 | 537 | 601.0 | A1L6I:60501 | Type1 | Inactive | DFGin | 6.842 | 15.41 | None | -119.38, -59.48 | -76.49, 94.24 | -100.04, 16.54 | 278.63, 76.93 | -66.67, -33.1 | in-in | in | 8.734 | Saltbr-in | 2.848 | HRD-in | -67.3, -42.38 | 69.63, -4.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.752 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.07, 173.43 | APE9-dihe-na | 69.88, 144.62 | APE8-dihe-in | -65.72, 149.7 | APE8-rot-in | 302.89 | APE67-dihe-in | -61.87, -38.72 | -60.58, -43.15 | APE12-dist-in | 12.537 | APE11-dist-in | 11.054 | APE10-dist-in | 6.618 | APE9-dist-in | 3.234 | None | PTR382 | PTR382 | XRAY | 3.2 | 0.233 | 0.276 | B | 407 | 387 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 9kqy | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DYRK2_HUMAN | AF-Q92630-K1A | Q92630 | 214 | 543 | 601.0 | No_ligand | No_ligand | Active | DFGin | 6.939 | 14.864 | BLAminus | -126.07, 177.15 | 62.42, 65.44 | -81.73, 10.25 | 284.63, 80.53 | -64.64, -17.85 | in-in | in | 8.728 | Saltbr-in | 2.723 | HRD-in | -66.96, -37.74 | 67.08, -16.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.848 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.84, 175.12 | APE9-dihe-na | 60.6, 144.79 | APE8-dihe-in | -65.13, 137.41 | APE8-rot-in | 294.19 | APE67-dihe-in | -65.52, -19.21 | -50.69, -46.33 | APE12-dist-in | 12.882 | APE11-dist-in | 11.334 | APE10-dist-in | 7.287 | APE9-dist-in | 3.021 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 330 | 330 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | AF-Q92630-K1 | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.8e-99 | 337.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | AF-Q92630-K3A | Q92630 | 214 | 543 | 601.0 | No_ligand | No_ligand | Active | DFGin | 6.623 | 14.471 | BLAminus | -128.09, 177.13 | 63.4, 64.99 | -80.7, 10.08 | 289.17, 77.94 | -66.05, -16.49 | in-in | in | 8.839 | Saltbr-in | 2.734 | HRD-in | -72.99, -34.76 | 62.62, -5.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.882 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.48, 175.5 | APE9-dihe-na | 61.64, 142.59 | APE8-dihe-in | -63.51, 134.37 | APE8-rot-in | 293.35 | APE67-dihe-in | -63.69, -20.47 | -54.61, -45.06 | APE12-dist-in | 12.796 | APE11-dist-in | 11.341 | APE10-dist-in | 7.03 | APE9-dist-in | 3.09 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 330 | 330 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | AF-Q92630-K3 | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.8e-99 | 337.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7EJVA | Q92630 | 151 | 537 | 601.0 | YK2:60501 | Type1 | Active | DFGin | 6.9 | 15.424 | BLAminus | -121.6, -175.71 | 52.95, 74.47 | -89.12, 21.12 | 283.92, 70.74 | -60.92, -24.61 | in-in | in | 8.982 | Saltbr-in | 3.13 | HRD-in | -72.41, -42.76 | 75.36, 0.64 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.755 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.92, 162.27 | APE9-dihe-na | 76.47, 145.84 | APE8-dihe-in | -66.78, 142.47 | APE8-rot-in | 275.38 | APE67-dihe-in | -56.79, -30.59 | -58.46, -46.41 | APE12-dist-in | 12.918 | APE11-dist-in | 11.297 | APE10-dist-in | 6.969 | APE9-dist-in | 3.304 | None | PTR382 | PTR382 | XRAY | 2.5 | 0.202 | 0.246 | A | 387 | 385 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7ejv | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 8HLTA | Q92630 | 151 | 535 | 601.0 | XSE:60501 | Type1 | Active | DFGin | 7.153 | 15.661 | BLAminus | -128.03, -174.41 | 42.45, 74.99 | -83.08, 17.4 | 279.93, 74.95 | -62.5, -19.89 | in-in | in | 9.177 | Saltbr-in | 2.717 | HRD-in | -71.74, -44.48 | 73.83, 0.55 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.747 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.16, 170.0 | APE9-dihe-na | 71.16, 164.17 | APE8-dihe-in | -84.62, 135.53 | APE8-rot-in | 250.25 | APE67-dihe-in | -56.1, -31.76 | -49.25, -50.28 | APE12-dist-in | 13.315 | APE11-dist-in | 11.966 | APE10-dist-in | 7.57 | APE9-dist-in | 3.21 | None | PTR382 | PTR382 | XRAY | 2.8 | 0.213 | 0.267 | A | 393 | 385 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 8hlt | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7AKHA | Q92630 | 146 | 535 | 601.0 | RK8:60601 | Type1 | Active | DFGin | 6.926 | 15.074 | BLAminus | -121.6, -171.14 | 52.21, 81.66 | -96.01, 25.36 | 287.39, 72.64 | -67.66, -23.05 | in-in | in | 9.121 | Saltbr-in | 2.705 | HRD-in | -56.66, -58.54 | 81.07, -0.93 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.821 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.43, 168.94 | APE9-dihe-na | 72.6, 150.47 | APE8-dihe-in | -61.43, 140.56 | APE8-rot-in | 278.26 | APE67-dihe-in | -62.31, -24.44 | -52.56, -49.45 | APE12-dist-in | 12.815 | APE11-dist-in | 11.442 | APE10-dist-in | 6.914 | APE9-dist-in | 3.229 | None | SEP232,PTR382,SEP458 | SEP232,PTR382,SEP458 | XRAY | 2.85 | 0.188 | 0.245 | A | 429 | 390 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7akh | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 3K2LA | Q92630 | 146 | 543 | 601.0 | No_ligand | No_ligand | Inactive | DFGin | 7.095 | 15.241 | BLAminus | -127.38, 178.65 | 61.29, 89.71 | -107.22, 23.8 | 277.85, 81.5 | -75.9, -16.57 | in-in | in | 8.858 | Saltbr-in | 2.965 | HRD-in | -80.34, -48.51 | 75.91, -1.73 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.974 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.89, 168.99 | APE9-dihe-na | 66.37, 164.94 | APE8-dihe-in | -92.92, 137.86 | APE8-rot-out | 183.76 | APE67-dihe-in | -63.43, -18.18 | -49.75, -48.38 | APE12-dist-in | 12.59 | APE11-dist-in | 11.884 | APE10-dist-in | 7.261 | APE9-dist-in | 3.098 | None | SEP232,TPO381,PTR382,SEP442,SEP458 | SEP232,TPO381,PTR382,SEP442,SEP458 | XRAY | 2.36 | 0.228 | 0.288 | A | 429 | 397 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 3k2l | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DG4A | Q92630 | 215 | 538 | 601.0 | H5R:601 | Type1 | Inactive | DFGin | 7.076 | 15.315 | BLAminus | -112.18, -176.63 | 54.26, 82.32 | -95.55, 24.49 | 281.35, 68.71 | -70.68, -16.69 | in-in | in | 9.062 | Saltbr-in | 2.632 | HRD-in | -72.69, -45.13 | 72.43, 4.61 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.829 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -123.35, 168.65 | APE9-dihe-na | 72.59, 152.62 | APE8-dihe-in | -75.5, 133.34 | APE8-rot-out | 190.89 | APE67-dihe-in | -53.88, -27.24 | -50.74, -49.3 | APE12-dist-in | 13.02 | APE11-dist-in | 11.794 | APE10-dist-in | 7.365 | APE9-dist-in | 3.357 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.58 | 0.206 | 0.249 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dg4 | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DH9A | Q92630 | 215 | 538 | 601.0 | H7F:601 | Type1 | Inactive | DFGin | 6.955 | 15.393 | BLAminus | -118.25, -176.44 | 52.33, 72.66 | -86.4, 22.32 | 285.5, 71.17 | -68.46, -16.6 | in-in | in | 9.091 | Saltbr-in | 2.818 | HRD-in | -67.52, -48.86 | 77.78, -1.