CAMK_CHEK2 (Serine/threonine-protein kinase Chk2)

Total number of chains: 46
Active chains: 2
Uniprot: CHK2_HUMAN
Kinase Domain Residues: 220 - 486
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 40 87.0% AF-O96017-K1A
DFGin None 5 10.9% 3I6UB
DFGin BLAplus 1 2.2% 3I6UA

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CHEK2 AF-O96017-K1A O96017 212 494 543.0 No_ligand No_ligand Active DFGin 6.5446 14.1254 BLAminus -134.29, 178.07 63.36, 67.46 -81.42, 12.79 286.94, 80.33 -62.36, -24.52 in-in in 9.1985 Saltbr-in 2.7666 HRD-in -73.96, -47.53 67.01, -6.66 in-in-in SNCiii in-in ActLoopNT-in 2.9216 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.75, 160.77 APE9-dihe-na 92.75, 178.13 APE8-dihe-in -87.23, 123.5 APE8-rot-in 297.99 APE67-dihe-in -58.52, -25.91 -46.52, -43.3 APE12-dist-in 9.1546 APE11-dist-in 11.3986 APE10-dist-in 5.5917 APE9-dist-in 4.172 None None None AF2 -1.0 1.0 1.0 A 283.0 283.0 0 27 27 0 [[220, 486]] 1.0 AF-O96017-K1 CAMK_CHEK2_HUMAN CAMK 1.2e-85 292.8 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 AF-O96017-K3A O96017 212 494 543.0 No_ligand No_ligand Active DFGin 6.4611 14.0711 BLAminus -134.66, -179.17 61.2, 67.72 -80.09, 11.6 287.9, 83.97 -61.23, -22.88 in-in in 9.0586 Saltbr-in 2.7426 HRD-in -76.36, -47.81 68.82, -4.77 in-in-in SNCiii in-in ActLoopNT-in 2.9525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.66, 145.05 APE9-dihe-na 102.94, 172.88 APE8-dihe-in -82.21, 128.17 APE8-rot-in 302.29 APE67-dihe-in -66.9, -22.16 -48.63, -42.33 APE12-dist-in 9.52 APE11-dist-in 11.4179 APE10-dist-in 5.9336 APE9-dist-in 3.4485 None None None AF2 -1.0 1.0 1.0 A 283.0 283.0 0 27 27 0 [[220, 486]] 1.0 AF-O96017-K3 CAMK_CHEK2_HUMAN CAMK 1.2e-85 292.8 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2CN5A O96017 209 504 543.0 ADP:61509 ATPlike Inactive DFGin 6.789 14.4943 BLAminus -135.2, 179.16 64.2, 79.37 -102.1, 20.75 283.06, 77.6 -58.46, -25.36 in-out in 9.9172 Saltbr-out 4.3439 HRD-in -79.96, -48.23 69.59, 1.14 out-in-out SNCoio in-out ActLoopNT-in 2.8477 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_oooo APE10-dihe-na -76.74, 7.44 APE9-dihe-na -76.93, 179.76 APE8-dihe-out 76.66, 47.76 APE8-rot-out 216.78 APE67-dihe-in -44.78, -36.74 -82.05, -7.37 APE12-dist-out 25.3627 APE11-dist-out 27.5187 APE10-dist-out 29.8721 APE9-dist-out 32.7677 None None None XRAY 2.25 0.201 0.24 A 329.0 282.0 14 27 27 0 [[220, 486]] 1.0 2cn5 CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2XK9A O96017 211 510 543.0 XK9:1511 Type1 Inactive DFGin 6.7012 14.7137 BLAminus -130.91, 176.22 68.06, 85.61 -101.66, 24.39 282.26, 77.18 -65.19, -20.58 out-out out 10.5552 Saltbr-out 8.5436 HRD-in -73.65, -51.71 72.1, 1.84 out-in-out SNCoio in-out ActLoopNT-in 2.8971 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -86.23, -28.13 APE9-dihe-na -86.5, 175.56 APE8-dihe-in -74.63, 134.78 APE8-rot-in 304.51 APE67-dihe-in -34.66, -41.42 -81.19, 19.55 APE12-dist-out 25.3556 APE11-dist-out 27.3446 APE10-dist-out 29.6169 APE9-dist-out 33.2765 None None None XRAY 2.35 0.2 0.249 A 322.0 284.0 16 27 27 0 [[220, 486]] 1.0 2xk9 CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2YCFA O96017 210 510 543.0 YCF:600 Type1 Inactive DFGin 6.6505 14.4245 BLAminus -133.14, 179.08 68.92, 89.26 -105.02, 26.49 290.18, 77.38 -65.99, -23.19 in-out in 9.994 Saltbr-out 8.5603 HRD-in -70.72, -52.98 75.15, -0.9 out-in-out SNCoio in-out ActLoopNT-in 2.9054 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -72.28, -26.54 APE9-dihe-na -96.81, -179.54 APE8-dihe-in -85.38, 132.85 APE8-rot-in 297.44 APE67-dihe-in -44.53, -40.92 -82.1, 28.65 APE12-dist-out 25.2308 APE11-dist-out 27.2893 APE10-dist-out 29.3634 APE9-dist-out 33.1045 None None None XRAY 1.77 0.197 0.218 A 322.0 286.0 15 27 27 0 [[220, 486]] 1.0 2ycf CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2W0JA O96017 210 510 543.0 ZAT:1511 Type1 Inactive DFGin 6.6763 14.674 BLAminus -128.11, -176.55 62.13, 84.81 -102.97, 25.22 285.55, 71.63 -69.13, -14.74 out-out out 10.2545 Saltbr-out 8.5376 HRD-in -76.58, -49.8 74.39, -1.67 out-in-out SNCoio in-out ActLoopNT-in 2.9166 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_oooo APE10-dihe-na -90.12, -18.5 APE9-dihe-na -73.0, 168.81 APE8-dihe-out 50.61, 79.46 APE8-rot-out 58.92 APE67-dihe-in -42.13, -44.63 -89.18, 29.26 APE12-dist-out 25.3177 APE11-dist-out 27.3939 APE10-dist-out 29.7732 APE9-dist-out 33.2675 None None None XRAY 2.05 0.217 0.246 A 323.0 280.0 20 27 25 2 [[220, 486]] 1.0 2w0j CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2W7XA O96017 210 510 543.0 D1A:601 Type1 Inactive DFGin 6.5977 14.7428 BLAminus -129.99, -177.26 60.9, 85.9 -97.87, 22.55 286.87, 67.24 -60.05, -24.16 out-out out 10.6926 Saltbr-out 8.8493 HRD-in -75.1, -54.18 74.96, 3.75 out-in-out SNCoio in-out ActLoopNT-in 2.8954 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -72.97, -29.05 APE9-dihe-na -92.97, -167.36 APE8-dihe-in -99.64, 134.31 APE8-rot-in 294.25 APE67-dihe-in -46.4, -41.23 -85.41, 31.83 APE12-dist-out 25.5223 APE11-dist-out 27.1759 APE10-dist-out 29.2583 APE9-dist-out 32.8571 None None None XRAY 2.07 0.195 0.22 A 323.0 285.0 16 27 27 0 [[220, 486]] 1.0 2w7x CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2YCQA O96017 211 510 543.0 UPX:600 Type1 Inactive DFGin 6.6497 14.8765 BLAminus -132.8, -177.16 59.34, 84.42 -98.28, 22.3 281.1, 67.21 -59.37, -26.91 out-out out 10.8358 Saltbr-out 8.9182 HRD-in -78.37, -53.37 73.84, 4.72 out-in-out SNCoio in-out ActLoopNT-in 2.9185 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -72.61, -26.15 APE9-dihe-na -92.03, 178.24 APE8-dihe-in -85.71, 133.17 APE8-rot-out 186.97 APE67-dihe-in -42.38, -41.08 -83.93, 27.59 APE12-dist-out 25.6689 APE11-dist-out 27.2596 APE10-dist-out 29.2586 APE9-dist-out 32.6899 None None None XRAY 2.05 0.211 0.247 A 323.0 285.0 15 27 27 0 [[220, 486]] 1.0 2ycq CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2YCSA O96017 210 510 543.0 NXP:600 Type1 Inactive DFGin 6.7247 14.7134 BLAminus -132.88, -179.1 64.96, 82.34 -101.44, 26.5 282.68, 78.61 -68.86, -18.9 out-out out 10.3484 Saltbr-out 8.6099 HRD-in -79.87, -54.24 74.54, 0.09 out-in-out SNCoio in-out ActLoopNT-in 2.8448 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -83.09, -21.7 APE9-dihe-na -88.87, 176.25 APE8-dihe-in -80.2, 140.31 APE8-rot-in 301.82 APE67-dihe-in -38.14, -42.58 -89.14, 27.52 APE12-dist-out 25.5639 APE11-dist-out 27.5169 APE10-dist-out 29.8073 APE9-dist-out 33.3517 None None None XRAY 2.35 0.202 0.239 A 323.0 281.0 20 27 25 2 [[220, 486]] 1.0 2ycs CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2YIQA O96017 211 510 543.0 YIQ:600 Type1 Inactive DFGin 6.5619 14.3133 BLAminus -133.88, 178.0 71.17, 87.99 -103.54, 29.21 291.07, 76.61 -70.84, -18.27 out-out out 10.0924 Saltbr-out 8.3626 HRD-in -73.68, -53.29 74.71, -0.67 out-in-out SNCoio in-out ActLoopNT-in 2.8857 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -78.28, -22.51 APE9-dihe-na -99.37, 177.03 APE8-dihe-in -80.23, 129.9 APE8-rot-in 306.71 APE67-dihe-in -42.88, -42.2 -82.08, 29.5 APE12-dist-out 25.2483 APE11-dist-out 27.176 APE10-dist-out 29.4082 APE9-dist-out 33.0205 None None None XRAY 1.89 0.199 0.234 A 323.0 280.0 20 27 27 0 [[220, 486]] 1.0 2yiq CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2YIRA O96017 210 509 543.0 YIR:600 Type1 Inactive DFGin 6.5659 14.9663 BLAminus -130.93, -176.93 59.85, 86.3 -99.62, 21.86 282.71, 67.25 -65.17, -21.28 out-out out 10.9052 Saltbr-out 9.0659 HRD-in -77.38, -52.19 70.37, 4.14 out-in-out SNCoio in-out ActLoopNT-in 2.9859 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -62.64, 100.76 APE9-dihe-na -47.9, -163.01 APE8-dihe-in -110.87, 147.89 APE8-rot-out 79.27 APE67-dihe-in -47.35, -40.76 -83.01, 30.27 APE12-dist-out 25.5808 APE11-dist-out 27.1838 APE10-dist-out 29.4784 APE9-dist-out 32.8341 None None None XRAY 2.1 0.197 0.225 A 323.0 286.0 14 27 27 0 [[220, 486]] 1.0 2yir CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2YCRA O96017 211 510 543.0 HCW:600 Type1 Inactive DFGin 6.6543 14.6075 BLAminus -133.62, 179.45 64.45, 83.31 -100.07, 25.98 284.45, 71.85 -69.21, -20.46 out-out out 10.2792 Saltbr-out 8.4869 HRD-in -78.07, -55.38 77.02, -0.95 out-in-out SNCoio in-out ActLoopNT-in 2.9075 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -77.27, -21.77 APE9-dihe-na -96.08, 172.08 APE8-dihe-in -73.99, 132.07 APE8-rot-in 308.16 APE67-dihe-in -43.16, -44.09 -85.85, 32.09 APE12-dist-out 25.4342 APE11-dist-out 27.3345 APE10-dist-out 29.5684 APE9-dist-out 33.0882 None None None XRAY 2.2 0.202 0.233 A 323.0 282.0 18 27 27 0 [[220, 486]] 1.0 2ycr CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2CN8A O96017 212 503 543.0 DBQ:1506 Type1 Inactive DFGin 6.6829 14.0259 BLAminus -126.23, -176.93 68.63, 82.3 -102.35, 19.5 293.05, 94.64 -53.78, -39.11 in-out in 9.1023 Saltbr-out 4.864 HRD-in -79.47, -58.42 90.84, -5.13 out-in-out SNCoio in-out ActLoopNT-in 2.8431 ActLoopCT-out nonTYR APEdihe_aannn APEdist_ooon APE10-dihe-na -88.18, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -60.25, 2.43 999.0, -77.69 APE12-dist-out 23.072 APE11-dist-out 26.6802 APE10-dist-out 29.5924 APE9-dist-none 999.0 None None None XRAY 2.7 0.207 0.271 A 329.0 266.0 26 27 23 4 [[220, 486]] 1.0 2cn8 CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2WTCA O96017 211 512 543.0 VGM:1513 Type1 Inactive DFGin 6.96 14.5977 BLAminus -142.89, 177.82 62.27, 76.17 -93.52, 17.14 286.37, 80.54 -50.13, -44.16 in-in in 9.2308 Saltbr-in 3.0766 HRD-in -65.77, -51.7 71.75, -2.65 in-in-out SNCiio in-out ActLoopNT-in 2.9166 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -71.55, 70.47 APE9-dihe-na -164.95, -154.3 APE8-dihe-in -85.46, 92.16 APE8-rot-in 343.35 APE67-dihe-in -39.77, -41.29 -73.1, -9.9 APE12-dist-out 24.8852 APE11-dist-out 27.0184 APE10-dist-out 30.3343 APE9-dist-out 32.6458 None None None XRAY 3.0 0.183 0.237 A 329.0 284.0 18 27 25 2 [[220, 486]] 1.0 2wtc CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2WTDA O96017 210 512 543.0 ZZK:1513 Type1 Inactive DFGin 6.8682 14.3859 BLAminus -134.38, 170.12 69.53, 79.32 -99.08, 23.68 290.8, 77.12 -56.21, -43.36 in-in in 9.51 Saltbr-in 2.9336 HRD-in -64.83, -58.62 82.47, -13.48 in-in-out SNCiio in-out ActLoopNT-in 2.9305 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oooo APE10-dihe-na -94.4, -11.95 APE9-dihe-na -102.11, 165.57 APE8-dihe-in -61.96, 131.04 APE8-rot-none 999.0 APE67-dihe-out 58.6, -51.68 -61.18, -83.01 APE12-dist-out 25.4917 APE11-dist-out 27.032 APE10-dist-out 29.7743 APE9-dist-out 33.0877 None None None XRAY 2.75 0.194 0.258 A 329.0 285.0 18 27 25 2 [[220, 486]] 1.0 2wtd CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2WTIA O96017 210 512 543.0 WTI:1513 Type1 Inactive DFGin 6.8035 14.4413 BLAminus -139.27, 171.02 71.57, 81.35 -101.15, 19.03 289.19, 81.34 -57.41, -38.09 in-in in 9.2929 Saltbr-in 2.7818 HRD-in -65.33, -55.65 78.76, -5.44 in-in-out SNCiio in-out ActLoopNT-in 2.8903 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -75.65, 126.85 APE9-dihe-na 95.81, 162.84 APE8-dihe-in -79.24, 139.59 APE8-rot-out 183.86 APE67-dihe-in -45.66, -43.39 -86.32, 25.78 APE12-dist-out 25.5709 APE11-dist-out 27.4276 APE10-dist-out 29.631 APE9-dist-out 33.4469 None None None XRAY 2.5 0.197 0.243 A 329.0 286.0 17 27 26 1 [[220, 486]] 1.0 2wti CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2WTJA O96017 209 512 543.0 WTJ:1513 Type1 Inactive DFGin 6.7682 14.3968 BLAminus -143.21, -175.71 63.88, 70.96 -94.85, 21.39 287.09, 79.29 -65.13, -27.57 in-in in 9.2009 Saltbr-in 2.8037 HRD-in -83.11, -47.4 72.91, -5.26 in-in-out SNCiio in-out ActLoopNT-in 2.9834 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -81.47, 86.19 APE9-dihe-na -179.27, -179.27 APE8-dihe-in -66.27, 96.5 APE8-rot-in 325.12 APE67-dihe-in -39.81, -42.18 -60.31, -27.07 APE12-dist-out 25.1497 APE11-dist-out 27.516 APE10-dist-out 29.727 APE9-dist-out 32.4164 None None None XRAY 2.1 0.189 0.217 A 329.0 287.0 17 27 26 1 [[220, 486]] 1.0 2wtj CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2XBJA O96017 211 512 543.0 XBJ:1513 Type1 Inactive DFGin 6.925 14.5707 BLAminus -129.3, -178.28 67.17, 77.45 -97.3, 21.01 288.34, 74.07 -62.67, -27.58 in-out in 9.7477 Saltbr-out 4.5246 HRD-in -69.81, -57.72 79.35, 2.86 out-in-out SNCoio in-out ActLoopNT-in 2.9152 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -67.84, -26.11 APE9-dihe-na -100.1, -172.89 APE8-dihe-in -86.59, 135.42 APE8-rot-in 298.39 APE67-dihe-in -36.76, -45.01 -82.11, 14.62 APE12-dist-out 25.5753 APE11-dist-out 27.4122 APE10-dist-out 29.6606 APE9-dist-out 33.0343 None None None XRAY 2.3 0.196 0.243 A 329.0 286.0 16 27 25 2 [[220, 486]] 1.0 2xbj CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2XM8A O96017 211 503 543.0 B4W:1504 Type1 Inactive DFGin 6.3422 12.9218 BLAminus -125.52, -159.17 52.75, 71.91 -93.76, 25.93 289.45, 88.03 -69.47, -21.5 in-none in 7.9766 Saltbr-none 999.0 HRD-in -75.42, -46.87 67.16, 2.71 none-in-out SNCnio in-out ActLoopNT-in 3.0805 ActLoopCT-out nonTYR APEdihe_aannn APEdist_oooo APE10-dihe-na 38.83, 60.44 APE9-dihe-na -174.64, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-out 24.9584 APE11-dist-out 27.8567 APE10-dist-out 31.0396 APE9-dist-out 32.6679 None None None XRAY 3.4 0.266 0.323 A 329.0 265.0 28 27 22 5 [[220, 486]] 1.0 2xm8 CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2XM9A O96017 211 512 543.0 LWH:1513 Type1 Inactive DFGin 6.8803 14.3779 BLAminus -125.43, -173.87 60.76, 67.11 -91.78, 18.27 285.7, 76.49 -56.15, -47.29 in-in in 8.996 Saltbr-in 2.8196 HRD-in -71.54, -54.2 78.98, -8.38 in-in-out SNCiio in-out ActLoopNT-in 2.958 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -87.82, -22.14 APE9-dihe-na -97.37, -176.91 APE8-dihe-in -89.66, 136.87 APE8-rot-out 72.73 APE67-dihe-in -35.47, -45.2 -82.47, 21.28 APE12-dist-out 25.7732 APE11-dist-out 27.5535 APE10-dist-out 29.8482 APE9-dist-out 33.2789 None None None XRAY 2.5 0.189 0.238 A 329.0 287.0 15 27 27 0 [[220, 486]] 1.0 2xm9 CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4A9RA O96017 210 513 543.0 RU5:1514 Type1 Inactive DFGin 6.7628 14.2999 BLAminus -147.21, -178.58 61.61, 81.41 -102.74, 28.88 295.59, 85.94 -69.84, -27.47 in-in in 9.3431 Saltbr-in 2.8354 HRD-in -63.8, -57.24 81.3, -12.46 in-in-out SNCiio in-out ActLoopNT-in 2.8411 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -74.06, -26.96 APE9-dihe-na -96.58, 164.45 APE8-dihe-in -71.01, 133.8 APE8-rot-out 188.13 APE67-dihe-in -40.81, -51.82 -88.38, 20.75 APE12-dist-out 25.8231 APE11-dist-out 27.3195 APE10-dist-out 29.6705 APE9-dist-out 32.6522 None None None XRAY 2.85 0.186 0.235 A 329.0 286.0 18 27 27 0 [[220, 486]] 1.0 4a9r CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4A9SA O96017 211 513 543.0 RU9:1515 Type1 Inactive DFGin 6.8633 14.2743 BLAminus -146.52, 173.61 72.14, 88.16 -109.62, 21.75 290.51, 89.55 -55.8, -40.77 in-in in 9.0664 Saltbr-in 2.5188 HRD-in -64.11, -53.18 75.3, 0.11 in-in-out SNCiio in-out