| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIA | P11362 | 458 | 764 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.058 | 13.4362 | BLAplus | -111.91, 163.26 | 62.65, 26.85 | -80.22, -19.74 | 58.59, 88.0 | -94.12, 4.52 | in-in | in | 8.2512 | Saltbr-in | 2.8878 | HRD-in | -74.14, -50.3 | 78.02, -11.1 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.5114 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -88.77, 149.44 | APE9-dihe-in | -108.01, 98.39 | APE8-dihe-out | -63.46, -15.87 | APE8-rot-na | 3.35 | APE67-dihe-in | -71.69, -10.38 | -55.45, -26.93 | APE12-dist-na | 17.216 | APE11-dist-na | 19.6718 | APE10-dist-na | 16.6848 | APE9-dist-out | 11.0826 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | A | 310.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 9uhi | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIB | P11362 | 458 | 763 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.2132 | 12.7377 | BLAplus | -108.15, 164.77 | 66.41, 24.28 | -84.34, -17.16 | 58.96, 83.83 | -89.87, -8.4 | in-in | in | 7.7681 | Saltbr-in | 3.4492 | HRD-in | -77.39, -52.67 | 76.89, -15.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -74.45, 132.66 | APE9-dihe-in | -102.74, 93.19 | APE8-dihe-out | -60.68, -21.29 | APE8-rot-na | 332.28 | APE67-dihe-in | -72.11, -2.38 | -56.87, -27.58 | APE12-dist-na | 17.3515 | APE11-dist-na | 20.6822 | APE10-dist-na | 16.9654 | APE9-dist-out | 11.3637 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | B | 310.0 | 286.0 | 20 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 9uhi | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIA | P11362 | 458 | 764 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.058 | 13.4362 | BLAplus | -111.91, 163.26 | 62.65, 26.85 | -80.22, -19.74 | 58.59, 88.0 | -94.12, 4.52 | in-in | in | 8.2512 | Saltbr-in | 2.8878 | HRD-in | -74.14, -50.3 | 78.02, -11.1 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.5114 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -88.77, 149.44 | APE9-dihe-in | -108.01, 98.39 | APE8-dihe-out | -63.46, -15.87 | APE8-rot-na | 3.35 | APE67-dihe-in | -71.69, -10.38 | -55.45, -26.93 | APE12-dist-na | 17.216 | APE11-dist-na | 19.6718 | APE10-dist-na | 16.6848 | APE9-dist-out | 11.0826 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | A | 310.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 9uhi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 9UHIB | P11362 | 458 | 763 | 822.0 | A1EPF:60801 | Type1 | Inactive | DFGin | 5.2132 | 12.7377 | BLAplus | -108.15, 164.77 | 66.41, 24.28 | -84.34, -17.16 | 58.96, 83.83 | -89.87, -8.4 | in-in | in | 7.7681 | Saltbr-in | 3.4492 | HRD-in | -77.39, -52.67 | 76.89, -15.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -74.45, 132.66 | APE9-dihe-in | -102.74, 93.19 | APE8-dihe-out | -60.68, -21.29 | APE8-rot-na | 332.28 | APE67-dihe-in | -72.11, -2.38 | -56.87, -27.58 | APE12-dist-na | 17.3515 | APE11-dist-na | 20.6822 | APE10-dist-na | 16.9654 | APE9-dist-out | 11.3637 | None | None | None | XRAY | 1.76 | 0.163 | 0.197 | B | 310.0 | 286.0 | 20 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 9uhi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|