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.826 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.21, 165.64 | APE9-dihe-na | 77.26, 152.01 | APE8-dihe-in | -71.35, 136.19 | APE8-rot-out | 186.16 | APE67-dihe-in | -56.24, -27.47 | -53.15, -48.91 | APE12-dist-in | 13.085 | APE11-dist-in | 11.935 | APE10-dist-in | 7.588 | APE9-dist-in | 3.308 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.194 | 0.19 | 0.218 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dh9 | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DHCA | Q92630 | 215 | 538 | 601.0 | H99:601 | Type1 | Inactive | DFGin | 6.897 | 15.183 | BLAminus | -120.85, -173.65 | 54.47, 76.85 | -89.75, 13.16 | 285.05, 71.42 | -59.73, -14.3 | in-in | in | 9.165 | Saltbr-in | 2.836 | HRD-in | -67.26, -47.7 | 73.48, 5.77 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.79 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -124.28, 171.52 | APE9-dihe-na | 72.07, 147.78 | APE8-dihe-in | -70.3, 140.28 | APE8-rot-out | 189.19 | APE67-dihe-in | -57.12, -25.22 | -59.04, -44.86 | APE12-dist-in | 13.016 | APE11-dist-in | 11.9 | APE10-dist-in | 7.482 | APE9-dist-in | 3.275 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.592 | 0.17 | 0.217 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhc | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DHHA | Q92630 | 215 | 538 | 601.0 | H7L:601 | Type1 | Inactive | DFGin | 7.002 | 15.315 | BLAminus | -121.49, -175.98 | 53.38, 75.83 | -90.0, 17.27 | 285.73, 67.63 | -60.12, -17.2 | in-in | in | 9.069 | Saltbr-in | 2.831 | HRD-in | -72.48, -43.45 | 72.8, 3.03 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.934 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -112.98, 162.3 | APE9-dihe-na | 71.38, 148.19 | APE8-dihe-in | -71.4, 141.57 | APE8-rot-out | 161.34 | APE67-dihe-in | -65.17, -19.89 | -55.14, -43.22 | APE12-dist-in | 12.9 | APE11-dist-in | 11.849 | APE10-dist-in | 7.619 | APE9-dist-in | 3.387 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.486 | 0.195 | 0.245 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhh | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DHKA | Q92630 | 215 | 538 | 601.0 | H7O:601 | Type1 | Inactive | DFGin | 7.052 | 15.35 | BLAminus | -117.35, 177.72 | 56.81, 75.07 | -85.18, 19.92 | 283.41, 63.05 | -63.85, -33.36 | in-in | in | 9.196 | Saltbr-in | 2.644 | HRD-in | -71.37, -46.63 | 75.15, -1.94 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.906 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -118.3, 166.48 | APE9-dihe-na | 68.65, 147.66 | APE8-dihe-in | -62.61, 137.42 | APE8-rot-out | 200.1 | APE67-dihe-in | -57.5, -27.74 | -53.83, -48.57 | APE12-dist-in | 12.955 | APE11-dist-in | 11.738 | APE10-dist-in | 7.593 | APE9-dist-in | 3.202 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.341 | 0.199 | 0.257 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhk | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DHNA | Q92630 | 215 | 538 | 601.0 | H7R:601 | Type1 | Inactive | DFGin | 6.943 | 15.204 | BLAminus | -121.26, -177.62 | 55.21, 78.31 | -90.06, 20.47 | 287.34, 73.71 | -59.07, -25.63 | in-out | in | 9.064 | Saltbr-out | 3.683 | HRD-in | -71.04, -47.07 | 70.57, 6.17 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.681 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.33, 167.28 | APE9-dihe-na | 70.26, 153.99 | APE8-dihe-in | -74.79, 138.71 | APE8-rot-out | 162.7 | APE67-dihe-in | -57.15, -24.62 | -55.14, -47.5 | APE12-dist-in | 13.035 | APE11-dist-in | 11.859 | APE10-dist-in | 7.473 | APE9-dist-in | 3.339 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.38 | 0.187 | 0.223 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhn | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DHOA | Q92630 | 215 | 538 | 601.0 | H7U:601 | Type1 | Inactive | DFGin | 7.024 | 15.384 | BLAminus | -119.43, -172.42 | 42.56, 78.27 | -84.62, 15.62 | 281.95, 67.94 | -55.62, -33.56 | in-in | in | 9.274 | Saltbr-in | 2.624 | HRD-in | -82.16, -38.69 | 68.11, 7.67 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.83 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -109.77, 178.86 | APE9-dihe-na | 69.78, 147.69 | APE8-dihe-in | -69.75, 134.88 | APE8-rot-out | 211.6 | APE67-dihe-in | -60.55, -23.47 | -49.02, -52.25 | APE12-dist-in | 12.813 | APE11-dist-in | 11.959 | APE10-dist-in | 7.417 | APE9-dist-in | 3.473 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 3.29 | 0.188 | 0.259 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dho | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DJOA | Q92630 | 215 | 538 | 601.0 | H80:601 | Type1 | Inactive | DFGin | 6.825 | 15.46 | BLAminus | -127.28, -171.08 | 53.55, 75.01 | -93.19, 14.88 | 276.88, 71.94 | -62.8, -14.89 | in-in | in | 9.123 | Saltbr-in | 2.61 | HRD-in | -68.11, -47.05 | 70.53, 3.02 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.794 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -112.85, 165.38 | APE9-dihe-na | 72.88, 157.2 | APE8-dihe-in | -82.18, 142.51 | APE8-rot-out | 184.87 | APE67-dihe-in | -72.03, -23.08 | -61.29, -39.89 | APE12-dist-in | 12.99 | APE11-dist-in | 11.881 | APE10-dist-in | 7.591 | APE9-dist-in | 3.376 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.499 | 0.184 | 0.234 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7djo | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DL6A | Q92630 | 215 | 538 | 601.0 | H96:601 | Type1 | Inactive | DFGin | 7.152 | 15.218 | BLAminus | -117.62, -177.39 | 53.85, 78.98 | -93.5, 18.12 | 285.84, 68.07 | -63.99, -13.06 | in-in | in | 9.043 | Saltbr-in | 2.543 | HRD-in | -67.53, -45.24 | 75.47, 0.91 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.92 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -125.16, 165.64 | APE9-dihe-na | 68.7, 158.66 | APE8-dihe-in | -84.48, 139.38 | APE8-rot-out | 172.15 | APE67-dihe-in | -59.22, -22.44 | -52.23, -48.32 | APE12-dist-in | 13.001 | APE11-dist-in | 11.777 | APE10-dist-in | 7.505 | APE9-dist-in | 3.173 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.648 | 0.177 | 0.232 | A | 324 | 324 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dl6 | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.4e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DH3A | Q92630 | 213 | 538 | 601.0 | H7C:601 | Type1 | Inactive | DFGin | 7.045 | 15.26 | BLAminus | -119.08, -179.53 | 58.29, 74.58 | -88.67, 21.96 | 286.19, 71.25 | -64.16, -21.81 | in-in | in | 8.924 | Saltbr-in | 3.399 | HRD-in | -71.55, -47.36 | 71.56, 3.54 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.739 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -134.02, 171.08 | APE9-dihe-na | 72.29, 151.84 | APE8-dihe-in | -71.94, 135.94 | APE8-rot-out | 194.0 | APE67-dihe-in | -56.42, -28.28 | -53.31, -46.8 | APE12-dist-in | 13.015 | APE11-dist-in | 11.909 | APE10-dist-in | 7.475 | APE9-dist-in | 3.347 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.33 | 0.195 | 0.217 | A | 326 | 326 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dh3 | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.5e-99 | 337.1 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7DHVA | Q92630 | 212 | 538 | 601.0 | H7X:601 | Type1 | Inactive | DFGin | 7.004 | 15.218 | BLAminus | -128.46, -170.28 | 43.26, 83.31 | -95.73, 25.21 | 286.23, 69.56 | -68.03, -32.6 | in-in | in | 8.932 | Saltbr-in | 2.635 | HRD-in | -77.4, -41.95 | 73.79, 2.