ActLoopNT-in 2.8965 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -75.09, -19.69 APE9-dihe-na -101.6, 161.25 APE8-dihe-in -74.31, 127.17 APE8-rot-out 170.54 APE67-dihe-in -46.9, -37.89 -82.94, 32.22 APE12-dist-out 25.7232 APE11-dist-out 27.3869 APE10-dist-out 29.6102 APE9-dist-out 32.5358 None None None XRAY 2.66 0.189 0.234 A 329.0 283.0 20 27 25 2 [[220, 486]] 1.0 4a9s CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4A9TA O96017 210 513 543.0 A9T:61514 Type1 Inactive DFGin 6.6133 14.044 BLAminus -140.55, 174.91 73.55, 81.79 -103.33, 21.84 296.3, 86.84 -59.13, -31.93 in-in in 9.266 Saltbr-in 2.7918 HRD-in -65.19, -48.64 77.36, -3.1 in-in-out SNCiio in-out ActLoopNT-in 2.9218 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -66.79, -23.76 APE9-dihe-na -96.24, 179.33 APE8-dihe-in -79.09, 144.87 APE8-rot-out 196.37 APE67-dihe-in -45.41, -43.5 -98.69, 25.4 APE12-dist-out 25.6471 APE11-dist-out 27.4126 APE10-dist-out 29.4803 APE9-dist-out 32.5223 None None None XRAY 2.7 0.191 0.218 A 329.0 289.0 15 27 27 0 [[220, 486]] 1.0 4a9t CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4A9UA O96017 210 513 543.0 A9U:61516 Type1 Inactive DFGin 6.5498 14.1102 BLAminus -142.4, 175.14 71.78, 86.2 -106.33, 25.7 296.4, 87.76 -63.02, -27.27 in-in in 9.156 Saltbr-in 2.6937 HRD-in -67.75, -58.54 79.15, -0.8 in-in-out SNCiio in-out ActLoopNT-in 2.874 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -67.1, -23.4 APE9-dihe-na -98.7, 178.68 APE8-dihe-in -79.95, 138.74 APE8-rot-out 189.39 APE67-dihe-in -40.75, -43.99 -91.72, 18.98 APE12-dist-out 25.5355 APE11-dist-out 27.3233 APE10-dist-out 29.5523 APE9-dist-out 32.6821 None None None XRAY 2.48 0.185 0.214 A 329.0 287.0 17 27 25 2 [[220, 486]] 1.0 4a9u CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDAA O96017 210 512 543.0 VFB:61515 Type1 Inactive DFGin 6.886 14.4626 BLAminus -132.25, -173.99 57.22, 71.24 -86.72, 12.36 287.47, 84.02 -55.8, -30.5 in-in in 9.8498 Saltbr-in 3.1773 HRD-in -66.73, -51.09 75.92, -3.51 in-in-out SNCiio in-out ActLoopNT-in 2.8481 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -68.48, -27.3 APE9-dihe-na -86.39, 178.98 APE8-dihe-in -83.88, 128.17 APE8-rot-none 999.0 APE67-dihe-in -40.46, -44.57 -79.99, 21.04 APE12-dist-out 25.4951 APE11-dist-out 27.5508 APE10-dist-out 29.8285 APE9-dist-out 32.8545 None None None XRAY 2.6 0.183 0.236 A 329.0 283.0 20 27 26 1 [[220, 486]] 1.0 4bda CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDBA O96017 210 513 543.0 ODO:61515 Type1 Inactive DFGin 6.7742 14.8029 BLAminus -136.35, 178.52 66.56, 72.83 -88.8, 15.73 282.83, 82.64 -59.07, -39.67 out-none out 10.0602 Saltbr-none 999.0 HRD-in -69.66, -55.49 76.85, -6.7 none-in-out SNCnio in-out ActLoopNT-in 2.8767 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -64.7, -26.78 APE9-dihe-na -91.52, -174.61 APE8-dihe-in -86.59, 133.65 APE8-rot-none 999.0 APE67-dihe-in -42.37, -42.55 -81.43, 19.5 APE12-dist-out 25.2858 APE11-dist-out 27.3516 APE10-dist-out 29.5173 APE9-dist-out 32.9691 None None None XRAY 2.5 0.192 0.224 A 329.0 283.0 21 27 26 1 [[220, 486]] 1.0 4bdb CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDCA O96017 210 512 543.0 ODH:1513 Type1 Inactive DFGin 6.8094 14.7096 BLAminus -121.85, 179.33 58.65, 81.14 -99.04, 25.33 285.47, 81.08 -60.15, -42.76 in-none in 9.8736 Saltbr-none 999.0 HRD-in -63.39, -48.96 72.38, -9.76 none-in-out SNCnio in-out ActLoopNT-in 3.0032 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -65.73, -25.1 APE9-dihe-na -88.24, 177.42 APE8-dihe-in -91.65, 130.28 APE8-rot-in 280.04 APE67-dihe-in -46.0, -49.87 -76.43, 30.07 APE12-dist-out 25.5638 APE11-dist-out 27.5547 APE10-dist-out 29.7408 APE9-dist-out 32.6052 None None None XRAY 3.0 0.17 0.213 A 329.0 283.0 20 27 26 1 [[220, 486]] 1.0 4bdc CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDDA O96017 210 512 543.0 Z0O:61514 Type1 Inactive DFGin 6.8173 14.6485 BLAminus -132.93, -178.51 62.81, 71.23 -90.6, 15.21 285.85, 82.33 -56.39, -37.94 out-none out 10.1332 Saltbr-none 999.0 HRD-in -68.43, -50.93 76.06, -9.67 none-in-out SNCnio in-out ActLoopNT-in 2.9224 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -72.29, -34.04 APE9-dihe-na -87.58, 175.4 APE8-dihe-in -77.29, 130.46 APE8-rot-none 999.0 APE67-dihe-in -44.92, -49.08 -83.02, 28.4 APE12-dist-out 25.54 APE11-dist-out 27.3591 APE10-dist-out 29.7354 APE9-dist-out 32.9752 None None None XRAY 2.67 0.188 0.22 A 329.0 280.0 23 27 25 2 [[220, 486]] 1.0 4bdd CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDEA O96017 210 513 543.0 CWS:61515 Type1 Inactive DFGin 6.7778 14.2958 BLAminus -131.6, -178.28 58.9, 74.03 -89.63, 22.66 291.98, 82.31 -63.69, -26.8 in-none in 9.7287 Saltbr-none 999.0 HRD-in -67.95, -51.51 74.87, -6.35 none-in-out SNCnio in-out ActLoopNT-in 2.8902 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -64.7, -34.93 APE9-dihe-na -83.4, 175.42 APE8-dihe-in -77.39, 136.48 APE8-rot-out 183.08 APE67-dihe-in -39.74, -49.29 -84.29, 23.06 APE12-dist-out 25.3602 APE11-dist-out 27.4204 APE10-dist-out 29.7116 APE9-dist-out 32.8905 None None None XRAY 2.55 0.186 0.215 A 329.0 283.0 21 27 25 2 [[220, 486]] 1.0 4bde CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDFA O96017 210 512 543.0 H3R:61513 Type1 Inactive DFGin 6.7834 14.4018 BLAminus -125.44, 175.49 63.53, 80.46 -98.42, 23.13 291.77, 82.6 -62.25, -35.46 in-none in 9.8908 Saltbr-none 999.0 HRD-in -62.58, -48.43 71.21, -3.61 none-in-out SNCnio in-out ActLoopNT-in 2.7955 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -72.78, -21.33 APE9-dihe-na -88.28, -178.11 APE8-dihe-in -86.27, 138.16 APE8-rot-out 190.73 APE67-dihe-in -42.2, -47.8 -89.14, 16.34 APE12-dist-out 25.4494 APE11-dist-out 27.4024 APE10-dist-out 29.6311 APE9-dist-out 32.4861 None None None XRAY 2.7 0.183 0.233 A 329.0 284.0 19 27 27 0 [[220, 486]] 1.0 4bdf CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDGA O96017 210 512 543.0 P3J:61513 Type1 Inactive DFGin 6.8712 14.401 BLAminus -128.46, -179.27 57.5, 78.39 -93.56, 21.21 287.69, 84.04 -57.6, -46.72 in-none in 9.8501 Saltbr-none 999.0 HRD-in -58.86, -48.1 72.95, -15.51 none-in-out SNCnio in-out ActLoopNT-in 2.872 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -69.01, -13.44 APE9-dihe-na -106.22, 172.52 APE8-dihe-in -76.2, 130.88 APE8-rot-none 999.0 APE67-dihe-in -40.87, -48.07 -84.34, 27.3 APE12-dist-out 25.3338 APE11-dist-out 27.2171 APE10-dist-out 29.4918 APE9-dist-out 32.5247 None None None XRAY 2.84 0.188 0.227 A 329.0 285.0 18 27 27 0 [[220, 486]] 1.0 4bdg CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDHA O96017 210 513 543.0 WVI:1514 Type1 Inactive DFGin 6.794 14.6838 BLAminus -135.07, 178.29 66.95, 74.06 -95.2, 22.2 285.38, 80.12 -69.45, -24.52 in-none in 9.6448 Saltbr-none 999.0 HRD-in -67.85, -48.22 72.37, -7.17 none-in-out SNCnio in-out ActLoopNT-in 2.7838 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -63.77, -37.18 APE9-dihe-na -81.92, 173.91 APE8-dihe-in -78.09, 132.72 APE8-rot-none 999.0 APE67-dihe-in -42.66, -45.46 -85.31, 24.54 APE12-dist-out 25.5261 APE11-dist-out 27.3667 APE10-dist-out 29.703 APE9-dist-out 32.8103 None None None XRAY 2.7 0.179 0.225 A 329.0 283.0 21 27 27 0 [[220, 486]] 1.0 4bdh CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDIA O96017 210 515 543.0 HAU:61516 Type1 Inactive DFGin 6.8406 14.3562 BLAminus -137.43, -178.59 62.59, 75.88 -93.64, 21.11 289.33, 82.1 -63.95, -34.38 in-none in 9.3436 Saltbr-none 999.0 HRD-in -71.64, -51.74 72.08, -2.17 none-in-out