| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8S16A | P10721 | 566 | 932 | 976.0 | STI:61001 | Type2 | Inactive | DFGout | 16.1561 | 10.6327 | BBAminus | -135.66, -175.47 | -146.5, 109.21 | -66.07, -39.1 | 278.01, 69.44 | 60.83, -124.1 | in-in | in | 7.9119 | Saltbr-in | 2.9645 | HRD-in | -69.14, -53.88 | 78.27, -9.6 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.0214 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.16, 109.76 | APE9-dihe-in | -124.4, 150.42 | APE8-dihe-in | -79.68, 69.89 | APE8-rot-na | 33.56 | APE67-dihe-in | -69.51, -13.06 | -61.98, -37.06 | APE12-dist-na | 16.4365 | APE11-dist-na | 13.1795 | APE10-dist-na | 11.1209 | APE9-dist-in | 7.7908 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.177 | 0.207 | A | 327.0 | 289.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s16 | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S16B | P10721 | 578 | 931 | 976.0 | STI:61001 | Type2 | Inactive | DFGout | 15.8879 | 10.5227 | BBAminus | -137.35, -173.79 | -154.74, 102.74 | -60.21, -39.63 | 280.81, 66.69 | 55.03, -114.07 | in-in | in | 7.8423 | Saltbr-in | 2.8528 | HRD-in | -70.27, -58.28 | 86.53, -13.22 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.1216 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.71, 104.25 | APE9-dihe-in | -123.97, 149.57 | APE8-dihe-in | -79.76, 65.91 | APE8-rot-na | 34.81 | APE67-dihe-in | -69.88, -14.71 | -57.96, -38.02 | APE12-dist-na | 17.0837 | APE11-dist-na | 13.8991 | APE10-dist-na | 11.4361 | APE9-dist-in | 7.9103 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.177 | 0.207 | B | 327.0 | 276.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s16 | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | KIT | KIT_HUMAN | 8S16A | P10721 | 566 | 932 | 976.0 | STI:61001 | Type2 | Inactive | DFGout | 16.1561 | 10.6327 | BBAminus | -135.66, -175.47 | -146.5, 109.21 | -66.07, -39.1 | 278.01, 69.44 | 60.83, -124.1 | in-in | in | 7.9119 | Saltbr-in | 2.9645 | HRD-in | -69.14, -53.88 | 78.27, -9.6 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.0214 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -116.16, 109.76 | APE9-dihe-in | -124.4, 150.42 | APE8-dihe-in | -79.68, 69.89 | APE8-rot-na | 33.56 | APE67-dihe-in | -69.51, -13.06 | -61.98, -37.06 | APE12-dist-na | 16.4365 | APE11-dist-na | 13.1795 | APE10-dist-na | 11.1209 | APE9-dist-in | 7.7908 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.177 | 0.207 | A | 327.0 | 289.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s16 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| TYR | KIT | KIT_HUMAN | 8S16B | P10721 | 578 | 931 | 976.0 | STI:61001 | Type2 | Inactive | DFGout | 15.8879 | 10.5227 | BBAminus | -137.35, -173.79 | -154.74, 102.74 | -60.21, -39.63 | 280.81, 66.69 | 55.03, -114.07 | in-in | in | 7.8423 | Saltbr-in | 2.8528 | HRD-in | -70.27, -58.28 | 86.53, -13.22 | in-out-in | SNCioi | out-in | ActLoopNT-out | 16.1216 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.71, 104.25 | APE9-dihe-in | -123.97, 149.57 | APE8-dihe-in | -79.76, 65.91 | APE8-rot-na | 34.81 | APE67-dihe-in | -69.88, -14.71 | -57.96, -38.02 | APE12-dist-na | 17.0837 | APE11-dist-na | 13.8991 | APE10-dist-na | 11.4361 | APE9-dist-in | 7.9103 | I563S,V569S,Y609Q,L631S,M651E,I662H,D768H,R804N,V825D,C844S,L890S,H894Y,L912D,L923D | None | None | XRAY | 1.85 | 0.177 | 0.207 | B | 327.0 | 276.0 | 0 | 30 | 30 | 0 | [[589, 926]] | 1.0 | 8s16 | Homo sapiens | TYR_KIT_HUMAN | TYR | 2.3e-104 | 354.3 | 1.0 | 261.0 | 261.0 | 809 | 810 | 811 | 813 | 815 | 623 | 640 | 644 | 789 | 791 | 790 | 792.0 | 851 | 839 | 834 | 833 | 832 | 831 | 830 | 829 | 828 | 671 | Mast/stem cell growth factor receptor Kit |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|