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.712 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -125.51, 169.17 | APE9-dihe-na | 70.62, 163.65 | APE8-dihe-in | -91.1, 137.8 | APE8-rot-out | 165.09 | APE67-dihe-in | -63.71, -20.64 | -53.82, -42.56 | APE12-dist-in | 12.705 | APE11-dist-in | 11.639 | APE10-dist-in | 7.382 | APE9-dist-in | 3.329 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.679 | 0.193 | 0.249 | A | 327 | 327 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7dhv | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.6e-99 | 337.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 4AZFA | Q92630 | 146 | 536 | 601.0 | 3RA:60600 | Type1 | Inactive | DFGin | 6.995 | 15.39 | BLAminus | -118.77, 179.61 | 61.33, 77.52 | -93.54, 30.44 | 283.47, 77.53 | -76.64, -12.42 | in-in | in | 9.082 | Saltbr-in | 2.733 | HRD-in | -73.11, -47.79 | 80.4, -7.32 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.921 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -141.82, 174.61 | APE9-dihe-na | 70.03, 158.03 | APE8-dihe-in | -81.89, 134.84 | APE8-rot-out | 174.41 | APE67-dihe-in | -64.03, -20.73 | -38.64, -55.03 | APE12-dist-in | 10.247 | APE11-dist-in | 11.617 | APE10-dist-in | 7.116 | APE9-dist-in | 3.212 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.55 | 0.2 | 0.255 | A | 417 | 389 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 4azf | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.3e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7EJVB | Q92630 | 153 | 543 | 601.0 | YK2:60501 | Type1 | Inactive | DFGin | 7.155 | 15.775 | BLAminus | -119.43, -178.81 | 52.81, 76.66 | -89.1, 19.14 | 283.4, 73.64 | -64.56, -23.63 | in-out | in | 8.918 | Saltbr-out | 3.623 | HRD-in | -70.75, -42.53 | 75.19, 1.74 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.874 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.05, 163.39 | APE9-dihe-na | 74.33, 145.19 | APE8-dihe-in | -65.87, 144.25 | APE8-rot-in | 282.1 | APE67-dihe-in | -56.42, -28.58 | -55.11, -50.7 | APE12-dist-in | 13.028 | APE11-dist-in | 11.768 | APE10-dist-in | 7.569 | APE9-dist-in | 3.367 | None | PTR382 | PTR382 | XRAY | 2.5 | 0.202 | 0.246 | B | 391 | 391 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7ejv | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 3KVWA | Q92630 | 146 | 536 | 601.0 | IRB:60001 | Type1 | Inactive | DFGin | 6.948 | 15.117 | BLAminus | -111.07, -179.04 | 64.3, 75.68 | -93.62, 22.45 | 282.14, 79.62 | -72.21, -11.84 | in-in | in | 9.088 | Saltbr-in | 2.684 | HRD-in | -73.11, -47.89 | 78.54, -3.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.901 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -142.44, 168.47 | APE9-dihe-na | 69.36, 159.88 | APE8-dihe-in | -78.87, 139.14 | APE8-rot-out | 177.13 | APE67-dihe-in | -55.72, -26.97 | -53.0, -51.24 | APE12-dist-in | 13.447 | APE11-dist-in | 11.708 | APE10-dist-in | 7.236 | APE9-dist-in | 3.158 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.28 | 0.211 | 0.26 | A | 429 | 389 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 3kvw | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 5ZTNA | Q92630 | 146 | 536 | 601.0 | CUR:60501 | Type1 | Inactive | DFGin | 7.044 | 14.917 | BLAminus | -121.02, -170.84 | 55.37, 74.14 | -90.27, 24.89 | 284.91, 71.59 | -68.02, -21.72 | in-in | in | 9.038 | Saltbr-in | 3.201 | HRD-in | -75.34, -43.05 | 70.76, 4.