SNCnio in-out ActLoopNT-in 2.8765 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -72.96, -19.96 APE9-dihe-na -100.2, 177.47 APE8-dihe-in -80.99, 134.81 APE8-rot-out 179.62 APE67-dihe-in -45.43, -42.87 -86.02, 25.2 APE12-dist-out 25.2421 APE11-dist-out 27.3013 APE10-dist-out 29.4002 APE9-dist-out 32.537 None None None XRAY 2.32 0.19 0.221 A 329.0 289.0 17 27 27 0 [[220, 486]] 1.0 4bdi CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDJA O96017 211 513 543.0 Z2M:1514 Type1 Inactive DFGin 6.8972 14.848 BLAminus -128.8, -172.27 57.43, 67.48 -85.28, 22.35 287.38, 81.36 -58.43, -49.41 in-none in 9.9585 Saltbr-none 999.0 HRD-in -59.56, -48.03 73.4, -19.9 none-in-out SNCnio in-out ActLoopNT-in 2.9466 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -62.93, -27.44 APE9-dihe-na -88.34, 169.56 APE8-dihe-in -81.49, 123.4 APE8-rot-in 304.23 APE67-dihe-in -39.18, -46.45 -71.01, 19.97 APE12-dist-out 25.3516 APE11-dist-out 27.236 APE10-dist-out 29.5786 APE9-dist-out 32.4102 None None None XRAY 3.01 0.179 0.215 A 329.0 282.0 21 27 26 1 [[220, 486]] 1.0 4bdj CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 4BDKA O96017 211 513 543.0 RQQ:1514 Type1 Inactive DFGin 6.996 14.8025 BLAminus -128.37, -174.72 53.22, 75.18 -89.98, 17.32 277.81, 90.45 -55.79, -43.6 in-none in 9.5584 Saltbr-none 999.0 HRD-in -60.35, -51.11 73.62, -12.31 none-in-out SNCnio in-out ActLoopNT-in 2.883 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_oooo APE10-dihe-na -63.43, -31.74 APE9-dihe-na -86.23, 175.01 APE8-dihe-in -83.22, 121.69 APE8-rot-out 179.06 APE67-dihe-out -64.51, -46.04 -77.96, 50.49 APE12-dist-out 25.2813 APE11-dist-out 27.0305 APE10-dist-out 29.5359 APE9-dist-out 32.5104 None None None XRAY 3.3 0.171 0.233 A 329.0 286.0 17 27 27 0 [[220, 486]] 1.0 4bdk CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 2YITA O96017 211 510 543.0 YIT:600 Type1.5_Back Inactive DFGin 6.7249 14.8959 BLAminus -133.34, -177.92 62.96, 85.15 -102.27, 23.57 279.85, 70.04 -62.49, -22.93 out-out out 10.5148 Saltbr-out 8.3353 HRD-in -77.93, -52.92 73.62, -0.76 out-in-out SNCoio in-out ActLoopNT-in 3.0008 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -83.45, -20.34 APE9-dihe-na -95.61, -175.75 APE8-dihe-in -92.19, 134.54 APE8-rot-in 294.55 APE67-dihe-in -44.05, -39.15 -88.49, 32.62 APE12-dist-out 25.6333 APE11-dist-out 27.4042 APE10-dist-out 29.5055 APE9-dist-out 33.0757 None None None XRAY 2.2 0.196 0.226 A 323.0 286.0 14 27 27 0 [[220, 486]] 1.0 2yit CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6UA O96017 89 501 543.0 No_ligand No_ligand Inactive DFGin 6.3728 13.8281 BLAplus -145.58, 171.6 61.21, 49.14 -102.23, -43.96 37.5, 82.48 -103.81, -9.28 out-none out 13.9661 Saltbr-none 999.0 HRD-in -61.53, -58.97 79.71, -12.85 none-out-none SNCnon out-none ActLoopNT-out 7.5635 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -48.02, -23.93 999.0, -21.46 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.0 0.247 0.28 A 419.0 390.0 23 27 16 11 [[220, 486]] 1.0 3i6u CAMK_CHEK2_HUMAN CAMK 6.3e-84 287.4 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6UB O96017 89 501 543.0 No_ligand No_ligand Inactive DFGin 6.1563 12.4796 None -142.78, 168.99 70.83, 76.16 -115.43, 999.0 26.14, 78.04 999.0, 999.0 out-none out 13.9532 Saltbr-none 999.0 HRD-in -61.77, -58.18 77.91, -11.36 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -48.92, -23.0 999.0, -21.53 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.0 0.247 0.28 B 419.0 376.0 37 27 9 18 [[220, 486]] 1.0 3i6u CAMK_CHEK2_HUMAN CAMK 6.3e-84 287.4 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WA O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.3486 13.5162 None -131.02, -176.1 64.38, 89.31 -97.7, 999.0 302.36, 133.8 999.0, 999.0 out-none out 13.0764 Saltbr-none 999.0 HRD-in -64.4, -41.66 75.43, -23.93 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.49, -47.48 999.0, -37.14 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 A 443.0 369.0 41 27 9 18 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WC O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.5775 13.998 None -131.8, -178.23 63.57, 98.9 -117.45, 999.0 335.54, 98.66 999.0, 999.0 out-none out 13.0805 Saltbr-none 999.0 HRD-in -63.6, -43.12 77.0, -24.17 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.04, -46.8 999.0, -37.07 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 C 443.0 368.0 42 27 9 18 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WE O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.5459 13.6974 None -130.93, -177.05 65.38, 105.03 -130.22, 999.0 325.6, 106.63 999.0, 999.0 out-none out 13.0915 Saltbr-none 999.0 HRD-in -61.69, -42.13 73.77, -23.14 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.57, -46.22 999.0, -36.71 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 E 443.0 368.0 42 27 9 18 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WG O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.5136 13.8031 None -131.95, -176.65 65.29, 79.69 -111.56, 999.0 332.1, 109.83 999.0, 999.0 out-none out 13.0784 Saltbr-none 999.0 HRD-in -62.8, -42.52 74.63, -23.4 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.54, -46.24 999.0, -36.98 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 G 443.0 369.0 41 27 9 18 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WB O96017 92 501 543.0 No_ligand No_ligand None DFGin 6.749 14.2708 BLAminus -132.31, -176.87 65.1, 94.3 -111.58, 28.46 301.82, 101.23 -75.68, -15.25 out-none out 12.8234 Saltbr-none 999.0 HRD-in -62.32, -42.81 74.92, -23.29 none-in-none SNCnin in-none ActLoopNT-in 3.0593 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -68.9, -14.83 999.0, -25.18 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 B 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WD O96017 92 501 543.0 No_ligand No_ligand None DFGin 7.1208 14.4732 BLAminus -130.43, -175.81 63.91, 79.02 -93.96, 27.08 301.9, 101.65 -74.68, -15.75 out-none out 12.8406 Saltbr-none 999.0 HRD-in -63.78, -41.36 74.21, -23.95 none-in-none SNCnin in-none ActLoopNT-in 2.8167 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -68.71, -15.0 999.0, -25.14 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 D 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WF O96017 92 501 543.0 No_ligand No_ligand None DFGin 7.0122 14.1916 BLAminus -131.41, -176.41 64.86, 90.78 -109.15, 26.06 302.9, 101.84 -74.04, -16.03 out-none out 12.8713 Saltbr-none 999.0 HRD-in -63.34, -41.92 73.76, -23.06 none-in-none SNCnin in-none ActLoopNT-in 2.9844 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -68.91, -15.1 999.0, -24.96 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 F 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 3I6WH O96017 92 501 543.0 No_ligand No_ligand None DFGin 6.8741 14.2536 BLAminus -131.53, -176.78 65.02, 88.11 -104.7, 27.13 303.5, 101.73 -74.81, -16.38 out-none out 12.8827 Saltbr-none 999.0 HRD-in -62.35, -41.54 74.34, -23.8 none-in-none SNCnin in-none ActLoopNT-in 3.0871 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -69.26, -15.11 999.0, -24.78 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 H 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2

CAMK_CHEK2 (Serine/threonine-protein kinase Chk2)

Total number of chains: 46
Active chains: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 40 87.0% AF-O96017-K1A
DFGin None 5 10.9% 3I6UB
DFGin BLAplus 1 2.2% 3I6UA

Hover over column headers for tooltip help.

Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CHEK2 CHK2_HUMAN AF-O96017-K1A O96017 212 494 543.0 No_ligand No_ligand Active DFGin 6.5446 14.1254 BLAminus -134.29, 178.07 63.36, 67.46 -81.42, 12.79 286.94, 80.33 -62.36, -24.52 in-in in 9.1985 Saltbr-in 2.7666 HRD-in -73.96, -47.53 67.01, -6.66 in-in-in SNCiii in-in ActLoopNT-in 2.9216 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.75, 160.77 APE9-dihe-na 92.75, 178.13 APE8-dihe-in -87.23, 123.5 APE8-rot-in 297.99 APE67-dihe-in -58.52, -25.91 -46.52, -43.3 APE12-dist-in 9.1546 APE11-dist-in 11.3986 APE10-dist-in 5.5917 APE9-dist-in 4.172 None None None AF2 -1.0 1.0 1.0 A 283.0 283.0 0 27 27 0 [[220, 486]] 1.0 AF-O96017-K1 Homo sapiens CAMK_CHEK2_HUMAN CAMK 1.2e-85 292.8 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN AF-O96017-K3A O96017 212 494 543.0 No_ligand No_ligand Active DFGin 6.4611 14.0711 BLAminus -134.66, -179.17 61.2, 67.72 -80.09, 11.6 287.9, 83.97 -61.23, -22.88 in-in in 9.0586 Saltbr-in 2.7426 HRD-in -76.36, -47.81 68.82, -4.77 in-in-in SNCiii in-in ActLoopNT-in 2.9525 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.66, 145.05 APE9-dihe-na 102.94, 172.88 APE8-dihe-in -82.21, 128.17 APE8-rot-in 302.29 APE67-dihe-in -66.9, -22.16 -48.63, -42.33 APE12-dist-in 9.52 APE11-dist-in 11.4179 APE10-dist-in 5.9336 APE9-dist-in 3.4485 None None None AF2 -1.0 1.0 1.0 A 283.0 283.0 0 27 27 0 [[220, 486]] 1.0 AF-O96017-K3 Homo sapiens CAMK_CHEK2_HUMAN CAMK 1.2e-85 292.8 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2CN5A O96017 209 504 543.0 ADP:61509 ATPlike Inactive DFGin 6.789 14.4943 BLAminus -135.2, 179.16 64.2, 79.37 -102.1, 20.75 283.06, 77.6 -58.46, -25.36 in-out in 9.9172 Saltbr-out 4.3439 HRD-in -79.96, -48.23 69.59, 1.14 out-in-out SNCoio in-out ActLoopNT-in 2.8477 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_oooo APE10-dihe-na -76.74, 7.44 APE9-dihe-na -76.93, 179.76 APE8-dihe-out 76.66, 47.76 APE8-rot-out 216.78 APE67-dihe-in -44.78, -36.74 -82.05, -7.37 APE12-dist-out 25.3627 APE11-dist-out 27.5187 APE10-dist-out 29.8721 APE9-dist-out 32.7677 None None None XRAY 2.25 0.201 0.24 A 329.0 282.0 14 27 27 0 [[220, 486]] 1.0 2cn5 Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2XK9A O96017 211 510 543.0 XK9:1511 Type1 Inactive DFGin 6.7012 14.7137 BLAminus -130.91, 176.22 68.06, 85.61 -101.66, 24.39 282.26, 77.18 -65.19, -20.58 out-out out 10.5552 Saltbr-out 8.5436 HRD-in -73.65, -51.71 72.1, 1.84 out-in-out SNCoio in-out ActLoopNT-in 2.8971 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -86.23, -28.13 APE9-dihe-na -86.5, 175.56 APE8-dihe-in -74.63, 134.78 APE8-rot-in 304.51 APE67-dihe-in -34.66, -41.42 -81.19, 19.55 APE12-dist-out 25.3556 APE11-dist-out 27.3446 APE10-dist-out 29.6169 APE9-dist-out 33.2765 None None None XRAY 2.35 0.2 0.249 A 322.0 284.0 16 27 27 0 [[220, 486]] 1.0 2xk9 Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2YCFA O96017 210 510 543.0 YCF:600 Type1 Inactive DFGin 6.6505 14.4245 BLAminus -133.14, 179.08 68.92, 89.26 -105.02, 26.49 290.18, 77.38 -65.99, -23.19 in-out in 9.994 Saltbr-out 8.5603 HRD-in -70.72, -52.98 75.15, -0.9 out-in-out SNCoio in-out ActLoopNT-in 2.9054 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -72.28, -26.54 APE9-dihe-na -96.81, -179.54 APE8-dihe-in -85.38, 132.85 APE8-rot-in 297.44 APE67-dihe-in -44.53, -40.92 -82.1, 28.65 APE12-dist-out 25.2308 APE11-dist-out 27.2893 APE10-dist-out 29.3634 APE9-dist-out 33.1045 None None None XRAY 1.77 0.197 0.218 A 322.0 286.0 15 27 27 0 [[220, 486]] 1.0 2ycf Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2W0JA O96017 210 510 543.0 ZAT:1511 Type1 Inactive DFGin 6.6763 14.674 BLAminus -128.11, -176.55 62.13, 84.81 -102.97, 25.22 285.55, 71.63 -69.13, -14.74 out-out out 10.2545 Saltbr-out 8.5376 HRD-in -76.58, -49.8 74.39, -1.67 out-in-out SNCoio in-out ActLoopNT-in 2.9166 ActLoopCT-out nonTYR APEdihe_aaooi APEdist_oooo APE10-dihe-na -90.12, -18.5 APE9-dihe-na -73.0, 168.81 APE8-dihe-out 50.61, 79.46 APE8-rot-out 58.92 APE67-dihe-in -42.13, -44.63 -89.18, 29.26 APE12-dist-out 25.3177 APE11-dist-out 27.3939 APE10-dist-out 29.7732 APE9-dist-out 33.2675 None None None XRAY 2.05 0.217 0.246 A 323.0 280.0 20 27 25 2 [[220, 486]] 1.0 2w0j Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2W7XA O96017 210 510 543.0 D1A:601 Type1 Inactive DFGin 6.5977 14.7428 BLAminus -129.99, -177.26 60.9, 85.9 -97.87, 22.55 286.87, 67.24 -60.05, -24.16 out-out out 10.6926 Saltbr-out 8.8493 HRD-in -75.1, -54.18 74.96, 3.75 out-in-out SNCoio in-out ActLoopNT-in 2.8954 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -72.97, -29.05 APE9-dihe-na -92.97, -167.36 APE8-dihe-in -99.64, 134.31 APE8-rot-in 294.25 APE67-dihe-in -46.4, -41.23 -85.41, 31.83 APE12-dist-out 25.5223 APE11-dist-out 27.1759 APE10-dist-out 29.2583 APE9-dist-out 32.8571 None None None XRAY 2.07 0.195 0.22 A 323.0 285.0 16 27 27 0 [[220, 486]] 1.0 2w7x Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2YCQA O96017 211 510 543.0 UPX:600 Type1 Inactive DFGin 6.6497 14.8765 BLAminus -132.8, -177.16 59.34, 84.42 -98.28, 22.3 281.1, 67.21 -59.37, -26.91 out-out out 10.8358 Saltbr-out 8.9182 HRD-in -78.37, -53.37 73.84, 4.72 out-in-out SNCoio in-out ActLoopNT-in 2.9185 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -72.61, -26.15 APE9-dihe-na -92.03, 178.24 APE8-dihe-in -85.71, 133.17 APE8-rot-out 186.97 APE67-dihe-in -42.38, -41.08 -83.93, 27.59 APE12-dist-out 25.6689 APE11-dist-out 27.2596 APE10-dist-out 29.2586 APE9-dist-out 32.6899 None None None XRAY 2.05 0.211 0.247 A 323.0 285.0 15 27 27 0 [[220, 486]] 1.0 2ycq Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2YCSA O96017 210 510 543.0 NXP:600 Type1 Inactive DFGin 6.7247 14.7134 BLAminus -132.88, -179.1 64.96, 82.34 -101.44, 26.5 282.68, 78.61 -68.86, -18.9 out-out out 10.3484 Saltbr-out 8.6099 HRD-in -79.87, -54.24 74.54, 0.09 out-in-out SNCoio in-out ActLoopNT-in 2.8448 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -83.09, -21.7 APE9-dihe-na -88.87, 176.25 APE8-dihe-in -80.2, 140.31 APE8-rot-in 301.82 APE67-dihe-in -38.14, -42.58 -89.14, 27.52 APE12-dist-out 25.5639 APE11-dist-out 27.5169 APE10-dist-out 29.8073 APE9-dist-out 33.3517 None None None XRAY 2.35 0.202 0.239 A 323.0 281.0 20 27 25 2 [[220, 486]] 1.0 2ycs Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2YIQA O96017 211 510 543.0 YIQ:600 Type1 Inactive DFGin 6.5619 14.3133 BLAminus -133.88, 178.0 71.17, 87.99 -103.54, 29.21 291.07, 76.61 -70.84, -18.27 out-out out 10.0924 Saltbr-out 8.3626 HRD-in -73.68, -53.29 74.71, -0.67 out-in-out SNCoio in-out ActLoopNT-in 2.8857 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -78.28, -22.51 APE9-dihe-na -99.37, 177.03 APE8-dihe-in -80.23, 129.9 APE8-rot-in 306.71 APE67-dihe-in -42.88, -42.2 -82.08, 29.5 APE12-dist-out 25.2483 APE11-dist-out 27.176 APE10-dist-out 29.4082 APE9-dist-out 33.0205 None None None XRAY 1.89 0.199 0.234 A 323.0 280.0 20 27 27 0 [[220, 486]] 1.0 2yiq Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2YIRA O96017 210 509 543.0 YIR:600 Type1 Inactive DFGin 6.5659 14.9663 BLAminus -130.93, -176.93 59.85, 86.3 -99.62, 21.86 282.71, 67.25 -65.17, -21.28 out-out out 10.9052 Saltbr-out 9.0659 HRD-in -77.38, -52.19 70.37, 4.14 out-in-out SNCoio in-out ActLoopNT-in 2.9859 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -62.64, 100.76 APE9-dihe-na -47.9, -163.01 APE8-dihe-in -110.87, 147.89 APE8-rot-out 79.27 APE67-dihe-in -47.35, -40.76 -83.01, 30.27 