CAMK_CAMK2A (Calcium/calmodulin-dependent protein kinase type II subunit alpha)

Total number of chains: 27
Active chains: 19
Family: CAMK
Uniprot: KCC2A_HUMAN
Kinase Domain Residues: 13 - 271
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 24 88.9% AF-Q9UQM7-K1A
DFGinter None 3 11.1% 3SOAA

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PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
7UJSA 7 274 478.0 ADP:301 ATPlike Active DFGin 6.209 15.164 BLAminus -142.86, -173.92 52.2, 80.06 -100.62, 24.47 291.74, 81.6 -63.11, -26.23 in-in in 9.512 Saltbr-in 3.444 HRD-in -76.47, -52.69 80.52, -7.0 in-in-in SNCiii in-in ActLoopNT-in 2.952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.88, 140.41 APE9-dihe-na 133.49, -148.09 APE8-dihe-in -128.43, 117.33 APE8-rot-in 305.05 APE67-dihe-in -59.07, -26.67 -36.29, -54.08 APE12-dist-in 10.197 APE11-dist-in 11.505 APE10-dist-in 5.779 APE9-dist-in 3.683 Q223K None None XRAY 2.75 0.201 0.262 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujs CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UIRA 7 274 478.0 ATP:302 ATPlike Active DFGin 6.045 15.107 BLAminus -137.0, 179.68 44.28, 101.28 -106.42, 24.78 295.79, 81.95 -53.14, -27.06 in-in in 9.85 Saltbr-in 3.466 HRD-in -74.22, -43.69 67.52, 3.92 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.48, 156.41 APE9-dihe-na 131.95, -156.1 APE8-dihe-in -122.09, 129.91 APE8-rot-in 298.28 APE67-dihe-in -55.12, -36.11 -51.43, -40.3 APE12-dist-in 10.333 APE11-dist-in 11.793 APE10-dist-in 6.056 APE9-dist-in 3.425 D135N,Q223K None None XRAY 3.1 0.234 0.274 A 268 268 0 0 0 0 [[13, 271]] 1.0 7uir CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UIRB 7 273 478.0 ATP:301 ATPlike Active DFGin 6.093 14.463 BLAminus -136.84, -179.4 43.86, 99.82 -105.8, 24.57 296.99, 81.24 -56.04, -26.17 in-in in 9.403 Saltbr-in 3.027 HRD-in -74.93, -42.65 67.84, 3.24 in-in-in SNCiii in-in ActLoopNT-in 2.915 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.86, 157.92 APE9-dihe-na 132.59, -155.55 APE8-dihe-in -122.09, 129.05 APE8-rot-in 298.73 APE67-dihe-in -54.7, -35.97 -51.63, -40.47 APE12-dist-in 10.303 APE11-dist-in 11.733 APE10-dist-in 5.989 APE9-dist-in 3.504 D135N,Q223K None None XRAY 3.1 0.234 0.274 B 268 261 6 0 0 0 [[13, 271]] 1.0 7uir CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UJPA 7 274 478.0 ADP:301 ATPlike Active DFGin 6.775 14.64 BLAminus -129.88, 174.11 65.35, 73.67 -96.28, 29.41 284.7, 81.79 -65.3, -26.47 in-in in 8.527 Saltbr-in 2.903 HRD-in -76.38, -51.72 77.74, -11.0 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.94, 142.69 APE9-dihe-na 139.08, -169.53 APE8-dihe-in -115.65, 123.25 APE8-rot-in 308.77 APE67-dihe-in -69.44, -15.11 -33.38, -56.34 APE12-dist-in 10.469 APE11-dist-in 11.397 APE10-dist-in 5.657 APE9-dist-in 3.521 D135N,Q223K None None XRAY 2.56 0.234 0.281 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujp CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UJPB 7 273 478.0 ATP:301 ATPlike Active DFGin 6.942 14.313 BLAminus -133.64, 174.92 62.39, 75.15 -97.38, 27.07 283.14, 81.65 -64.42, -25.12 in-in in 8.558 Saltbr-in 2.783 HRD-in -76.01, -51.46 77.74, -9.31 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.94, 139.06 APE9-dihe-na 146.74, -166.31 APE8-dihe-in -115.05, 124.1 APE8-rot-in 308.42 APE67-dihe-in -69.31, -14.12 -35.51, -54.36 APE12-dist-in 10.25 APE11-dist-in 11.592 APE10-dist-in 5.843 APE9-dist-in 3.572 D135N,Q223K None None XRAY 2.56 0.234 0.281 B 268 267 0 0 0 0 [[13, 271]] 1.0 7ujp CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
AF-Q9UQM7-K1A 5 279 478.0 No_ligand No_ligand Active DFGin 6.488 14.315 BLAminus -125.02, 173.38 53.51, 80.22 -85.69, 18.65 289.06, 79.25 -60.63, -25.38 in-in in 8.898 Saltbr-in 2.702 HRD-in -73.35, -47.46 65.63, -1.47 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.72, 148.09 APE9-dihe-na 125.54, 170.94 APE8-dihe-in -88.92, 132.18 APE8-rot-in 302.3 APE67-dihe-in -70.6, -10.42 -44.59, -50.01 APE12-dist-in 10.478 APE11-dist-in 11.531 APE10-dist-in 5.755 APE9-dist-in 3.456 None None None AF2 -1.0 1.0 1.0 A 275 275 0 0 0 0 [[13, 271]] 1.0 AF-Q9UQM7-K1 CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
AF-Q9UQM7-K3A 5 279 478.0 No_ligand No_ligand Active DFGin 6.191 13.905 BLAminus -129.09, 176.81 54.38, 73.99 -79.35, 15.21 294.98, 88.86 -61.22, -26.9 in-in in 9.017 Saltbr-in 2.715 HRD-in -74.96, -46.17 66.01, -1.86 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.93, 151.74 APE9-dihe-na 116.08, 172.73 APE8-dihe-in -91.09, 134.45 APE8-rot-in 297.0 APE67-dihe-in -70.49, -13.14 -45.84, -50.34 APE12-dist-in 10.43 APE11-dist-in 11.27 APE10-dist-in 5.606 APE9-dist-in 3.191 None None None AF2 -1.0 1.0 1.0 A 275 275 0 0 0 0 [[13, 271]] 1.0 AF-Q9UQM7-K3 CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
6VZKA 7 274 478.0 No_ligand No_ligand Active DFGin 6.351 13.943 BLAminus -134.11, -178.17 51.67, 87.56 -98.04, 20.59 282.85, 84.39 -60.3, -28.86 in-in in 9.088 Saltbr-in 3.136 HRD-in -72.72, -60.29 84.66, -3.19 in-in-in SNCiii in-in ActLoopNT-in 2.811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.77, 146.91 APE9-dihe-na 134.03, -157.81 APE8-dihe-in -109.96, 122.28 APE8-rot-in 299.52 APE67-dihe-in -55.05, -26.94 -35.18, -55.5 APE12-dist-in 10.16 APE11-dist-in 11.717 APE10-dist-in 5.949 APE9-dist-in 3.748 D135N,Q223K None None XRAY 2.55 0.214 0.294 A 268 258 10 0 0 0 [[13, 271]] 1.0 6vzk CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7KL1A 7 274 478.0 No_ligand No_ligand Active DFGin 6.741 14.476 BLAminus -129.89, 173.99 62.82, 73.66 -90.36, 22.61 284.03, 81.93 -59.26, -32.92 in-in in 8.517 Saltbr-in 2.62 HRD-in -74.19, -47.29 75.62, -9.98 in-in-in SNCiii in-in ActLoopNT-in 2.835 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.66, 145.5 APE9-dihe-na 146.44, -167.15 APE8-dihe-in -115.44, 124.28 APE8-rot-in 304.29 APE67-dihe-in -62.08, -17.44 -33.31, -60.62 APE12-dist-in 10.743 APE11-dist-in 11.382 APE10-dist-in 5.755 APE9-dist-in 3.722 D135N,Q223K None None XRAY 2.4 0.208 0.258 A 268 268 0 0 0 0 [[13, 271]] 1.0 7kl1 CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7KL1B 7 274 478.0 No_ligand No_ligand Active DFGin 6.876 13.994 BLAminus -133.07, 175.01 58.84, 76.6 -91.98, 17.74 279.67, 81.85 -58.73, -30.25 in-in in 8.475 Saltbr-in 2.747 HRD-in -76.2, -48.57 73.65, -5.41 in-in-in SNCiii in-in ActLoopNT-in 2.838 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.02, 138.2 APE9-dihe-na 146.36, -168.65 APE8-dihe-in -114.66, 124.72 APE8-rot-in 303.9 APE67-dihe-in -60.87, -18.94 -37.1, -55.74 APE12-dist-in 10.312 APE11-dist-in 11.652 APE10-dist-in 6.031 APE9-dist-in 3.745 D135N,Q223K None None XRAY 2.4 0.208 0.258 B 268 268 0 0 0 0 [[13, 271]] 1.0 7kl1 CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UIQA 7 274 478.0 No_ligand No_ligand Active DFGin 6.449 15.084 BLAminus -140.43, -178.97 55.68, 69.33 -81.32, 13.56 293.24, 82.91 -55.86, -14.59 in-in in 9.369 Saltbr-in 3.241 HRD-in -63.79, -57.12 80.21, -18.13 in-in-in SNCiii in-in ActLoopNT-in 2.95 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.13, 162.67 APE9-dihe-na 124.48, -161.06 APE8-dihe-in -101.59, 135.95 APE8-rot-in 309.11 APE67-dihe-in -59.39, -26.36 -49.73, -52.37 APE12-dist-in 10.776 APE11-dist-in 11.902 APE10-dist-in 6.319 APE9-dist-in 3.925 D135N,Q223K None None XRAY 3.11 0.261 0.309 A 268 268 0 0 0 0 [[13, 271]] 1.0 7uiq CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UIQB 8 273 478.0 No_ligand No_ligand Active DFGin 6.354 14.86 BLAminus -135.8, -173.94 47.0, 72.56 -81.17, 12.3 291.45, 79.85 -57.12, -13.89 in-in in 9.302 Saltbr-in 3.162 HRD-in -71.21, -53.55 83.02, -20.81 in-in-in SNCiii in-in ActLoopNT-in 3.012 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.85, 162.27 APE9-dihe-na 122.54, -165.04 APE8-dihe-in -104.82, 139.66 APE8-rot-in 306.2 APE67-dihe-in -59.16, -25.74 -56.75, -47.86 APE12-dist-in 10.807 APE11-dist-in 11.867 APE10-dist-in 6.301 APE9-dist-in 4.027 D135N,Q223K None None XRAY 3.11 0.261 0.309 B 268 261 5 0 0 0 [[13, 271]] 1.0 7uiq CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
2VZ6A 9 299 478.0 FEF:60600 Type1 Active DFGin 7.124 13.93 BLAminus -130.3, 144.9 77.59, 104.3 -118.45, 37.91 281.19, 70.53 -60.86, -31.43 in-in in 9.032 Saltbr-in 2.623 HRD-in -71.43, -45.76 75.34, -9.9 in-in-in SNCiii in-in ActLoopNT-in 2.805 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.76, 148.02 APE9-dihe-na 132.07, -168.34 APE8-dihe-in -120.79, 126.49 APE8-rot-in 299.71 APE67-dihe-in -63.07, -18.83 -35.01, -58.7 APE12-dist-in 10.327 APE11-dist-in 11.819 APE10-dist-in 5.993 APE9-dist-in 3.832 None None None XRAY 2.3 0.165 0.203 A 313 289 2 0 0 0 [[13, 271]] 1.0 2vz6 CAMK_CAMK2A_HUMAN CAMK 1.6e-96 328.7 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
2VZ6B 9 300 478.0 FEF:60600 Type1 Active DFGin 6.865 14.032 BLAminus -131.92, 139.26 77.54, 110.88 -122.08, 32.95 286.68, 71.96 -61.55, -26.54 in-in in 9.31 Saltbr-in 2.931 HRD-in -73.12, -44.65 73.93, -20.22 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.21, 149.78 APE9-dihe-na 143.11, -171.05 APE8-dihe-in -118.3, 128.44 APE8-rot-in 303.95 APE67-dihe-in -66.72, -18.78 -39.97, -52.82 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None XRAY 2.3 0.165 0.203 B 313 292 0 0 0 0 [[13, 271]] 1.0 2vz6 CAMK_CAMK2A_HUMAN CAMK 1.6e-96 328.7 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7KL0A 7 274 478.0 UZD:301 Type1 Active DFGin 6.77 14.532 BLAminus -136.67, 172.68 63.72, 78.54 -95.13, 23.83 289.55, 78.47 -63.68, -26.92 in-in in 8.456 Saltbr-in 2.845 HRD-in -73.15, -49.92 78.5, -7.4 in-in-in SNCiii in-in ActLoopNT-in 2.823 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.88, 144.1 APE9-dihe-na 136.1, -171.7 APE8-dihe-in -113.97, 130.36 APE8-rot-in 302.39 APE67-dihe-in -62.47, -20.95 -39.79, -54.85 APE12-dist-in 10.297 APE11-dist-in 11.423 APE10-dist-in 5.714 APE9-dist-in 3.654 D135N,Q223K None None XRAY 2.4 0.209 0.258 A 268 268 0 0 0 0 [[13, 271]] 1.0 7kl0 CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7KL0B 7 274 478.0 UZD:301 Type1 Active DFGin 6.749 14.557 BLAminus -135.5, 169.63 63.85, 78.98 -95.27, 24.21 290.21, 80.29 -65.31, -21.38 in-in in 8.502 Saltbr-in 2.899 HRD-in -76.54, -48.6 76.75, -5.26 in-in-in SNCiii in-in ActLoopNT-in 2.835 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.75, 146.84 APE9-dihe-na 143.82, -168.2 APE8-dihe-in -112.24, 128.47 APE8-rot-in 302.73 APE67-dihe-in -64.12, -18.13 -40.1, -53.96 APE12-dist-in 10.262 APE11-dist-in 11.385 APE10-dist-in 5.689 APE9-dist-in 3.705 D135N,Q223K None None XRAY 2.4 0.209 0.258 B 268 268 0 0 0 0 [[13, 271]] 1.0 7kl0 CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UJQA 7 274 478.0 UZD:301 Type1 Active DFGin 6.71 14.596 BLAminus -130.29, 166.42 66.39, 83.92 -99.29, 27.12 288.6, 77.85 -63.43, -28.99 in-in in 8.503 Saltbr-in 2.716 HRD-in -69.37, -48.63 77.68, -9.72 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.38, 146.4 APE9-dihe-na 132.63, -170.13 APE8-dihe-in -113.98, 127.54 APE8-rot-in 302.91 APE67-dihe-in -64.79, -16.69 -37.21, -55.42 APE12-dist-in 10.39 APE11-dist-in 11.413 APE10-dist-in 5.693 APE9-dist-in 3.661 D135N,Q223K None None XRAY 2.25 0.222 0.271 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujq CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UJQB 7 274 478.0 UZD:301 Type1 Active DFGin 6.776 14.527 BLAminus -130.71, 166.51 65.49, 84.45 -98.57, 27.04 288.12, 79.65 -65.11, -27.34 in-in in 8.514 Saltbr-in 2.74 HRD-in -69.76, -48.69 76.31, -7.39 in-in-in SNCiii in-in ActLoopNT-in 2.91 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.35, 149.36 APE9-dihe-na 136.2, -166.91 APE8-dihe-in -112.91, 126.09 APE8-rot-in 303.49 APE67-dihe-in -63.04, -16.99 -38.33, -54.23 APE12-dist-in 10.355 APE11-dist-in 11.469 APE10-dist-in 5.743 APE9-dist-in 3.69 D135N,Q223K None None XRAY 2.25 0.222 0.271 B 268 268 0 0 0 0 [[13, 271]] 1.0 7ujq CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
6X5GA 7 274 478.0 BCN:303 Type1.5_Back Active DFGin 6.275 15.29 BLAminus -137.39, 173.54 61.4, 81.65 -93.04, 16.42 283.75, 82.3 -58.37, -20.82 in-in in 9.287 Saltbr-in 3.494 HRD-in -74.17, -48.17 75.9, -4.37 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.51, 141.58 APE9-dihe-na 134.3, -159.12 APE8-dihe-in -120.77, 126.02 APE8-rot-in 299.57 APE67-dihe-in -64.67, -15.46 -38.22, -55.61 APE12-dist-in 10.635 APE11-dist-in 11.558 APE10-dist-in 5.946 APE9-dist-in 3.621 D135N,Q223K None None XRAY 1.85 0.189 0.227 A 268 268 0 0 0 0 [[13, 271]] 1.0 6x5g CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UJTA 7 274 478.0 ATP:301 ATPlike Inactive DFGin 5.793 15.871 BLAminus -136.06, 173.98 63.2, 83.03 -96.5, 26.66 288.93, 81.42 -61.86, -26.9 out-out out 10.354 Saltbr-out 4.962 HRD-in -68.86, -51.05 77.4, -6.28 out-in-in SNCoii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.17, 142.76 APE9-dihe-na 138.67, -159.02 APE8-dihe-in -111.71, 119.97 APE8-rot-in 304.14 APE67-dihe-in -65.52, -19.91 -39.43, -49.22 APE12-dist-in 10.406 APE11-dist-in 11.791 APE10-dist-in 5.962 APE9-dist-in 3.835 D135N,Q223K None None XRAY 2.1 0.205 0.246 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujt CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UJRA 7 274 478.0 No_ligand No_ligand Inactive DFGin 5.546 15.912 BLAminus -138.72, 175.62 54.3, 83.24 -93.75, 23.98 285.53, 77.02 -59.87, -27.58 out-out out 10.003 Saltbr-out 4.876 HRD-in -70.69, -48.57 80.32, -8.63 out-in-in SNCoii in-in ActLoopNT-in 2.907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.03, 145.84 APE9-dihe-na 136.24, -161.73 APE8-dihe-in -116.25, 126.46 APE8-rot-in 299.42 APE67-dihe-in -64.43, -22.59 -42.96, -51.59 APE12-dist-in 10.209 APE11-dist-in 11.469 APE10-dist-in 5.732 APE9-dist-in 3.751 Q223K None None XRAY 1.95 0.211 0.252 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujr CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
