1H1W

PDPK1 (3-phosphoinositide-dependent protein kinase 1)
Group: AGC
Uniprot: PDPK1_HUMAN
Organism: Homo sapiens
Domain boundary: 82 - 342
Resolu: 2.0

Chain id Activity_label Spatial_label Dihedral_label Chelix-SaltBridge ActLoopNT-ActLoopCT Ligand Type Residues in structure Unresolved residues in A-loop
A Active DFGin BLAminus in-in in-in ATP Type1 71 - 359 4
Representative sequence - Chain A
80 90 100 110
PPQPRKKRPE DFKFGKILGE GSFSTVVLAR ELATSREYAI
120 130 140 150
KILEKRHIIK ENKVPYVTRE RDVMSRLDHP FFVKLYFTFQ
160 170 180 190
DDEKLYFGLS YAKNGELLKY IRKIGSFDET CTRFYTAEIV
200 210 220 230
SALEYLHGKG IIHRDLKPEN ILLNEDMHIQ ITDFGTAKVL
240 250 260 270
SPeskqARAN SFVGTAQYVS PELLTEKSAC KSSDLWALGC
280 290 300 310
IIYQLVAGLP PFRAGNEYLI FQKIIKLEYD FPEKFFPKAR
320 330 340 350
DLVEKLLVLD ATKRLGCEEM EGYGPLKAHP FFESVTWENL

HQQTPPKLT
Lower-case residues are disordered in structure.
Mutations: None
Phosphorylation: X241