APE12-dist-out 25.5808 APE11-dist-out 27.1838 APE10-dist-out 29.4784 APE9-dist-out 32.8341 None None None XRAY 2.1 0.197 0.225 A 323.0 286.0 14 27 27 0 [[220, 486]] 1.0 2yir Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2YCRA O96017 211 510 543.0 HCW:600 Type1 Inactive DFGin 6.6543 14.6075 BLAminus -133.62, 179.45 64.45, 83.31 -100.07, 25.98 284.45, 71.85 -69.21, -20.46 out-out out 10.2792 Saltbr-out 8.4869 HRD-in -78.07, -55.38 77.02, -0.95 out-in-out SNCoio in-out ActLoopNT-in 2.9075 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -77.27, -21.77 APE9-dihe-na -96.08, 172.08 APE8-dihe-in -73.99, 132.07 APE8-rot-in 308.16 APE67-dihe-in -43.16, -44.09 -85.85, 32.09 APE12-dist-out 25.4342 APE11-dist-out 27.3345 APE10-dist-out 29.5684 APE9-dist-out 33.0882 None None None XRAY 2.2 0.202 0.233 A 323.0 282.0 18 27 27 0 [[220, 486]] 1.0 2ycr Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2CN8A O96017 212 503 543.0 DBQ:1506 Type1 Inactive DFGin 6.6829 14.0259 BLAminus -126.23, -176.93 68.63, 82.3 -102.35, 19.5 293.05, 94.64 -53.78, -39.11 in-out in 9.1023 Saltbr-out 4.864 HRD-in -79.47, -58.42 90.84, -5.13 out-in-out SNCoio in-out ActLoopNT-in 2.8431 ActLoopCT-out nonTYR APEdihe_aannn APEdist_ooon APE10-dihe-na -88.18, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -60.25, 2.43 999.0, -77.69 APE12-dist-out 23.072 APE11-dist-out 26.6802 APE10-dist-out 29.5924 APE9-dist-none 999.0 None None None XRAY 2.7 0.207 0.271 A 329.0 266.0 26 27 23 4 [[220, 486]] 1.0 2cn8 Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2WTCA O96017 211 512 543.0 VGM:1513 Type1 Inactive DFGin 6.96 14.5977 BLAminus -142.89, 177.82 62.27, 76.17 -93.52, 17.14 286.37, 80.54 -50.13, -44.16 in-in in 9.2308 Saltbr-in 3.0766 HRD-in -65.77, -51.7 71.75, -2.65 in-in-out SNCiio in-out ActLoopNT-in 2.9166 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -71.55, 70.47 APE9-dihe-na -164.95, -154.3 APE8-dihe-in -85.46, 92.16 APE8-rot-in 343.35 APE67-dihe-in -39.77, -41.29 -73.1, -9.9 APE12-dist-out 24.8852 APE11-dist-out 27.0184 APE10-dist-out 30.3343 APE9-dist-out 32.6458 None None None XRAY 3.0 0.183 0.237 A 329.0 284.0 18 27 25 2 [[220, 486]] 1.0 2wtc Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2WTDA O96017 210 512 543.0 ZZK:1513 Type1 Inactive DFGin 6.8682 14.3859 BLAminus -134.38, 170.12 69.53, 79.32 -99.08, 23.68 290.8, 77.12 -56.21, -43.36 in-in in 9.51 Saltbr-in 2.9336 HRD-in -64.83, -58.62 82.47, -13.48 in-in-out SNCiio in-out ActLoopNT-in 2.9305 ActLoopCT-out nonTYR APEdihe_aaino APEdist_oooo APE10-dihe-na -94.4, -11.95 APE9-dihe-na -102.11, 165.57 APE8-dihe-in -61.96, 131.04 APE8-rot-none 999.0 APE67-dihe-out 58.6, -51.68 -61.18, -83.01 APE12-dist-out 25.4917 APE11-dist-out 27.032 APE10-dist-out 29.7743 APE9-dist-out 33.0877 None None None XRAY 2.75 0.194 0.258 A 329.0 285.0 18 27 25 2 [[220, 486]] 1.0 2wtd Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2WTIA O96017 210 512 543.0 WTI:1513 Type1 Inactive DFGin 6.8035 14.4413 BLAminus -139.27, 171.02 71.57, 81.35 -101.15, 19.03 289.19, 81.34 -57.41, -38.09 in-in in 9.2929 Saltbr-in 2.7818 HRD-in -65.33, -55.65 78.76, -5.44 in-in-out SNCiio in-out ActLoopNT-in 2.8903 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -75.65, 126.85 APE9-dihe-na 95.81, 162.84 APE8-dihe-in -79.24, 139.59 APE8-rot-out 183.86 APE67-dihe-in -45.66, -43.39 -86.32, 25.78 APE12-dist-out 25.5709 APE11-dist-out 27.4276 APE10-dist-out 29.631 APE9-dist-out 33.4469 None None None XRAY 2.5 0.197 0.243 A 329.0 286.0 17 27 26 1 [[220, 486]] 1.0 2wti Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2WTJA O96017 209 512 543.0 WTJ:1513 Type1 Inactive DFGin 6.7682 14.3968 BLAminus -143.21, -175.71 63.88, 70.96 -94.85, 21.39 287.09, 79.29 -65.13, -27.57 in-in in 9.2009 Saltbr-in 2.8037 HRD-in -83.11, -47.4 72.91, -5.26 in-in-out SNCiio in-out ActLoopNT-in 2.9834 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -81.47, 86.19 APE9-dihe-na -179.27, -179.27 APE8-dihe-in -66.27, 96.5 APE8-rot-in 325.12 APE67-dihe-in -39.81, -42.18 -60.31, -27.07 APE12-dist-out 25.1497 APE11-dist-out 27.516 APE10-dist-out 29.727 APE9-dist-out 32.4164 None None None XRAY 2.1 0.189 0.217 A 329.0 287.0 17 27 26 1 [[220, 486]] 1.0 2wtj Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2XBJA O96017 211 512 543.0 XBJ:1513 Type1 Inactive DFGin 6.925 14.5707 BLAminus -129.3, -178.28 67.17, 77.45 -97.3, 21.01 288.34, 74.07 -62.67, -27.58 in-out in 9.7477 Saltbr-out 4.5246 HRD-in -69.81, -57.72 79.35, 2.86 out-in-out SNCoio in-out ActLoopNT-in 2.9152 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -67.84, -26.11 APE9-dihe-na -100.1, -172.89 APE8-dihe-in -86.59, 135.42 APE8-rot-in 298.39 APE67-dihe-in -36.76, -45.01 -82.11, 14.62 APE12-dist-out 25.5753 APE11-dist-out 27.4122 APE10-dist-out 29.6606 APE9-dist-out 33.0343 None None None XRAY 2.3 0.196 0.243 A 329.0 286.0 16 27 25 2 [[220, 486]] 1.0 2xbj Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2XM8A O96017 211 503 543.0 B4W:1504 Type1 Inactive DFGin 6.3422 12.9218 BLAminus -125.52, -159.17 52.75, 71.91 -93.76, 25.93 289.45, 88.03 -69.47, -21.5 in-none in 7.9766 Saltbr-none 999.0 HRD-in -75.42, -46.87 67.16, 2.71 none-in-out SNCnio in-out ActLoopNT-in 3.0805 ActLoopCT-out nonTYR APEdihe_aannn APEdist_oooo APE10-dihe-na 38.83, 60.44 APE9-dihe-na -174.64, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, 999.0 999.0, 999.0 APE12-dist-out 24.9584 APE11-dist-out 27.8567 APE10-dist-out 31.0396 APE9-dist-out 32.6679 None None None XRAY 3.4 0.266 0.323 A 329.0 265.0 28 27 22 5 [[220, 486]] 1.0 2xm8 Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2XM9A O96017 211 512 543.0 LWH:1513 Type1 Inactive DFGin 6.8803 14.3779 BLAminus -125.43, -173.87 60.76, 67.11 -91.78, 18.27 285.7, 76.49 -56.15, -47.29 in-in in 8.996 Saltbr-in 2.8196 HRD-in -71.54, -54.2 78.98, -8.38 in-in-out SNCiio in-out ActLoopNT-in 2.958 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -87.82, -22.14 APE9-dihe-na -97.37, -176.91 APE8-dihe-in -89.66, 136.87 APE8-rot-out 72.73 APE67-dihe-in -35.47, -45.2 -82.47, 21.28 APE12-dist-out 25.7732 APE11-dist-out 27.5535 APE10-dist-out 29.8482 APE9-dist-out 33.2789 None None None XRAY 2.5 0.189 0.238 A 329.0 287.0 15 27 27 0 [[220, 486]] 1.0 2xm9 Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4A9RA O96017 210 513 543.0 RU5:1514 Type1 Inactive DFGin 6.7628 14.2999 BLAminus -147.21, -178.58 61.61, 81.41 -102.74, 28.88 295.59, 85.94 -69.84, -27.47 in-in in 9.3431 Saltbr-in 2.8354 HRD-in -63.8, -57.24 81.3, -12.46 in-in-out SNCiio in-out ActLoopNT-in 2.8411 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -74.06, -26.96 APE9-dihe-na -96.58, 164.45 APE8-dihe-in -71.01, 133.8 APE8-rot-out 188.13 APE67-dihe-in -40.81, -51.82 -88.38, 20.75 APE12-dist-out 25.8231 APE11-dist-out 27.3195 APE10-dist-out 29.6705 APE9-dist-out 32.6522 None None None XRAY 2.85 0.186 0.235 A 329.0 286.0 18 27 27 0 [[220, 486]] 1.0 4a9r Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4A9SA O96017 211 513 543.0 RU9:1515 Type1 Inactive DFGin 6.8633 14.2743 BLAminus -146.52, 173.61 72.14, 88.16 -109.62, 21.75 290.51, 89.55 -55.8, -40.77 in-in in 9.0664 Saltbr-in 2.5188 HRD-in -64.11, -53.18 75.3, 0.11 in-in-out SNCiio in-out ActLoopNT-in 2.8965 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -75.09, -19.69 APE9-dihe-na -101.6, 161.25 APE8-dihe-in -74.31, 127.17 APE8-rot-out 170.54 APE67-dihe-in -46.9, -37.89 -82.94, 32.22 APE12-dist-out 25.7232 APE11-dist-out 