| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK4 | GRK4_HUMAN | AF-P32298-K1A | P32298 | 179 | 457 | 578.0 | No_ligand | No_ligand | Active | DFGin | 6.124 | 12.8326 | BLAminus | -120.03, -175.56 | 45.08, 74.96 | -87.72, 22.25 | 285.66, 73.41 | -59.0, -38.27 | in-in | in | 8.7678 | Saltbr-in | 2.6596 | HRD-in | -81.72, -44.96 | 67.52, -0.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8739 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.15, 151.54 | APE9-dihe-na | 127.86, 174.63 | APE8-dihe-in | -80.28, 134.89 | APE8-rot-in | 301.77 | APE67-dihe-inflip | 97.33, -20.86 | -54.78, 131.24 | APE12-dist-in | 10.4793 | APE11-dist-in | 12.2528 | APE10-dist-in | 6.2546 | APE9-dist-in | 3.5753 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[187, 449]] | 1.0 | AF-P32298-K1 | AGC_GRK4_HUMAN | AGC | 8.7e-85 | 289.8 | 1.0 | 260.0 | 260.0 | 329 | 330 | 331 | 333 | 335 | 216 | 235 | 239 | 309 | 311 | 310 | 312.0 | 368 | 356 | 351 | 350 | 349 | 348 | 347 | 346 | 345 | 265 | G protein-coupled receptor kinase 4 |
| AGC | GRK4 | GRK4_HUMAN | AF-P32298-K3A | P32298 | 179 | 457 | 578.0 | No_ligand | No_ligand | Active | DFGin | 6.0992 | 12.7677 | BLAminus | -126.56, 178.75 | 48.35, 61.02 | -72.83, 20.71 | 294.75, 76.46 | -64.12, -27.65 | in-in | in | 8.8853 | Saltbr-in | 2.619 | HRD-in | -85.16, -47.19 | 67.94, 0.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.923 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.65, 150.99 | APE9-dihe-na | 125.92, -171.45 | APE8-dihe-in | -98.43, 134.52 | APE8-rot-in | 298.92 | APE67-dihe-inflip | 98.38, -17.84 | -56.69, 129.66 | APE12-dist-in | 10.1996 | APE11-dist-in | 11.8575 | APE10-dist-in | 5.8719 | APE9-dist-in | 3.2346 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[187, 449]] | 1.0 | AF-P32298-K3 | AGC_GRK4_HUMAN | AGC | 8.7e-85 | 289.8 | 1.0 | 260.0 | 260.0 | 329 | 330 | 331 | 333 | 335 | 216 | 235 | 239 | 309 | 311 | 310 | 312.0 | 368 | 356 | 351 | 350 | 349 | 348 | 347 | 346 | 345 | 265 | G protein-coupled receptor kinase 4 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK4 | GRK4_HUMAN | AF-P32298-K1A | P32298 | 179 | 457 | 578.0 | No_ligand | No_ligand | Active | DFGin | 6.124 | 12.8326 | BLAminus | -120.03, -175.56 | 45.08, 74.96 | -87.72, 22.25 | 285.66, 73.41 | -59.0, -38.27 | in-in | in | 8.7678 | Saltbr-in | 2.6596 | HRD-in | -81.72, -44.96 | 67.52, -0.44 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8739 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.15, 151.54 | APE9-dihe-na | 127.86, 174.63 | APE8-dihe-in | -80.28, 134.89 | APE8-rot-in | 301.77 | APE67-dihe-inflip | 97.33, -20.86 | -54.78, 131.24 | APE12-dist-in | 10.4793 | APE11-dist-in | 12.2528 | APE10-dist-in | 6.2546 | APE9-dist-in | 3.5753 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[187, 449]] | 1.0 | AF-P32298-K1 | Homo sapiens | AGC_GRK4_HUMAN | AGC | 8.7e-85 | 289.8 | 1.0 | 260.0 | 260.0 | 329 | 330 | 331 | 333 | 335 | 216 | 235 | 239 | 309 | 311 | 310 | 312.0 | 368 | 356 | 351 | 350 | 349 | 348 | 347 | 346 | 345 | 265 | G protein-coupled receptor kinase 4 |
| AGC | GRK4 | GRK4_HUMAN | AF-P32298-K3A | P32298 | 179 | 457 | 578.0 | No_ligand | No_ligand | Active | DFGin | 6.0992 | 12.7677 | BLAminus | -126.56, 178.75 | 48.35, 61.02 | -72.83, 20.71 | 294.75, 76.46 | -64.12, -27.65 | in-in | in | 8.8853 | Saltbr-in | 2.619 | HRD-in | -85.16, -47.19 | 67.94, 0.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.923 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -132.65, 150.99 | APE9-dihe-na | 125.92, -171.45 | APE8-dihe-in | -98.43, 134.52 | APE8-rot-in | 298.92 | APE67-dihe-inflip | 98.38, -17.84 | -56.69, 129.66 | APE12-dist-in | 10.1996 | APE11-dist-in | 11.8575 | APE10-dist-in | 5.8719 | APE9-dist-in | 3.2346 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 279.0 | 279.0 | 0 | 27 | 27 | 0 | [[187, 449]] | 1.0 | AF-P32298-K3 | Homo sapiens | AGC_GRK4_HUMAN | AGC | 8.7e-85 | 289.8 | 1.0 | 260.0 | 260.0 | 329 | 330 | 331 | 333 | 335 | 216 | 235 | 239 | 309 | 311 | 310 | 312.0 | 368 | 356 | 351 | 350 | 349 | 348 | 347 | 346 | 345 | 265 | G protein-coupled receptor kinase 4 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|