6X5QA 8 274 478.0 No_ligand No_ligand Inactive DFGin 6.527 15.58 BLAminus -134.71, 170.87 63.66, 75.98 -85.8, 23.34 287.77, 83.34 -69.43, -20.49 out-out out 10.091 Saltbr-out 4.613 HRD-in -66.38, -51.39 77.93, -13.96 out-in-in SNCoii in-in ActLoopNT-in 2.9 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.68, 160.55 APE9-dihe-na 122.71, -155.88 APE8-dihe-in -122.94, 126.71 APE8-rot-in 300.44 APE67-dihe-in -67.88, -13.13 -40.28, -55.54 APE12-dist-in 10.177 APE11-dist-in 11.654 APE10-dist-in 5.988 APE9-dist-in 3.653 D135N,Q223K None None XRAY 2.14 0.192 0.235 A 268 267 0 0 0 0 [[13, 271]] 1.0 6x5q CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7KL2A 7 274 478.0 No_ligand No_ligand Inactive DFGin 6.167 15.536 BLAminus -137.58, -175.58 55.42, 91.02 -111.73, 21.35 287.14, 75.27 -57.86, -27.26 in-out in 9.294 Saltbr-out 3.795 HRD-in -93.15, -40.87 70.97, 4.12 out-in-in SNCoii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.48, 148.08 APE9-dihe-na 123.82, -145.05 APE8-dihe-in -132.54, 127.88 APE8-rot-in 291.51 APE67-dihe-in -61.08, -41.89 -37.96, -52.4 APE12-dist-in 10.253 APE11-dist-in 11.685 APE10-dist-in 5.966 APE9-dist-in 3.556 D135N,Q223K None None XRAY 2.56 0.247 0.293 A 268 268 0 0 0 0 [[13, 271]] 1.0 7kl2 CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
7UISA 7 273 478.0 No_ligand No_ligand Inactive DFGin 6.159 15.598 BLAminus -136.09, 172.3 56.68, 85.32 -101.07, 15.7 288.59, 76.16 -50.93, -32.03 in-out in 9.621 Saltbr-out 4.074 HRD-in -70.04, -54.24 82.99, -21.09 out-in-in SNCoii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.26, 146.81 APE9-dihe-na 126.81, -168.25 APE8-dihe-in -110.56, 126.2 APE8-rot-in 308.0 APE67-dihe-in -57.13, -31.77 -46.02, -45.83 APE12-dist-in 10.335 APE11-dist-in 11.661 APE10-dist-in 5.986 APE9-dist-in 4.094 D135N,Q223K None None XRAY 2.58 0.22 0.268 A 268 267 0 0 0 0 [[13, 271]] 1.0 7uis CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
6W4OO 7 301 478.0 No_ligand No_ligand Inactive DFGinter 10.806 10.238 None -98.81, 109.81 -79.77, 114.68 -136.99, 147.47 315.53, 123.33 104.37, -23.29 in-na in 8.798 Saltbr-na 999.0 HRD-in -73.78, -41.7 68.26, -19.24 na-in-in SNCaii in-in ActLoopNT-in 3.181 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.12, 161.52 APE9-dihe-na 103.65, -177.0 APE8-dihe-in -98.82, 133.37 APE8-rot-in 301.51 APE67-dihe-in -73.83, -31.08 -42.99, -42.18 APE12-dist-in 9.829 APE11-dist-in 10.848 APE10-dist-in 5.275 APE9-dist-in 3.989 K42M None None EM 4.8 999.0 999.0 O 473 293 2 0 0 0 [[13, 271]] 1.0 6w4o CAMK_CAMK2A_HUMAN CAMK 3.3e-93 318.2 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
6W4PH 7 301 478.0 No_ligand No_ligand Inactive DFGinter 10.806 10.237 None -98.91, 109.73 -79.66, 114.62 -137.0, 147.49 315.5, 123.34 104.35, -23.19 in-na in 8.799 Saltbr-na 999.0 HRD-in -73.79, -41.59 68.22, -19.25 na-in-in SNCaii in-in ActLoopNT-in 3.181 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.15, 161.56 APE9-dihe-na 103.69, -177.07 APE8-dihe-in -98.77, 133.22 APE8-rot-in 301.62 APE67-dihe-in -73.83, -31.05 -42.85, -42.28 APE12-dist-in 9.829 APE11-dist-in 10.849 APE10-dist-in 5.276 APE9-dist-in 3.988 K42M None None EM 6.6 999.0 999.0 H 473 293 2 0 0 0 [[13, 271]] 1.0 6w4p CAMK_CAMK2A_HUMAN CAMK 3.3e-93 318.2 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
3SOAA 7 474 478.0 DB8:60445 Type1 Inactive DFGinter 10.807 10.237 None -98.86, 109.77 -79.7, 114.69 -137.02, 147.48 315.53, 123.27 104.35, -23.23 in-na in 8.799 Saltbr-na 999.0 HRD-in -73.81, -41.57 68.14, -19.19 na-in-in SNCaii in-in ActLoopNT-in 3.181 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.13, 161.55 APE9-dihe-na 103.67, -177.05 APE8-dihe-in -98.78, 133.3 APE8-rot-in 301.55 APE67-dihe-in -73.82, -31.03 -42.95, -42.2 APE12-dist-in 9.829 APE11-dist-in 10.848 APE10-dist-in 5.275 APE9-dist-in 3.989 K42M,D135N,T306V None None XRAY 3.55 0.279 0.327 A 444 436 2 0 0 0 [[13, 271]] 1.0 3soa CAMK_CAMK2A_HUMAN CAMK 2.8e-93 318.5 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha

CAMK_CAMK2A (Calcium/calmodulin-dependent protein kinase type II subunit alpha)

Total number of chains: 42
Active chains: 34
Family: CAMK
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 39 92.9% AF-Q9UQM7-K1A
DFGinter None 3 7.1% 3SOAA

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
KCC2A_HUMAN 7UJSA Q9UQM7 7 274 478.0 ADP:301 ATPlike Active DFGin 6.209 15.164 BLAminus -142.86, -173.92 52.2, 80.06 -100.62, 24.47 291.74, 81.6 -63.11, -26.23 in-in in 9.512 Saltbr-in 3.444 HRD-in -76.47, -52.69 80.52, -7.0 in-in-in SNCiii in-in ActLoopNT-in 2.952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.88, 140.41 APE9-dihe-na 133.49, -148.09 APE8-dihe-in -128.43, 117.33 APE8-rot-in 305.05 APE67-dihe-in -59.07, -26.67 -36.29, -54.08 APE12-dist-in 10.197 APE11-dist-in 11.505 APE10-dist-in 5.779 APE9-dist-in 3.683 Q223K None None XRAY 2.75 0.201 0.262 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujs Homo sapiens CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UIRA Q9UQM7 7 274 478.0 ATP:302 ATPlike Active DFGin 6.045 15.107 BLAminus -137.0, 179.68 44.28, 101.28 -106.42, 24.78 295.79, 81.95 -53.14, -27.06 in-in in 9.85 Saltbr-in 3.466 HRD-in -74.22, -43.69 67.52, 3.92 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.48, 156.41 APE9-dihe-na 131.95, -156.1 APE8-dihe-in -122.09, 129.91 APE8-rot-in 298.28 APE67-dihe-in -55.12, -36.11 -51.43, -40.3 APE12-dist-in 10.333 APE11-dist-in 11.793 APE10-dist-in 6.056 APE9-dist-in 3.425 D135N,Q223K None None XRAY 3.1 0.234 0.274 A 268 268 0 0 0 0 [[13, 271]] 1.0 7uir Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UIRB Q9UQM7 7 273 478.0 ATP:301 ATPlike Active DFGin 6.093 14.463 BLAminus -136.84, -179.4 43.86, 99.82 -105.8, 24.57 296.99, 81.24 -56.04, -26.17 in-in in 9.403 Saltbr-in 3.027 HRD-in -74.93, -42.65 67.84, 3.24 in-in-in SNCiii in-in ActLoopNT-in 2.915 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.86, 157.92 APE9-dihe-na 132.59, -155.55 APE8-dihe-in -122.09, 129.05 APE8-rot-in 298.73 APE67-dihe-in -54.7, -35.97 -51.63, -40.47 APE12-dist-in 10.303 APE11-dist-in 11.733 APE10-dist-in 5.989 APE9-dist-in 3.504 D135N,Q223K None None XRAY 3.1 0.234 0.274 B 268 261 6 0 0 0 [[13, 271]] 1.0 7uir Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UJPA Q9UQM7 7 274 478.0 ADP:301 ATPlike Active DFGin 6.775 14.64 BLAminus -129.88, 174.11 65.35, 73.67 -96.28, 29.41 284.7, 81.79 -65.3, -26.47 in-in in 8.527 Saltbr-in 2.903 HRD-in -76.38, -51.72 77.74, -11.0 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.94, 142.69 APE9-dihe-na 139.08, -169.53 APE8-dihe-in -115.65, 123.25 APE8-rot-in 308.77 APE67-dihe-in -69.44, -15.11 -33.38, -56.34 APE12-dist-in 10.469 APE11-dist-in 11.397 APE10-dist-in 5.657 APE9-dist-in 3.521 D135N,Q223K None None XRAY 2.56 0.234 0.281 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujp Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UJPB Q9UQM7 7 273 478.0 ATP:301 ATPlike Active DFGin 6.942 14.313 BLAminus -133.64, 174.92 62.39, 75.15 -97.38, 27.07 283.14, 81.65 -64.42, -25.12 in-in in 8.558 Saltbr-in 2.783 HRD-in -76.01, -51.46 77.74, -9.31 in-in-in SNCiii in-in ActLoopNT-in 2.871 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.94, 139.06 APE9-dihe-na 146.74, -166.31 APE8-dihe-in -115.05, 124.1 APE8-rot-in 308.42 APE67-dihe-in -69.31, -14.12 -35.51, -54.36 APE12-dist-in 10.25 APE11-dist-in 11.592 APE10-dist-in 5.843 APE9-dist-in 3.572 D135N,Q223K None None XRAY 2.56 0.234 0.281 B 268 267 0 0 0 0 [[13, 271]] 1.0 7ujp Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN AF-Q9UQM7-K1A Q9UQM7 5 279 478.0 No_ligand No_ligand Active DFGin 6.488 14.315 BLAminus -125.02, 173.38 53.51, 80.22 -85.69, 18.65 289.06, 79.25 -60.63, -25.38 in-in in 8.898 Saltbr-in 2.702 HRD-in -73.35, -47.46 65.63, -1.47 in-in-in SNCiii in-in ActLoopNT-in 2.981 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.72, 148.09 APE9-dihe-na 125.54, 170.94 APE8-dihe-in -88.92, 132.18 APE8-rot-in 302.3 APE67-dihe-in -70.6, -10.42 -44.59, -50.01 APE12-dist-in 10.478 APE11-dist-in 11.531 APE10-dist-in 5.755 APE9-dist-in 3.456 None None None AF2 -1.0 1.0 1.0 A 275 275 0 0 0 0 [[13, 271]] 1.0 AF-Q9UQM7-K1 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN AF-Q9UQM7-K3A Q9UQM7 5 279 478.0 No_ligand No_ligand Active DFGin 6.191 13.905 BLAminus -129.09, 176.81 54.38, 73.99 -79.35, 15.21 294.98, 88.86 -61.22, -26.9 in-in in 9.017 Saltbr-in 2.715 HRD-in -74.96, -46.17 66.01, -1.86 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.93, 151.74 APE9-dihe-na 116.08, 172.73 APE8-dihe-in -91.09, 134.45 APE8-rot-in 297.0 APE67-dihe-in -70.49, -13.14 -45.84, -50.34 APE12-dist-in 10.43 APE11-dist-in 11.27 APE10-dist-in 5.606 APE9-dist-in 3.191 None None None AF2 -1.0 1.0 1.0 A 275 275 0 0 0 0 [[13, 271]] 1.0 AF-Q9UQM7-K3 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 6VZKA Q9UQM7 7 274 478.0 No_ligand No_ligand Active DFGin 6.351 13.943 BLAminus -134.11, -178.17 51.67, 87.56 -98.04, 20.59 282.85, 84.39 -60.3, -28.86 in-in in 9.088 Saltbr-in 3.136 HRD-in -72.72, -60.29 84.66, -3.19 in-in-in SNCiii in-in ActLoopNT-in 2.811 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -142.77, 146.91 APE9-dihe-na 134.03, -157.81 APE8-dihe-in -109.96, 122.28 APE8-rot-in 299.52 APE67-dihe-in -55.05, -26.94 -35.18, -55.5 APE12-dist-in 10.16 APE11-dist-in 11.717 APE10-dist-in 5.949 APE9-dist-in 3.748 D135N,Q223K None None XRAY 2.55 0.214 0.294 A 268 258 10 0 0 0 [[13, 271]] 1.0 6vzk Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7KL1A Q9UQM7 7 274 478.0 No_ligand No_ligand Active DFGin 6.741 14.476 BLAminus -129.89, 173.99 62.82, 73.66 -90.36, 22.61 284.03, 81.93 -59.26, -32.92 in-in in 8.517 Saltbr-in 2.62 HRD-in -74.19, -47.29 75.62, -9.98 in-in-in SNCiii in-in ActLoopNT-in 2.835 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.66, 145.5 APE9-dihe-na 146.44, -167.15 APE8-dihe-in -115.44, 124.28 APE8-rot-in 304.29 APE67-dihe-in -62.08, -17.44 -33.31, -60.62 APE12-dist-in 10.743 APE11-dist-in 11.382 APE10-dist-in 5.755 APE9-dist-in 3.722 D135N,Q223K None None XRAY 2.4 0.208 0.258 A 268 268 0 0 0 0 [[13, 271]] 1.0 7kl1 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7KL1B Q9UQM7 7 274 478.0 No_ligand No_ligand Active DFGin 6.876 13.994 BLAminus -133.07, 175.01 58.84, 76.6 -91.98, 17.74 279.67, 81.85 -58.73, -30.25 in-in in 8.475 Saltbr-in 2.747 HRD-in -76.2, -48.57 73.65, -5.41 in-in-in SNCiii in-in ActLoopNT-in 2.838 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.02, 138.2 APE9-dihe-na 146.36, -168.65 APE8-dihe-in -114.66, 124.72 APE8-rot-in 303.9 APE67-dihe-in -60.87, -18.94 -37.1, -55.74 APE12-dist-in 10.312 APE11-dist-in 11.652 APE10-dist-in 6.031 APE9-dist-in 3.745 D135N,Q223K None None XRAY 2.4 0.208 0.258 B 268 268 0 0 0 0 [[13, 271]] 1.0 7kl1 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UIQA Q9UQM7 7 274 478.0 No_ligand No_ligand Active DFGin 6.449 15.084 BLAminus -140.43, -178.97 55.68, 69.33 -81.32, 13.56 293.24, 82.91 -55.86, -14.59 in-in in 9.369 Saltbr-in 3.241 HRD-in -63.79, -57.12 80.21, -18.13 in-in-in SNCiii in-in ActLoopNT-in 2.95 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -156.13, 162.67 APE9-dihe-na 124.48, -161.06 APE8-dihe-in -101.59, 135.95 APE8-rot-in 309.11 APE67-dihe-in -59.39, -26.36 -49.73, -52.37 APE12-dist-in 10.776 APE11-dist-in 11.902 APE10-dist-in 6.319 APE9-dist-in 3.925 D135N,Q223K None None XRAY 3.11 0.261 0.309 A 268 268 0 0 0 0 [[13, 271]] 1.0 7uiq Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UIQB Q9UQM7 8 273 478.0 No_ligand No_ligand Active DFGin 6.354 14.86 BLAminus -135.8, -173.94 47.0, 72.56 -81.17, 12.3 291.45, 79.85 -57.12, -13.89 in-in in 9.302 Saltbr-in 3.162 HRD-in -71.21, -53.55 83.02, -20.81 in-in-in SNCiii in-in ActLoopNT-in 3.012 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.85, 162.27 APE9-dihe-na 122.54, -165.04 APE8-dihe-in -104.82, 139.66 APE8-rot-in 306.2 APE67-dihe-in -59.16, -25.74 -56.75, -47.86 APE12-dist-in 10.807 APE11-dist-in 11.867 APE10-dist-in 6.301 APE9-dist-in 4.027 D135N,Q223K None None XRAY 3.11 0.261 0.309 B 268 261 5 0 0 0 [[13, 271]] 1.0 7uiq Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 2VZ6A Q9UQM7 9 299 478.0 FEF:60600 Type1 Active DFGin 7.124 13.93 BLAminus -130.3, 144.9 77.59, 104.3 -118.45, 37.91 281.19, 70.53 -60.86, -31.43 in-in in 9.032 Saltbr-in 2.623 HRD-in -71.43, -45.76 75.34, -9.9 in-in-in SNCiii in-in ActLoopNT-in 2.805 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.76, 148.02 APE9-dihe-na 132.07, -168.34 APE8-dihe-in -120.79, 126.49 APE8-rot-in 299.71 APE67-dihe-in -63.07, -18.83 -35.01, -58.7 APE12-dist-in 10.327 APE11-dist-in 11.819 APE10-dist-in 5.993 APE9-dist-in 3.832 None None None XRAY 2.3 0.165 0.203 A 313 289 2 0 0 0 [[13, 271]] 1.0 2vz6 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 1.6e-96 328.7 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 2VZ6B Q9UQM7 9 300 478.0 FEF:60600 Type1 Active DFGin 6.865 14.032 BLAminus -131.92, 139.26 77.54, 110.88 -122.08, 32.95 286.68, 71.96 -61.55, -26.54 in-in in 9.31 Saltbr-in 2.931 HRD-in -73.12, -44.65 