27.3869 APE10-dist-out 29.6102 APE9-dist-out 32.5358 None None None XRAY 2.66 0.189 0.234 A 329.0 283.0 20 27 25 2 [[220, 486]] 1.0 4a9s Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4A9TA O96017 210 513 543.0 A9T:61514 Type1 Inactive DFGin 6.6133 14.044 BLAminus -140.55, 174.91 73.55, 81.79 -103.33, 21.84 296.3, 86.84 -59.13, -31.93 in-in in 9.266 Saltbr-in 2.7918 HRD-in -65.19, -48.64 77.36, -3.1 in-in-out SNCiio in-out ActLoopNT-in 2.9218 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -66.79, -23.76 APE9-dihe-na -96.24, 179.33 APE8-dihe-in -79.09, 144.87 APE8-rot-out 196.37 APE67-dihe-in -45.41, -43.5 -98.69, 25.4 APE12-dist-out 25.6471 APE11-dist-out 27.4126 APE10-dist-out 29.4803 APE9-dist-out 32.5223 None None None XRAY 2.7 0.191 0.218 A 329.0 289.0 15 27 27 0 [[220, 486]] 1.0 4a9t Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4A9UA O96017 210 513 543.0 A9U:61516 Type1 Inactive DFGin 6.5498 14.1102 BLAminus -142.4, 175.14 71.78, 86.2 -106.33, 25.7 296.4, 87.76 -63.02, -27.27 in-in in 9.156 Saltbr-in 2.6937 HRD-in -67.75, -58.54 79.15, -0.8 in-in-out SNCiio in-out ActLoopNT-in 2.874 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -67.1, -23.4 APE9-dihe-na -98.7, 178.68 APE8-dihe-in -79.95, 138.74 APE8-rot-out 189.39 APE67-dihe-in -40.75, -43.99 -91.72, 18.98 APE12-dist-out 25.5355 APE11-dist-out 27.3233 APE10-dist-out 29.5523 APE9-dist-out 32.6821 None None None XRAY 2.48 0.185 0.214 A 329.0 287.0 17 27 25 2 [[220, 486]] 1.0 4a9u Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDAA O96017 210 512 543.0 VFB:61515 Type1 Inactive DFGin 6.886 14.4626 BLAminus -132.25, -173.99 57.22, 71.24 -86.72, 12.36 287.47, 84.02 -55.8, -30.5 in-in in 9.8498 Saltbr-in 3.1773 HRD-in -66.73, -51.09 75.92, -3.51 in-in-out SNCiio in-out ActLoopNT-in 2.8481 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -68.48, -27.3 APE9-dihe-na -86.39, 178.98 APE8-dihe-in -83.88, 128.17 APE8-rot-none 999.0 APE67-dihe-in -40.46, -44.57 -79.99, 21.04 APE12-dist-out 25.4951 APE11-dist-out 27.5508 APE10-dist-out 29.8285 APE9-dist-out 32.8545 None None None XRAY 2.6 0.183 0.236 A 329.0 283.0 20 27 26 1 [[220, 486]] 1.0 4bda Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDBA O96017 210 513 543.0 ODO:61515 Type1 Inactive DFGin 6.7742 14.8029 BLAminus -136.35, 178.52 66.56, 72.83 -88.8, 15.73 282.83, 82.64 -59.07, -39.67 out-none out 10.0602 Saltbr-none 999.0 HRD-in -69.66, -55.49 76.85, -6.7 none-in-out SNCnio in-out ActLoopNT-in 2.8767 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -64.7, -26.78 APE9-dihe-na -91.52, -174.61 APE8-dihe-in -86.59, 133.65 APE8-rot-none 999.0 APE67-dihe-in -42.37, -42.55 -81.43, 19.5 APE12-dist-out 25.2858 APE11-dist-out 27.3516 APE10-dist-out 29.5173 APE9-dist-out 32.9691 None None None XRAY 2.5 0.192 0.224 A 329.0 283.0 21 27 26 1 [[220, 486]] 1.0 4bdb Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDCA O96017 210 512 543.0 ODH:1513 Type1 Inactive DFGin 6.8094 14.7096 BLAminus -121.85, 179.33 58.65, 81.14 -99.04, 25.33 285.47, 81.08 -60.15, -42.76 in-none in 9.8736 Saltbr-none 999.0 HRD-in -63.39, -48.96 72.38, -9.76 none-in-out SNCnio in-out ActLoopNT-in 3.0032 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -65.73, -25.1 APE9-dihe-na -88.24, 177.42 APE8-dihe-in -91.65, 130.28 APE8-rot-in 280.04 APE67-dihe-in -46.0, -49.87 -76.43, 30.07 APE12-dist-out 25.5638 APE11-dist-out 27.5547 APE10-dist-out 29.7408 APE9-dist-out 32.6052 None None None XRAY 3.0 0.17 0.213 A 329.0 283.0 20 27 26 1 [[220, 486]] 1.0 4bdc Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDDA O96017 210 512 543.0 Z0O:61514 Type1 Inactive DFGin 6.8173 14.6485 BLAminus -132.93, -178.51 62.81, 71.23 -90.6, 15.21 285.85, 82.33 -56.39, -37.94 out-none out 10.1332 Saltbr-none 999.0 HRD-in -68.43, -50.93 76.06, -9.67 none-in-out SNCnio in-out ActLoopNT-in 2.9224 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -72.29, -34.04 APE9-dihe-na -87.58, 175.4 APE8-dihe-in -77.29, 130.46 APE8-rot-none 999.0 APE67-dihe-in -44.92, -49.08 -83.02, 28.4 APE12-dist-out 25.54 APE11-dist-out 27.3591 APE10-dist-out 29.7354 APE9-dist-out 32.9752 None None None XRAY 2.67 0.188 0.22 A 329.0 280.0 23 27 25 2 [[220, 486]] 1.0 4bdd Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDEA O96017 210 513 543.0 CWS:61515 Type1 Inactive DFGin 6.7778 14.2958 BLAminus -131.6, -178.28 58.9, 74.03 -89.63, 22.66 291.98, 82.31 -63.69, -26.8 in-none in 9.7287 Saltbr-none 999.0 HRD-in -67.95, -51.51 74.87, -6.35 none-in-out SNCnio in-out ActLoopNT-in 2.8902 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -64.7, -34.93 APE9-dihe-na -83.4, 175.42 APE8-dihe-in -77.39, 136.48 APE8-rot-out 183.08 APE67-dihe-in -39.74, -49.29 -84.29, 23.06 APE12-dist-out 25.3602 APE11-dist-out 27.4204 APE10-dist-out 29.7116 APE9-dist-out 32.8905 None None None XRAY 2.55 0.186 0.215 A 329.0 283.0 21 27 25 2 [[220, 486]] 1.0 4bde Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDFA O96017 210 512 543.0 H3R:61513 Type1 Inactive DFGin 6.7834 14.4018 BLAminus -125.44, 175.49 63.53, 80.46 -98.42, 23.13 291.77, 82.6 -62.25, -35.46 in-none in 9.8908 Saltbr-none 999.0 HRD-in -62.58, -48.43 71.21, -3.61 none-in-out SNCnio in-out ActLoopNT-in 2.7955 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -72.78, -21.33 APE9-dihe-na -88.28, -178.11 APE8-dihe-in -86.27, 138.16 APE8-rot-out 190.73 APE67-dihe-in -42.2, -47.8 -89.14, 16.34 APE12-dist-out 25.4494 APE11-dist-out 27.4024 APE10-dist-out 29.6311 APE9-dist-out 32.4861 None None None XRAY 2.7 0.183 0.233 A 329.0 284.0 19 27 27 0 [[220, 486]] 1.0 4bdf Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDGA O96017 210 512 543.0 P3J:61513 Type1 Inactive DFGin 6.8712 14.401 BLAminus -128.46, -179.27 57.5, 78.39 -93.56, 21.21 287.69, 84.04 -57.6, -46.72 in-none in 9.8501 Saltbr-none 999.0 HRD-in -58.86, -48.1 72.95, -15.51 none-in-out SNCnio in-out ActLoopNT-in 2.872 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -69.01, -13.44 APE9-dihe-na -106.22, 172.52 APE8-dihe-in -76.2, 130.88 APE8-rot-none 999.0 APE67-dihe-in -40.87, -48.07 -84.34, 27.3 APE12-dist-out 25.3338 APE11-dist-out 27.2171 APE10-dist-out 29.4918 APE9-dist-out 32.5247 None None None XRAY 2.84 0.188 0.227 A 329.0 285.0 18 27 27 0 [[220, 486]] 1.0 4bdg Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDHA O96017 210 513 543.0 WVI:1514 Type1 Inactive DFGin 6.794 14.6838 BLAminus -135.07, 178.29 66.95, 74.06 -95.2, 22.2 285.38, 80.12 -69.45, -24.52 in-none in 9.6448 Saltbr-none 999.0 HRD-in -67.85, -48.22 72.37, -7.17 none-in-out SNCnio in-out ActLoopNT-in 2.7838 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -63.77, -37.18 APE9-dihe-na -81.92, 173.91 APE8-dihe-in -78.09, 132.72 APE8-rot-none 999.0 APE67-dihe-in -42.66, -45.46 -85.31, 24.54 APE12-dist-out 25.5261 APE11-dist-out 27.3667 APE10-dist-out 29.703 APE9-dist-out 32.8103 None None None XRAY 2.7 0.179 0.225 A 329.0 283.0 21 27 27 0 [[220, 486]] 1.0 4bdh Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDIA O96017 210 515 543.0 HAU:61516 Type1 Inactive DFGin 6.8406 14.3562 BLAminus -137.43, -178.59 62.59, 75.88 -93.64, 21.11 289.33, 82.1 -63.95, -34.38 in-none in 9.3436 Saltbr-none 999.0 HRD-in -71.64, -51.74 72.08, -2.17 none-in-out SNCnio in-out ActLoopNT-in 2.8765 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -72.96, -19.96 APE9-dihe-na -100.2, 177.47 APE8-dihe-in -80.99, 134.81 APE8-rot-out 179.62 APE67-dihe-in -45.43, -42.87 -86.02, 25.2 APE12-dist-out 25.2421 