| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 8XLOA | P11362 | 462 | 764 | 822.0 | A1LVQ:60801 | Type1.5_Back | Inactive | DFGin | 5.3499 | 13.4604 | BLAplus | -120.07, 167.95 | 56.19, 37.83 | -98.04, 4.56 | 56.68, 90.6 | -112.93, 25.35 | in-in | in | 7.9829 | Saltbr-in | 3.258 | HRD-out | -75.5, 142.74 | -82.57, -37.38 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.2004 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -113.57, 158.46 | APE9-dihe-in | -97.47, 110.21 | APE8-dihe-out | -58.39, -18.54 | APE8-rot-na | 19.21 | APE67-dihe-in | -81.65, 0.42 | -62.39, -18.82 | APE12-dist-na | 20.741 | APE11-dist-na | 21.9456 | APE10-dist-na | 20.2119 | APE9-dist-out | 11.7779 | C584S | None | None | XRAY | 2.36 | 0.21 | 0.255 | A | 310.0 | 293.0 | 10 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 8xlo | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 8XLOB | P11362 | 458 | 763 | 822.0 | A1LVQ:60801 | Type1.5_Back | Inactive | DFGin | 5.5876 | 13.1874 | BLAplus | -122.66, 168.69 | 59.17, 27.93 | -79.17, -12.14 | 48.47, 88.63 | -115.21, 3.75 | in-in | in | 7.7683 | Saltbr-in | 2.8826 | HRD-out | -89.09, 129.19 | -58.3, -36.38 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.09, 159.35 | APE9-dihe-in | -98.63, 108.84 | APE8-dihe-out | -54.34, -25.08 | APE8-rot-na | 331.75 | APE67-dihe-in | -70.85, 2.53 | -59.01, -24.97 | APE12-dist-na | 19.448 | APE11-dist-na | 20.7383 | APE10-dist-na | 19.2996 | APE9-dist-out | 11.7119 | C584S | None | None | XRAY | 2.36 | 0.21 | 0.255 | B | 310.0 | 287.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 8xlo | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 8XLOA | P11362 | 462 | 764 | 822.0 | A1LVQ:60801 | Type1.5_Back | Inactive | DFGin | 5.3499 | 13.4604 | BLAplus | -120.07, 167.95 | 56.19, 37.83 | -98.04, 4.56 | 56.68, 90.6 | -112.93, 25.35 | in-in | in | 7.9829 | Saltbr-in | 3.258 | HRD-out | -75.5, 142.74 | -82.57, -37.38 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.2004 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -113.57, 158.46 | APE9-dihe-in | -97.47, 110.21 | APE8-dihe-out | -58.39, -18.54 | APE8-rot-na | 19.21 | APE67-dihe-in | -81.65, 0.42 | -62.39, -18.82 | APE12-dist-na | 20.741 | APE11-dist-na | 21.9456 | APE10-dist-na | 20.2119 | APE9-dist-out | 11.7779 | C584S | None | None | XRAY | 2.36 | 0.21 | 0.255 | A | 310.0 | 293.0 | 10 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 8xlo | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 8XLOB | P11362 | 458 | 763 | 822.0 | A1LVQ:60801 | Type1.5_Back | Inactive | DFGin | 5.5876 | 13.1874 | BLAplus | -122.66, 168.69 | 59.17, 27.93 | -79.17, -12.14 | 48.47, 88.63 | -115.21, 3.75 | in-in | in | 7.7683 | Saltbr-in | 2.8826 | HRD-out | -89.09, 129.19 | -58.3, -36.38 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.09, 159.35 | APE9-dihe-in | -98.63, 108.84 | APE8-dihe-out | -54.34, -25.08 | APE8-rot-na | 331.75 | APE67-dihe-in | -70.85, 2.53 | -59.01, -24.97 | APE12-dist-na | 19.448 | APE11-dist-na | 20.7383 | APE10-dist-na | 19.2996 | APE9-dist-out | 11.7119 | C584S | None | None | XRAY | 2.36 | 0.21 | 0.255 | B | 310.0 | 287.0 | 19 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 8xlo | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|