| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 8JMZA | P11362 | 460 | 765 | 822.0 | UKI:60801 | Type1 | Inactive | DFGin | 5.1589 | 13.2886 | BLAplus | -113.58, 162.96 | 62.0, 28.58 | -83.36, -13.84 | 56.58, 89.17 | -102.65, 12.75 | in-in | in | 7.8587 | Saltbr-in | 2.8351 | HRD-in | -72.3, -51.47 | 78.17, -4.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9805 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -88.22, 148.56 | APE9-dihe-in | -107.32, 99.52 | APE8-dihe-out | -56.46, -18.86 | APE8-rot-na | 328.17 | APE67-dihe-in | -74.96, -9.03 | -56.04, -27.86 | APE12-dist-na | 16.4248 | APE11-dist-na | 18.9969 | APE10-dist-na | 16.2227 | APE9-dist-out | 11.0211 | C584S | None | None | XRAY | 1.988 | 0.166 | 0.205 | A | 310.0 | 306.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 8jmz | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 8JMZB | P11362 | 458 | 763 | 822.0 | UKI:60801 | Type1 | Inactive | DFGin | 5.259 | 13.0071 | BLAplus | -114.88, 158.62 | 61.68, 33.22 | -84.25, -18.02 | 53.38, 88.43 | -92.93, -0.34 | in-in | in | 7.7668 | Saltbr-in | 2.9243 | HRD-in | -72.45, -50.78 | 74.31, -4.23 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3535 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -137.73, 168.34 | APE9-dihe-in | -103.17, 113.28 | APE8-dihe-out | -51.14, -25.22 | APE8-rot-na | 328.21 | APE67-dihe-in | -74.28, -2.47 | -57.8, -24.89 | APE12-dist-na | 20.439 | APE11-dist-na | 21.4008 | APE10-dist-na | 20.0649 | APE9-dist-out | 11.5011 | C584S | None | None | XRAY | 1.988 | 0.166 | 0.205 | B | 310.0 | 290.0 | 16 | 30 | 27 | 3 | [[478, 756]] | 1.0 | 8jmz | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 8JMZA | P11362 | 460 | 765 | 822.0 | UKI:60801 | Type1 | Inactive | DFGin | 5.1589 | 13.2886 | BLAplus | -113.58, 162.96 | 62.0, 28.58 | -83.36, -13.84 | 56.58, 89.17 | -102.65, 12.75 | in-in | in | 7.8587 | Saltbr-in | 2.8351 | HRD-in | -72.3, -51.47 | 78.17, -4.24 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9805 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -88.22, 148.56 | APE9-dihe-in | -107.32, 99.52 | APE8-dihe-out | -56.46, -18.86 | APE8-rot-na | 328.17 | APE67-dihe-in | -74.96, -9.03 | -56.04, -27.86 | APE12-dist-na | 16.4248 | APE11-dist-na | 18.9969 | APE10-dist-na | 16.2227 | APE9-dist-out | 11.0211 | C584S | None | None | XRAY | 1.988 | 0.166 | 0.205 | A | 310.0 | 306.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 8jmz | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 8JMZB | P11362 | 458 | 763 | 822.0 | UKI:60801 | Type1 | Inactive | DFGin | 5.259 | 13.0071 | BLAplus | -114.88, 158.62 | 61.68, 33.22 | -84.25, -18.02 | 53.38, 88.43 | -92.93, -0.34 | in-in | in | 7.7668 | Saltbr-in | 2.9243 | HRD-in | -72.45, -50.78 | 74.31, -4.23 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3535 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -137.73, 168.34 | APE9-dihe-in | -103.17, 113.28 | APE8-dihe-out | -51.14, -25.22 | APE8-rot-na | 328.21 | APE67-dihe-in | -74.28, -2.47 | -57.8, -24.89 | APE12-dist-na | 20.439 | APE11-dist-na | 21.4008 | APE10-dist-na | 20.0649 | APE9-dist-out | 11.5011 | C584S | None | None | XRAY | 1.988 | 0.166 | 0.205 | B | 310.0 | 290.0 | 16 | 30 | 27 | 3 | [[478, 756]] | 1.0 | 8jmz | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|