4TND

GRK5 (G protein-coupled receptor kinase 5)
Group: AGC
Uniprot: GRK5_HUMAN
Organism: Homo sapiens
Domain boundary: 186 - 448
Resolu: 1.802

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in ANP Type1 15 - 543 0
Representative sequence - Chain A
10 20 30 40
melenivant vllkAREGGG GKRKGKSKKW KEILKFPHIS
50 60 70 80
QCEDLRRTID RDYCSLCDKQ PIGRLLFRQF CETRPGLECY
90 100 110 120
IQFLDSVAEY EVTPDEKLGE KGKKIMTKYL TPKSPVFIAQ
130 140 150 160
VGQDLVSQTE EKLLQKPCKE LFSACAQSVH EYLRGEPFHE
170 180 190 200
YLDSMFFDRF LQWKWLERQP VTKNTFRQYR VLGKGGFGEV
210 220 230 240
CACQVRATGK MYACKRLEKK RIKKRKGESM ALNEKQILEK
250 260 270 280
VNSQFVVNLA YAYETKDALC LVLTIMNGGD LKFHIYNMGN
290 300 310 320
PGFEEERALF YAAEILCGLE DLHHENTVYR DLKPENILLD
330 340 350 360
DYGHIRISDL GLAVKIPEGD LIRGRVGTVG YMAPEVLNNQ
370 380 390 400
RYGLSPDYWG LGCLIYEMIE GQSPFRGRKE KVKREEVDRR
410 420 430 440
VLETEEVYSH KFSEEAKSIC KMLLTKDAKQ RLGCQEEEAA
450 460 470 480
EVKRHPFFRN MNFKRLEAGM LDPPFVPDPR AVYCKDVLDI
490 500 510 520
EQFSTVKGVN LDHTDDDFYS KFSTGSVSIP WQNEMIETEC
530 540 550 560
FKELNVFGPN GTLPPDLNRN HPPeppkkgl lqrlfkrqhq
570 580 590
nnsksspssk tsfnhhinsn hvssnstgss
Lower-case residues are disordered in structure.
Mutations: None
Phosphorylation: None