| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8STGA | P21802 | 461 | 764 | 821.0 | WCJ:801 | Type1 | Inactive | DFGin | 5.5904 | 12.8883 | BLAplus | -145.36, 157.52 | 90.77, 4.11 | -67.5, -2.28 | 57.4, 70.91 | -126.28, 999.0 | in-out | in | 8.1835 | Saltbr-out | 4.6059 | HRD-out | -102.42, 117.61 | -61.0, -55.0 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -15.95 | APE9-dihe-in | -134.91, 146.08 | APE8-dihe-in | -92.36, 82.18 | APE8-rot-na | 24.23 | APE67-dihe-in | -66.95, -23.69 | -61.29, -38.8 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.9073 | None | None | None | XRAY | 3.79 | 0.307 | 0.311 | A | 317.0 | 277.0 | 27 | 30 | 13 | 17 | [[481, 759]] | 1.0 | 8stg | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8STGB | P21802 | 472 | 765 | 821.0 | WCJ:801 | Type1.5_Back | Inactive | DFGin | 5.7481 | 12.473 | None | -146.69, 51.17 | -166.05, 99.26 | -159.05, 129.25 | 42.24, 92.9 | -129.91, 121.06 | in-out | in | 7.5175 | Saltbr-out | 4.9612 | HRD-out | -109.82, 96.26 | -71.43, -48.73 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 71.23, -15.79 | APE9-dihe-in | -138.41, 153.88 | APE8-dihe-in | -76.95, 77.58 | APE8-rot-na | 30.06 | APE67-dihe-in | -68.25, -27.71 | -60.57, -41.19 | APE12-dist-na | 23.5958 | APE11-dist-na | 24.2264 | APE10-dist-na | 21.8134 | APE9-dist-in | 7.3025 | None | None | None | XRAY | 3.79 | 0.307 | 0.311 | B | 317.0 | 274.0 | 20 | 30 | 20 | 10 | [[481, 759]] | 1.0 | 8stg | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 8STGA | P21802 | 461 | 764 | 821.0 | WCJ:801 | Type1 | Inactive | DFGin | 5.5904 | 12.8883 | BLAplus | -145.36, 157.52 | 90.77, 4.11 | -67.5, -2.28 | 57.4, 70.91 | -126.28, 999.0 | in-out | in | 8.1835 | Saltbr-out | 4.6059 | HRD-out | -102.42, 117.61 | -61.0, -55.0 | out-none-none | SNConn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, -15.95 | APE9-dihe-in | -134.91, 146.08 | APE8-dihe-in | -92.36, 82.18 | APE8-rot-na | 24.23 | APE67-dihe-in | -66.95, -23.69 | -61.29, -38.8 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.9073 | None | None | None | XRAY | 3.79 | 0.307 | 0.311 | A | 317.0 | 277.0 | 27 | 30 | 13 | 17 | [[481, 759]] | 1.0 | 8stg | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 8STGB | P21802 | 472 | 765 | 821.0 | WCJ:801 | Type1.5_Back | Inactive | DFGin | 5.7481 | 12.473 | None | -146.69, 51.17 | -166.05, 99.26 | -159.05, 129.25 | 42.24, 92.9 | -129.91, 121.06 | in-out | in | 7.5175 | Saltbr-out | 4.9612 | HRD-out | -109.82, 96.26 | -71.43, -48.73 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 71.23, -15.79 | APE9-dihe-in | -138.41, 153.88 | APE8-dihe-in | -76.95, 77.58 | APE8-rot-na | 30.06 | APE67-dihe-in | -68.25, -27.71 | -60.57, -41.19 | APE12-dist-na | 23.5958 | APE11-dist-na | 24.2264 | APE10-dist-na | 21.8134 | APE9-dist-in | 7.3025 | None | None | None | XRAY | 3.79 | 0.307 | 0.311 | B | 317.0 | 274.0 | 20 | 30 | 20 | 10 | [[481, 759]] | 1.0 | 8stg | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.6e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|