3R21

AURKA (Aurora kinase A)
Group: CAMK
Uniprot: AURKA_HUMAN
Organism: Homo sapiens
Domain boundary: 133 - 383
Resolu: 2.9

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Inactive DFGin BLAminus out-out in-out D36 Type1 127 - 389 9
Representative sequence - Chain A
130 140 150 160
gplgsrQWAL EDFEIGRPLG KGKFGNVYLA REKQSKFILA
170 180 190 200
LKVLFKAQLE KAGVEHQLRR EVEIQSHLRH PNILRLYGYF
210 220 230 240
HDATRVYLIL EYAPLGTVYR ELQKLSKFDE QRTATYITEL
250 260 270 280
ANALSYCHSK RVIHRDIKPE NLLLGSAGEL KIADFGWSVh
290 300 310 320
apssrrddLC GTLDYLPPEM IEGRMHDEKV DLWSLGVLCY
330 340 350 360
EFLVGKPPFE ANTYQETYKR ISRVEFTFPD FVTEGARDLI
370 380 390
SRLLKHNPSQ RPMLREVLEH PWITANSSKp s
Lower-case residues are disordered in structure.
Mutations: T287D,T288D
Phosphorylation: None