4YHJ

GRK4 (G protein-coupled receptor kinase 4)
Group: AGC
Uniprot: GRK4_HUMAN
Organism: Homo sapiens
Domain boundary: 187 - 449
Resolu: 2.6

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in AN2 Type1 25 - 525 0
B Active DFGin BLAminus in-in in-in AN2 Type1 25 - 527 0
Representative sequence - Chain B
10 20 30 40
melenivans lllkarqggy gkksGRSKKW KEILTLPPVS
50 60 70 80
QCSELRHSIE KDYSSLCDKQ PIGRRLFRQF CDTKPTLKRH
90 100 110 120
IEFLDAVAEY EVADDEDRSD CGLSILDRFF NDKLAAPLPE
130 140 150 160
IPPDVVTECR LGLKEENPSK KAFEECTRVA HNYLRGEPFE
170 180 190 200
EYQESSYFSQ FLQWKWLERQ PVTKNTFRHY RVLGKGGFGE
210 220 230 240
VCACQVRATG KMYACKKLQK KRIKKRKGEA MALNEKRILE
250 260 270 280
KVQSRFVVSL AYAYETKDAL CLVLTIMNGG DLKFHIYNLG
290 300 310 320
NPGFDEQRAV FYAAELCCGL EDLQRERIVY RDLKPENILL
330 340 350 360
DDRGHIRISD LGLATEIPEG QRVRGRVGTV GYMAPEVVNN
370 380 390 400
EKYTFSPDWW GLGCLIYEMI QGHSPFKKYK EKVKWEEVDQ
410 420 430 440
RIKNDTEEYS EKFSEDAKSI CRMLLTKNPS KRLGCRGEGA
450 460 470 480
AGVKQHPVFK DINFRRLEAN MLEPPFCPDP HAVYCkdvld
490 500 510 520
ieqfsvvkGI YLDTADEDFY ARFATGCVSI PWQNEMIESG
530 540 550 560
CFKDINKses eealpldldk nihtpvsrpn rgffyrlfrr
570 -
ggsltmvpse kevepkqsen lyfq
Lower-case residues are disordered in structure.
Mutations: C563S,C578S
Phosphorylation: None