| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK6 | GRK6_HUMAN | AF-P43250-K1A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.2157 | 12.749 | BLAminus | -123.11, -178.58 | 47.67, 74.06 | -87.65, 23.59 | 291.93, 77.77 | -58.68, -35.83 | in-in | in | 8.7118 | Saltbr-in | 2.6653 | HRD-in | -82.84, -44.36 | 66.32, 2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9261 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.32, 157.5 | APE9-dihe-na | 121.0, 172.74 | APE8-dihe-in | -78.3, 135.32 | APE8-rot-in | 301.62 | APE67-dihe-inflip | 93.32, -20.35 | -55.72, 131.85 | APE12-dist-in | 10.366 | APE11-dist-in | 12.1373 | APE10-dist-in | 6.1395 | APE9-dist-in | 3.4895 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K1 | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| AGC | GRK6 | GRK6_HUMAN | AF-P43250-K3A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.0455 | 12.2821 | BLAminus | -130.79, 178.36 | 51.08, 64.04 | -74.31, 18.83 | 302.42, 178.07 | -60.87, -31.76 | in-in | in | 8.6239 | Saltbr-in | 2.6188 | HRD-in | -87.79, -47.34 | 67.55, 3.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9098 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.34, 159.69 | APE9-dihe-na | 109.39, -175.73 | APE8-dihe-in | -92.28, 133.79 | APE8-rot-in | 298.55 | APE67-dihe-inflip | 96.49, -17.7 | -57.25, 129.59 | APE12-dist-in | 10.5252 | APE11-dist-in | 11.9519 | APE10-dist-in | 5.9894 | APE9-dist-in | 3.1921 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K3 | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK6 | GRK6_HUMAN | AF-P43250-K1A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.2157 | 12.749 | BLAminus | -123.11, -178.58 | 47.67, 74.06 | -87.65, 23.59 | 291.93, 77.77 | -58.68, -35.83 | in-in | in | 8.7118 | Saltbr-in | 2.6653 | HRD-in | -82.84, -44.36 | 66.32, 2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9261 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.32, 157.5 | APE9-dihe-na | 121.0, 172.74 | APE8-dihe-in | -78.3, 135.32 | APE8-rot-in | 301.62 | APE67-dihe-inflip | 93.32, -20.35 | -55.72, 131.85 | APE12-dist-in | 10.366 | APE11-dist-in | 12.1373 | APE10-dist-in | 6.1395 | APE9-dist-in | 3.4895 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K1 | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| AGC | GRK6 | GRK6_HUMAN | AF-P43250-K3A | P43250 | 178 | 456 | 576.0 | No_ligand | No_ligand | Active | DFGin | 6.0455 | 12.2821 | BLAminus | -130.79, 178.36 | 51.08, 64.04 | -74.31, 18.83 | 302.42, 178.07 | -60.87, -31.76 | in-in | in | 8.6239 | Saltbr-in | 2.6188 | HRD-in | -87.79, -47.34 | 67.55, 3.73 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9098 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.34, 159.69 | APE9-dihe-na | 109.39, -175.73 | APE8-dihe-in | -92.28, 133.79 | APE8-rot-in | 298.55 | APE67-dihe-inflip | 96.49, -17.7 | -57.25, 129.59 | APE12-dist-in | 10.5252 | APE11-dist-in | 11.9519 | APE10-dist-in | 5.9894 | APE9-dist-in | 3.1921 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P43250-K3 | Homo sapiens | AGC_GRK6_HUMAN | AGC | 2.2e-86 | 295.0 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 6 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|