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.991 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.75, -1.92 | APE9-dihe-na | -118.6, 178.64 | APE8-dihe-in | -75.97, 135.26 | APE8-rot-out | 181.93 | APE67-dihe-in | -60.16, -23.88 | -54.39, -47.99 | APE12-dist-in | 13.019 | APE11-dist-in | 11.6 | APE10-dist-in | 7.156 | APE9-dist-in | 3.639 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.496 | 0.2 | 0.244 | A | 429 | 384 | 7 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5ztn | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 5ZTNB | Q92630 | 146 | 536 | 601.0 | CUR:60501 | Type1 | Inactive | DFGin | 6.985 | 14.938 | BLAminus | -121.23, -170.26 | 54.62, 73.44 | -89.58, 24.17 | 284.13, 70.16 | -67.88, -20.27 | in-in | in | 9.125 | Saltbr-in | 3.318 | HRD-in | -75.96, -42.97 | 70.51, 4.22 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.915 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -132.98, -2.03 | APE9-dihe-na | -118.4, 178.1 | APE8-dihe-in | -73.54, 134.92 | APE8-rot-out | 181.22 | APE67-dihe-in | -60.19, -23.13 | -53.91, -47.68 | APE12-dist-in | 13.056 | APE11-dist-in | 11.551 | APE10-dist-in | 7.147 | APE9-dist-in | 3.663 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.496 | 0.2 | 0.244 | B | 429 | 384 | 7 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5ztn | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 6HDPA | Q92630 | 146 | 542 | 601.0 | FZ5:60501 | Type1 | Inactive | DFGin | 6.931 | 15.235 | BLAminus | -114.28, 179.49 | 62.03, 77.41 | -96.04, 25.56 | 278.7, 72.31 | -76.29, -11.59 | in-in | in | 9.224 | Saltbr-in | 3.383 | HRD-in | -70.91, -50.83 | 77.22, 0.35 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.763 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -141.94, 167.37 | APE9-dihe-na | 71.47, 153.79 | APE8-dihe-in | -72.94, 137.06 | APE8-rot-out | 179.54 | APE67-dihe-in | -60.52, -24.48 | -51.62, -50.78 | APE12-dist-in | 13.278 | APE11-dist-in | 11.659 | APE10-dist-in | 7.064 | APE9-dist-in | 3.22 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.3 | 0.186 | 0.238 | A | 429 | 397 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 6hdp | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 6HDRA | Q92630 | 146 | 536 | 601.0 | CC9:60501 | Type1 | Inactive | DFGin | 6.939 | 14.832 | BLAminus | -116.98, -175.8 | 60.97, 77.21 | -96.77, 23.88 | 280.67, 81.52 | -78.88, -6.9 | in-in | in | 9.328 | Saltbr-in | 3.505 | HRD-in | -71.46, -52.99 | 79.25, 3.29 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.804 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -130.88, 167.44 | APE9-dihe-na | 70.73, 153.88 | APE8-dihe-in | -70.98, 134.66 | APE8-rot-out | 177.54 | APE67-dihe-in | -61.24, -20.91 | -50.8, -48.3 | APE12-dist-in | 12.885 | APE11-dist-in | 11.357 | APE10-dist-in | 6.899 | APE9-dist-in | 3.222 | None | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.2 | 0.192 | 0.243 | A | 429 | 389 | 2 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 6hdr | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 7AKFA | Q92630 | 146 | 535 | 601.0 | RK5:60601 | Type1 | Inactive | DFGin | 6.785 | 14.751 | BLAminus | -116.54, -178.37 | 61.83, 93.06 | -112.09, 28.57 | 283.6, 77.78 | -86.48, 0.57 | in-in | in | 8.763 | Saltbr-in | 2.658 | HRD-in | -67.66, -54.85 | 75.7, 9.17 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.989 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -135.94, 166.25 | APE9-dihe-na | 63.8, 156.1 | APE8-dihe-in | -67.55, 128.45 | APE8-rot-out | 225.46 | APE67-dihe-in | -65.91, -25.18 | -38.34, -48.5 | APE12-dist-in | 12.873 | APE11-dist-in | 11.166 | APE10-dist-in | 6.714 | APE9-dist-in | 3.342 | None | SEP232,PTR382,SEP458 | SEP232,PTR382,SEP458 | XRAY | 2.6 | 0.192 | 0.259 | A | 429 | 390 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 7akf | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.5e-98 | 335.