73.93, -20.22 in-in-in SNCiii in-in ActLoopNT-in 2.874 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.21, 149.78 APE9-dihe-na 143.11, -171.05 APE8-dihe-in -118.3, 128.44 APE8-rot-in 303.95 APE67-dihe-in -66.72, -18.78 -39.97, -52.82 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None XRAY 2.3 0.165 0.203 B 313 292 0 0 0 0 [[13, 271]] 1.0 2vz6 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 1.6e-96 328.7 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7KL0A Q9UQM7 7 274 478.0 UZD:301 Type1 Active DFGin 6.77 14.532 BLAminus -136.67, 172.68 63.72, 78.54 -95.13, 23.83 289.55, 78.47 -63.68, -26.92 in-in in 8.456 Saltbr-in 2.845 HRD-in -73.15, -49.92 78.5, -7.4 in-in-in SNCiii in-in ActLoopNT-in 2.823 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.88, 144.1 APE9-dihe-na 136.1, -171.7 APE8-dihe-in -113.97, 130.36 APE8-rot-in 302.39 APE67-dihe-in -62.47, -20.95 -39.79, -54.85 APE12-dist-in 10.297 APE11-dist-in 11.423 APE10-dist-in 5.714 APE9-dist-in 3.654 D135N,Q223K None None XRAY 2.4 0.209 0.258 A 268 268 0 0 0 0 [[13, 271]] 1.0 7kl0 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7KL0B Q9UQM7 7 274 478.0 UZD:301 Type1 Active DFGin 6.749 14.557 BLAminus -135.5, 169.63 63.85, 78.98 -95.27, 24.21 290.21, 80.29 -65.31, -21.38 in-in in 8.502 Saltbr-in 2.899 HRD-in -76.54, -48.6 76.75, -5.26 in-in-in SNCiii in-in ActLoopNT-in 2.835 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.75, 146.84 APE9-dihe-na 143.82, -168.2 APE8-dihe-in -112.24, 128.47 APE8-rot-in 302.73 APE67-dihe-in -64.12, -18.13 -40.1, -53.96 APE12-dist-in 10.262 APE11-dist-in 11.385 APE10-dist-in 5.689 APE9-dist-in 3.705 D135N,Q223K None None XRAY 2.4 0.209 0.258 B 268 268 0 0 0 0 [[13, 271]] 1.0 7kl0 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UJQA Q9UQM7 7 274 478.0 UZD:301 Type1 Active DFGin 6.71 14.596 BLAminus -130.29, 166.42 66.39, 83.92 -99.29, 27.12 288.6, 77.85 -63.43, -28.99 in-in in 8.503 Saltbr-in 2.716 HRD-in -69.37, -48.63 77.68, -9.72 in-in-in SNCiii in-in ActLoopNT-in 2.909 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -151.38, 146.4 APE9-dihe-na 132.63, -170.13 APE8-dihe-in -113.98, 127.54 APE8-rot-in 302.91 APE67-dihe-in -64.79, -16.69 -37.21, -55.42 APE12-dist-in 10.39 APE11-dist-in 11.413 APE10-dist-in 5.693 APE9-dist-in 3.661 D135N,Q223K None None XRAY 2.25 0.222 0.271 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujq Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UJQB Q9UQM7 7 274 478.0 UZD:301 Type1 Active DFGin 6.776 14.527 BLAminus -130.71, 166.51 65.49, 84.45 -98.57, 27.04 288.12, 79.65 -65.11, -27.34 in-in in 8.514 Saltbr-in 2.74 HRD-in -69.76, -48.69 76.31, -7.39 in-in-in SNCiii in-in ActLoopNT-in 2.91 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -153.35, 149.36 APE9-dihe-na 136.2, -166.91 APE8-dihe-in -112.91, 126.09 APE8-rot-in 303.49 APE67-dihe-in -63.04, -16.99 -38.33, -54.23 APE12-dist-in 10.355 APE11-dist-in 11.469 APE10-dist-in 5.743 APE9-dist-in 3.69 D135N,Q223K None None XRAY 2.25 0.222 0.271 B 268 268 0 0 0 0 [[13, 271]] 1.0 7ujq Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 6X5GA Q9UQM7 7 274 478.0 BCN:303 Type1.5_Back Active DFGin 6.275 15.29 BLAminus -137.39, 173.54 61.4, 81.65 -93.04, 16.42 283.75, 82.3 -58.37, -20.82 in-in in 9.287 Saltbr-in 3.494 HRD-in -74.17, -48.17 75.9, -4.37 in-in-in SNCiii in-in ActLoopNT-in 2.881 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -149.51, 141.58 APE9-dihe-na 134.3, -159.12 APE8-dihe-in -120.77, 126.02 APE8-rot-in 299.57 APE67-dihe-in -64.67, -15.46 -38.22, -55.61 APE12-dist-in 10.635 APE11-dist-in 11.558 APE10-dist-in 5.946 APE9-dist-in 3.621 D135N,Q223K None None XRAY 1.85 0.189 0.227 A 268 268 0 0 0 0 [[13, 271]] 1.0 6x5g Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UJTA Q9UQM7 7 274 478.0 ATP:301 ATPlike Inactive DFGin 5.793 15.871 BLAminus -136.06, 173.98 63.2, 83.03 -96.5, 26.66 288.93, 81.42 -61.86, -26.9 out-out out 10.354 Saltbr-out 4.962 HRD-in -68.86, -51.05 77.4, -6.28 out-in-in SNCoii in-in ActLoopNT-in 2.865 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.17, 142.76 APE9-dihe-na 138.67, -159.02 APE8-dihe-in -111.71, 119.97 APE8-rot-in 304.14 APE67-dihe-in -65.52, -19.91 -39.43, -49.22 APE12-dist-in 10.406 APE11-dist-in 11.791 APE10-dist-in 5.962 APE9-dist-in 3.835 D135N,Q223K None None XRAY 2.1 0.205 0.246 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujt Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UJRA Q9UQM7 7 274 478.0 No_ligand No_ligand Inactive DFGin 5.546 15.912 BLAminus -138.72, 175.62 54.3, 83.24 -93.75, 23.98 285.53, 77.02 -59.87, -27.58 out-out out 10.003 Saltbr-out 4.876 HRD-in -70.69, -48.57 80.32, -8.63 out-in-in SNCoii in-in ActLoopNT-in 2.907 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.03, 145.84 APE9-dihe-na 136.24, -161.73 APE8-dihe-in -116.25, 126.46 APE8-rot-in 299.42 APE67-dihe-in -64.43, -22.59 -42.96, -51.59 APE12-dist-in 10.209 APE11-dist-in 11.469 APE10-dist-in 5.732 APE9-dist-in 3.751 Q223K None None XRAY 1.95 0.211 0.252 A 268 268 0 0 0 0 [[13, 271]] 1.0 7ujr Homo sapiens CAMK_CAMK2A_HUMAN CAMK 1e-96 329.1 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 6X5QA Q9UQM7 8 274 478.0 No_ligand No_ligand Inactive DFGin 6.527 15.58 BLAminus -134.71, 170.87 63.66, 75.98 -85.8, 23.34 287.77, 83.34 -69.43, -20.49 out-out out 10.091 Saltbr-out 4.613 HRD-in -66.38, -51.39 77.93, -13.96 out-in-in SNCoii in-in ActLoopNT-in 2.9 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.68, 160.55 APE9-dihe-na 122.71, -155.88 APE8-dihe-in -122.94, 126.71 APE8-rot-in 300.44 APE67-dihe-in -67.88, -13.13 -40.28, -55.54 APE12-dist-in 10.177 APE11-dist-in 11.654 APE10-dist-in 5.988 APE9-dist-in 3.653 D135N,Q223K None None XRAY 2.14 0.192 0.235 A 268 267 0 0 0 0 [[13, 271]] 1.0 6x5q Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7KL2A Q9UQM7 7 274 478.0 No_ligand No_ligand Inactive DFGin 6.167 15.536 BLAminus -137.58, -175.58 55.42, 91.02 -111.73, 21.35 287.14, 75.27 -57.86, -27.26 in-out in 9.294 Saltbr-out 3.795 HRD-in -93.15, -40.87 70.97, 4.12 out-in-in SNCoii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -152.48, 148.08 APE9-dihe-na 123.82, -145.05 APE8-dihe-in -132.54, 127.88 APE8-rot-in 291.51 APE67-dihe-in -61.08, -41.89 -37.96, -52.4 APE12-dist-in 10.253 APE11-dist-in 11.685 APE10-dist-in 5.966 APE9-dist-in 3.556 D135N,Q223K None None XRAY 2.56 0.247 0.293 A 268 268 0 0 0 0 [[13, 271]] 1.0 7kl2 Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 7UISA Q9UQM7 7 273 478.0 No_ligand No_ligand Inactive DFGin 6.159 15.598 BLAminus -136.09, 172.3 56.68, 85.32 -101.07, 15.7 288.59, 76.16 -50.93, -32.03 in-out in 9.621 Saltbr-out 4.074 HRD-in -70.04, -54.24 82.99, -21.09 out-in-in SNCoii in-in