| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 8BZPA | P53779 | 46 | 400 | 464.0 | SWM:501,C15:512 | Type1,Allosteric | Inactive | DFGin | 3.9487 | 13.914 | ABAminus | -89.43, -27.22 | -142.11, 175.41 | -118.21, 7.54 | 305.21, 97.74 | 61.64, -136.69 | in-none | in | 9.3247 | Saltbr-none | 999.0 | HRD-in | -70.92, -54.64 | 68.45, -3.99 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 5.6131 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_onno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 153.19 | APE8-dihe-in | -106.65, 112.81 | APE8-rot-in | 284.72 | APE67-dihe-in | -67.36, -13.74 | -110.92, 6.88 | APE12-dist-out | 16.0093 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.8464 | None | None | None | XRAY | 1.86 | 0.19 | 0.216 | A | 364.0 | 350.0 | 5 | 27 | 22 | 5 | [[64, 359]] | 1.0 | 8bzp | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.1 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 8BZPB | P53779 | 47 | 400 | 464.0 | SWM:502,C15:509,C15:510 | Type1,Type1,Allosteric | Inactive | DFGin | 3.8943 | 14.3724 | ABAminus | -88.61, -25.41 | -141.39, 172.54 | -107.56, 12.73 | 298.48, 92.43 | 76.94, -166.0 | in-out | in | 9.4701 | Saltbr-out | 3.7104 | HRD-in | -75.07, -55.95 | 68.9, 0.04 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 128.71 | APE8-rot-out | 62.47 | APE67-dihe-in | -67.38, -8.49 | -119.38, 11.72 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.86 | 0.19 | 0.216 | B | 364.0 | 326.0 | 19 | 27 | 12 | 15 | [[64, 359]] | 1.0 | 8bzp | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.1 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 8BZPA | P53779 | 46 | 400 | 464.0 | SWM:501,C15:512 | Type1,Allosteric | Inactive | DFGin | 3.9487 | 13.914 | ABAminus | -89.43, -27.22 | -142.11, 175.41 | -118.21, 7.54 | 305.21, 97.74 | 61.64, -136.69 | in-none | in | 9.3247 | Saltbr-none | 999.0 | HRD-in | -70.92, -54.64 | 68.45, -3.99 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 5.6131 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_onno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 153.19 | APE8-dihe-in | -106.65, 112.81 | APE8-rot-in | 284.72 | APE67-dihe-in | -67.36, -13.74 | -110.92, 6.88 | APE12-dist-out | 16.0093 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.8464 | None | None | None | XRAY | 1.86 | 0.19 | 0.216 | A | 364.0 | 350.0 | 5 | 27 | 22 | 5 | [[64, 359]] | 1.0 | 8bzp | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.1 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 8BZPB | P53779 | 47 | 400 | 464.0 | SWM:502,C15:509,C15:510 | Type1,Type1,Allosteric | Inactive | DFGin | 3.8943 | 14.3724 | ABAminus | -88.61, -25.41 | -141.39, 172.54 | -107.56, 12.73 | 298.48, 92.43 | 76.94, -166.0 | in-out | in | 9.4701 | Saltbr-out | 3.7104 | HRD-in | -75.07, -55.95 | 68.9, 0.04 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | nonTYR | APEdihe_aanoi | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 128.71 | APE8-rot-out | 62.47 | APE67-dihe-in | -67.38, -8.49 | -119.38, 11.72 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.86 | 0.19 | 0.216 | B | 364.0 | 326.0 | 19 | 27 | 12 | 15 | [[64, 359]] | 1.0 | 8bzp | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.1 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|