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 5LXCA | Q92630 | 153 | 536 | 601.0 | 7AA:60501 | Type1 | Inactive | DFGin | 7.077 | 15.396 | BLAminus | -127.7, 168.29 | 65.71, 89.28 | -103.99, 15.3 | 281.54, 81.72 | -66.81, -20.15 | in-in | in | 8.692 | Saltbr-in | 2.893 | HRD-in | -69.9, -43.78 | 75.48, 2.4 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.899 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.55, 166.23 | APE9-dihe-na | 72.78, 145.6 | APE8-dihe-in | -76.68, 135.17 | APE8-rot-out | 177.09 | APE67-dihe-in | -59.77, -30.24 | -44.95, -46.79 | APE12-dist-in | 13.342 | APE11-dist-in | 11.748 | APE10-dist-in | 7.517 | APE9-dist-in | 3.286 | None | PTR382 | PTR382 | XRAY | 2.15 | 0.208 | 0.254 | A | 408 | 384 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxc | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 5LXCB | Q92630 | 153 | 538 | 601.0 | 7AA:60501 | Type1 | Inactive | DFGin | 7.058 | 15.351 | BLAminus | -125.13, 171.0 | 62.64, 89.27 | -105.23, 19.5 | 281.52, 82.75 | -66.91, -27.57 | in-in | in | 8.807 | Saltbr-in | 2.978 | HRD-in | -70.76, -50.91 | 83.26, -7.25 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.943 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -139.21, 164.87 | APE9-dihe-na | 72.46, 149.37 | APE8-dihe-in | -74.96, 138.82 | APE8-rot-out | 175.15 | APE67-dihe-in | -59.45, -29.64 | -49.5, -49.1 | APE12-dist-in | 13.348 | APE11-dist-in | 11.697 | APE10-dist-in | 7.461 | APE9-dist-in | 3.137 | None | PTR382 | PTR382 | XRAY | 2.15 | 0.208 | 0.254 | B | 408 | 386 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxc | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 5LXDA | Q92630 | 153 | 538 | 601.0 | 7A7:60501 | Type1 | Inactive | DFGin | 7.044 | 15.038 | BLAminus | -123.98, 173.69 | 67.75, 85.87 | -103.32, 20.02 | 290.69, 80.27 | -60.79, -26.58 | in-in | in | 8.985 | Saltbr-in | 2.718 | HRD-in | -78.02, -45.82 | 73.2, 0.43 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.933 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.87, 166.87 | APE9-dihe-na | 75.57, 144.69 | APE8-dihe-in | -63.57, 135.03 | APE8-rot-out | 186.77 | APE67-dihe-in | -56.98, -18.46 | -55.94, -51.68 | APE12-dist-in | 13.257 | APE11-dist-in | 12.121 | APE10-dist-in | 7.648 | APE9-dist-in | 3.33 | None | PTR382 | PTR382 | XRAY | 2.58 | 0.2 | 0.253 | A | 408 | 386 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxd | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 5LXDB | Q92630 | 153 | 538 | 601.0 | 7A7:60501 | Type1 | Inactive | DFGin | 7.017 | 15.002 | BLAminus | -125.15, 174.13 | 66.86, 85.87 | -102.41, 18.55 | 290.97, 80.01 | -60.53, -24.71 | in-in | in | 8.991 | Saltbr-in | 2.786 | HRD-in | -79.02, -46.62 | 74.88, 2.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.867 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -136.84, 168.16 | APE9-dihe-na | 73.17, 145.14 | APE8-dihe-in | -63.72, 133.94 | APE8-rot-out | 182.75 | APE67-dihe-in | -55.28, -20.15 | -52.56, -53.24 | APE12-dist-in | 13.282 | APE11-dist-in | 12.127 | APE10-dist-in | 7.665 | APE9-dist-in | 3.299 | None | PTR382 | PTR382 | XRAY | 2.58 | 0.2 | 0.253 | B | 408 | 386 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 5lxd | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 6K0JA | Q92630 | 212 | 536 | 601.0 | CQO:60601 | Type1 | Inactive | DFGin | 7.065 | 15.359 | BLAminus | -116.77, 179.78 | 59.52, 75.88 | -89.73, 24.44 | 286.49, 66.6 | -65.24, -18.56 | in-in | in | 9.258 | Saltbr-in | 2.849 | HRD-in | -66.29, -47.14 | 70.83, 1.