ActLoopNT-in 2.888 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -160.26, 146.81 APE9-dihe-na 126.81, -168.25 APE8-dihe-in -110.56, 126.2 APE8-rot-in 308.0 APE67-dihe-in -57.13, -31.77 -46.02, -45.83 APE12-dist-in 10.335 APE11-dist-in 11.661 APE10-dist-in 5.986 APE9-dist-in 4.094 D135N,Q223K None None XRAY 2.58 0.22 0.268 A 268 267 0 0 0 0 [[13, 271]] 1.0 7uis Homo sapiens CAMK_CAMK2A_HUMAN CAMK 9.3e-96 326.0 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 6W4OO Q9UQM7 7 301 478.0 No_ligand No_ligand Inactive DFGinter 10.806 10.238 None -98.81, 109.81 -79.77, 114.68 -136.99, 147.47 315.53, 123.33 104.37, -23.29 in-na in 8.798 Saltbr-na 999.0 HRD-in -73.78, -41.7 68.26, -19.24 na-in-in SNCaii in-in ActLoopNT-in 3.181 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.12, 161.52 APE9-dihe-na 103.65, -177.0 APE8-dihe-in -98.82, 133.37 APE8-rot-in 301.51 APE67-dihe-in -73.83, -31.08 -42.99, -42.18 APE12-dist-in 9.829 APE11-dist-in 10.848 APE10-dist-in 5.275 APE9-dist-in 3.989 K42M None None EM 4.8 999.0 999.0 O 473 293 2 0 0 0 [[13, 271]] 1.0 6w4o Homo sapiens CAMK_CAMK2A_HUMAN CAMK 3.3e-93 318.2 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 6W4PH Q9UQM7 7 301 478.0 No_ligand No_ligand Inactive DFGinter 10.806 10.237 None -98.91, 109.73 -79.66, 114.62 -137.0, 147.49 315.5, 123.34 104.35, -23.19 in-na in 8.799 Saltbr-na 999.0 HRD-in -73.79, -41.59 68.22, -19.25 na-in-in SNCaii in-in ActLoopNT-in 3.181 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.15, 161.56 APE9-dihe-na 103.69, -177.07 APE8-dihe-in -98.77, 133.22 APE8-rot-in 301.62 APE67-dihe-in -73.83, -31.05 -42.85, -42.28 APE12-dist-in 9.829 APE11-dist-in 10.849 APE10-dist-in 5.276 APE9-dist-in 3.988 K42M None None EM 6.6 999.0 999.0 H 473 293 2 0 0 0 [[13, 271]] 1.0 6w4p Homo sapiens CAMK_CAMK2A_HUMAN CAMK 3.3e-93 318.2 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_HUMAN 3SOAA Q9UQM7 7 474 478.0 DB8:60445 Type1 Inactive DFGinter 10.807 10.237 None -98.86, 109.77 -79.7, 114.69 -137.02, 147.48 315.53, 123.27 104.35, -23.23 in-na in 8.799 Saltbr-na 999.0 HRD-in -73.81, -41.57 68.14, -19.19 na-in-in SNCaii in-in ActLoopNT-in 3.181 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.13, 161.55 APE9-dihe-na 103.67, -177.05 APE8-dihe-in -98.78, 133.3 APE8-rot-in 301.55 APE67-dihe-in -73.82, -31.03 -42.95, -42.2 APE12-dist-in 9.829 APE11-dist-in 10.848 APE10-dist-in 5.275 APE9-dist-in 3.989 K42M,D135N,T306V None None XRAY 3.55 0.279 0.327 A 444 436 2 0 0 0 [[13, 271]] 1.0 3soa Homo sapiens CAMK_CAMK2A_HUMAN CAMK 2.8e-93 318.5 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_MOUSE 7B56B P11798 5 307 478.0 ANP:60401 ATPlike Active DFGin 6.729 14.232 BLAminus -127.69, 175.68 61.5, 79.97 -89.44, 23.96 289.95, 77.46 -66.33, -24.14 in-in in 8.963 Saltbr-in 2.797 HRD-in -75.83, -42.64 71.61, -6.11 in-in-in SNCiii in-in ActLoopNT-in 2.891 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.35, 145.48 APE9-dihe-na 136.45, -166.63 APE8-dihe-in -115.36, 130.21 APE8-rot-in 297.52 APE67-dihe-in -66.37, -13.84 -48.36, -50.63 APE12-dist-in 10.406 APE11-dist-in 11.67 APE10-dist-in 5.883 APE9-dist-in 3.799 T305A,T306A None None XRAY 1.45 0.191 0.215 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b56 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_MOUSE 7B57B P11798 5 307 478.0 ADP:603 ATPlike Active DFGin 6.612 14.081 BLAminus -127.42, 175.73 58.47, 86.34 -93.82, 26.41 288.57, 77.62 -63.18, -29.51 in-in in 8.79 Saltbr-in 2.799 HRD-in -66.41, -49.66 65.98, 1.57 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.13, 142.7 APE9-dihe-na 131.67, 177.43 APE8-dihe-in -91.43, 131.98 APE8-rot-in 302.75 APE67-dihe-in -62.31, -16.39 -48.04, -47.99 APE12-dist-in 10.368 APE11-dist-in 11.44 APE10-dist-in 5.743 APE9-dist-in 3.998 T305A,T306A None None XRAY 1.95 0.206 0.247 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b57 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_MOUSE 7B55B P11798 5 312 478.0 No_ligand No_ligand Active DFGin 6.737 14.001 BLAminus -130.59, 167.68 65.62, 87.9 -96.05, 24.95 289.73, 74.39 -58.3, -31.88 in-in in 8.775 Saltbr-in 2.744 HRD-in -69.98, -47.5 67.83, 2.57 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.09, 141.72 APE9-dihe-na 131.6, 179.58 APE8-dihe-in -96.74, 130.32 APE8-rot-in 288.79 APE67-dihe-in -62.69, -14.11 -44.5, -51.15 APE12-dist-in 10.443 APE11-dist-in 11.496 APE10-dist-in 5.795 APE9-dist-in 4.059 T305A,T306A None None XRAY 1.6 0.198 0.214 B 317 308 0 0 0 0 [[13, 271]] 1.0 7b55 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YA P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.86, 139.31 77.49, 110.85 -122.06, 32.93 286.68, 71.99 -61.48, -26.61 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.13, -44.6 73.87, -20.22 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.25, 149.7 APE9-dihe-na 143.17, -171.02 APE8-dihe-in -118.35, 128.47 APE8-rot-in 303.96 APE67-dihe-in -66.76, -18.7 -40.04, -52.83 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 A 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YB P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.032 BLAminus -131.95, 139.31 77.48, 110.85 -122.06, 32.98 286.65, 71.96 -61.49, -26.64 in-in in 9.311 Saltbr-in 2.93 HRD-in -73.09, -44.73 74.01, -20.3 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.28, 149.66 APE9-dihe-na 143.24, -170.9 APE8-dihe-in -118.43, 128.46 APE8-rot-in 303.94 APE67-dihe-in -66.75, -18.73 -40.11, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.757 APE10-dist-in 5.996 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 B 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YC P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.96, 139.34 77.44, 110.96 -122.08, 32.86 286.64, 72.06 -61.52, -26.54 in-in in 9.31 Saltbr-in 2.931 HRD-in -73.14, -44.67 73.9, -20.21 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.22, 149.66 APE9-dihe-na 143.26, -171.08 APE8-dihe-in -118.34, 128.48 APE8-rot-in 303.98 APE67-dihe-in -66.83, -18.67 -40.06, -52.78 APE12-dist-in 10.251 APE11-dist-in 11.755 APE10-dist-in 5.995 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 C 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YD P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.032 BLAminus -131.91, 139.34 77.49, 110.87 -122.11, 32.91 286.66, 71.93 -61.43, -26.54 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.12, -44.58 73.75, -20.14 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.2, 149.78 APE9-dihe-na 143.1, -171.01 APE8-dihe-in -118.32, 128.47 APE8-rot-in 303.98 APE67-dihe-in -66.82, -18.71 -40.07, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.995 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 D 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YE