4PRJ

AURKA (Aurora kinase A)
Group: CAMK
Uniprot: AURKA_HUMAN
Organism: Homo sapiens
Domain boundary: 133 - 383
Resolu: 2.8

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Inactive DFGin None in-in in-out 2VU Type1 125 - 388 10
Representative sequence - Chain A
132 142 152 162
maKRQWALED FEIGRPLGKG kfgNVYLARE KNSKFILALK
172 182 192 202
VLFKAQLEKA GVEHQLRREV EIQSHLRHPN ILRLYGYFHD
212 222 232 242
STRVYLILEY APLGTVYREL QKLSKFDEQR TATYITELAN
252 262 272 282
ALSYCHSKKV IHRDIKPENL LLGSAGELKI ADFGWSVhap
292 302 312 322
ssrraalCGT LDYLPPEMIE GRMHDEKVDL WSLGVLCYEF
332 342 352 362
LVGKPPFEAN TYQDTYKRIS RVEFTFPDFV TEGARDLISR
372 382
LLKHNPSQRP MLREVLEHPW ITANSSkps
Lower-case residues are disordered in structure.
Mutations: K124A,Q154N,A203S,R251K,T287A,T288A,E336D
Phosphorylation: None