| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK5 | GRK5_HUMAN | AF-P34947-K1A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 5.488 | 12.6736 | BLAminus | -115.97, -177.38 | 48.25, 67.07 | -77.66, 16.16 | 284.97, 107.27 | -63.58, -32.29 | in-in | in | 8.9664 | Saltbr-in | 2.674 | HRD-in | -81.4, -44.95 | 66.95, -1.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.35, 159.3 | APE9-dihe-na | 118.39, -174.52 | APE8-dihe-in | -94.59, 137.57 | APE8-rot-in | 303.09 | APE67-dihe-inflip | 95.72, -15.07 | -56.34, 127.54 | APE12-dist-in | 10.5047 | APE11-dist-in | 12.2476 | APE10-dist-in | 6.2146 | APE9-dist-in | 3.7811 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K1 | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | GRK5 | GRK5_HUMAN | AF-P34947-K3A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 6.0217 | 12.0992 | BLAminus | -130.04, 178.69 | 50.56, 62.08 | -71.61, 20.06 | 306.44, 6.94 | -60.07, -35.44 | in-in | in | 8.5425 | Saltbr-in | 2.6154 | HRD-in | -88.42, -48.64 | 68.04, 5.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9566 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.09, 156.11 | APE9-dihe-na | 120.9, -174.14 | APE8-dihe-in | -94.05, 138.77 | APE8-rot-in | 297.52 | APE67-dihe-inflip | 92.74, -12.69 | -58.9, 127.55 | APE12-dist-in | 10.5409 | APE11-dist-in | 11.9762 | APE10-dist-in | 5.9613 | APE9-dist-in | 3.3122 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K3 | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK5 | GRK5_HUMAN | AF-P34947-K1A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 5.488 | 12.6736 | BLAminus | -115.97, -177.38 | 48.25, 67.07 | -77.66, 16.16 | 284.97, 107.27 | -63.58, -32.29 | in-in | in | 8.9664 | Saltbr-in | 2.674 | HRD-in | -81.4, -44.95 | 66.95, -1.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8959 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.35, 159.3 | APE9-dihe-na | 118.39, -174.52 | APE8-dihe-in | -94.59, 137.57 | APE8-rot-in | 303.09 | APE67-dihe-inflip | 95.72, -15.07 | -56.34, 127.54 | APE12-dist-in | 10.5047 | APE11-dist-in | 12.2476 | APE10-dist-in | 6.2146 | APE9-dist-in | 3.7811 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K1 | Homo sapiens | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| AGC | GRK5 | GRK5_HUMAN | AF-P34947-K3A | P34947 | 178 | 456 | 590.0 | No_ligand | No_ligand | Active | DFGin | 6.0217 | 12.0992 | BLAminus | -130.04, 178.69 | 50.56, 62.08 | -71.61, 20.06 | 306.44, 6.94 | -60.07, -35.44 | in-in | in | 8.5425 | Saltbr-in | 2.6154 | HRD-in | -88.42, -48.64 | 68.04, 5.72 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9566 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -129.09, 156.11 | APE9-dihe-na | 120.9, -174.14 | APE8-dihe-in | -94.05, 138.77 | APE8-rot-in | 297.52 | APE67-dihe-inflip | 92.74, -12.69 | -58.9, 127.55 | APE12-dist-in | 10.5409 | APE11-dist-in | 11.9762 | APE10-dist-in | 5.9613 | APE9-dist-in | 3.3122 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[186, 448]] | 1.0 | AF-P34947-K3 | Homo sapiens | AGC_GRK5_HUMAN | AGC | 6e-85 | 290.4 | 1.0 | 260.0 | 260.0 | 328 | 329 | 330 | 332 | 334 | 215 | 234 | 238 | 308 | 310 | 309 | 311.0 | 367 | 355 | 350 | 349 | 348 | 347 | 346 | 345 | 344 | 264 | G protein-coupled receptor kinase 5 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|