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.859 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -133.01, 167.62 | APE9-dihe-na | 74.56, 150.55 | APE8-dihe-in | -69.83, 137.05 | APE8-rot-out | 181.49 | APE67-dihe-in | -55.27, -26.64 | -53.33, -50.0 | APE12-dist-in | 13.006 | APE11-dist-in | 11.846 | APE10-dist-in | 7.514 | APE9-dist-in | 3.362 | E256N,L349A | PTR382,SEP458 | PTR382,SEP458 | XRAY | 2.352 | 0.175 | 0.209 | A | 327 | 325 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 6k0j | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 5.6e-98 | 333.8 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 9KQYA | Q92630 | 151 | 537 | 601.0 | No_ligand | No_ligand | Inactive | DFGin | 6.559 | 15.306 | None | -118.46, -58.2 | -76.39, 93.69 | -100.84, 14.42 | 280.8, 85.79 | -66.94, -30.92 | in-in | in | 8.842 | Saltbr-in | 2.954 | HRD-in | -69.15, -42.93 | 69.8, -4.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.747 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.16, 173.73 | APE9-dihe-na | 69.18, 145.61 | APE8-dihe-in | -65.57, 148.39 | APE8-rot-in | 308.71 | APE67-dihe-in | -62.63, -39.04 | -60.44, -42.14 | APE12-dist-in | 13.024 | APE11-dist-in | 11.654 | APE10-dist-in | 7.133 | APE9-dist-in | 3.15 | None | PTR382 | PTR382 | XRAY | 3.2 | 0.233 | 0.276 | A | 407 | 387 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 9kqy | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 8HLTB | Q92630 | 151 | 537 | 601.0 | XSE:60501 | Type1 | Inactive | DFGin | 6.677 | 15.172 | None | -123.1, -45.42 | -92.76, 76.97 | -82.13, 19.07 | 287.19, 77.16 | -64.05, -27.16 | in-in | in | 8.966 | Saltbr-in | 2.975 | HRD-in | -75.54, -44.65 | 72.51, -4.12 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.784 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -135.69, 168.46 | APE9-dihe-na | 73.66, 156.43 | APE8-dihe-in | -77.8, 146.18 | APE8-rot-in | 309.51 | APE67-dihe-in | -59.07, -35.58 | -50.16, -47.35 | APE12-dist-in | 12.987 | APE11-dist-in | 11.623 | APE10-dist-in | 7.106 | APE9-dist-in | 3.124 | None | PTR382 | PTR382 | XRAY | 2.8 | 0.213 | 0.267 | B | 393 | 387 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 8hlt | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.1e-98 | 336.2 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| DYRK2_HUMAN | 9KQYB | Q92630 | 151 | 537 | 601.0 | A1L6I:60501 | Type1 | Inactive | DFGin | 6.842 | 15.41 | None | -119.38, -59.48 | -76.49, 94.24 | -100.04, 16.54 | 278.63, 76.93 | -66.67, -33.1 | in-in | in | 8.734 | Saltbr-in | 2.848 | HRD-in | -67.3, -42.38 | 69.63, -4.95 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.752 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -120.07, 173.43 | APE9-dihe-na | 69.88, 144.62 | APE8-dihe-in | -65.72, 149.7 | APE8-rot-in | 302.89 | APE67-dihe-in | -61.87, -38.72 | -60.58, -43.15 | APE12-dist-in | 12.537 | APE11-dist-in | 11.054 | APE10-dist-in | 6.618 | APE9-dist-in | 3.234 | None | PTR382 | PTR382 | XRAY | 3.2 | 0.233 | 0.276 | B | 407 | 387 | 0 | 0 | 0 | 0 | [[222, 535]] | 1.0 | 9kqy | Homo sapiens | CMGC_DYRK2_HUMAN | CMGC | 1.2e-98 | 336.0 | 1 | 301 | 301 | 367 | 368 | 369 | 371 | 373 | 251 | 266 | 270 | 345 | 347 | 346 | 348 | 404 | 392 | 387 | 386 | 385 | 384 | 383 | 382 | 381 | 302 | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
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