| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8S18A | P10721 | 568 | 931 | 976.0 | A1H4U:61001 | Type2 | Inactive | DFGout | 14.3583 | 9.8464 | BBAminus | -136.5, 172.4 | -143.71, 96.71 | -74.26, -23.47 | 290.48, 134.1 | 43.91, -111.27 | in-in | in | 7.7684 | Saltbr-in | 2.8325 | HRD-in | -78.51, -51.56 | 81.82, -15.01 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.2359 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -125.06, 109.89 | APE9-dihe-in | -125.76, 152.89 | APE8-dihe-in | -81.62, 69.52 | APE8-rot-na | 33.63 | APE67-dihe-in | -66.18, -17.82 | -59.01, -39.86 | APE12-dist-na | 16.4919 | APE11-dist-na | 13.1016 | APE10-dist-na | 11.2511 | APE9-dist-in | 7.7736 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.1 | 0.194 | 0.218 | A | 327.0 | 286.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s18 | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S18B | P10721 | 578 | 931 | 976.0 | A1H4U:61001 | Type2 | Inactive | DFGout | 14.1082 | 9.4757 | BBAminus | -139.33, 158.91 | -137.25, 115.01 | -87.55, -17.15 | 295.29, 118.72 | 51.85, -119.38 | in-in | in | 7.955 | Saltbr-in | 2.7671 | HRD-in | -75.32, -56.82 | 85.0, -9.46 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.856 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -124.84, 113.28 | APE9-dihe-in | -126.85, 149.08 | APE8-dihe-in | -82.57, 70.64 | APE8-rot-na | 34.25 | APE67-dihe-in | -68.54, -17.43 | -60.68, -37.6 | APE12-dist-na | 16.6629 | APE11-dist-na | 13.3739 | APE10-dist-na | 11.5603 | APE9-dist-in | 7.7784 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.1 | 0.194 | 0.218 | B | 327.0 | 276.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s18 | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8S18A | P10721 | 568 | 931 | 976.0 | A1H4U:61001 | Type2 | Inactive | DFGout | 14.3583 | 9.8464 | BBAminus | -136.5, 172.4 | -143.71, 96.71 | -74.26, -23.47 | 290.48, 134.1 | 43.91, -111.27 | in-in | in | 7.7684 | Saltbr-in | 2.8325 | HRD-in | -78.51, -51.56 | 81.82, -15.01 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.2359 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -125.06, 109.89 | APE9-dihe-in | -125.76, 152.89 | APE8-dihe-in | -81.62, 69.52 | APE8-rot-na | 33.63 | APE67-dihe-in | -66.18, -17.82 | -59.01, -39.86 | APE12-dist-na | 16.4919 | APE11-dist-na | 13.1016 | APE10-dist-na | 11.2511 | APE9-dist-in | 7.7736 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.1 | 0.194 | 0.218 | A | 327.0 | 286.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s18 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S18B | P10721 | 578 | 931 | 976.0 | A1H4U:61001 | Type2 | Inactive | DFGout | 14.1082 | 9.4757 | BBAminus | -139.33, 158.91 | -137.25, 115.01 | -87.55, -17.15 | 295.29, 118.72 | 51.85, -119.38 | in-in | in | 7.955 | Saltbr-in | 2.7671 | HRD-in | -75.32, -56.82 | 85.0, -9.46 | in-out-in | SNCioi | out-in | ActLoopNT-out | 15.856 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -124.84, 113.28 | APE9-dihe-in | -126.85, 149.08 | APE8-dihe-in | -82.57, 70.64 | APE8-rot-na | 34.25 | APE67-dihe-in | -68.54, -17.43 | -60.68, -37.6 | APE12-dist-na | 16.6629 | APE11-dist-na | 13.3739 | APE10-dist-na | 11.5603 | APE9-dist-in | 7.7784 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 2.1 | 0.194 | 0.218 | B | 327.0 | 276.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s18 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|