P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.93, 139.32 77.45, 110.92 -122.11, 33.05 286.68, 71.92 -61.6, -26.5 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.04, -44.67 73.88, -20.22 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.16, 149.72 APE9-dihe-na 143.17, -171.04 APE8-dihe-in -118.33, 128.47 APE8-rot-in 303.95 APE67-dihe-in -66.81, -18.72 -40.11, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.757 APE10-dist-in 5.997 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 E 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YF P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.032 BLAminus -131.93, 139.32 77.42, 110.87 -122.1, 32.98 286.71, 71.94 -61.53, -26.5 in-in in 9.311 Saltbr-in 2.932 HRD-in -73.09, -44.66 73.92, -20.32 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.26, 149.65 APE9-dihe-na 143.17, -171.02 APE8-dihe-in -118.33, 128.42 APE8-rot-in 304.0 APE67-dihe-in -66.75, -18.74 -40.02, -52.76 APE12-dist-in 10.251 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.962 None None None EM 20.0 999.0 999.0 F 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YG P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.032 BLAminus -131.85, 139.33 77.48, 110.87 -122.11, 32.96 286.62, 72.03 -61.49, -26.59 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.18, -44.61 73.91, -20.27 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.24, 149.76 APE9-dihe-na 143.06, -171.13 APE8-dihe-in -118.25, 128.47 APE8-rot-in 304.07 APE67-dihe-in -66.77, -18.8 -40.08, -52.75 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 G 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YH P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.032 BLAminus -131.88, 139.32 77.5, 110.88 -122.07, 32.96 286.74, 71.95 -61.56, -26.5 in-in in 9.311 Saltbr-in 2.932 HRD-in -73.06, -44.63 73.85, -20.24 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.2, 149.67 APE9-dihe-na 143.16, -171.09 APE8-dihe-in -118.29, 128.44 APE8-rot-in 303.93 APE67-dihe-in -66.72, -18.73 -40.03, -52.81 APE12-dist-in 10.253 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 H 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YI P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.88, 139.32 77.51, 110.82 -122.03, 32.96 286.72, 72.01 -61.6, -26.54 in-in in 9.311 Saltbr-in 2.93 HRD-in -73.14, -44.59 73.89, -20.24 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.18, 149.76 APE9-dihe-na 143.1, -170.97 APE8-dihe-in -118.34, 128.48 APE8-rot-in 304.0 APE67-dihe-in -66.74, -18.77 -40.07, -52.78 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 I 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YJ P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.864 14.031 BLAminus -131.96, 139.32 77.43, 110.94 -122.11, 32.97 286.66, 72.03 -61.61, -26.48 in-in in 9.311 Saltbr-in 2.932 HRD-in -73.06, -44.6 73.89, -20.28 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.26, 149.71 APE9-dihe-na 143.13, -170.97 APE8-dihe-in -118.31, 128.48 APE8-rot-in 304.0 APE67-dihe-in -66.76, -18.72 -40.1, -52.77 APE12-dist-in 10.252 APE11-dist-in 11.757 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 J 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YK P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.033 BLAminus -131.9, 139.29 77.45, 110.86 -122.02, 32.92 286.62, 72.03 -61.54, -26.54 in-in in 9.311 Saltbr-in 2.93 HRD-in -73.15, -44.63 73.76, -20.13 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.25, 149.7 APE9-dihe-na 143.13, -171.07 APE8-dihe-in -118.27, 128.49 APE8-rot-in 303.97 APE67-dihe-in -66.81, -18.77 -40.05, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 K 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YL P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.92, 139.31 77.56, 110.83 -122.08, 32.9 286.66, 71.99 -61.46, -26.52 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.09, -44.69 73.91, -20.23 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.24, 149.66 APE9-dihe-na 143.13, -170.99 APE8-dihe-in -118.31, 128.48 APE8-rot-in 303.97 APE67-dihe-in -66.81, -18.73 -40.08, -52.69 APE12-dist-in 10.252 APE11-dist-in 11.755 APE10-dist-in 5.995 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 L 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha

CAMK_CAMK2A (Calcium/calmodulin-dependent protein kinase type II subunit alpha)

Total number of chains: 15
Active chains: 15
Family: CAMK
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 15 100.0% 7B56B

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
KCC2A_MOUSE 7B56B P11798 5 307 478.0 ANP:60401 ATPlike Active DFGin 6.729 14.232 BLAminus -127.69, 175.68 61.5, 79.97 -89.44, 23.96 289.95, 77.46 -66.33, -24.14 in-in in 8.963 Saltbr-in 2.797 HRD-in -75.83, -42.64 71.61, -6.11 in-in-in SNCiii in-in ActLoopNT-in 2.891 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -146.35, 145.48 APE9-dihe-na 136.45, -166.63 APE8-dihe-in -115.36, 130.21 APE8-rot-in 297.52 APE67-dihe-in -66.37, -13.84 -48.36, -50.63 APE12-dist-in 10.406 APE11-dist-in 11.67 APE10-dist-in 5.883 APE9-dist-in 3.799 T305A,T306A None None XRAY 1.45 0.191 0.215 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b56 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_MOUSE 7B57B P11798 5 307 478.0 ADP:603 ATPlike Active DFGin 6.612 14.081 BLAminus -127.42, 175.73 58.47, 86.34 -93.82, 26.41 288.57, 77.62 -63.18, -29.51 in-in in 8.79 Saltbr-in 2.799 HRD-in -66.41, -49.66 65.98, 1.57 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -154.13, 142.7 APE9-dihe-na 131.67, 177.43 APE8-dihe-in -91.43, 131.98 APE8-rot-in 302.75 APE67-dihe-in -62.31, -16.39 -48.04, -47.99 APE12-dist-in 10.368 APE11-dist-in 11.44 APE10-dist-in 5.743 APE9-dist-in 3.998 T305A,T306A None None XRAY 1.95 0.206 0.247 B 317 303 0 0 0 0 [[13, 271]] 1.0 7b57 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_MOUSE 7B55B P11798 5 312 478.0 No_ligand No_ligand Active DFGin 6.737 14.001 BLAminus -130.59, 167.68 65.62, 87.9 -96.05, 24.95 289.73, 74.39 -58.3, -31.88 in-in in 8.775 Saltbr-in 2.744 HRD-in -69.98, -47.5 67.83, 2.57 in-in-in SNCiii in-in ActLoopNT-in 2.933 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.09, 141.72 APE9-dihe-na 131.6, 179.58 APE8-dihe-in -96.74, 130.32 APE8-rot-in 288.79 APE67-dihe-in -62.69, -14.11 -44.5, -51.15 APE12-dist-in 10.443 APE11-dist-in 11.496 APE10-dist-in 5.795 APE9-dist-in 4.059 T305A,T306A None None XRAY 1.6 0.198 0.214 B 317 308 0 0 0 0 [[13, 271]] 1.0 7b55 Mus musculus CAMK_CAMK2A_MOUSE CAMK 1.7e-96 328.6 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YA P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.86, 139.31 77.49, 110.85 -122.06, 32.93 286.68, 71.99 -61.48, -26.61 