1UU9

PDPK1 (3-phosphoinositide-dependent protein kinase 1)
Group: AGC
Uniprot: PDPK1_HUMAN
Organism: Homo sapiens
Domain boundary: 82 - 342
Resolu: 1.95

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in BI3 Type1 72 - 357 9
Representative sequence - Chain A
81 91 101 111
PQPRKKRPED FKFGKILGEG SFSTVVLARE LATSREYAIK
121 131 141 151
ILEKRHIIKE NKVPYVTRER DVMSRLDHPF FVKLYFTFQD
161 171 181 191
DEKLYFGLSY AKNGELLKYI RKIGSFDETC TRFYTAEIVS
201 211 221 231
ALEYLHGKGI IHRDLKPENI LLNEDMHIQI TDFGTAKVLs
241 251 261 271
peskqaraNS FVGTAQYVSP ELLTEKSACK SSDLWALGCI
281 291 301 311
IYQLVAGLPP FRAGNEYLIF QKIIKLEYDF PEKFFPKARD
321 331 341 351
LVEKLLVLDA TKRLGCEEME GYGPLKAHPF FESVTWENLH

QQTPPK
Lower-case residues are disordered in structure.
Mutations: None
Phosphorylation: X241