APE11-dist-out 27.3013 APE10-dist-out 29.4002 APE9-dist-out 32.537 None None None XRAY 2.32 0.19 0.221 A 329.0 289.0 17 27 27 0 [[220, 486]] 1.0 4bdi Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDJA O96017 211 513 543.0 Z2M:1514 Type1 Inactive DFGin 6.8972 14.848 BLAminus -128.8, -172.27 57.43, 67.48 -85.28, 22.35 287.38, 81.36 -58.43, -49.41 in-none in 9.9585 Saltbr-none 999.0 HRD-in -59.56, -48.03 73.4, -19.9 none-in-out SNCnio in-out ActLoopNT-in 2.9466 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -62.93, -27.44 APE9-dihe-na -88.34, 169.56 APE8-dihe-in -81.49, 123.4 APE8-rot-in 304.23 APE67-dihe-in -39.18, -46.45 -71.01, 19.97 APE12-dist-out 25.3516 APE11-dist-out 27.236 APE10-dist-out 29.5786 APE9-dist-out 32.4102 None None None XRAY 3.01 0.179 0.215 A 329.0 282.0 21 27 26 1 [[220, 486]] 1.0 4bdj Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 4BDKA O96017 211 513 543.0 RQQ:1514 Type1 Inactive DFGin 6.996 14.8025 BLAminus -128.37, -174.72 53.22, 75.18 -89.98, 17.32 277.81, 90.45 -55.79, -43.6 in-none in 9.5584 Saltbr-none 999.0 HRD-in -60.35, -51.11 73.62, -12.31 none-in-out SNCnio in-out ActLoopNT-in 2.883 ActLoopCT-out nonTYR APEdihe_aaioo APEdist_oooo APE10-dihe-na -63.43, -31.74 APE9-dihe-na -86.23, 175.01 APE8-dihe-in -83.22, 121.69 APE8-rot-out 179.06 APE67-dihe-out -64.51, -46.04 -77.96, 50.49 APE12-dist-out 25.2813 APE11-dist-out 27.0305 APE10-dist-out 29.5359 APE9-dist-out 32.5104 None None None XRAY 3.3 0.171 0.233 A 329.0 286.0 17 27 27 0 [[220, 486]] 1.0 4bdk Homo sapiens CAMK_CHEK2_HUMAN CAMK 2.1e-85 292.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 2YITA O96017 211 510 543.0 YIT:600 Type1.5_Back Inactive DFGin 6.7249 14.8959 BLAminus -133.34, -177.92 62.96, 85.15 -102.27, 23.57 279.85, 70.04 -62.49, -22.93 out-out out 10.5148 Saltbr-out 8.3353 HRD-in -77.93, -52.92 73.62, -0.76 out-in-out SNCoio in-out ActLoopNT-in 3.0008 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -83.45, -20.34 APE9-dihe-na -95.61, -175.75 APE8-dihe-in -92.19, 134.54 APE8-rot-in 294.55 APE67-dihe-in -44.05, -39.15 -88.49, 32.62 APE12-dist-out 25.6333 APE11-dist-out 27.4042 APE10-dist-out 29.5055 APE9-dist-out 33.0757 None None None XRAY 2.2 0.196 0.226 A 323.0 286.0 14 27 27 0 [[220, 486]] 1.0 2yit Homo sapiens CAMK_CHEK2_HUMAN CAMK 2e-85 292.2 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6UA O96017 89 501 543.0 No_ligand No_ligand Inactive DFGin 6.3728 13.8281 BLAplus -145.58, 171.6 61.21, 49.14 -102.23, -43.96 37.5, 82.48 -103.81, -9.28 out-none out 13.9661 Saltbr-none 999.0 HRD-in -61.53, -58.97 79.71, -12.85 none-out-none SNCnon out-none ActLoopNT-out 7.5635 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -48.02, -23.93 999.0, -21.46 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.0 0.247 0.28 A 419.0 390.0 23 27 16 11 [[220, 486]] 1.0 3i6u Homo sapiens CAMK_CHEK2_HUMAN CAMK 6.3e-84 287.4 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6UB O96017 89 501 543.0 No_ligand No_ligand Inactive DFGin 6.1563 12.4796 None -142.78, 168.99 70.83, 76.16 -115.43, 999.0 26.14, 78.04 999.0, 999.0 out-none out 13.9532 Saltbr-none 999.0 HRD-in -61.77, -58.18 77.91, -11.36 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -48.92, -23.0 999.0, -21.53 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.0 0.247 0.28 B 419.0 376.0 37 27 9 18 [[220, 486]] 1.0 3i6u Homo sapiens CAMK_CHEK2_HUMAN CAMK 6.3e-84 287.4 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WA O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.3486 13.5162 None -131.02, -176.1 64.38, 89.31 -97.7, 999.0 302.36, 133.8 999.0, 999.0 out-none out 13.0764 Saltbr-none 999.0 HRD-in -64.4, -41.66 75.43, -23.93 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.49, -47.48 999.0, -37.14 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 A 443.0 369.0 41 27 9 18 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WC O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.5775 13.998 None -131.8, -178.23 63.57, 98.9 -117.45, 999.0 335.54, 98.66 999.0, 999.0 out-none out 13.0805 Saltbr-none 999.0 HRD-in -63.6, -43.12 77.0, -24.17 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.04, -46.8 999.0, -37.07 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 C 443.0 368.0 42 27 9 18 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WE O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.5459 13.6974 None -130.93, -177.05 65.38, 105.03 -130.22, 999.0 325.6, 106.63 999.0, 999.0 out-none out 13.0915 Saltbr-none 999.0 HRD-in -61.69, -42.13 73.77, -23.14 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.57, -46.22 999.0, -36.71 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 E 443.0 368.0 42 27 9 18 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WG O96017 92 501 543.0 No_ligand No_ligand Inactive DFGin 7.5136 13.8031 None -131.95, -176.65 65.29, 79.69 -111.56, 999.0 332.1, 109.83 999.0, 999.0 out-none out 13.0784 Saltbr-none 999.0 HRD-in -62.8, -42.52 74.63, -23.4 none-none-none SNCnnn none-none ActLoopNT-none 999.0 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -53.54, -46.24 999.0, -36.98 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 G 443.0 369.0 41 27 9 18 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WB O96017 92 501 543.0 No_ligand No_ligand None DFGin 6.749 14.2708 BLAminus -132.31, -176.87 65.1, 94.3 -111.58, 28.46 301.82, 101.23 -75.68, -15.25 out-none out 12.8234 Saltbr-none 999.0 HRD-in -62.32, -42.81 74.92, -23.29 none-in-none SNCnin in-none ActLoopNT-in 3.0593 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -68.9, -14.83 999.0, -25.18 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 B 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WD O96017 92 501 543.0 No_ligand No_ligand None DFGin 7.1208 14.4732 BLAminus -130.43, -175.81 63.91, 79.02 -93.96, 27.08 301.9, 101.65 -74.68, -15.75 out-none out 12.8406 Saltbr-none 999.0 HRD-in -63.78, -41.36 74.21, -23.95 none-in-none SNCnin in-none ActLoopNT-in 2.8167 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -68.71, -15.0 999.0, -25.14 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 D 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WF O96017 92 501 543.0 No_ligand No_ligand None DFGin 7.0122 14.1916 BLAminus -131.41, -176.41 64.86, 90.78 -109.15, 26.06 302.9, 101.84 -74.04, -16.03 out-none out 12.8713 Saltbr-none 999.0 HRD-in -63.34, -41.92 73.76, -23.06 none-in-none SNCnin in-none ActLoopNT-in 2.9844 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -68.91, -15.1 999.0, -24.96 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 F 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2
CHEK2 CHK2_HUMAN 3I6WH O96017 92 501 543.0 No_ligand No_ligand None DFGin 6.8741 14.2536 BLAminus -131.53, -176.78 65.02, 88.11 -104.7, 27.13 303.5, 101.73 -74.81, -16.38 out-none out 12.8827 Saltbr-none 999.0 HRD-in -62.35, -41.54 74.34, -23.8 none-in-none SNCnin in-none ActLoopNT-in 3.0871 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -69.26, -15.11 999.0, -24.78 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 K249R None None XRAY 3.25 0.252 0.287 H 443.0 382.0 28 27 22 5 [[220, 486]] 1.0 3i6w Homo sapiens CAMK_CHEK2_HUMAN CAMK 7.4e-84 287.1 1.0 256.0 256.0 367 368 369 371 373 249 273 277 344 346 345 347.0 409 394 389 388 387 386 385 384 383 302 Serine/threonine-protein kinase Chk2

CAMK_CHEK2 (Serine/threonine-protein kinase Chk2)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name