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.13, -44.6 73.87, -20.22 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.25, 149.7 APE9-dihe-na 143.17, -171.02 APE8-dihe-in -118.35, 128.47 APE8-rot-in 303.96 APE67-dihe-in -66.76, -18.7 -40.04, -52.83 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 A 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YB P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.032 BLAminus -131.95, 139.31 77.48, 110.85 -122.06, 32.98 286.65, 71.96 -61.49, -26.64 in-in in 9.311 Saltbr-in 2.93 HRD-in -73.09, -44.73 74.01, -20.3 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.28, 149.66 APE9-dihe-na 143.24, -170.9 APE8-dihe-in -118.43, 128.46 APE8-rot-in 303.94 APE67-dihe-in -66.75, -18.73 -40.11, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.757 APE10-dist-in 5.996 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 B 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YC P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.96, 139.34 77.44, 110.96 -122.08, 32.86 286.64, 72.06 -61.52, -26.54 in-in in 9.31 Saltbr-in 2.931 HRD-in -73.14, -44.67 73.9, -20.21 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.22, 149.66 APE9-dihe-na 143.26, -171.08 APE8-dihe-in -118.34, 128.48 APE8-rot-in 303.98 APE67-dihe-in -66.83, -18.67 -40.06, -52.78 APE12-dist-in 10.251 APE11-dist-in 11.755 APE10-dist-in 5.995 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 C 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YD P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.032 BLAminus -131.91, 139.34 77.49, 110.87 -122.11, 32.91 286.66, 71.93 -61.43, -26.54 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.12, -44.58 73.75, -20.14 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.2, 149.78 APE9-dihe-na 143.1, -171.01 APE8-dihe-in -118.32, 128.47 APE8-rot-in 303.98 APE67-dihe-in -66.82, -18.71 -40.07, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.995 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 D 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YE P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.93, 139.32 77.45, 110.92 -122.11, 33.05 286.68, 71.92 -61.6, -26.5 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.04, -44.67 73.88, -20.22 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.16, 149.72 APE9-dihe-na 143.17, -171.04 APE8-dihe-in -118.33, 128.47 APE8-rot-in 303.95 APE67-dihe-in -66.81, -18.72 -40.11, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.757 APE10-dist-in 5.997 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 E 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YF P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.032 BLAminus -131.93, 139.32 77.42, 110.87 -122.1, 32.98 286.71, 71.94 -61.53, -26.5 in-in in 9.311 Saltbr-in 2.932 HRD-in -73.09, -44.66 73.92, -20.32 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.26, 149.65 APE9-dihe-na 143.17, -171.02 APE8-dihe-in -118.33, 128.42 APE8-rot-in 304.0 APE67-dihe-in -66.75, -18.74 -40.02, -52.76 APE12-dist-in 10.251 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.962 None None None EM 20.0 999.0 999.0 F 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YG P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.032 BLAminus -131.85, 139.33 77.48, 110.87 -122.11, 32.96 286.62, 72.03 -61.49, -26.59 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.18, -44.61 73.91, -20.27 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.24, 149.76 APE9-dihe-na 143.06, -171.13 APE8-dihe-in -118.25, 128.47 APE8-rot-in 304.07 APE67-dihe-in -66.77, -18.8 -40.08, -52.75 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 G 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YH P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.032 BLAminus -131.88, 139.32 77.5, 110.88 -122.07, 32.96 286.74, 71.95 -61.56, -26.5 in-in in 9.311 Saltbr-in 2.932 HRD-in -73.06, -44.63 73.85, -20.24 in-in-in SNCiii in-in ActLoopNT-in 2.876 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.2, 149.67 APE9-dihe-na 143.16, -171.09 APE8-dihe-in -118.29, 128.44 APE8-rot-in 303.93 APE67-dihe-in -66.72, -18.73 -40.03, -52.81 APE12-dist-in 10.253 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 H 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YI P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.88, 139.32 77.51, 110.82 -122.03, 32.96 286.72, 72.01 -61.6, -26.54 in-in in 9.311 Saltbr-in 2.93 HRD-in -73.14, -44.59 73.89, -20.24 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.18, 149.76 APE9-dihe-na 143.1, -170.97 APE8-dihe-in -118.34, 128.48 APE8-rot-in 304.0 APE67-dihe-in -66.74, -18.77 -40.07, -52.78 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 I 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YJ P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.864 14.031 BLAminus -131.96, 139.32 77.43, 110.94 -122.11, 32.97 286.66, 72.03 -61.61, -26.48 in-in in 9.311 Saltbr-in 2.932 HRD-in -73.06, -44.6 73.89, -20.28 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.26, 149.71 APE9-dihe-na 143.13, -170.97 APE8-dihe-in -118.31, 128.48 APE8-rot-in 304.0 APE67-dihe-in -66.76, -18.72 -40.1, -52.77 APE12-dist-in 10.252 APE11-dist-in 11.757 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 J 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YK P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.866 14.033 BLAminus -131.9, 139.29 77.45, 110.86 -122.02, 32.92 286.62, 72.03 -61.54, -26.54 in-in in 9.311 Saltbr-in 2.93 HRD-in -73.15, -44.63 73.76, -20.13 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.25, 149.7 APE9-dihe-na 143.13, -171.07 APE8-dihe-in -118.27, 128.49 APE8-rot-in 303.97 APE67-dihe-in -66.81, -18.77 -40.05, -52.72 APE12-dist-in 10.252 APE11-dist-in 11.756 APE10-dist-in 5.996 APE9-dist-in 3.963 None None None EM 20.0 999.0 999.0 K 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha
KCC2A_RAT 5U6YL P11275 13 472 478.0 No_ligand No_ligand Active DFGin 6.865 14.031 BLAminus -131.92, 139.31 77.56, 110.83 -122.08, 32.9 286.66, 71.99 -61.46, -26.52 in-in in 9.311 Saltbr-in 2.931 HRD-in -73.09, -44.69 73.91, -20.23 in-in-in SNCiii in-in ActLoopNT-in 2.875 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -148.24, 149.66 APE9-dihe-na 143.13, -170.99 APE8-dihe-in -118.31, 128.48 APE8-rot-in 303.97 APE67-dihe-in -66.81, -18.73 -40.08, -52.69 APE12-dist-in 10.252 APE11-dist-in 11.755 APE10-dist-in 5.995 APE9-dist-in 3.964 None None None EM 20.0 999.0 999.0 L 461 458 0 0 0 0 [[13, 271]] 1.0 5u6y Rattus norvegicus CAMK_CAMK2A_RAT CAMK 5.4e-96 327.3 1 256 256 155 156 157 159 161 42 60 64 132 134 133 135 195 183 178 177 176 175 174 173 172 90 Calcium/calmodulin-dependent protein kinase type II subunit alpha