4WNK

GRK5 (G protein-coupled receptor kinase 5)
Group: AGC
Uniprot: GRK5_BOVIN
Organism: Bos taurus
Domain boundary: 186 - 448
Resolu: 2.42

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Inactive DFGin ABAminus in-in in-in 453 Type1.5_Front 24 - 541 0
Representative sequence - Chain A
10 20 30 40
melenivant vllkareggg gkrKGKSKKW KEILKFPHIN
50 60 70 80
QCEDLRRTID RDYCSLCDKQ PVGRLLFRQF CETRPGLESY
90 100 110 120
IQFLDSVAEY EVTPDEKLGE KGKEIMTKYL TPKSPVFITQ
130 140 150 160
VGRDLVSQTE EKLLQKPCKE LFSACVQSVH DYLRGEPFHE
170 180 190 200
YLDSMYFDRF LQWKWLERQP VTKNTFRQYR VLGKGGFGEV
210 220 230 240
CACQVRATGK MYACKRLEKK RIKKRKGESM ALNEKQILEK
250 260 270 280
VNSRFVVNLA YAYETKDALC LVLTIMNGGD LKFHIYNMGN
290 300 310 320
PGFEEERALF YAAEILCGLE DLHHENIVYR DLKPENILLD
330 340 350 360
DYGHIRISDL GLAVKIPEGD LIRGRVGTVG YMAPEVLNNQ
370 380 390 400
RYGLSPDYWG LGCLIYEMIE GQSPFRGRKE KVKREEVDRR
410 420 430 440
VLETEEVYSH KFSEEAKSIC KMLLTKDAKQ RLGCQEEGAA
450 460 470 480
EVKRHPFFRN MNFKRLEAGM LDPPFVPDPR AVYckdvldi
490 500 510 520
eqfstvkgvn ldHTDDDFYS KFSTGSVPIP WQSEMIETEC
530 540 550 560
FKELNVFGPH GTLSPDLNRS Hppeppkkgl lqrlfkrqhq
570 580 590
nnsksspnsk tsfnhhinsn hvssnstgss vdhhhhhh
Lower-case residues are disordered in structure.
Mutations: None
Phosphorylation: None